Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 3517
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Graphical contents list| 2007
- 3531
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Design, docking, and synthesis of novel indeno[1,2-c]isoquinolines for the development of antitumor agents as topoisomerase I inhibitorsCho, Won-Jea / Le, Quynh Manh / My Van, Hue Thi et al. | 2007
- 3535
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Development of piperazine-tethered heterodimers as potent antimalarials against chloroquine-resistant P. falciparum strains. Synthesis and molecular modelingGemma, Sandra / Kukreja, Gagan / Campiani, Giuseppe et al. | 2007
- 3540
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Synthesis and antibacterial activity of 5-deoxy-5-episubstituted arbekacin derivativesHiraiwa, Yukiko / Usui, Takayuki / Akiyama, Yoshihisa et al. | 2007
- 3544
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Structure–activity relationships of SERMs optimized for uterine antagonism and ovarian safetyRichardson, Timothy I. / Frank, Scott A. / Wang, Minmin et al. | 2007
- 3550
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Novel inhibitors of VEGF receptors-1 and -2 based on azole-5-carboxamide templatesKiselyov, Alexander S. / Milligan, Daniel / Ouyang, Xiaohu et al. | 2007
- 3558
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Synthesis and SAR studies of potent imidazopyridine anticoccidial agentsLiang, Gui-Bai / Qian, Xiaoxia / Feng, Dennis et al. | 2007
- 3562
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Synthesis and SAR of thiophene containing kinesin spindle protein (KSP) inhibitorsPinkerton, Anthony B. / Lee, Tom T. / Hoffman, Timothy Z. et al. | 2007
- 3570
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Benzopyrans as selective estrogen receptor β agonists (SERBAs). Part 2: Structure–activity relationship studies on the benzopyran scaffoldRichardson, Timothy I. / Norman, Bryan H. / Lugar, Charles W. et al. | 2007
- 3570
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Benzopyrans as selective estrogen receptor b agonists (SERBAs). Part 2: Structure-activity relationship studies on the benzopyran scaffoldRichardson, T. I. / Norman, B. H. / Lugar, C. W. et al. | 2007
- 3575
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Discovery of 6-ethyl-2,4-diaminopyrimidine-based small molecule renin inhibitorsHolsworth, Daniel D. / Jalaie, Mehran / Belliotti, Thomas et al. | 2007
- 3581
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Radioiodinated aza-diphenylacetylenes as potential SPECT imaging agents for β-amyloid plaque detectionQu, Wenchao / Kung, Mei-Ping / Hou, Catherine et al. | 2007
- 3581
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Radioiodinated aza-diphenylacetylenes as potential SPECT imaging agents for b-amyloid plaque detectionQu, W. / Kung, M. P. / Hou, C. et al. | 2007
- 3585
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Carbonic anhydrase inhibitors: The b-carbonic anhydrase from Helicobacter pylori is a new target for sulfonamide and sulfamate inhibitorsNishimori, I. / Minakuchi, T. / Kohsaki, T. et al. | 2007
- 3585
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Carbonic anhydrase inhibitors: The β-carbonic anhydrase from Helicobacter pylori is a new target for sulfonamide and sulfamate inhibitorsNishimori, Isao / Minakuchi, Tomoko / Kohsaki, Takuhiro et al. | 2007
- 3595
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Design, synthesis, and structure–activity relationship of carbamate-tethered aryl propanoic acids as novel PPARα/γ dual agonistsKim, Nam-Jung / Lee, Kwang-Ok / Koo, Bon-Woong et al. | 2007
- 3595
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Design, synthesis, and structure-activity relationship of carbamate-tethered aryl propanoic acids as novel PPARa/g dual agonistsKim, N. J. / Lee, K. O. / Koo, B. W. et al. | 2007
- 3599
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A novel artemisinin–quinine hybrid with potent antimalarial activityWalsh, John J. / Coughlan, David / Heneghan, Nicola et al. | 2007
- 3603
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Evaluation of 4prime-substituted bicyclic pyridones as non-steroidal inhibitors of steroid 5a-reductaseMcCarthy, A. R. / Hartmann, R. W. / Abell, A. D. et al. | 2007
- 3603
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Evaluation of 4′-substituted bicyclic pyridones as non-steroidal inhibitors of steroid 5α-reductaseMcCarthy, Anna R. / Hartmann, Rolf W. / Abell, Andrew D. et al. | 2007
- 3608
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Bradykinin B1 antagonists: Biphenyl SAR studies in the cyclopropanecarboxamide seriesKuduk, Scott D. / DiPardo, Robert M. / Chang, Ronald K. et al. | 2007
- 3613
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Novel potent antimitotic heterocyclic ketones: Synthesis, antiproliferative activity, and structure–activity relationshipsHu, Laixing / Jiang, Jian-dong / Qu, Jinrong et al. | 2007
- 3618
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1,4-Dihydroindeno[1,2-c]pyrazoles as potent checkpoint kinase 1 inhibitors: Extended exploration on phenyl ring substitutions and preliminary ADME/PK studiesTong, Yunsong / Claiborne, Akiyo / Pyzytulinska, Magdalena et al. | 2007
- 3624
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Discovery of highly potent and selective benzyloxybenzyl-based peroxisome proliferator-activator receptor (PPAR) δ agonistsBratton, Larry D. / Filzen, Gary F. / Geyer, Andrew et al. | 2007
- 3624
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Discovery of highly potent and selective benzyloxybenzyl-based peroxisome proliferator-activator receptor (PPAR) d agonistsBratton, L. D. / Filzen, G. F. / Geyer, A. et al. | 2007
- 3630
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Synthesis and SAR of selective benzothiophene, benzofuran, and indole-based peroxisome proliferator-activated receptor d agonistsFilzen, G. F. / Bratton, L. / Cheng, X. M. et al. | 2007
- 3630
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Synthesis and SAR of selective benzothiophene, benzofuran, and indole-based peroxisome proliferator-activated receptor δ agonistsFilzen, Gary F. / Bratton, Larry / Cheng, Xue-Min et al. | 2007
- 3636
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3-Amino-1-alkyl-cyclopentane carboxamides as small molecule antagonists of the human and murine CC chemokine receptor 2Butora, Gabor / Jiao, Richard / Parsons, William H. et al. | 2007
- 3642
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Paclitaxel C-10 carbamates: Potential candidates for the treatment of neurodegenerative tauopathiesBallatore, Carlo / Hyde, Edward / Deiches, Robert F. et al. | 2007
- 3647
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Himbacine derived thrombin receptor antagonists: Discovery of a new tricyclic coreClasby, Martin C. / Chackalamannil, Samuel / Czarniecki, Michael et al. | 2007
- 3652
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Biaryl cannabinoid mimetics—Synthesis and structure–activity relationshipWorm, Karin / Zhou, Q. Jean / Stabley, Gabriel J. et al. | 2007
- 3657
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Highly potent growth hormone secretagoguesLu, Zhijian / Tata, James R. / Cheng, Kang et al. | 2007
- 3660
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Hit-to-lead studies on benzimidazole inhibitors of ITK: Discovery of a novel class of kinase inhibitorsSnow, Roger J. / Abeywardane, Asitha / Campbell, Scot et al. | 2007
- 3666
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Design, synthesis, and anti-HIV activity of 2prime,3prime-didehydro-2prime,3prime-dideoxyuridine (d4U), 2prime,3prime-dideoxyuridine (ddU) phosphoramidate `ProTide' derivativesMehellou, Y. / McGuigan, C. / Brancale, A. et al. | 2007
- 3666
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Design, synthesis, and anti-HIV activity of 2′,3′-didehydro-2′,3′-dideoxyuridine (d4U), 2′,3′-dideoxyuridine (ddU) phosphoramidate ‘ProTide’ derivativesMehellou, Youcef / McGuigan, Christopher / Brancale, Andrea et al. | 2007
- 3670
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A new class of histamine H3 receptor antagonists derived from ligand based designRoche, Olivier / Rodríguez Sarmiento, Rosa María et al. | 2007
- 3676
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Cytotoxic effects of C-glycosides in HOS and HeLa cell linesSanhueza, Carlos A. / Mayato, Carlos / Machı´n, Rubén P. et al. | 2007
- 3682
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Improvement of base selectivity and binding affinity by controlling hydrogen bonding motifs between nucleobases and isoxanthopterin: Application to the detection of T/C mutationRajendar, Burki / Sato, Yusuke / Nishizawa, Seiichi et al. | 2007
- 3686
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Synthesis and antifungal activities of new fluconazole analogues with azaheterocycle moietyLebouvier, Nicolas / Pagniez, Fabrice / Duflos, Muriel et al. | 2007
- 3690
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Synthesis and anthelmintic activity of cyclohexadepsipeptides with cyclohexylmethyl side chainsJeschke, Peter / Harder, Achim / Etzel, Winfried et al. | 2007
- 3696
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2-Phenyl-2,3-dihydro-1H-imidazo[1,2-b]pyrazole derivatives: New potent inhibitors of fMLP-induced neutrophil chemotaxisBruno, Olga / Brullo, Chiara / Bondavalli, Francesco et al. | 2007
- 3702
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Antitumor anthraquinones from an endophytic actinomycete Micromonospora lupini sp. nov.Igarashi, Yasuhiro / Trujillo, Martha E. / Martínez-Molina, Eustoquio et al. | 2007
- 3706
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Boswellic acids and glucosamine show synergistic effect in preclinical anti-inflammatory study in ratsSingh, Surjeet / Khajuria, Anamika / Taneja, Subhash Chandra et al. | 2007
- 3712
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Synthesis and anticonvulsant activity of 4-(2-(2,6-dimethylphenylamino)-2-oxoethylamino)-N-(substituted)butanamides: A pharmacophoric hybrid approachYogeeswari, Perumal / Sriram, Dharmarajan / Sahitya, Puppala et al. | 2007
- 3716
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Docking-based 3D-QSAR study for selectivity of DPP4, DPP8, and DPP9 inhibitorsKang, Nam Sook / Ahn, Jin Hee / Kim, Sung Soo et al. | 2007
- 3722
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Synthesis and structure–activity relationships of taxuyunnanine C derivatives as multidrug resistance modulator in MDR cancer cellsHasegawa, Toshiaki / Bai, Jiao / Dai, Jungui et al. | 2007
- 3729
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Structure–activity relationship, kinetic mechanism, and selectivity for a new class of ubiquitin C-terminal hydrolase-L1 (UCH-L1) inhibitorsMermerian, Ara H. / Case, April / Stein, Ross L. et al. | 2007
- 3733
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Synthesis and local anesthetic activity of fluoro-substituted imipramine and its analoguesLi, Wen / You, Qidong et al. | 2007
- 3736
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Synthesis and evaluation of isoxazole derivatives as lysophosphatidic acid (LPA) antagonistsYamamoto, Takashi / Fujita, Koichi / Asari, Sayaka et al. | 2007
- 3741
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Synthesis and biological evaluation of analogues of the anti-tumor alkaloid naamidine AAberle, Nicholas / Catimel, Jenny / Nice, Edouard C. et al. | 2007
- 3745
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Phosphonic acid analogs of GABA through reductive dealkylation of phosphonic diesters with lithium trialkylborohydridesChowdhury, Sarwat / Muni, Niraj J. / Greenwood, Nicholas P. et al. | 2007
- 3749
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N-(3-Triethoxysilylpropyl)-4-(Nprime-maleimidylmethyl)cyclohexanamide (TPMC): A heterobifunctional reagent for immobilization of oligonucleotides on glass surfaceMisra, A. et al. | 2007
- 3749
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N-(3-Triethoxysilylpropyl)-4-(N′-maleimidylmethyl)cyclohexanamide (TPMC): A heterobifunctional reagent for immobilization of oligonucleotides on glass surfaceMisra, Arvind et al. | 2007
- 3754
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Design and synthesis of novel hydantoin-containing melanin-concentrating hormone receptor antagonistsBalavoine, Fabrice / Malabre, Patrice / Alleaume, Thierry et al. | 2007
- 3760
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Optimization of triaryl bis-sulfones as cannabinoid-2 receptor ligandsLavey, Brian J. / Kozlowski, Joseph A. / Shankar, Bandarpalle B. et al. | 2007
- 3765
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Derivatives of oxoisoaporphine alkaloids: A novel class of selective acetylcholinesterase inhibitorsTang, Huang / Ning, Fang-Xian / Wei, Yong-Biao et al. | 2007
- 3769
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Synthesis and biological evaluation of (R)-N-(diarylmethylthio/sulfinyl)ethyl/propyl-piperidine-3-carboxylic acid hydrochlorides as novel GABA uptake inhibitorsZhang, Jiange / Zhang, Pei / Liu, Xianbo et al. | 2007
- 3774
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The crystal structures of copper(II), manganese(II), and nickel(II) complexes of a (Z)-2-hydroxy-N′-(2-oxoindolin-3-ylidene) benzohydrazide—potential antitumor agentsZhong, Xia / Wei, Hu-Lai / Liu, Wei-Sheng et al. | 2007
- 3774
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The crystal structures of copper(II), manganese(II), and nickel(II) complexes of a (Z)-2-hydroxy-Nprime-(2-oxoindolin-3-ylidene) benzohydrazide-potential antitumor agentsZhong, X. / Wei, H. L. / Liu, W. S. et al. | 2007
- 3778
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C(4)-alkyl substituted furanyl cyclobutenediones as potent, orally bioavailable CXCR2 and CXCR1 receptor antagonistsChao, Jianhua / Taveras, Arthur G. / Chao, Jianping et al. | 2007
- 3784
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Synthesis, bioactivity, theoretical and molecular docking study of 1-cyano-N-substituted-cyclopropanecarboxamide as ketol-acid reductoisomerase inhibitorLiu, Xing-Hai / Chen, Pei-Quan / Wang, Bao-Lei et al. | 2007
- 3789
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Ortho-azo substituted phenylboronic acids for colorimetric sugar sensorsEgawa, Yuya / Gotoh, Ryota / Niina, Satoshi et al. | 2007
- 3793
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Design, synthesis, and binding studies of bidentate Zn-chelating peptidic inhibitors of glyoxalase-IMore, Swati S. / Vince, Robert et al. | 2006
- I
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Instructions to contributors| 2007
- IFC
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Editorial board| 2007