Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 4251
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Graphical Abstracts| 2003
- 4265
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Announcement—new Editor for Tetrahedron Letters| 2003
- 4267
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Phenolics with PPAR-g ligand-Binding activity obtained from licorice (Glycyrrhiza uralensis Roots) and ameliorative effects of glycyrin on genetically diabetic KK-Ay miceKuroda, Minpei et al. | 2003
- 4267
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Phenolics with PPAR-γ ligand-Binding activity obtained from licorice (Glycyrrhiza uralensis Roots) and ameliorative effects of glycyrin on genetically diabetic KK-Ay miceKuroda, Minpei / Mimaki, Yoshihiro / Sashida, Yutaka et al. | 2003
- 4273
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KMI-008, a novel b-Secretase inhibitor containing a hydroxymethylcarbonyl isostere as a transition-State mimic: design and synthesis of substrate-based octapeptidesShuto, Daisuke et al. | 2003
- 4273
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KMI-008, a novel β-Secretase inhibitor containing a hydroxymethylcarbonyl isostere as a transition-State mimic: design and synthesis of substrate-based octapeptidesShuto, Daisuke / Kasai, Soko / Kimura, Tooru et al. | 2003
- 4277
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A simple stereoselective synthesis and biological evaluation of FR181157: orally active prostacyclin mimeticHattori, Kouji / Tabuchi, Seiichiro / Okitsu, Osamu et al. | 2003
- 4281
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B-Ring unsaturated estrogens: biological evaluation of 17α-Dihydroequilein and novel B-Nor-6-thiaequilenins as tissue selective estrogensLugar, Charles W III / Magee, David / Adrian, Mary D et al. | 2003
- 4281
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B-Ring unsaturated estrogens: biological evaluation of 17a-Dihydroequilein and novel B-Nor-6-thiaequilenins as tissue selective estrogensLugar, Charles W. et al. | 2003
- 4285
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Non-peptide avb3 antagonists: Identification of potent, chain-shortened RGD mimetics that incorporate a central pyrrolidinone constraintPerkins, James J. et al. | 2003
- 4285
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Non-peptide αvβ3 antagonists: Identification of potent, chain-shortened RGD mimetics that incorporate a central pyrrolidinone constraintPerkins, James J / Duong, L.T / Fernandez-Metzler, Carmen et al. | 2003
- 4289
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Lysine sulfonamides as novel HIV-Protease inhibitors: optimization of the Ne-acyl-phenyl spacerStranix, Brent R. et al. | 2003
- 4289
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Lysine sulfonamides as novel HIV-Protease inhibitors: optimization of the Nε-acyl-phenyl spacerStranix, Brent R. / Sauvé, Gilles / Bouzide, Abderrahim et al. | 2003
- 4293
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Rational design, synthesis and structure-Activity relationships of a cyclic succinate series of TNF-a converting enzyme inhibitors. Part 1: lead identificationXue, Chu-Biao et al. | 2003
- 4293
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Rational design, synthesis and structure–Activity relationships of a cyclic succinate series of TNF-α converting enzyme inhibitors. Part 1: lead identificationXue, Chu-Biao / He, Xiaohua / Roderick, John et al. | 2003
- 4299
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Rational design, synthesis and structure-activity relationships of a cyclic succinate series of TNF-a converting enzyme inhibitors. Part 2: lead optimizationXue, Chu-Biao et al. | 2003
- 4299
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Rational design, synthesis and structure–activity relationships of a cyclic succinate series of TNF-α converting enzyme inhibitors. Part 2: lead optimizationXue, Chu-Biao / He, Xiaohua / Roderick, John et al. | 2003
- 4305
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Fluorescence resonance energy transfer in a novel cyclodextrin–Peptide conjugate for detecting steroid moleculesHossain, Mohammed Akhter / Mihara, Hisakazu / Ueno, Akihiko et al. | 2003
- 4309
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3-Iodo-4-phenoxypyridinones (IOPY's), a new family of highly potent non-nucleoside inhibitors of HIV-1 reverse transcriptaseBenjahad, Abdellah / Guillemont, Jérôme / Andries, Koen et al. | 2003
- 4313
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6-(2-Adamantan-2-ylidene-hydroxybenzoxazole)-O-sulfamate: A potent non-steroidal irreversible inhibitor of human steroid sulfataseSchreiner, Erwin P. / Wolff, Barbara / Winiski, Anthony P. et al. | 2003
- 4317
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4-(4-Alkylpiperazin-1-yl)phenyl group: A novel class of basic side chains for selective estrogen receptor modulatorsWatanabe, Nobuhide / Nakagawa, Hiroshi / Ikeno, Akihisa et al. | 2003
- 4321
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Novel histone deacetylase inhibitors: design, synthesis, enzyme inhibition, and binding mode study of SAHA-Based non-hydroxamatesSuzuki, Takayoshi / Nagano, Yuki / Matsuura, Azusa et al. | 2003
- 4327
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Synthesis and analgesic activity of hydrochlorides and quaternary ammoniums of epibatidine incorporated with amino acid esterDong, Jing-Chao / Wang, Xin / Li, Run-Tao et al. | 2003
- 4331
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Catechol-Substituted l-Chicoric acid analogues as HIV integrase inhibitorsLee, Jae Yeol / Yoon, Kwon Joong / Lee, Yong Sup et al. | 2003
- 4335
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Design and synthesis of statine-Containing BACE inhibitorsHu, Jingdan / Cwi, Cynthia L / Smiley, David L et al. | 2003
- 4341
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b-Alanine dipeptides as MC4R agonistsRuel, Réjean et al. | 2003
- 4341
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β-Alanine dipeptides as MC4R agonistsRuel, Réjean / Herpin, Timothy F. / Iben, Lawrence et al. | 2003
- 4345
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New cerebrosides from Euphorbia peplis L.: antimicrobial activity evaluationCateni, Francesca / Zilic, Jelena / Falsone, Gioacchino et al. | 2003
- 4351
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DAPI derivative: A fluorescent DNA dye that Can be covalently attached to biomoleculesLi, Min / Wu, Robert S. / Tsai, Jane S.C. et al. | 2003
- 4355
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Successful shape-Based virtual screening: The discovery of a potent inhibitor of the type I TGFb receptor kinase (TbRI)Singh, Juswinder et al. | 2003
- 4355
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Successful shape-Based virtual screening: The discovery of a potent inhibitor of the type I TGFβ receptor kinase (TβRI)Singh, Juswinder / Chuaqui, Claudio E. / Boriack-Sjodin, P.Ann et al. | 2003
- 4361
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4-Methyl-1,2,4-triazol-3-yl heterocycle as an alternative to the 1-methylimidazol-5-yl moiety in the Farnesyltransferase inhibitor ZARNESTRAtradeAngibaud, Patrick et al. | 2003
- 4361
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4-Methyl-1,2,4-triazol-3-yl heterocycle as an alternative to the 1-methylimidazol-5-yl moiety in the Farnesyltransferase inhibitor ZARNESTRA™Angibaud, Patrick / Saha, Ashis K. / Bourdrez, Xavier et al. | 2003
- 4365
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Substituted azoloquinolines and -quinazolines as new potent farnesyl protein transferase inhibitorsAngibaud, Patrick / Bourdrez, Xavier / End, David W. et al. | 2003
- 4371
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Synthesis and antiviral evaluation of 3-hydroxy-2-methylpyridin-4-one dideoxynucleoside derivativesBarral, Karine / Hider, Robert C / Balzarini, Jan et al. | 2003
- 4375
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3D-QSAR Studies on natural acetylcholinesterase inhibitors of Sarcococca saligna by comparative molecular field analysis (CoMFA)Zaheer-ul-Haq / Wellenzohn, Bernd / Tonmunphean, Somsak et al. | 2003
- 4381
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Heterocyclic aminopyrrolidine derivatives as melatoninergic agentsSun, Li-Qiang / Chen, Jie / Mattson, Ronald J. et al. | 2003
- 4385
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Novel 3,4-Dihydroquinolin-2(1H)-one inhibitors of human glycogen phosphorylase aRosauer, Keith G. / Ogawa, Anthony K. / Willoughby, Chris A. et al. | 2003
- 4389
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Novel non-vanilloid VR1 antagonist of high analgesic effects and its structural requirement for VR1 antagonistic effectsSuh, Young-Ger / Lee, Yong-Sil / Min, Kyung-Hoon et al. | 2003
- 4395
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Antibacterial and antiproliferative activity of cationic fullerene derivativesMashino, Tadahiko / Nishikawa, Dai / Takahashi, Kyoko et al. | 2003
- 4399
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Synthesis and biological activity of novel 1b-Methylcarbapenems with oxyiminopyrrolidinylamide moietyLee, Ji Hoon et al. | 2003
- 4399
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Synthesis and biological activity of novel 1β-Methylcarbapenems with oxyiminopyrrolidinylamide moietyLee, Ji Hoon / Lee, Kyung Seok / Kang, Yong Koo et al. | 2003
- 4405
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Stable analogues of geranylgeranyl diphosphate possessing improved geranylgeranyl versus farnesyl protein transferase inhibitory selectivityMinutolo, Filippo / Bertini, Simone / Betti, Laura et al. | 2003
- 4409
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Design, synthesis and biological activity of novel dimethyl-{2-[6-substituted-indol-1-yl]-ethyl}-amine as potent, selective, and orally-Bioavailable 5-HT1D agonistsIsaac, Methvin / Slassi, Malik / Xin, Tao et al. | 2003
- 4415
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Synthesis of non-immunosuppressive cyclophilin-Binding cyclosporin A derivatives as potential anti-HIV-1 drugsEvers, Michel / Barrière, Jean-Claude / Bashiardes, Georges et al. | 2003
- 4421
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Binding of b-Carbolines at 5-HT2 serotonin receptorsGrella, Brian et al. | 2003
- 4421
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Binding of β-Carbolines at 5-HT2 serotonin receptorsGrella, Brian / Teitler, Milt / Smith, Carol et al. | 2003
- 4427
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1-Aryl-6,7-methylenedioxy-3H-quinazolin-4-ones as anticonvulsant agentsZappalà, Maria / Grasso, Silvana / Micale, Nicola et al. | 2003
- 4431
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Design and syntheses of melanocortin subtype-4 receptor agonists: evolution of the pyridazinone archetypeUjjainwalla, Feroze / Warner, Daniel / Walsh, Thomas F. et al. | 2003
- 4437
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Synthesis and Anti-HIV properties of new water-soluble bis-functionalized[60]fullerene derivativesBosi, Susanna / Da Ros, Tatiana / Spalluto, Giampiero et al. | 2003
- 4441
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O–N Intramolecular acyl migration strategy in water-soluble prodrugs of taxoidsSkwarczynski, Mariusz / Sohma, Youhei / Kimura, Maiko et al. | 2003
- 4445
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Potent anti-metastatic activity of dimeric sesquiterpene thioalkaloids from the rhizome of Nuphar pumilumMatsuda, Hisashi / Morikawa, Toshio / Oda, Mamiko et al. | 2003
- 4451
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Synthesis of new 3-Arylisoquinolinamines: effect on topoisomerase I inhibition and cytotoxicityCho, Won-Jea / Min, Sun Young / Le, Thanh Nguyen et al. | 2003
- 4455
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Synthesis and evaluation of optically pure dioxolanes as inhibitors of hepatitis C virus RNA replicationBera, Sanjib / Malik, Leila / Bhat, Balkrishen et al. | 2003
- 4459
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trans-3,4-Dimethyl-4-(3-carboxamidophenyl)piperidines: A novel class of (micro)-Selective opioid antagonistsLe Bourdonnec, Bertrand et al. | 2003
- 4459
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trans-3,4-Dimethyl-4-(3-carboxamidophenyl)piperidines: A novel class of m-Selective opioid antagonistsLe Bourdonnec, B. / Belanger, S. / Cassel, J. A. et al. | 2003
- 4459
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trans-3,4-Dimethyl-4-(3-carboxamidophenyl)piperidines: A novel class of μ-Selective opioid antagonistsLe Bourdonnec, Bertrand / Belanger, Serge / Cassel, Joel A. et al. | 2003
- 4463
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Ureas of 5-aminopyrazole and 2-aminothiazole inhibit growth of gram-positive bacteriaKane, John L. Jr. / Hirth, Bradford H. / Liang, Beirong et al. | 2003
- 4467
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Tripeptidyl-peptidase II (TPP II) inhibitory activity of (S)-2,3-dihydro-2-(1H-imidazol-2-yl)-1H-indoles, a systematic SAR evaluation. Part 2Breslin, Henry J. / Miskowski, Tamara A. / Kukla, Michael J. et al. | 2003
- 4473
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1,3-Dihydrobenzo[c]furan nucleoside analogues: additional studies of the thymine derivativeEgron, David / Périgaud, Christian / Gosselin, Gilles et al. | 2003
- 4477
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Duloxetine (Cymbalta™), a dual inhibitor of serotonin and norepinephrine reuptakeBymaster, F.P. / Beedle, E.E. / Findlay, J. et al. | 2003
- 4477
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Duloxetine (Cymbaltatrade), a dual inhibitor of serotonin and norepinephrine reuptakeBymaster, F.P. et al. | 2003
- 4481
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Conicamin, a novel histamine antagonist from the mediterranean tunicate Aplidium conicumAiello, Anna / Borrelli, Francesca / Capasso, Raffaele et al. | 2003
- 4485
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Exploration of the bicyclo[3.3.1]nonane system as a template for the development of new ligands for the estrogen receptorMuthyala, Rajeev S / Carlson, Kathryn E / Katzenellenbogen, John A et al. | 2003
- 4489
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Novel mechanism of inhibiting b-Lactamases by sulfonylation using b-SultamsPage, Michael I. et al. | 2003
- 4489
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Novel mechanism of inhibiting β-Lactamases by sulfonylation using β-SultamsPage, Michael I / Hinchliffe, Paul S / Wood, J.Matthew et al. | 2003
- 4493
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Microbial transformation of baccatin VI and 1β-Hydroxy baccatin I by aspergillus nigerShen, Ya-Ching / Lo, Kuang-Liang / Lin, Chun-Ling et al. | 2003
- 4493
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Microbial transformation of baccatin VI and 1b-Hydroxy baccatin I by aspergillus nigerShen, Ya-Ching et al. | 2003
- 4497
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N-Acyl 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline: The first orexin-2 receptor selective non-peptidic antagonistHirose, Masaaki / Egashira, Shin-ichiro / Goto, Yasuhiro et al. | 2003
- 4501
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Structure–activity relationships of indole cytosolic phospholipase A2α inhibitors: substrate mimeticsMcKew, John C / Lovering, Frank / Clark, James D et al. | 2003
- 4501
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Structure-activity relationships of indole cytosolic phospholipase A2a inhibitors: substrate mimeticsMckew, John C. et al. | 2003
- 4505
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Design and pharmacology of peptoids and peptide–peptoid hybrids based on the melanocortin agonists core tetrapeptide sequenceHolder, Jerry Ryan / Bauzo, Rayna M / Xiang, Zhimin et al. | 2003
- 4511
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Novel bicyclic furanopyrimidines with dual anti-VZV and -HCMV activityMcGuigan, Christopher / Brancale, Andrea / Andrei, Graciela et al. | 2003
- 4515
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An unnatural hydrophobic base, 4-propynylpyrrole-2-carbaldehyde, as an efficient pairing partner of 9-methylimidazo[(4,5)-b]pyridineMitsui, Tsuneo / Kimoto, Michiko / Sato, Akira et al. | 2003
- 4519
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Corrigendum to “Bone-Targeted Src Kinase Inhibitors: Novel Pyrrolo- and Pyrazolopyrimidine Analogues”[Bioorg. Med. Chem. Lett. 13 (2003) 3063]Sundaramoorthi, Raji / Shakespeare, William C / Keenan, Terence P et al. | 2003
- 4521
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Erratum to "Aryloxazolidinediones: Identification of Potent Orally Active PPAR Dual a/g Agonists"Desai, R. C. / Gratale, D. F. / Han, W. et al. | 2003
- 4521
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Erratum to “Aryloxazolidinediones: Identification of Potent Orally Active PPAR Dual α/γ Agonists”Desai, Ranjit C. / Gratale, Dominick F. / Han, Wei et al. | 2003
- 4521
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Erratum to "Aryloxazolidinediones: Identification of Potent Orally Active PPAR Dual a-g Agonists" - (Bioorg. Med. Chem. Lett. 13 (2003) 3541)Desai, Ranjit C. et al. | 2003
- CO2
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Editorial Board| 2003
- I
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Instructions to Contributors| 2003
- iii
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Contents List| 2003
- V
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Author Index| 2003
- vii
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Contributors to this Issue| 2003
- XLV
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Volume Contents| 2003