Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 1245
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Graphical contents list| 2008
- 1260
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Radiosyntheses of two positron emission tomography probes: [11C]Oseltamivir and its active metabolite [11C]Ro 64-0802Konno, Fujiko / Arai, Takuya / Zhang, Ming-Rong et al. | 2008
- 1264
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Synthesis and evaluation of [123I] labeled iodovinyl amino acids syn-, anti-1-amino-3-[2-iodoethenyl]-cyclobutane-1-carboxylic acid, and 1-amino-3-iodomethylene-cyclobutane-1-carboxylic acid as potential SPECT brain tumor imaging agentsYu, Weiping / Williams, Larry / Malveaux, Eugene et al. | 2008
- 1269
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2,6-Diaryl-4-phenacylaminopyrimidines as potent and selective adenosine A2A antagonists with reduced hERG liabilityMoorjani, Manisha / Zhang, Xiaohu / Chen, Yongsheng et al. | 2008
- 1274
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Development of Pyridopyrimidines as Potent Akt1/2 InhibitorsWu, Zhicai / Hartnett, John C. / Neilson, Lou Anne et al. | 2008
- 1280
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The discovery of adamantyl-derived, inhaled, long acting β2-adrenoreceptor agonistsBrown, Alan D. / Bunnage, Mark E. / Glossop, Paul A. et al. | 2008
- 1280
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The discovery of adamantyl-derived, inhaled, long acting b2-adrenoreceptor agonistsBrown, A. D. / Bunnage, M. E. / Glossop, P. A. et al. | 2008
- 1284
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Inhaled adenosine A2A receptor agonists for the treatment of chronic obstructive pulmonary diseaseMantell, Simon J. / Stephenson, Peter T. / Monaghan, Sandra M. et al. | 2008
- 1288
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α,β-Cyclic-β-benzamido hydroxamic acids: Novel oxaspiro[4.4]nonane templates for the discovery of potent, selective, orally bioavailable inhibitors of tumor necrosis factor-α converting enzyme (TACE)Ott, Gregory R. / Asakawa, Naoyuki / Liu, Rui-Qin et al. | 2008
- 1288
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a,b-Cyclic-b-benzamido hydroxamic acids: Novel oxaspiro[4.4]nonane templates for the discovery of potent, selective, orally bioavailable inhibitors of tumor necrosis factor-a converting enzyme (TACE)Ott, G. R. / Asakawa, N. / Liu, R. Q. et al. | 2008
- 1293
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Synthesis of pyrimidine and quinolone conjugates as a scaffold for dual inhibitors of HIV reverse transcriptase and integraseWang, Zhengqiang / Vince, Robert et al. | 2008
- 1297
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Identification of a potent new chemotype for the selective inhibition of PDE4Skoumbourdis, Amanda P. / Huang, Ruili / Southall, Noel et al. | 2008
- 1304
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Tyramine fragment binding to BACE-1Kuglstatter, Andreas / Stahl, Martin / Peters, Jens-Uwe et al. | 2008
- 1308
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Synthesis and biological evaluation of novel 1,3,5-triazine derivatives as antimicrobial agentsZhou, Chunhui / Min, Jaeki / Liu, Zhigang et al. | 2008
- 1312
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1H-Pyrazolo[3,4-g]hexahydro-isoquinolines as selective glucocorticoid receptor antagonists with high functional activityClark, Robin D. / Ray, Nicholas C. / Williams, Karen et al. | 2008
- 1318
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Synthesis and structure–activity relationships of heteroaryl substituted-3,4-diamino-3-cyclobut-3-ene-1,2-dione CXCR2/CXCR1 receptor antagonistsYu, Younong / Dwyer, Michael P. / Chao, Jianping et al. | 2008
- 1323
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QSAR studies on CCR2 antagonists with chiral sensitive hologram descriptorsNair, Pramod C. / Srikanth, K. / Sobhia, M. Elizabeth et al. | 2008
- 1331
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Synthesis and SAR of pyridazinone-substituted phenylalanine amide α4 integrin antagonistsGong, Yong / Kent Barbay, J. / Kimball, Edward S. et al. | 2008
- 1331
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Synthesis and SAR of pyridazinone-substituted phenylalanine amide a4 integrin antagonistsGong, Y. / Kent Barbay, J. / Kimball, E. S. et al. | 2008
- 1336
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Design and synthesis of 1,3-diarylurea derivatives as selective cyclooxygenase (COX-2) inhibitorsZarghi, Afshin / Kakhgi, Samaneh / Hadipoor, Atefeh et al. | 2008
- 1340
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Discovery of novel inhibitors of 11b-hydroxysteroid dehydrogenase type 1 by docking and pharmacophore modelingYang, H. / Dou, W. / Lou, J. et al. | 2008
- 1340
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Discovery of novel inhibitors of 11β-hydroxysteroid dehydrogenase type 1 by docking and pharmacophore modelingYang, Huaiyu / Dou, Wei / Lou, Jing et al. | 2008
- 1346
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Studies on the SAR and pharmacophore of milnacipran derivatives as monoamine transporter inhibitorsChen, Chen / Dyck, Brian / Fleck, Beth A. et al. | 2008
- 1350
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Novel highly potent μ-opioid receptor antagonist based on endomorphin-2 structureFichna, Jakub / do-Rego, Jean-Claude / Janecki, Tomasz et al. | 2008
- 1350
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Novel highly potent m-opioid receptor antagonist based on endomorphin-2 structureFichna, J. / do-Rego, J. C. / Janecki, T. et al. | 2008
- 1354
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Synthesis, SAR, and Evaluation of 4-[2,4-Difluoro-5-(cyclopropylcarbamoyl)phenylamino]pyrrolo[2,1-f][1,2,4]triazine-based VEGFR-2 kinase inhibitorsCai, Zhen-wei / Wei, Donna / Borzilleri, Robert M. et al. | 2008
- 1359
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Synthesis and anticancer activity studies of cyclopamine derivativesZhang, Jianjun / Garrossian, Massoud / Gardner, Dale et al. | 2008
- 1364
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Syntheses of N3-substituted thymine acyclic nucleoside phosphonates and a comparison of their inhibitory effect towards thymidine phosphorylasePomeisl, Karel / Holý, Antonín / Votruba, Ivan et al. | 2008
- 1368
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Synthesis and evaluation of PSSRI-based inhibitors of Staphylococcus aureus multidrug efflux pumpsGerman, Nadezhda / Kaatz, Glenn W. / Kerns, Robert J. et al. | 2008
- 1374
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Conformational studies of 3-amino-1-alkyl-cyclopentane carboxamide CCR2 antagonists leading to new spirocyclic antagonistsPasternak, Alexander / Goble, Stephen D. / Doss, George A. et al. | 2008
- 1378
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Cryptolepine analogues containing basic aminoalkyl side-chains at C-11: Synthesis, antiplasmodial activity, and cytotoxicityLavrado, João / Paulo, Alexandra / Gut, Jiri et al. | 2008
- 1382
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Design and synthesis of benzo-lipoxin A4 analogs with enhanced stability and potent anti-inflammatory propertiesPetasis, Nicos A. / Keledjian, Raquel / Sun, Yee-Ping et al. | 2008
- 1388
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Tricyclic HIV integrase inhibitors: Potent and orally bioavailable C5-aza analogsJin, Haolun / Wright, Matthew / Pastor, Richard et al. | 2008
- 1392
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Novel three-component synthesis and antiproliferative properties of diversely functionalized pyrrolinesMagedov, Igor V. / Luchetti, Giovanni / Evdokimov, Nikolai M. et al. | 2008
- 1397
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Selective, high affinity A2B adenosine receptor antagonists: N-1 monosubstituted 8-(pyrazol-4-yl)xanthinesKalla, Rao V. / Elzein, Elfatih / Perry, Thao et al. | 2008
- 1402
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Potent, selective MCH-1 receptor antagonistsErickson, Shawn D. / Banner, Bruce / Berthel, Steven et al. | 2008
- 1407
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Design, synthesis, and biological evaluation of 8-biarylquinolines: A novel class of PDE4 inhibitorsGallant, Michel / Chauret, Nathalie / Claveau, David et al. | 2008
- 1413
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Novel HCV NS5B polymerase inhibitors derived from 4-(1′,1′-dioxo-1′,4′-dihydro-1′λ6-benzo[1′,2′,4′]thiadiazin-3′-yl)-5-hydroxy-2H-pyridazin-3-ones. Part 1: Exploration of 7′-substitution of benzothiadiazineZhou, Yuefen / Webber, Stephen E. / Murphy, Douglas E. et al. | 2008
- 1413
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Novel HCV NS5B polymerase inhibitors derived from 4-(1prime,1prime-dioxo-1prime,4prime-dihydro-1primel6-benzo[1prime,2prime,4prime]thiadiazin-3prime-yl)-5-hydroxy-2H-pyridazin-3-ones. Part 1: Exploration of 7prime-substitution of benzothiadiazineZhou, Y. / Webber, S. E. / Murphy, D. E. et al. | 2008
- 1419
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Novel HCV NS5B polymerase inhibitors derived from 4-(1′,1′-dioxo-1′,4′-dihydro-1′λ6-benzo[1′,2′,4′]thiadiazin-3′-yl)-5-hydroxy-2H-pyridazin-3-ones. Part 2: Variation of the 2- and 6-pyridazinone substituentsZhou, Yuefen / Li, Lian-Sheng / Dragovich, Peter S. et al. | 2008
- 1419
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Novel HCV NS5B polymerase inhibitors derived from 4-(1prime,1prime-dioxo-1prime,4prime-dihydro-1primel6-benzo[1prime,2prime,4prime]thiadiazin-3prime-yl)-5-hydroxy-2H-pyridazin-3-ones. Part 2: Variation of the 2- and 6-pyridazinone substituentsZhou, Y. / Li, L. S. / Dragovich, P. S. et al. | 2008
- 1425
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Proline bis-amides as potent dual orexin receptor antagonistsBergman, Jeffrey M. / Roecker, Anthony J. / Mercer, Swati P. et al. | 2008
- 1431
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Implications for selectivity of 3,4-diarylquinolinones as p38αMAP kinase inhibitorsPeifer, Christian / Urich, Robert / Schattel, Verena et al. | 2007
- 1431
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Implications for selectivity of 3,4-diarylquinolinones as p38aMAP kinase inhibitorsPeifer, C. / Urich, R. / Schattel, V. et al. | 2008
- 1436
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Orally active esters of dihydroartemisinin: Synthesis and antimalarial activity against multidrug-resistant Plasmodium yoelii in miceSingh, Chandan / Chaudhary, Sandeep / Puri, Sunil K. et al. | 2007
- 1442
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Synthesis and biological evaluation of 99mTc, Re-monoamine-monoamide conjugated to 2-(4-aminophenyl)benzothiazole as potential probes for β-amyloid plaques in the brainChen, Xiangji / Yu, Pingrong / Zhang, Lianfeng et al. | 2007
- 1442
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Synthesis and biological evaluation of 99mTc, Re-monoamine-monoamide conjugated to 2-(4-aminophenyl)benzothiazole as potential probes for b-amyloid plaques in the brainChen, X. / Yu, P. / Zhang, L. et al. | 2008
- 1446
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Synthesis, thermal stability, antimalarial activity of symmetrically and asymmetrically substituted tetraoxanesAtheaya, Himanshu / Khan, Shabana I. / Mamgain, Ritu et al. | 2007
- 1450
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Probing the structural and topological requirements for CCR2 antagonism: Holographic QSAR for indolopiperidine derivativesSrikanth, K. / Nair, Pramod C. / Sobhia, M. Elizabeth et al. | 2007
- 1457
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Anticancer activity of (1,2,3,5-tetrahydro-4,1-benzoxazepine-3-yl)-pyrimidines and -purines against the MCF-7 cell line: Preliminary cDNA microarray studiesDíaz-Gavilán, Mónica / Gómez-Vidal, José A. / Rodríguez-Serrano, Fernando et al. | 2007
- 1461
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SAR study of 2,3,4,14b-tetrahydro-1H-dibenzo[b,f]pyrido[1,2-d][1,4]oxazepines as progesterone receptor agonistsDols, Paul P.M.A. / Folmer, Brigitte J.B. / Hamersma, Hans et al. | 2007
- 1468
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Synthesis of 1,2,3-triazole-linked pyrrolobenzodiazepine conjugates employing ‘click’ chemistry: DNA-binding affinity and anticancer activityKamal, Ahmed / Shankaraiah, N. / Devaiah, V. et al. | 2007
- 1474
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Novel echinocandin antifungals. Part 1: Novel side-chain analogs of the natural product FR901379Tomishima, Masaki / Ohki, Hidenori / Yamada, Akira et al. | 2007
- 1478
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5-Aryl-imidazolin-2-ones as a scaffold for potent antioxidant and memory-improving activityWatanabe, Kazutoshi / Morinaka, Yasuhiro / Hayashi, Yoshio et al. | 2007
- 1484
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Synthesis and cytotoxic activity of a new series of topoisomerase I inhibitorsDallavalle, Sabrina / Gattinoni, Sonia / Mazzini, Stefania et al. | 2007
- 1490
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A new family of H3 receptor antagonists based on the natural product ConessineSantora, Vincent J. / Covel, Jonathan A. / Hayashi, Rena et al. | 2007
- 1495
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Lysianadioic acid, a carboxypeptidase B inhibitor from Lysiana subfalcataBuchanan, Malcolm S. / Carroll, Anthony R. / Edser, Annette et al. | 2007
- 1498
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Anti-HIV-1 entry optimization of novel imidazopiperidine-tropane CCR5 antagonistsErnst, Justin / Dahl, Russell / Lum, Christopher et al. | 2007
- 1502
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4-(Heteroarylaminomethyl)-N-(2-aminophenyl)-benzamides and their analogs as a novel class of histone deacetylase inhibitorsFréchette, Sylvie / Leit, Silvana / Woo, Soon Hyung et al. | 2007
- 1507
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Synthesis of and evaluation of lipid A modification by 4-substituted 4-deoxy arabinose analogs as potential inhibitors of bacterial polymyxin resistanceKline, T. / Trent, M.S. / Stead, C.M. et al. | 2007
- 1511
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In vitro anti-inflammatory activity of 3-O-methyl-flavones isolated from Siegesbeckia glabrescensKim, Jae Yeon / Lim, Hyo Jin / Ryu, Jae-Ha et al. | 2007
- 1515
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Total synthesis and evaluation of [18F]MHMZHerth, Matthias M. / Debus, Fabian / Piel, Markus et al. | 2007
- 1520
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New insight for fluoroquinophenoxazine derivatives as possibly new potent topoisomerase I inhibitorKang, Da-Hye / Kim, Jung-Sook / Jung, Mi-Ja et al. | 2007
- 1525
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Synthesis and anti-inflammatory activities of mono-carbonyl analogues of curcuminLiang, Guang / Li, Xiaokun / Chen, Li et al. | 2007
- 1530
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Investigation of the alkenyldiarylmethane non-nucleoside reverse transcriptase inhibitors as potential cAMP phosphodiesterase-4B2 inhibitorsCullen, Matthew D. / Cheung, York-Fong / Houslay, Miles D. et al. | 2007
- 1534
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Synthesis and evaluation of stilbenylbenzoxazole and stilbenylbenzothiazole derivatives for detecting β-amyloid fibrilsLee, Ji Hoon / Byeon, Seong Rim / Lim, Soo Jeong et al. | 2007
- 1534
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Synthesis and evaluation of stilbenylbenzoxazole and stilbenylbenzothiazole derivatives for detecting b-amyloid fibrilsLee, J. H. / Byeon, S. R. / Lim, S. J. et al. | 2008
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Instructions to contributors| 2008
- IFC
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Editorial board| 2008