Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 4425
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Graphical contents list| 2006
- 4440
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Selective COX-2 inhibitors. Part 1: Synthesis and biological evaluation of phenylazobenzenesulfonamidesTsai, Wei-Jern / Shiao, Young-Ji / Lin, Shwu-Jiuan et al. | 2006
- 4444
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Tri-substituted triazoles as potent non-nucleoside inhibitors of the HIV-1 reverse transcriptaseDe La Rosa, Martha / Kim, Hong Woo / Gunic, Esmir et al. | 2006
- 4450
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Synthesis and structure–activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 1Rowbottom, Martin W. / Vickers, Troy D. / Dyck, Brian et al. | 2006
- 4458
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Structure of a new cyclic nonapeptide, segetalin F, and vasorelaxant activity of segetalins from Vaccaria segetalisMorita, Hiroshi / Eda, Michiko / Iizuka, Toru et al. | 2006
- 4462
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Tetrahydrofluorenones with conformationally restricted side chains as selective estrogen receptor beta ligandsWildonger, Kenneth J. / Ratcliffe, Ronald W. / Mosley, Ralph T. et al. | 2006
- 4467
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Comparative QSAR modeling of CCR5 receptor binding affinity of substituted 1-(3,3-diphenylpropyl)-piperidinyl amides and ureasThomas Leonard, J. / Roy, Kunal et al. | 2006
- 4475
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Metabolism investigation leading to novel drug design 2: Orally active prostacyclin mimetics. Part 5Takamura, Fujiko / Tanaka, Akira / Takasugi, Hisashi et al. | 2006
- 4479
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An efficient one-pot synthesis of octahydroquinazolinone derivatives using catalytic amount of H2SO4 in waterHassani, Zahra / Islami, Mohammad Reza / Kalantari, Maryam et al. | 2006
- 4483
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Design and synthesis of new water-soluble tetrazolide derivatives of celecoxib and rofecoxib as selective cyclooxygenase-2 (COX-2) inhibitorsNavidpour, Latifeh / Amini, Mohsen / Shafaroodi, Hamed et al. | 2006
- 4488
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Fluorogenic ester substrates to assess proteolytic activityMugherli, Laurent / Burchak, Olga N. / Chatelain, François et al. | 2006
- 4492
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Development of first photoresponsive prodrug of paclitaxelSkwarczynski, Mariusz / Noguchi, Mayo / Hirota, Shun et al. | 2006
- 4497
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Cyclopentane-based human NK1 antagonists. Part 1: Discovery and initial SARFinke, Paul E. / Meurer, Laura C. / Levorse, Dorothy A. et al. | 2006
- 4504
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Cyclopentane-based human NK1 antagonists. Part 2: Development of potent, orally active, water-soluble derivativesMeurer, Laura C. / Finke, Paul E. / Owens, Karen A. et al. | 2006
- 4512
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Antifungal anthraquinones from Saprosma fragransSingh, D.N. / Verma, N. / Raghuwanshi, S. et al. | 2006
- 4515
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Synthesis of a red-shifted fluorescence polarization probe for Hsp90Moulick, Kamalika / Clement, Cristina C. / Aguirre, Julia et al. | 2006
- 4519
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Synthesis, biochemical evaluation and rationalisation of the inhibitory activity of a series of 4-hydroxyphenyl ketones as potential inhibitors of 17b-hydroxysteroid dehydrogenase type 3 (17b-HSD3)Lota, Rupinder K. et al. | 2006
- 4519
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Synthesis, biochemical evaluation and rationalisation of the inhibitory activity of a series of 4-hydroxyphenyl ketones as potential inhibitors of 17β-hydroxysteroid dehydrogenase type 3 (17β-HSD3)Lota, Rupinder K. / Dhanani, Sachin / Owen, Caroline P. et al. | 2006
- 4523
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Dual-acting agents that possess free radical scavenging and antithrombotic activities: Design, synthesis, and evaluation of phenolic tetrahydro-b-carboline RGD peptide conjugatesBi, Wei et al. | 2006
- 4523
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Dual-acting agents that possess free radical scavenging and antithrombotic activities: Design, synthesis, and evaluation of phenolic tetrahydro-β-carboline RGD peptide conjugatesBi, Wei / Bi, Lanrong / Cai, Jianhui et al. | 2006
- 4528
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Studies towards the conception of new selective PPARβ/δ ligandsEkambomé Basséne, Carine / Suzenet, Franck / Hennuyer, Nathalie et al. | 2006
- 4528
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Studies towards the conception of new selective PPARb-δ ligandsEkambomé Basséne, Carine et al. | 2006
- 4528
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Studies towards the conception of new selective PPARb/d ligandsEkambome Bassene, C. / Suzenet, F. / Hennuyer, N. et al. | 2006
- 4533
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N-Tetrahydroquinolinyl, N-quinolinyl and N-isoquinolinyl biaryl carboxamides as antagonists of TRPV1Westaway, Susan M. / Chung, Ying-Kit / Davis, John B. et al. | 2006
- 4537
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Antibacterial activity of pyrrolopyridine-substituted oxazolidinones: synthesis and in vitro SAR of various C-5 acetamide replacementsPaget, Steven D. / Boggs, Christine M. / Foleno, Barbara D. et al. | 2006
- 4543
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Hydrazides of clozapine: A new class of D1 dopamine receptor subtype selective antagonistsSasikumar, T.K. / Burnett, D.A. / Zhang, H. et al. | 2006
- 4548
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Modification of the clozapine structure by parallel synthesisSu, Jing / Tang, Haiqun / McKittrick, Brian A. et al. | 2006
- 4554
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Discovery and structure–activity relationship of 2-phenyl-oxazole-4-carboxamide derivatives as potent apoptosis inducersTai, Vincent W.-F. / Sperandio, David / Shelton, Emma J. et al. | 2006
- 4559
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Synthesis and immunostimulatory activity of 8-substituted amino 9-benzyladenines as potent Toll-like receptor 7 agonistsJin, Guangyi / Wu, Christina C.N. / Tawatao, Rommel I. et al. | 2006
- 4564
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An expedient synthesis of N6-substituted-5′-modified adenosinesAshton, T.D. / Scammells, Peter J. et al. | 2006
- 4564
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An expedient synthesis of N6-substituted-5prime-modified adenosinesAshton, T. D. / Scammells, P. J. et al. | 2006
- 4567
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Potent 4-amino-5-azaindole factor VIIa inhibitorsHu, Huiyong / Kolesnikov, Aleksandr / Riggs, Jennifer R. et al. | 2006
- 4571
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Synthesis and evaluation of phenoxy acetic acid derivatives as anti-mycobacterial agentsyar, Mohammad Shahar / Siddiqui, Anees Ahmad / Ali, Mohamed Ashraf et al. | 2006
- 4575
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Tubeimoside V (1), a new cyclic bisdesmoside from tubers of Bolbostemma paniculatum, functions by inducing apoptosis in human glioblastoma U87MG cellsCheng, Guang / Zhang, Yun / Zhang, Xiang et al. | 2006
- 4581
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Synthesis and pharmacological study of novel pyrido-quinazolone analogues as anti-fungal, antibacterial, and anticancer agentsTiwari, Anjani K. / Mishra, A.K. / Bajpai, Aruna et al. | 2006
- 4586
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Two novel immunosuppressive pregnane glycosides from the roots of Stephanotis mucronataYe, Yiping / Chen, Fengyang / Sun, Hongxiang et al. | 2006
- 4592
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A practical and green approach toward synthesis of N3-substituted dihydropyrimidinones: Using Aza-Michael addition reaction catalyzed by KF/Al2O3Wang, Xicun / Quan, Zhengjun / Wang, Jun-Ke et al. | 2006
- 4596
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Synthesis and anti-angiogenesis activity of coumarin derivativesLee, Seokjoon / Sivakumar, Krishnamoorthy / Shin, Woon-Seob et al. | 2006
- 4600
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A novel iNOS and COX-2 inhibitor from the aerial parts of Rodgersia podophyllaChin, Young-Won / Park, Eun Young / Seo, Seung-Yong et al. | 2006
- 4603
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Synthesis of gallic acid based naphthophenone fatty acid amides as cathepsin D inhibitorsSrivastava, Vandana / Saxena, Hari Om / Shanker, Karuna et al. | 2006
- 4609
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Vasorelaxant activity of cyclic peptide, cyclosquamosin B, from Annona squamosaMorita, Hiroshi / Iizuka, Toru / Choo, Chee-Yan et al. | 2006
- 4612
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Synthesis of novel keto-ACE analogues as domain-selective angiotensin I-converting enzyme inhibitorsNchinda, Aloysius T. / Chibale, Kelly / Redelinghuys, Pierre et al. | 2006
- 4616
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Synthesis and molecular modeling of a lisinopril–tryptophan analogue inhibitor of angiotensin I-converting enzymeNchinda, Aloysius T. / Chibale, Kelly / Redelinghuys, Pierre et al. | 2006
- 4620
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3-Aryl-4-hydroxyquinolin-2(1H)-one derivatives as type I fatty acid synthase inhibitorsRivkin, Alexey / Kim, Yoona R. / Goulet, Mark T. et al. | 2006
- 4624
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Hepatoprotective activity of Schouwia thebica webbAwaad, Amani, S. / Maitland, D.J. / Soliman, G.A. et al. | 2006
- 4629
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Synthesis and evaluation of (2-phenethyl-2H-1,2,3-triazol-4-yl)(phenyl)methanones as Kv1.5 channel blockers for the treatment of atrial fibrillationBlass, Benjamin E. / Coburn, Keith / Lee, Wenlin et al. | 2006
- 4633
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Overcoming HERG affinity in the discovery of the CCR5 antagonist maravirocPrice, David A. / Armour, Duncan / de Groot, Marcel et al. | 2006
- 4638
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Benzimidazole-2-carboxamides as novel NR2B selective NMDA receptor antagonistsBorza, István / Kolok, Sándor / Gere, Anikó et al. | 2006
- 4641
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3,4-Dihydro-1H-[1,3]oxazino[4,5-c]acridines as a new family of cytotoxic drugsOuberai, Myriam / Asche, Christian / Carrez, Danièle et al. | 2006
- 4644
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Synthesis and anticonvulsant activity of new N-1′,N-3′-disubstituted-2′H,3H,5′H-spiro-(2-benzofuran-1,4′-imidazolidine)-2′,3,5′-trionesPatel, Hardik J. / Sarra, Joe / Caruso, Francesco et al. | 2006
- 4644
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Synthesis and anticonvulsant activity of new N-1prime,N-3prime-disubstituted-2primeH,3H,5primeH-spiro-(2-benzofuran-1,4prime-imidazolidine)-2prime,3,5prime-trionesPatel, H. J. / Sarra, J. / Caruso, F. et al. | 2006
- 4648
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The synthesis and nicotinic binding activity of (±)-epiquinamide and (±)-C(1)-epiepiquinamideKanakubo, Akira / Gray, Diane / Innocent, Neal et al. | 2006
- 4652
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Triazolo-tetrahydrofluorenones as selective estrogen receptor beta agonistsParker, Dann L. Jr. / Meng, Dongfang / Ratcliffe, Ronald W. et al. | 2006
- 4657
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Identification of small-molecule inhibitors of the Ab–ABAD interactionXie, Yuli et al. | 2006
- 4657
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Identification of small-molecule inhibitors of the Aβ–ABAD interactionXie, Yuli / Deng, Shixian / Chen, Zhenzhang et al. | 2006
- 4661
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Synthesis and monoamine transporter affinity of front bridged tricyclic 3b-(4prime-halo or 4prime-methyl)phenyltropanes bearing methylene or carbomethoxymethylene on the bridge to the 2b-positionZeng, F. / Jarkas, N. / Owens, M. J. et al. | 2006
- 4661
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Synthesis and monoamine transporter affinity of front bridged tricyclic 3b-(4′-halo or 4′-methyl)phenyltropanes bearing methylene or carbomethoxymethylene on the bridge to the 2b-positionZeng, Fanxing et al. | 2006
- 4661
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Synthesis and monoamine transporter affinity of front bridged tricyclic 3β-(4′-halo or 4′-methyl)phenyltropanes bearing methylene or carbomethoxymethylene on the bridge to the 2β-positionZeng, Fanxing / Jarkas, Nachwa / Owens, Michael J. et al. | 2006
- 4664
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High affinity inhibitors of the dopamine transporter (DAT): Novel biotinylated ligands for conjugation to quantum dotsTomlinson, Ian D. / Mason, John N. / Blakely, Randy D. et al. | 2006
- 4668
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Design and synthesis of potent and selective 1,3,4-trisubstituted-2-oxopiperazine based melanocortin-4 receptor agonistsTian, Xinrong / Mishra, Rajesh K. / Switzer, Adrian G. et al. | 2006
- 4674
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Arylpropionylpiperazines as antagonists of the human melanocortin-4 receptorJiang, Wanlong / Tucci, Fabio C. / Chen, Caroline W. et al. | 2006
- 4679
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Synthesis and in vitro evaluation of salvinorin A analogues: Effect of configuration at C(2) and substitution at C(18)Béguin, Cécile / Richards, Michele R. / Li, Jian-Guo et al. | 2006
- 4686
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Optimization and SAR for dual ErbB-1/ErbB-2 tyrosine kinase inhibition in the 6-furanylquinazoline seriesPetrov, Kimberly G. / Zhang, Yue-Mei / Carter, Malcolm et al. | 2006
- 4692
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Synthesis and antibacterial activity of C12 des-methyl ketolidesLin, Xiaodong / Rico, Alice C. / Chu, Daniel T. et al. | 2006
- 4697
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Small molecule inhibitors of IgE synthesisBrown, Alan / Henderson, Alan / Lane, Charlotte et al. | 2006
- 4700
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Corrigendum to "Development of N-2,4-pyrimidine-N-phenyl-Nprime-phenyl ureas as inhibitors of tumor necrosis factor alpha (TNF-a) synthesis. Part 1" [Bioorg. Med. Chem. Lett. 16 (2006) 3510-3513]Brugel, T. A. / Maier, J. A. / Clark, M. P. et al. | 2006
- 4700
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Corrigendum to “Development of N-2,4-pyrimidine-N-phenyl-N′-phenyl ureas as inhibitors of tumor necrosis factor alpha (TNF-α) synthesis. Part 1” [Bioorg. Med. Chem. Lett. 16 (2006) 3510–3513]Brugel, Todd A. / Maier, Jennifer A. / Clark, Michael P. et al. | 2006
- 4700
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Corrigendum to “Development of N-2,4-pyrimidine-N-phenyl-N′-phenyl ureas as inhibitors of tumor necrosis factor alpha (TNF-a) synthesis. Part 1” [Bioorg. Med. Chem. Lett. 16 (2006) 3510–3513]Brugel, Todd A. et al. | 2006
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Editorial board| 2006
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Instructions to contributors| 2006