Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 3115
-
Graphical Abstracts| 2003
- 3129
-
Discovery and SAR of novel, potent and selective protein tyrosine phosphatase 1B inhibitorsPei, Zhonghua / Li, Xiaofeng / Liu, Gang et al. | 2003
- 3133
-
Synthesis and SAR evaluation of oxadiazolopyrazines as selective Haemophilus influenzae antibacterial agentsBeebe, Xenia / Nilius, Angela M. / Merta, Philip J. et al. | 2003
- 3137
-
Synthesis and cytotoxic activity of a-ring modified betulinic acid derivativesYou, Young-Jae / Kim, Yong / Nam, Nguyen-Hai et al. | 2003
- 3141
-
Synthesis of S6-(2,4-dinitrophenyl)-6-thioguanosine phosphoramidite and its incorporation into oligoribonucleotidesZheng, Qinguo / Wang, Yang / Lattmann, Eric et al. | 2003
- 3145
-
Analysis of the Critical Structural Determinant(s) of Species-Selective Peroxisome Proliferator-Activated Receptor Alpha (PPARα)-Activation by Phenylpropanoic Acid-Type PPARα AgonistsMiyachi, Hiroyuki / Uchiki, Hideharu et al. | 2003
- 3145
-
Analysis of the Critical Structural Determinant(s) of Species-Selective Peroxisome Proliferator-Activated Receptor Alpha (PPARa)-Activation by Phenylpropanoic Acid-Type PPARa AgonistsMiyachi, Hiroyuki et al. | 2003
- 3151
-
Biological activities of a-mangostin derivatives against acidic sphingomyelinaseHamada, Motoko et al. | 2003
- 3151
-
Biological activities of α-mangostin derivatives against acidic sphingomyelinaseHamada, Motoko / Iikubo, Kazuhiko / Ishikawa, Yuichi et al. | 2003
- 3155
-
1-Benzyloxy-4,5-dihydro-1H-imidazol-2-yl-amines, a novel class of NR1/2B subtype selective NMDA receptor antagonistsAlanine, Alexander / Bourson, Anne / Büttelmann, Bernd et al. | 2003
- 3161
-
Reversed hydroxamate-Bearing thermolysin inhibitors mimic a high-energy intermediate along the enzyme-Catalyzed proteolytic reaction pathwayPark, Jung Dae / Kim, Dong H et al. | 2003
- 3167
-
De novo synthesis of two new cytotoxic tiazofurin analogues with modified sugar moietiesPopsavin, Mirjana / Torović, Ljilja / Kojić, Vesna et al. | 2003
- 3171
-
Selective 3-Amino-2-pyridinone acetamide thrombin inhibitors incorporating weakly basic partially saturated heterobicyclic P1-Arginine mimeticsPeterlin-Mašič, Lucija / Kranjc, Andreja / Marinko, Petra et al. | 2003
- 3177
-
Design and synthesis of new benzimidazole-arylpiperazine derivatives acting as mixed 5-HT1A/5-HT3 ligandsLópez-Rodrı́guez, Marı́a L. / Benhamú, Bellinda / Morcillo, Mª José et al. | 2003
- 3181
-
Regulation of gene expression by synthetic dimerizers with novel specificityYang, Wu / Keenan, Terence P. / Rozamus, Leonard W. et al. | 2003
- 3185
-
O-Arylmandelic acids as highly selective human PPAR a-g agonistsAdams, Alan D. et al. | 2003
- 3185
-
O-Arylmandelic acids as highly selective human PPAR α/γ agonistsAdams, Alan D / Hu, Zao / von Langen, Derek et al. | 2003
- 3191
-
Design and synthesis of fluorinated RXR modulatorsGernert, D.L. / Ajamie, R. / Ardecky, R.A. et al. | 2003
- 3197
-
Antiallergic principles from Alpinia galanga: structural requirements of phenylpropanoids for inhibition of degranulation and release of TNF-a and IL-4 in RBL-2H3 cellsMatsuda, Hisashi et al. | 2003
- 3197
-
Antiallergic principles from Alpinia galanga: structural requirements of phenylpropanoids for inhibition of degranulation and release of TNF-α and IL-4 in RBL-2H3 cellsMatsuda, Hisashi / Morikawa, Toshio / Managi, Hiromi et al. | 2003
- 3203
-
Design and synthesis of dimeric HIV-1 integrase inhibitory peptidesKrajewski, Krzysztof / Long, Ya-Qiu / Marchand, Christophe et al. | 2003
- 3207
-
The stability of pseudopeptides bearing sulfoximines as chiral backbone modifying element towards proteinase KBolm, Carsten / Müller, Dirk / Dalhoff, Christian et al. | 2003
- 3213
-
A convenient method for the computer-Aided molecular design of carborane containing compoundsJohnsamuel, Jayaseharan / Byun, Youngjoo / Jones, Thomas P. et al. | 2003
- 3217
-
Synthesis of a novel family of diterpenes and their evaluation as anti-inflammatory agentsLam, Thanh / Ling, Taotao / Chowdhury, Chinmay et al. | 2003
- 3223
-
Synthesis of methyl (5S,6R,7E,9E,11Z,13E,15S)-16-(4-fluorophenoxy)-5,6,15-trihydroxy-7,9,11,13-hexadecatetraenoate, an analogue of 15R-Lipoxin A4Phillips, Eifion D / Chang, Hui-Fang / Holmquist, Christopher R et al. | 2003
- 3227
-
Novel inhibitors of an emerging target in Mycobacterium tuberculosis; substituted thiazolidinones as inhibitors of dTDP-rhamnose synthesisBabaoglu, Kerim / Page, Mark A. / Jones, Victoria C. et al. | 2003
- 3231
-
Bisphosphonates derived from fatty acids are potent inhibitors of Trypanosoma cruzi farnesyl pyrophosphate synthaseSzajnman, Sergio H. / Montalvetti, Andrea / Wang, Youhong et al. | 2003
- 3237
-
Cyclohexanedione herbicides are inhibitors of rat heart acetyl-CoA carboxylaseSeng, Thomas W / Skillman, Tiffanie R / Yang, Nengyu et al. | 2003
- 3243
-
Synthesis and biological activity of piperazine-Based dual MMP-13 and TNF-a converting enzyme inhibitorsLetavic, Michael A. et al. | 2003
- 3243
-
Synthesis and biological activity of piperazine-Based dual MMP-13 and TNF-α converting enzyme inhibitorsLetavic, Michael A. / Barberia, John T. / Carty, Thomas J. et al. | 2003
- 3247
-
Design and parallel synthesis of piperidine libraries targeting the nociceptin (N/OFQ) receptorChen, Zhengming / Miller, Wendy S / Shan, Shen et al. | 2003
- 3253
-
2-Piperidin-4-yl-benzimidazoles with broad spectrum antibacterial activitiesHe, Yun / Wu, Baogen / Yang, Jun et al. | 2003
- 3257
-
Structure of Plasmodium vivax dihydrofolate reductase determined by homology modeling and molecular dynamics refinementRastelli, Giulio / Pacchioni, Sara / Parenti, Marco Daniele et al. | 2003
- 3261
-
Electrostatic interaction of p-Acidic amides with hydrogen-Bond acceptorsLi, Yi et al. | 2003
- 3261
-
Electrostatic interaction of π-Acidic amides with hydrogen-Bond acceptorsLi, Yi / Snyder, Lawrence B. / Langley, David R. et al. | 2003
- 3267
-
Xylylated dimers of putrescine and polyamines: influence of the polyamine backbone on spermidine transport inhibitionCovassin, Laurence / Desjardins, Michel / Soulet, Denis et al. | 2003
- 3273
-
Synthesis and PDF inhibitory activities of novel benzothiazolylidenehydroxamic acid derivativesTakayama, Wataru / Shirasaki, Yoshihisa / Sakai, Yusuke et al. | 2003
- 3277
-
Bicyclo[2.2.1]heptanes as novel triple re-uptake inhibitors for the treatment of depressionAxford, Lorraine / Boot, John R. / Hotten, Terrence M. et al. | 2003
- 3281
-
Glycidol-carbohydrate hybrids: a new family of DNA alkylating agentsToshima, Kazunobu / Okuno, Yukiko / Matsumura, Shuichi et al. | 2003
- 3285
-
Synthesis and anthelmintic activity of cyclohexadepsipeptides with (S,S,S,R,S,R)-configurationJeschke, Peter / Benet-Buchholz, Jordi / Harder, Achim et al. | 2003
- 3289
-
Detection of 1270 nm emission from singlet oxygen and photocytotoxic property of sugar-Pendant [60] fullerenesMikata, Yuji / Takagi, Satowa / Tanahashi, Maki et al. | 2003
- 3293
-
Stereocontrolled dopamine receptor binding and subtype selectivity of clebopride analogues synthesized from aspartic acidEinsiedel, Jürgen / Weber, Klaus / Thomas, Christoph et al. | 2003
- 3297
-
Synthesis of pyrimidinopyridine–triazene conjugates targeted to abl tyrosine kinaseRachid, Zakaria / Katsoulas, Athanasia / Brahimi, Fouad et al. | 2003
- 3301
-
Arachidonylsulfonyl derivatives as cannabinoid CB1 receptor and fatty acid amide hydrolase inhibitorsSegall, Yoffi / Quistad, Gary B. / Nomura, Daniel K. et al. | 2003
- 3305
-
Synthetic dihydropacidamycin antibioticsBoojamra, Constantine G. / Lemoine, Rémy C. / Blais, Johanne et al. | 2003
- 3305
-
Synthetic dihydropacidamycin antibiotics - A modified spectrum of activity for the pacidamycin classBoojamra, Constantine G. et al. | 2003
- 3311
-
Synthesis and Structure–Activity relationships of 1-arylmethyl-3-(2-aminopropyl)-5-aryl-6-methyluracils as potent GnRH receptor antagonistsGuo, Zhiqiang / Zhu, Yun-Fei / Tucci, Fabio C. et al. | 2003
- 3317
-
Synthesis and Structure–activity relationships of 1-arylmethyl-3-(1-methyl-2-amino)ethyl-5-aryl-6-methyluracils as antagonists of the human GnRH ReceptorTucci, Fabio C. / Zhu, Yun-Fei / Guo, Zhiqiang et al. | 2003
- 3323
-
HIV-1 protease inhibitors with picomolar potency against PI-resistant HIV-1 by modification of the P1′ substituentDuffy, Joseph L. / Kirk, Brian A. / Kevin, Nancy J. et al. | 2003
- 3323
-
HIV-1 protease inhibitors with picomolar potency against PI-resistant HIV-1 by modification of the P1prime substituentDuffy, J. L. / Kirk, B. A. / Kevin, N. J. et al. | 2003
- 3327
-
Structure activity studies of a novel cytotoxic benzodiazepineBoitano, Anthony / Emal, Cory D / Leonetti, Francesco et al. | 2003
- 3331
-
α-Keto amides as inhibitors of histone deacetylaseWada, Carol K. / Frey, Robin R. / Ji, Zhiqin et al. | 2003
- 3331
-
a-Keto amides as inhibitors of histone deacetylaseWada, Carol K. et al. | 2003
- 3337
-
Activity predictions for efavirenz analogues with the K103N mutant of HIV reverse transcriptaseUdier-Blagović, Marina / Watkins, Edward K. / Tirado-Rives, Julian et al. | 2003
- 3341
-
Further SAR studies on novel small molecule inhibitors of the hepatitis C (HCV) NS5B polymeraseReddy, T.Jagadeeswar / Chan, Laval / Turcotte, Nathalie et al. | 2003
- 3345
-
Muraymycins, novel peptidoglycan biosynthesis inhibitors: synthesis and SAR of their analoguesYamashita, Ayako / Norton, Emily / Petersen, Peter J et al. | 2003
- 3351
-
Stereoselective synthesis of phosphoramidate a(2-6)Sialyltransferase transition-State analogue inhibitorsSkropeta, Danielle et al. | 2003
- 3351
-
Stereoselective synthesis of phosphoramidate α(2-6)Sialyltransferase transition-State analogue inhibitorsSkropeta, Danielle / Schwörer, Ralf / Schmidt, Richard R. et al. | 2003
- 3355
-
N1-Benzenesulfonylgramine and N1-benzenesulfonylskatole: novel 5-HT6 receptor ligand templatesPullagurla, Manik R. / Dukat, Małgorzata / Setola, Vincent et al. | 2003
- 3361
-
Synthesis and biological evaluation of menthol-based derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1)Ye, Bin / Bauer, Shawn / Buckman, Brad O. et al. | 2003
- 3367
-
Synthesis of 3-phenylpyrazolo[4,3-b]pyridines via a convenient synthesis of 4-amino-3-arylpyrazoles and SAR of corticotropin-Releasing factor receptor type-1 antagonistsWilcoxen, Keith / Huang, Charles Q / McCarthy, James R et al. | 2003
- 3371
-
Synthesis of 1-methyl-3-phenylpyrazolo[4,3-b]pyridines via a methylation of 4-phthalimino-3-phenylpyrazoles and optimization toward highly potent corticotropin-releasing factor type-1 antagonistsHuang, Charles Q. / Wilcoxen, Keith / McCarthy, James R. et al. | 2003
- 3375
-
Synthesis and SAR of 8-Arylquinolines as potent corticotropin-Releasing factor1 (CRF1) receptor antagonistsHuang, Charles Q. / Wilcoxen, Keith / McCarthy, James R. et al. | 2003
- CO2
-
Editorial board| 2003
- I
-
Instructions to Contributors and GA example| 2003
- iii
-
Contents List| 2003
- vii
-
Contributors to this Issue| 2003