P04-76 EFFICIENT O-[^1^1C]METHYLATION WITH [^1^1C]METHYL TRIFLATE: SYNTHESIS OF ^1^1C-LABELED DIARYL SUBSTITUTED PYRAZOLE AND IMIDAZOLE CYCLOOXYGENASE INHIBITORS (English)
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JOURNAL OF LABELLED COMPOUNDS AND RADIOPHARMACEUTICALS
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48
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S206
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2005
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ISSN:
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Title:P04-76 EFFICIENT O-[^1^1C]METHYLATION WITH [^1^1C]METHYL TRIFLATE: SYNTHESIS OF ^1^1C-LABELED DIARYL SUBSTITUTED PYRAZOLE AND IMIDAZOLE CYCLOOXYGENASE INHIBITORS
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Contributors:Kawamura, K. ( author ) / Fujisaki, Y. ( author ) / Ishiwata, K. ( author ) / Yamamoto, F. ( author ) / Maeda, M. ( author )
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Publication date:2005-01-01
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Size:S206
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
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Table of contents – Volume 48
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1
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The synthesis of a benzamidine‐containing NR2B‐selective NMDA receptor ligand labelled with tritium or fluorine‐18Hamill, Terence G. / McCauley, John A. / Burns, H. Donald et al. | 2005
- 11
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Synthesis of [3H], [13C215N] and [14C]Sch 66336 (Sarasar™)Hesk, D. / Cesarz, D. / Magatti, C. / Voronin, K. / Lavey, C. / McNamara, P. / Koharski, D. / Saluja, S. / Hendershot, S. / Pham, H. et al. | 2005
- 25
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Stereoselective synthesis of radiolabelled avermectinsMcKillican, Bruce P. / Perine, Jeffrey W. / Simmons, Dana P. / Wilson, Timothy E. et al. | 2005
- 31
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N‐Arylation of indoles with 4‐[18F]fluoroiodobenzene: synthesis of 18F‐labelled σ2 receptor ligands for positron emission tomography (PET)Wüst, Frank R. / Kniess, Torsten et al. | 2005
- 31
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N-Arylation of indoles with 4-[^1^8F]fluoroiodobenzene: synthesis of ^1^8F-labelled sigma~2 receptor ligands for positron emission tomography (PET)Wust, F. R. / Kniess, T. et al. | 2005
- 45
-
Enzymatic synthesis of tritium‐labelled isotopomers of histaminePanufnik, E. / Kański, R. / Kańska, M. et al. | 2005
- 51
-
Fluorine‐18 labelling of PNAs functionalized at their pseudo‐peptidic backbone for imaging studies with PETKuhnast, B. / Hinnen, F. / Hamzavi, R. / Boisgard, R. / Tavitian, B. / Nielsen, P. E. / Dollé, F. et al. | 2005
- 63
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Synthesis and biological characterization of 99mTc(I) tricarbonyl cysteine complex, a potential diagnostic for assessment of renal functionPark, Sang Hyun / Jang, Beom Su / Park, Kyung Bae et al. | 2005
- 75
-
Labelling of anilines, benzylamines and some N‐heterocyclics using cycloocta‐1,5‐dienyliridium(I)‐1,1,1,5,5,5‐hexafluoro‐pentan‐2,4‐dionate and isotopic hydrogen gas in DMF or DMAGarman, R. N. / Hickey, M. J. / Kingston, L. P. / McAuley, B. / Jones, J. R. / Lockley, W. J. S. / Mather, A. N. / Wilkinson, D. J. et al. | 2005
- 85
-
Synthesis of 14C‐labeled and tritiated AMPA potentiator LY450108Czeskis, Boris A. / O'Bannon, Douglas D. / Wheeler, William J. / Clodfelter, Dean K. et al. | 2005
- 101
-
Synthesis of [123I]‐3‐(4‐iodobenzyl)‐1,2,3,4‐tetrahydro‐8‐hydroxychromeno[3,4‐c]pyridin‐5‐one, a potential dopamine D4 ligand for SPECT studiesStaelens, L. / Oltenfreiter, R. / Cornelissen, B. / Blanckaert, P. / De Vos, F. / Deforce, D. / Dierckx, R.A. / Slegers, G. et al. | 2005
- 109
-
Synthesis of 6‐acrylamido‐4‐(2‐[18F]fluoroanilino)quinazoline: a prospective irreversible EGFR binding probeVasdev, Neil / Dorff, Peter N. / Gibbs, Andrew R. / Nandanan, Erathodiyil / Reid, Leanne M. / O'Neil, James P. / VanBrocklin, Henry F. et al. | 2005
- 117
-
Synthesis of [13C4]furanVu, Choua C. / Peterson, Lisa A. et al. | 2005
- 123
-
Synthesis of 13C6‐labeled Reyataz™ (BMS‐232632)Burrell, Richard C. / Lago, Michael W. / Luke, George M. / Rinehart, J. Kent et al. | 2005
- 131
-
Synthesis of (4‐[18F]fluorophenyl)triphenylphosphonium as a potential imaging agent for mitochondrial dysfunctionCheng, Zhen / Subbarayan, Murugesan / Chen, Xiaoyuan / Gambhir, Sanjiv Sam et al. | 2005
- 139
-
The synthesis of carbon‐14 labeled (R)‐4‐(dipropylamino)‐1,3,4,5‐tetrahydrobenz[cd]indole‐6‐carboxamide hippurate. A partial ergoline with 5‐HT1A agonist activity and an 125I‐labeled analogWheeler, William J. / Swanson, Steven P. / Varie, David L. / O'Bannon, Douglas D. et al. | 2005
- 149
-
The synthesis of (S)‐di‐n‐propyl‐(8‐isoxazol‐5‐yl‐1,2,3,4‐tetrahydronaphthalen‐2‐yl)amine hydrochloride and its C‐14‐labeled isotopomerWheeler, William J. / O'Bannon, Douglas D. / Swanson, Steven / Gillespie, Todd A. / Varie, David L. et al. | 2005
- 165
-
Synthesis of [14C]‐imexonJagadish, Bhumasamudram / Iyengar, Bhashyam S. / Sólyom, Anikó M. / Remers, William A. / Dorr, Robert T. / Shin Yu, Jason / Gupta, Surendra / Mash, Eugene A. et al. | 2005
- 171
-
Synthesis of deuterium labelled 2‐bromobenzylamine by directed ortho‐metalation chemistryAtzrodt, Jens / Derdau, Volker et al. | 2005
- 179
-
Isotope labeled ‘HEA/HEE’ moiety in the synthesis of labeled HIV‐protease inhibitors—Part IIEkhato, I. Victor / Liao, Yuan / Plesescu, Mihaela et al. | 2005
- 195
-
Radiobromination of closo‐carboranes using palladium‐catalyzed halogen exchangeWinberg, Karl Johan / Mume, Eskender / Tolmachev, Vladimir / Sjöberg, Stefan et al. | 2005
- 203
-
Use of fluorous and solid‐phase electrophiles as scavengers for excess amine in the preparation of sulfur‐35 labelled radioligandsZhang, Andy Shiqiang / Elmore, Charles S. / Egan, Marjorie A. / Melillo, David G. / Dean, Dennis C. et al. | 2005
- 209
-
Efficient synthesis of deuterium‐labelled ferrocenesEvchenko, Svetlana V. / Kamounah, Fadhil S. / Schaumburg, Kjeld et al. | 2005
- 219
-
Synthesis of labelled N-(4-hydroxy-[^1^4C(U)]phenyl)-2-[2,3-dihydro-3-oxo-1,2-benzisothiazol-2-yl-1,1-dioxide]acetamideXu, L. / Trudell, M. L. et al. | 2005
- 219
-
Synthesis of labelled N‐(4‐hydroxy‐[14C(U)]phenyl)‐2‐[2,3‐dihydro‐3‐oxo‐l,2‐benzisothiazol‐2‐yl‐1,1‐dioxide]acetamideXu, Liang / Trudell, Mark L. et al. | 2005
- 223
-
Synthesis of 13C1‐pinonaldehydeDicus, Christopher W. / Willenbring, Dan / Nantz, Michael H. et al. | 2005
- 231
-
Preparation of [carboxy‐13C]4‐nitrophenylacetic acidCorrie, John E. T. / Munasinghe, V. Ranjit N. et al. | 2005
- 235
-
Enzymatic synthesis of tritium‐labelled isotopomers of L‐DOPAKozłowska, M. / Kański, R. / Kańska, M. et al. | 2005
- 241
-
Manufacturing I‐123‐labelled radiopharmaceuticals. Pitfalls and solutionsEersels, Jos L.H. / Travis, Michael J. / Herscheid, Jacobus D.M. et al. | 2005
- 259
-
Electrochemical radiofluorination. 3. Direct labeling of phenylalanine derivatives with [18F]fluoride after anodic oxidationKienzle, Gabriele J. / Reischl, Gerald / Machulla, H.‐Jürgen et al. | 2005
- 275
-
Synthesis of [35S]aryl sulfonyl chlorides from [35S]elemental sulfurWallace, Michael A. / Raab, Conrad E. / Dean, Dennis C. / Melillo, David G. et al. | 2005
- 285
-
An improved bidentate complex of iridium as a catalyst for hydrogen isotope exchangeHerbert, John M. / Kohler, Andrew D. / McNeill, Alan H. et al. | 2005
- 295
-
Synthesis of an iodine‐123‐labeled celecoxib analogue: a potential spect agentKabalka, George W. / Mereddy, Arjun R. / Schuller, Hildegard M. et al. | 2005
- 301
-
Synthesis and biological evaluation of S‐[11C]methylated mercaptoimidazole piperazinyl derivatives as potential radioligands for imaging 5‐HT1A receptors by positron emission tomography (PET)Garcia, Raquel / Xavier, Catarina / Paulo, António / Santos, Isabel / Kniess, Torsten / Bergmann, R. / Wüst, Frank et al. | 2005
- 317
-
The mediation of aryl ketone deuteration by [Ir(PPh3)3(cod)]+.BF4−Herbert, John M. et al. | 2005
- 323
-
Synthesis of C‐14‐labeled novel IKK inhibitor: 2‐[14C]‐N‐(6‐chloro‐9H‐pyrido [3,4‐b]indol‐8‐yl)‐3‐pyridinecarboxamideLi, Yuexian / Prakash, Shimoga R. et al. | 2005
- 331
-
Tritiation of CEP‐1347 at high specific activity using several methodsEgan, Judith A. / Filer, Crist N. / Pounds, Scot / Connors, Thomas / Knight, Ernest Jr / Hudkins, Robert L. et al. | 2005
- 337
-
Investigations into the C‐deuteriation of enol acetates derived from aryl alkyl ketonesBuksha, Svitlana / Coumbarides, Gregory S. / Dingjan, Marco / Eames, Jason / Suggate, Michael J. / Weerasooriya, Neluka et al. | 2005
- 353
-
Preparation of 14C2‐cis‐1,2‐dichloroethylene from 14C2‐trichloroethylene using a cobalt porphyrin catalystDeJournett, Todd D. / Fritsch, Joseph M. / McNeill, Kristopher / Arnold, William A. et al. | 2005
- 359
-
A facile synthesis of radioiodinated alkynyl iodides using potassium alkynyltrifluoroboratesKabalka, George W. / Mereddy, Arjun R. et al. | 2005
- 363
-
On the 99mTc‐labeling of isoniazid with different 99mTc coresSamuel, Grace / Kothari, Kanchan / Banerjee, Sharmila / Das, Tapas / Subramanian, Suresh / Kameshwaran, Mythili / Pillai, M. R. A. / Venkatesh, Meera et al. | 2005
- 379
-
Synthesis of the phytohormone [11C]methyl jasmonate via methylation on a C18 Sep Pak™ cartridgeHerth, Matthias M. / Thorpe, Michael R. / Ferrieri, Richard A. et al. | 2005
- 387
-
Synthesis, quality control and in vivo evaluation of [123I] rhTIMP‐2, a potential tumour‐imaging agentOltenfreiter, Ruth / Burvenich, Ingrid / Staelens, Ludovicus / Lejeune, Annabelle / Frankenne, Francis / Foidart, Jean‐Michel / Slegers, Guido et al. | 2005
- 397
-
The 14C, 13C and 15N syntheses of MON 37500, a sulfonylurea wheat herbicideMaxwell, Brad D. / Boyé, Olivier G. / Ohta, Kazunari et al. | 2005
- 407
-
Synthesis of beta~3 adrenergic receptor agonist LY377604 and its metabolite 4-hydroxycarbazole, labeled with carbon-14 and deuteriumCzeskis, B. A. / Wheeler, W. J. et al. | 2005
- 407
-
Synthesis of β3 adrenergic receptor agonist LY377604 and its metabolite 4‐hydroxycarbazole, labeled with carbon‐14 and deuteriumCzeskis, Boris A. / Wheeler, William J. et al. | 2005
- 421
-
Convenient methods for the synthesis of d4, d2 and d6 isotopomers of 4‐(4‐fluorobenzyl)piperidineProszenyák, Ágnes / Ágai, Béla / Tárkányi, Gábor / Vida, László / Faigl, Ferenc et al. | 2005
- 429
-
Tritium labelling of bromhexine via amide reduction with LiB3H4Larsen, Uffe S. / Begtrup, Mikael / Martiny, Lars et al. | 2005
- 435
-
Preparation of deuterated abscisic acid metabolites for use in mass spectrometry and feeding studiesZaharia, L. Irina / Galka, Marek M. / Ambrose, Stephen J. / Abrams, Suzanne R. et al. | 2005
- 447
-
Synthesis of deuterium‐, tritium‐, and carbon‐14‐labeled BILN2061, a potent hepatitis C virus protease inhibitorLatli, Bachir / Hrapchak, Matt / Gorys, Vida / Busacca, Carl A. / Senanayake, Chris et al. | 2005
- 457
-
Synthesis of [2H]‐labelled phase‐I‐metabolites using 1‐[2H]‐pyridinium hydrochlorideHeinkele, Georg / Mürdter, Thomas E. et al. | 2005
- 463
-
Simplified synthesis of N-(3-[^1^8F]fluoropropyl)-2beta-carbomethoxy-3beta-(4-fluorop henyl)nortropane ([^1^8F]beta-CFT-FP) using [^1^8F]fluoropropyl tosylate as the labelling reagentKoivula, T. / Perhola, O. / Kamarainen, E.-L. / Lipponen, T. / Vepsalainen, J. / Solin, O. et al. | 2005
- 463
-
Simplified synthesis of N‐(3‐[18F]fluoropropyl)‐2β‐carbomethoxy‐3β‐(4‐fluorophenyl)nortropane ([18F]β‐CFT‐FP) using [18F]fluoropropyl tosylate as the labelling reagentKoivula, Teija / Perhola, Outi / Kämäräinen, Eeva‐Liisa / Lipponen, Tiina / Vepsäläinen, Jouko / Solin, Olof et al. | 2005
- 473
-
The preparation of ^1^2^3^/^1^2^5I-clioquinol for the study of Abeta protein in Alzheimer's diseasePapazian, V. / Jackson, T. / Pham, T. / Liu, X. / Greguric, I. / Loc h, C. / Rowe, C. / Villemagne, V. / Masters, C. L. / Katsifis, A. et al. | 2005
- 473
-
The preparation of 123/125I‐clioquinol for the study of Aβ protein in Alzheimer's diseasePapazian, V. / Jackson, T. / Pham, T. / Liu, X. / Greguric, I. / Loc'h, C. / Rowe, C. / Villemagne, V. / Masters, C. L. / Katsifis, A. et al. | 2005
- 485
-
Syntheses of [14C] and [2H4]PD0205520, an inhibitor of the tyrosine kinase activity of the epidermal growth factor receptorZhang, Yinsheng / Huang, Yun / Huang, Che C. et al. | 2005
- 497
-
New radiolabelling chemistry: synthesis of phosphorus–[18F]fluorine compoundsStudenov, Andrei R. / Adam, Michael J. / Wilson, John S. / Ruth, Thomas J. et al. | 2005
- 501
-
Radiosynthesis of carbon‐11‐labelled GI181771, a new selective CCK‐A agonistDollé, F. / Martarello, L. / Bramoullé, Y. / Bottlaender, M. / Gee, A.D. et al. | 2005
- 515
-
14th International Isotope Society (UK group) symposiumAburel, P. S. / Aigbirhio, F. / Alexakis, E. / Audrain, H. / Austin, C. A. / Barry, C. / Bender, D. / Bushby, N. / Cable, K. / Carroll, M. A. et al. | 2005
- 547
-
Radiosynthesis and in vivo study of [18F]1‐(2‐fluoroethyl)‐4‐[(4‐cyanophenoxy)methyl]piperidine: a promising new sigma‐1 receptor ligandZhao, Jun / Chang, Raymond / Carambot, Patty / Waterhouse, Rikki N. et al. | 2005
- 557
-
Improved synthesis of [18F]fluoromethyl tosylate, a convenient reagent for radiofluoromethylationsNeal, Timothy R. / Apana, Scott / Berridge, Marc S. et al. | 2005
- 569
-
Fast and efficient tritium labelling of the nonsteroidal anti‐inflammatory drugs naproxen, tolmetin, and zomepiracJohansen, Steen K. / Sørensen, Lone / Martiny, Lars et al. | 2005
- 577
-
Synthesis of 1,1′ [11C]‐methylene‐di‐(2‐naphthol) ([11C]ST1859) for PET studies in humansLanger, Oliver / Krcal, Andreas / Schmid, Alexander / Abrahim, Aiman / Minetti, Patrizia / Celona, Diana / Roeda, Dirk / Dollé, Frédéric / Kletter, Kurt / Müller, Markus et al. | 2005
- 589
-
Tritiation of the cannabinoid receptor antagonist SR144528 involving lithium aluminum tritide reduction; assessment of the kinetic isotope effect by 3H‐NMRSeltzman, Herbert H. / Foster, Matthew C. / Wyrick, Christopher D. / Burgess, Jason P. / Ivy Carroll, F. et al. | 2005
- 597
-
Convenient synthesis of D‐threo‐[dichloroacetyl 1–14C] chloramphenicolSontakke, C. V. / Patil, S. P. / Unny, V. K. P. / Sivaprasad, N. et al. | 2005
- 605
-
The synthesis of isotopically labeled (+)‐2‐aminobicyclo[3.1.0]hexane‐2,6‐carboxylic acid and its 2‐oxa‐ and 2‐thia‐analogsWheeler, William J. / O'Bannon, Douglas D. / Kennedy, Joseph H. / Monn, James A. / Tharp‐Taylor, Roger W. / Valli, Matthew J. / Kuo, Fengjiun et al. | 2005
- 621
-
13C‐ and 14C‐labelling of N‐[1‐(4‐chlorophenyl)‐1H‐pyrrol‐2‐yl‐methyleneamino] guanidinium acetateAlmeida, Maria / Johannesson, Petra / Boman, Arne / Lundstedt, Torbjörn et al. | 2005
- 629
-
An improved synthesis of substituted [11C]toluenes via Suzuki coupling with [11C]methyl iodideHostetler, Eric D. / Terry, Garth E. / Donald Burns, H. et al. | 2005
- 635
-
Synthesis of 2‐[(2‐chloro‐2′‐[18F]fluoroethyl)amino]‐2H‐1,3,2‐oxazaphosphorinane‐2‐oxide (18F‐fluorocyclophosphamide), a potential tracer for breast tumor prognostic imaging with PETLacan, Goran / Kesner, Amanda L. / Gangloff, Anne / Zheng, Lei / Czernin, Johannes / Melega, William P. / Silverman, Daniel H. S. et al. | 2005
- 645
-
Synthesis of [14C]‐radiolabelled entecavirOgan, Marc D. / Kucera, David J. / Pendri, Yadagiri R. / Kent Rinehart, J. et al. | 2005
- 657
-
Synthesis and evaluation of [11C]RU40555, a selective glucocorticoid receptor antagonistMatsuya, Takahiro / Takamatsu, Hiroyuki / Murakami, Yoshihiro / Noda, Akihiro / Osoda, Kazuhiko / Ichise, Rikiya / Awaga, Yuji / Nishimura, Shintaro et al. | 2005
- 669
-
A novel method for the synthesis of carbon‐14‐labeled N‐[3‐(1‐methyl‐4‐piperidinyl)‐1H‐pyrrolo[3,2‐b]pyridin‐5‐yl]propanamide and its use in quantitative whole‐body autoradiography studiesWheeler, William J. / Chay, Sylvia H. / Herman, Jennifer L. / O'Bannon, Douglas D. et al. | 2005
- 683
-
Kit with technetium‐99m labelled antimicrobial peptide UBI 29‐41 for specific infection detectionWelling, Mick M. / Korsak, Agnieszka / Gorska, Barbara / Oliver, Patricia / Mikolajczak, Renata / Balter, Henia S. / Feitsma, Hans I. J. / Pauwels, Ernest K. J. et al. | 2005
- 693
-
Synthesis of deramciclane* labeled with tritium in various positionsSzammer, János / Simon‐Trompler, Edit / Banka, Zoltán / Szúnyog, József / Klebovich, Imre et al. | 2005
- 701
-
Utility of 1,3,4,6‐tetra‐O‐acetyl‐2‐deoxy‐2‐[18F]fluoro‐glucopyranoside for no‐carrier‐added 18F‐glycosylation of amino acidsMaschauer, Simone / Pischetsrieder, Monika / Kuwert, Torsten / Prante, Olaf et al. | 2005
- 721
-
Synthesis of (R)- and (S)-[O-methyl-^1^1C]N-[2-[3-(2-cyano-phenoxy)-2-hydroxy-propylamino]-ethyl]-N'-(4-methoxy-phenyl)-urea as candidate high affinity beta~1-adrenoceptor PET radioligandsWagner, S. / Law, M. P. / Riemann, B. / Pike, V. W. / Breyholz, H.-J. / Holtke, C. / Faust, A. / Schober, O. / Schafers, M. / Kopka, K. et al. | 2005
- 721
-
Synthesis of (R)‐ and (S)‐[O‐methyl‐11C]N‐[2‐[3‐(2‐cyano‐phenoxy)‐2‐hydroxy‐propylamino]‐ethyl]‐N′‐(4‐methoxy‐phenyl)‐urea as candidate high affinity β1‐adrenoceptor PET radioligandsWagner, Stefan / Law, Marilyn P. / Riemann, Burkhard / Pike, Victor W. / Breyholz, Hans‐Jörg / Höltke, Carsten / Faust, Andreas / Schober, Otmar / Schäfers, Michael / Kopka, Klaus et al. | 2005
- 735
-
Radiosyntheses and reactivities of novel [18F]2‐fluoroethyl arylsulfonatesMusachio, John L. / Shah, Jay / Pike, Victor W. et al. | 2005
- 749
-
Efficient methods for the synthesis of 5‐(4‐[18F]fluorophenyl)‐10,15,20‐tris(3‐methoxyphenyl)porphyrin as a potential imaging agent for tumorKavali, Rajesh R. / Chul Lee, Byung / Seok Moon, Byung / Dae Yang, Seung / Soo Chun, Kwon / Woon Choi, Chang / Lee, Chang‐Hee / Yoon Chi, Dae et al. | 2005
- 759
-
Microscale synthesis of isotopically labeled 6R‐N5, N10 methylene‐5, 6, 7, 8‐tetrahydrofolateHong, Baoyu / Kohen, Amnon et al. | 2005
- 771
-
Synthesis of [18F]fluoroalkyl esters of carfentanilHenriksen, Gjermund / Herz, Michael / Schwaiger, Markus / Wester, Hans‐Jürgen et al. | 2005
- 781
-
Preparation of isotopically labelled benzophenone‐containing lipid analoguesWang, Pingzhen / Spencer, Thomas A. et al. | 2005
- 789
-
Synthesis of tritium labelled CHS 828 and its prodrug EB 1627Schou, Søren Christian / Hunneche, Charlotte Schou / Binderup, Ernst / Grue‐Sørensen, Gunnar et al. | 2005
- 797
-
Syntheses of deuterated jasmonates for mass spectrometry and metabolism studiesGalka, Patrycja W. / Ambrose, Stephen J. / Ross, Andrew R. S. / Abrams, Suzanne R. et al. | 2005
- 811
-
Synthesis of 2H‐ and 3H‐labeled N‐cyclopropylmethyl‐7α‐[(R)‐1‐hydroxy‐1‐methyl‐3‐(2thienyl)‐propyl]‐6,14‐endoethano‐6,7,8,14‐tetrahydro nororipavineWu, Bo / Chen, Lanfu / Wang, Jingyan / Liu, Chunhe / Liu, He / Zhong, Bohua et al. | 2005
- 811
-
Synthesis of ^2H- and ^3H-labeled N-cyclopropylmethyl-7alpha-[(R)-1-hydroxy-1-methyl-3-(2thienyl)-propyl]-6,14-endoethano-6,7,8,14-tetrahydro nororipavineWu, B. / Chen, L. / Wang, J. / Liu, C. / Liu, H. / Zhong, B. et al. | 2005
- 819
-
Synthesis of an 18F‐fluorobenzoate idarubicin derivative as new potential PET radiotracer to predict chemotherapy resistanceSeimbille, Yann / Czernin, Johannes / Phelps, Michael E. / Silverman, Daniel H. S. et al. | 2005
- 829
-
Fluorine‐18 labeling of 6,7‐disubstituted anilinoquinazoline derivatives for positron emission tomography (PET) imaging of tyrosine kinase receptors: synthesis of 18F‐Iressa and related molecular probesSeimbille, Yann / Phelps, Michael E. / Czernin, Johannes / Silverman, Daniel H. S. et al. | 2005
- 845
-
Synthesis of [18F]‐6‐deoxy‐6‐fluoro‐D‐glucose ([18F]6FDG), a potential tracer of glucose transportNeal, Timothy R. / Schumann, William C. / Berridge, Marc S. / Landau, Bernard R. et al. | 2005
- 855
-
Synthesis and radioiodination of some 9‐aminoacridine derivatives for potential use in radionuclide therapyGhirmai, Senait / Mume, Eskender / Lundqvist, Hans / Tolmachev, Vladimir / Sjöberg, Stefan et al. | 2005
- 873
-
Improvement in radiolabelling proteins with the ^9^9^mTc-tricarbonyl-core [^9^9^mTc(CO)~3]^+, by thiol-derivatization with iminothiolane: application to gamma-globulins and annexin VBiechlin, M.-L. / d Hardemare, A. d. M. / Fraysse, M. / Gilly, F.-N. / Bonmartin, A. et al. | 2005
- 873
-
Improvement in radiolabelling proteins with the 99mTc‐tricarbonyl‐core [99mTc(CO)3]+, by thiol‐derivatization with iminothiolane: application to γ‐globulins and annexin VBiechlin, Marie‐Laure / d'Hardemare, Amaury du Moulinet / Fraysse, Marc / Gilly, François‐Noël / Bonmartin, Alain et al. | 2005
- 887
-
Synthesis of [11C]celecoxib: a potential PET probe for imaging COX‐2 expressionPrabhakaran, Jaya / Majo, Vattoly J. / Simpson, Norman R. / Van Heertum, Ronald L. / Mann, J. John / Kumar, J. S. Dileep et al. | 2005
- 897
-
The synthesis of [phenyl‐2H5]gluconasturtiin and its metabolites for metabolic studiesMorrison, John J. / Botting, Nigel P. et al. | 2005
- 909
-
Preparation and characterization of technetium‐99m complexes with new diphosphines containing polyether groupsValls, Esteve / Martin, David / Piera, Carlos / Suades, Joan et al. | 2005
- 923
-
A new synthesis of the labeling precursor for [18F]‐fluoromisonidazoleAdamsen, Tom C. H. / Grierson, John R. / Krohn, Kenneth A. et al. | 2005
- 929
-
Use of LC–MS–MS for the rapid, specific and sensitive quality control measurement of carrier in a PET radioligand: [18F]FECNTShetty, H. Umesha / Chin, Frederick T. / Musachio, John L. / Pike, Victor W. et al. | 2005
- 941
-
Synthesis of 3'-deoxy-3'-[^1^8F]fluoro-1-B-D-xylofuranosyluracil ([^1^8F]-FMXU) for petAlauddin, M. M. / Balatoni, J. / Gelovani, J. et al. | 2005
- 941
-
Synthesis of 3′‐deoxy‐3′‐[18F]fluoro‐1‐β‐D‐xylofuranosyluracil ([18F]‐FMXU) for PETAlauddin, M. M. / Balatoni, J. / Gelovani, J. et al. | 2005
- 951
-
The synthesis of multiply 13C‐labelled plant and mammalian lignans as internal standards for LC‐MS and GC‐MS analysisFryatt, Tara / Botting, Nigel P. et al. | 2005
- 971
-
Alternative methods for labeling the 5‐HT1A receptor agonist, 1‐[2‐(4‐fluorobenzoylamino)ethyl]‐4‐(7‐methoxynaphthyl)piperazine (S14506), with carbon‐11 or fluorine‐18Lu, Shui‐Yu / Hong, Jinsoo / Musachio, John L. / Chin, Frederick T. / Vermeulen, Erik S. / Wikström, Håkan V. / Pike, Victor W. et al. | 2005
- 983
-
^1^8F-FESB: Synthesis and Automated Radiofluorination of A Novel ^1^8F-Labelled PET Tracer for beta-Amyloid PlaquesKumar, P. / Zheng, W. / McQuarrie, S. A. / Jhamandas, J. H. / Wiebe, L. I. et al. | 2005
- 983
-
18F‐FESB: synthesis and automated radiofluorination of a novel 18F‐labeled pet tracer for β‐amyloid plaquesKumar, Piyush / Zheng, Weizhong / McQuarrie, Stephen A. / Jhamandas, Jack H. / Wiebe, Leonard I. et al. | 2005
- 997
-
High Specific Activity Tritium Labelling of Anti-Tumor Agent CEP-2563Filer, C. N. / Egan, J. A. / Hudkins, R. L. et al. | 2005
- 997
-
High specific activity tritium labeling of anti‐tumor agent CEP‐2563Egan, Judith A. / Filer, Crist N. / Hudkins, Robert L. et al. | 2005
- 1003
-
Preparation, characterisation and biological evaluation of ^9^9^m(CO)~3-labelled cyclic polyaminesVanbilloen, H. P. / Eraets, K. / Evens, N. / Terwinghe, C. / Rattat, D. / Bormans, G. / Mortelmans, L. / Verbruggen, A. M. et al. | 2005
- 1003
-
Preparation, characterization and biological evaluation of 99mTc(CO)3‐labelled cyclic polyaminesVanbilloen, H. P. / Eraets, K. / Evens, N. / Terwinghe, C. / Rattat, D. / Bormans, G. / Mortelmans, L. / Verbruggen, A. M. et al. | 2005
- 1013
-
High specific activity tritium labeling of vitamin D derivative RO275646de Keczer, Steve A. / Lane, Tim S. / Voronin, Tatyana / Masjedizadeh, Mohammad R. et al. | 2005
- 1025
-
Carbon‐14 labelling of selective H3 receptor antagonistsJohansen, Steen K. et al. | 2005
- 1031
-
Synthesis of labeled acrylamide and N‐methylolacrylamide (NMA): 15N‐acrylamide, 13C‐NMA, 15N‐NMA, and 13C,15N‐NMABrown, N. R. / Frazier, C. E. et al. | 2005
- 1041
-
A facile and efficient synthesis of d3‐labelled Reyataz™Zhang, Huiping / Bonacorsi, Samuel J. Jr / Chen, Bang‐Chi / Leith, Leslie W. / Kent Rinehart, J. / Balasubramanian, Balu / Barrish, Joel C. et al. | 2005
- 1049
-
An improved synthesis of UDP‐3‐O‐acyl‐N‐[3H‐acetyl]glucosamine: a probe for inhibitors of LpxC in gram‐negative bacteriaMaxwell, Brad D. / Bronstein, Joel C. et al. | 2005
- 1055
-
A facile synthesis of high specific activity sodium [1‐14C] lauryl sulphate under microwave irradiationRavi, S. / Mathew, K. M. / Unny, V. K. P. / Sivaprasad, N. et al. | 2005
- 1059
-
Cumulative compound index| 2005
- lv
-
Author index| 2005
- S1
-
Session 1: Neuroreceptors| 2005
- S12
-
Session 2: Radionuclide production| 2005
- S19
-
Session 3: Radiotherapy/pharmacy| 2005
- S24
-
Session 4: PET chemistry| 2005
- S30
-
Session 5: PET chemistry| 2005
- S36
-
Session 6: PET chemistry| 2005
- S40
-
Session 7: Amyloid plaque| 2005
- S44
-
Session 8: Technetium| 2005
- S49
-
Session 9: Technetium| 2005
- S51
-
Session 10: Other| 2005
- S55
-
Session 11: Other| 2005
- S61
-
Session 12: Miscellaneous| 2005
- S66
-
Session 13: Miscellaneous| 2005
- S70
-
P01 ‐ Neuroreceptors| 2005
- S106
-
P02 ‐ Radionuclide production| 2005
- S116
-
P03 ‐ Therapy/radiopharmacy| 2005
- S131
-
P04 ‐ PET chemistry| 2005
- S232
-
P05 ‐ Technetium| 2005
- S263
-
P06 ‐ Other receptors/metabolism/proliferation/apoptosis/angiogenesis/hypoxia‐oxidative stress/hormones/nuclear receptors| 2005
- S297
-
P07 ‐ Non‐PET chemistry| 2005
- S312
-
P08 ‐ Miscellaneous| 2005
- S341
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P08-30 SYNTHESIS AND IN VIVO VALIDATION OF [11C]MPT: A POTENTIAL AGONIST PET PROBE FOR IMAGING 5HT~1~A RECEPTORSKumar, J. S. D. / Majo, V. J. / Prabhakaran, J. / Simpson, N. R. / Arcement, J. / van Heertum, R. L. / Mann, J. J. / Parsey, R. V. et al. | 2005
- v
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Program Summary| 2005
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P04-16 METHODS FOR LABELING THE 5-HT~1~A RECEPTOR AGONIST, S14506, WITH A POSITRON-EMITTER AT ANY OF THREE ALTERNATIVE POSITIONSLu, S. Y. / Hong, J. / Musachio, J. L. / Chin, F. T. / Vermeulen, E. S. / Wikstrom, H. V. / Pike, V. W. et al. | 2005
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P04-34 EVALUATION OF Cu-ETS FOR USE AS A PET TRACER OF REGIONAL RENAL PERFUSIONGreen, M. A. / Mathias, C. J. / Willis, L. R. / Handa, R. K. / Miller, M. A. / Hutchins, G. D. et al. | 2005
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P04-59 FACILE SYNTHESIS OF L-[1-^1^1C]LEUCINE AS A PET RADIOTRACER FOR THE MEASUREMENT OF CEREBRAL PROTEIN SYNTHESISMu, F. / Mangner, T. J. / Chugani, H. T. et al. | 2005
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P04-83 QUALITY CONTROL STUDIES OF [^1^1C]METHYL IODIDE (^1^1CH~3I) PRODUCED IN LIQUID AND GAS PHASE SYNTHESIS MODULESSuehiro, M. / Kothari, P. J. / Vallabhajosula, S. et al. | 2005
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P05-15 ETHER LIGAND COMPLEXES OF Tc(CO)~3^+ FOR CARDIAC IMAGINGMaresca, K. P. / Keith, D. / Femia, F. J. / Kronauge, J. F. / Lazarova, N. / Zubieta, J. A. / Babich, J. W. et al. | 2005
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P06-03 NOVEL SOMATOSTATIN PEPTIDOMIMETICS AS SOMATOSTATIN RECEPTOR SUBTYPE-2 SPECIFIC IMAGING AGENTSHan, G. / Kung, H. F. / Choi, S. R. / Makonnen, S. / Lee, W. et al. | 2005
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P06-09 SYNTHESIS OF N-SUBSTITUTED 9-AZABICYCLO[3.3.1] NONAN-3alpha-YL PHENYLCARBAMATE ANALOGS AS SIGMA-2 RECEPTOR LIGANDSChu, W. / Xu, J. / Wheeler, K. T. / Mach, R. H. et al. | 2005
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P06-23 CASPASE-3 SUBSTRATES AS POTENTIAL APOPTOSIS IMAGING AGENTSBauer, C. / Bauder-Wuest, U. / Mier, W. / Haberkorn, U. / Eisenhut, M. et al. | 2005
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P06-28 SYNTHESIS AND BIODISTRIBUTION OF ^9^9^mTc(CO)~3-TRIDENTATE-LABELED INTEGRIN ANTAGONIST IN TUMOR BEARING MICEPark, S. H. / Jang, B. S. / Lim, E. / Bur, M. / Xie, J. / Le, N. / Danthi, N. / Dewanjee, M. / Li, K. C. / Carrasquillo, J. A. et al. | 2005
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P06-27 SYNTHESIS OF FLUORINE-18 LABELED GLUCOSE-Lys-Arg-Gly-Asp-D-Phe AS A POTENTIAL TUMOR IMAGING AGENTKim, J. S. / Lee, K. C. / Lee, B. C. / Moon, B. S. / Song, H. J. / Chun, K. S. / Chi, D. Y. et al. | 2005
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P08-04 DOSE DETERMINATION OF HIGH SPECIFIC ACTIVITY ^1^4^9Pm-DOTA-TYR3-OCTREOTATE IN RATSCutler, C. S. / Li, W. / Hsu, Y. N. / Engelbrecht, H. P. / Forbis, L. / Embree, M. F. / Ketring, A. R. / Anderson, C. J. / Miller, W. H. et al. | 2005
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THE EFFECT OF P-GLYCOPROTEIN (Pgp) MODULATION ON SPECIFIC UPTAKE OF SUBSTITUTED [^1^8F]MPPF DERIVATIVESde Vries, E. F. J. / Brattinga, N. S. / Elsinga, P. H. / Passchier, J. / van Waarde, A. et al. | 2005
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PET IMAGING AGENTS FOR THALAMIC AND EXTRATHALAMIC alpha4beta2 NICOTINIC RECEPTORSPichika, R. / Collins, D. / Christian, B. / Shi, B. / Narayanan, T. / Mukherjee, J. et al. | 2005
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ABSTRACT HAS BEEN MOVED TO A POSTER PRESENTATION AT THE REQUEST OF THE AUTHORS| 2005
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COMPARISON OF PRETARGET AND CONVENTIONAL CC49 RADIOIMMUNOTHERAPY USING ^1^4^9Pm, ^1^6^6Ho AND ^1^7^7LuMohsin, H. / Sivaguru, G. / Jia, F. / Bryan, J. N. / Cutler, C. S. / Ketring, A. R. / Athey, P. S. / Simon, J. / Frank, R. K. / Theodore, L. J. et al. | 2005
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VALIDATION OF PET RADIO-SYNTHESIS SYSTEMSSteel, C. / Turton, D. / Liow, E. / Crosby, P. / O Brien, A. / Luthra, S. et al. | 2005
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TARGETING PEPT1 FOR DETECTING PANCREAS CANCER WITH [^1^1C]GLY-SAR: MICROPET IMAGING OF NUDE MICE BEARING ASPC-1, CAPAN-2, and MPANC-96 XENOGRAFTSNabulsi, N. B. / Kilbourn, M. R. / Smith, D. E. / Snyder, S. E. / Hu, Y. et al. | 2005
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NOVEL DOTA CONJUGATED AMINO ACID BRIDGE CYCLIZED ALPHA-MELANOCYTE STIMULATING HORMONE PEPTIDE ANALOGS FOR MELANOMA TARGETINGMiao, Y. / Gallazzi, F. / Quinn, T. P. et al. | 2005
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P01-04 5-HT~1~A RECEPTOR IMAGING WITH [^1^1C](S)-RWAY IN RAT BRAIN SHOWS A STRIKING DIFFERENCE IN PGP EFFECT COMPARED TO IMAGING IN MONKEYMcCarron, J. A. / Zoghbi, S. S. / Liow, J. S. / Hong, J. / Lu, S. Y. / Vermeulen, E. S. / Wikstrom, H. V. / Seidel, J. / Innis, R. B. / Pike, V. W. et al. | 2005
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P01-24 SYNTHESIS AND RADIOIODINATION OF SELECTIVE LIGANDS FOR THE DOPAMINE D3 RECEPTOR SUBTYPEHocke, C. / Lober, S. / Hubner, H. / Gmeiner, P. / Kuwert, T. / Prante, O. et al. | 2005
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P01-27 EVALUATION OF A C-11 LABELED CONFORMATIONALLY-FLEXIBLE BENZAMIDE ANALOG AS A DOPAMINE D~3 RECEPTOR RADIOTRACERTu, Z. / Chu, W. / Xu, J. / Li, S. / Jones, L. A. / Dence, C. S. / Luedtke, R. R. / Mach, R. H. et al. | 2005
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P01-34 SUITABILITY OF A RAT ANIMAL MODEL OF CHOLINERGIC DEFICIENCY FOR THE EVALUATION OF NEW RADIOLIGANDS FOR THE VESICULAR ACETYLCHOLINE TRANSPORTER (VACHT) AS REVEALED BY IMMUNOCYTOCHEMISTRYGrossmann, U. / Hartig, W. / Sorger, D. / Kouznetsova, E. / Schliebs, R. / Scheunemann, M. / Steinbach, J. / Sabri, O. et al. | 2005
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P02-06 ROLE OF X-RAY SPECTROMETRY IN MEDICAL RADIONUCLIDE DEVELOPMENTQaim, S. M. / Sudar, S. / Skakun, Y. / Coenen, H. H. et al. | 2005
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P03-13 RADIOLABELING OF CATIONIC DEXTRAN WITH YTTRIUM-90Zhai, S. / He, C. / Du, J. et al. | 2005
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P04-05 ONE STEP SYNTHESIS OF [carbonyl-^1^1C]WAY-100635Itsenko, O. / Kihlberg, T. / Blom, E. / Langstrom, B. et al. | 2005
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P04-09 HPLC UV DETECTOR RESPONSE TO RADIOACTIVITY IN THE ANALYSIS OF PET RADIOTRACERSTurton, D. R. / Yau, K. et al. | 2005
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P04-08 SYNTHESIS AND INITIAL EVALUATION OF 2-[^1^8F]FLUORO-5-[2-(2-METHYLTHIAZOL-4-YL) ETHYNYL]PYRIDINE, A POTENTIAL PET LIGAND FOR THE METABOTROPIC GLUTAMATE SUBTYPE 5 RECEPTORYu, M. / Tueckmantel, W. / Wang, X. / Zhu, A. / Kozikowski, A. / Brownell, A.-L. et al. | 2005
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P04-11 RADIOSYNTHESIS OF [^1^1C]GI181771, A NEW SELECTIVE CCK-A AGONISTDolle, F. / Martarello, L. / Bramoulle, Y. / Bottlaender, M. / Gee, A. D. et al. | 2005
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DEVELOPMENT OF NOVEL ORGANOMETALLIC Tc-99m AND Re-188 FOLATE AND PTEROATE DERIVATIVES FOR TARGETED RADIONUCLIDE DIAGNOSIS AND THERAPYMueller, C. / Schibli, R. / Schubiger, A. P. et al. | 2005
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VASCULAR IMAGING OF SOLID TUMORS IN RATS WITH A RADIOACTIVE ARSENIC-LABELED ANTIBODY THAT BINDS ANIONIC PHOSPHOLIPIDSJennewein, M. / Hermanne, A. / Mason, R. P. / Thorpe, P. E. / Roesch, F. et al. | 2005
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MAO A AND B RADIOTRACERS SHOW A REDUCED ARTERIAL PLASMA INPUT FUNCTION, PROLONGED LUNG RETENTION AND REDUCED MAO IN SMOKERS vs NON-SMOKERSLogan, J. / Fowler, J. S. et al. | 2005
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P01-20 RADIOIODINATION OF BENZODIAZEPINE DERIVATIVES AS LIGANDS FOR GROUP II METABOTROPIC GLUTAMATE RECEPTORSKoren, A. O. / Da Costa, H. / Cosgrove, K. P. / Staley, J. K. / Amici, L. A. / Bois, F. / Baldwin, R. M. / Tamagnan, G. D. et al. | 2005
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P01-23 IN VITRO AND IN VIVO BINDING CHARACTERISTICS OF C-11 LABELED ANTAGONISTS FOR NR2B SUBUNIT OF NMDA RECEPTORSHaradahira, T. / Fuchigami, T. / Fujimoto, N. / Okauchi, T. / Maeda, J. / Suzuki, K. / Suhara, T. / Yamamoto, F. / Mukai, T. / Maeda, M. et al. | 2005
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P01-35 IDENTIFICATION OF A NOVEL TETRAHYDROPYRIDINE PHARMACOPHORE FOR DESIGN OF SELECTIVE PROBES FOR IMAGING OF THE SEROTONIN TRANSPORTERSSmith, M. P. / Keith, D. F. / Femia, F. J. / Babich, J. W. et al. | 2005
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P04-26 EVALUATION OF [^1^1C]FORMYL CHLORIDE AS A CARBON-11 FORMYLATION AGENT: SYNTHESIS OF N-(4-TOLYL)-[^1^1C]FORMAMIDE AS A MODEL REACTIONRoeda, D. / Dolle, F. et al. | 2005
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P04-27 EFFICIENT [^1^8F]FLUORINATION OF HYNIC-[TYR^3]-OCTREOTATE (HYNICTATE) VIA HYDRAZONE FORMATIONRennen, H. J. / Laverman, P. / Maecke, H. R. / Boerman, O. C. et al. | 2005
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P04-41 PALLADIUM-CATALYZED AMINOCARBONYLATION OF NITROGEN-CONTAINING ARYL HALIDES USING [^1^1C]BH~3CO AS SOURCE OF CARBON MONOXIDEBender, D. / Audrain, H. / Aburel, P. S. / Plisson, C. / Gee, A. D. / Martarello, L. et al. | 2005
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P04-42 SYNTHESIS AND C-11 LABELING OF THREE POTENT NOREPINEPHRINE TRANSPORTER SELECTIVE LIGANDS (LORTALAMINE, OXAPROTILINE AND (R)-NISOXETINE) FOR COMPARATIVE PET STUDIES IN BABOONSLin, K.-S. / Ding, Y.-S. et al. | 2005
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P04-40 SIGMA-2 SELECTIVE FLUORINATED LIGANDS: SYNTHETIC METHOD AND OPTIMIZATION OF DECARBONYLATION FOR RADIOLABELINGSeo, J. W. / Chi, D. Y. / Luyt, L. G. / Wuest, F. / Dence, C. S. / Sharp, T. L. / Mach, R. H. / Welch, M. J. / Katzenellenbogen, J. A. et al. | 2005
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P04-46 SYNTHESIS OF CARBON-11 LABELED CAMPTOTHECIN DERIVATIVES AS NOVEL PET TRACERS FOR IMAGING OF TOPOISOMERASE IN CANCERSGao, M. / Miller, K. D. / Sledge, G. W. / Zheng, Q.-H. et al. | 2005
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P04-52 A PREPARATIVE HPLC METHOD FOR ^1^1C-METHYLATED COMPOUNDS: CHANGING THE RETENTION ORDER OF PRODUCTS AND THEIR PRECURSORSLehel, S. / Madsen, J. / Soendergaard, K. / Gillings, N. et al. | 2005
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P04-50 RADIOSYNTHESIS OF [^1^8F]LBT-999, A SELECTIVE RADIOLIGAND FOR THE VISUALISATION OF THE DOPAMINE TRANSPORTER WITH PETDolle, F. / Emond, P. / Hinnen, F. / Mavel, S. / Mincheva, Z. / Saba, W. / Valette, H. / Chalon, S. / Halldin, C. / Helfenbein, J. et al. | 2005
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P04-55 SYNTHESIS, RADIOSYNTHESIS AND INITIAL BIOLOGICAL EVALUATION OF A NEW CLASS OF CANDIDATE BRAIN CANNABINOID TYPE-1 (CB~1) RECEPTOR RADIOLIGANDDonohue, S. / Halldin, C. / Brown, A. / Hong, J. / Musachio, J. L. / Bacher, J. / Innis, R. B. / Pike, V. W. et al. | 2005
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P04-70 BY-PRODUCT FORMATION DURING EVAPORATION WITH THE RADIOLYSIS SCAVENGER PROPYLENE GLYCOLArponen, E. / Helin, S. / Nagren, K. et al. | 2005
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P04-75 POTENTIAL PITFALLS OF [^1^1C]METHYL TRIFLATE AS A METHYLATION REAGENTMock, B. H. / Zheng, Q.-H. et al. | 2005
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P04-80 SIMPLIFIED METHOD FOR SYNTHESIS OF ^1^4O- AND ^1^5O-LABELLED BUTANOLMikecz, P. / Nemeth, E. / Lehel, S. / Horvath, G. / Tron, L. / Schweiger, L. / Dodd, M. / Craib, S. et al. | 2005
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P04-79 2'-[^1^8F]FLUORO-2'-DEOXYTHYMIDINE (2'-FTDR): A PET RADIOPHARMACEUTICAL TO MONITOR EXPRESSION OF HSV-1 TKSun, W. / Moharram, S. / Zhuo, A. / Hitt, M. / Kumar, P. / Knaus, E. E. / Wiebe, L. I. et al. | 2005
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P04-95 A MULTI-PURPOSE ^1^1C-RADIOSYNTHESIS SYSTEMMock, B. H. / Zheng, Q.-H. / DeGrado, T. R. et al. | 2005
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P05-04 DIRECT METAL-CYCLIZED SOMATOSTATIN ANALOGUES: SYNTHESIS, CHARACTERIZATION AND RECEPTOR BINDING STUDIESBigott, H. M. / Junnotula, S. / Gallazzi, F. / Lewis, M. R. / Jurisson, S. S. et al. | 2005
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P05-07 SYNTHESIS OF DICARBA ANALOGUES OF OCTREOTIDE USING TANDEM HOMOGENEOUS CATALYSISWhelan, A. N. / Elaridi, J. / Smith, S. V. / Mulder, R. J. / Robinson, A. J. / Sosabowski, J. et al. | 2005
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P06-01 SYNTHESIS AND EVALUATION OF THE SIGMA RECEPTORS LIGAND 4-((4-^1^2^3I]IODOPHENOXY)METHYL)-1-(2-FLUOROETHYL)PIPERIDINE IN ANIMAL TUMOUR MODELSKatsifis, A. / Mattner, F. / Pham, T. / Liu, X. / Berghofer, P. / Greguric, I. / Ballantyne, P. / Chapman, J. / Nguyen, V. / Homes, T. et al. | 2005
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P06-17 [6-OR 7-METHOXY-^1^1C]PD153035: DOES THE LABELING POSITION INFLUENCE THE LABELED METABOLITES GENERATED?Thorell, J.-O. / Fredriksson, A. / Samen, E. / Stone-Elander, S. et al. | 2005
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P07-04 RADIOCHEMISTRY AND IN VIVO EVALUATION OF THREE NOVEL ^6^4Cu-LABELED CROSS-BRIDGED MACROCYCLIC COMPLEXESWadas, T. J. / Sprague, J. E. / Weisman, G. R. / Wong, E. H. / Peng, Y. / Tranchemontagne, D. J. / Widger, P. C. B. / Anderson, C. J. et al. | 2005
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P08-06 DEVELOPMENT OF NEW NUCLEOSIDE ANALOGUES FOR THE PET IMAGING OF HSV1 tk GENE EXPRESSIONJohayem, A. / Ametamey, S. M. / Honer, M. / Malic, S. R. / Novak, I. / Scapozza, L. / Schubiger, A. P. et al. | 2005
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P08-14 QSAR STUDY OF STB SERIES OF IMAGING AGENTS FOR beta-AMYLOID PLAQUEChen, X. J. / Liu, B. L. / Kung, H. F. et al. | 2005
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P08-29 A NOVEL TECHNETIUM TRICARBONYL COMPLEX OF VITAMIN B12Knight, H. / Alberto, R. / Vries, E. / Kunze, S. / Mundwiler, S. et al. | 2005
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VISUALIZATION OF beta-AMYLOID DEPOSITS IN THE LIVING BRAIN OF A TRIPLE TRANSGENIC RAT MODEL OF beta-AMYLOID DEPOSITION USING [^1^8F] FDDNP-MICROPET IMAGINGKepe, V. / Cole, G. M. / Liu, J. / Flood, D. G. / Trusko, S. P. / Satyamurthy, N. / Huang, S.-C. / Small, G. W. / Petric, A. / Phelps, M. E. et al. | 2005
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TECHNETIUM(I) PYRAZOLYL BOMBESIN CONJUGATES: A CONCISE IN VITRO/IN VIVO STUDYSmith, C. J. / Alves, S. / Santos, I. / Sieckman, G. L. / Hoffman, T. J. / Rold, T. / Retzloff, L. / McCrate, J. / Prasanphanich, A. / Veerendra, B. et al. | 2005
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SYNTHESIS AND EVALUATION OF In-111 DOTA-POLYDIAMIDOPROPANOATE (PDAP) DENDRIMER-PNA-PEPTIDE CHIMERAS FOR NON-INVASIVE IMAGING OF CANCERAmirkhanov, N. / Aruva, M. R. / Zhang, K. / Mathew, B. / Thakur, M. L. / Wickstrom, E. et al. | 2005
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MULTIMERIZATION OF INTEGRIN ANTAGONISTS ALLOWS HIGH CONTRAST IMAGING OF alpha~vbeta~3 INTEGRINSPoethko, T. / Thumshirn, G. / Hersel, U. / Hauser, A. / Kessler, H. / Schwaiger, M. / Wester, H.-J. et al. | 2005
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COMPARISON OF HIGH RESOLUTION MOUSE PET/CT IMAGING AND CONVENTIONAL BIODISTRIBUTIONS OF COPPER-64-LABELLED ANTIBODIESLewis, M. R. / Bryan, J. N. / Jia, F. / Mohsin, H. / Sivaguru, G. / Miller, W. H. / Henry, C. J. / Anderson, C. J. et al. | 2005
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P01-07 RADIOSYNTHESIS OF ^1^8F-LABELLED PYRAZOLO[1,5a]PYRIDINES AND 5-CYANOINDOLES AS SUBTYPE SELECTIVE D4 RECEPTOR LIGANDS FOR PETPrante, O. / Hocke, C. / Tietze, R. / Lober, S. / Hubner, H. / Gmeiner, P. / Kuwert, T. et al. | 2005
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P01-12 SYNTHESIS, LABELLING AND EVALUATION OF A NEW FLUORINATED NMDA LIGAND TO STUDY GLUTAMATERGIC NEUROTRANSMISSION IN VIVOPiel, M. / Hoehnemann, S. / Jansen, M. / Schmitt, U. / Dannhardt, G. / Roesch, F. et al. | 2005
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P01-11 SYNTHESIS AND EVALUATION OF ^1^1C-LABELED METHYLVESAMICOLS AS A PET LIGAND FOR VESICULAR ACETYLCHOLINE TRANSPORTERS OR SIGMA RECEPTORSKawamura, K. / Shiba, K. / Yajima, K. / Ishiwata, K. et al. | 2005
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P01-22 2alpha,3beta - TROPANE-DERIVATIVES: NEW FLUORINATED LIGANDS FOR THE DOPAMINE TRANSPORTERDrewes, B. / Sihver, W. / Coenen, H. H. et al. | 2005
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P03-11 LABELING OF ANTI-CD20 WITH Re-188: THEORETICAL DOSIMETRY CONSIDERATIONSFerro-Flores, G. / Torres, E. / Garnica, H. / Rosales, J. et al. | 2005
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P04-03 ONE-POT SYNTHESIS OF [^1^1C]-UREAS VIA TRIPHENYLPHOSPHINIMINESvan Tilburg, E. W. / van der Mey, M. / Windhorst, A. D. / Herscheid, J. D. M. et al. | 2005
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P04-13 DOUBLE-TRACER TECHNIQUE FOR QUANTITATIVE AUTORADIOGRAPHY WITH SHORT-LIVED POSITRON EMITTERS USING A BIO IMAGING ANALYZER SYSTEMNoguchi, J. / Zhang, M.-R. / Suzuki, K. et al. | 2005
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P04-15 HYPERVALENT IODINE REAGENTS AS PRECURSORS FOR RADIOLABELLING PYRIMIDINES USING N.C.A. [^1^8F]FLUORIDERobins, E. G. / Brady, F. / Luthra, S. K. et al. | 2005
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P04-18 [^1^1C]AR-A014418: A RADIOLABELLED GLYCOGEN SYNTHASE KINASE 3-SPECIFIC INHIBITOR FOR PET STUDIESVasdev, N. / Garcia, A. / Meyer, J. H. / Stableford, W. T. / Houle, S. / Wilson, A. A. et al. | 2005
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P04-38 SYNTHESIS OF 5'-(2-[^1^8F]FLUOROPHENYL)-SPIRO[1-AZABICYCLO [2.2.2.]OCTANE]-3,2'(3'H)-FURO[2,3-b]PYRIDINE ([^1^8F]FPS), AN AGONIST AT THE alpha7 NICOTINIC ACETYLCHOLINE RECEPTORRavert, H. T. / Dorff, P. / Foss, C. A. / Fan, H. / Holmquist, C. R. / Phillips, E. / McCarthy, D. J. / Heyes, R. / Holt, D. / Dannals, R. F. et al. | 2005
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P04-39 SYNTHESIS, RESOLUTION, AND STABILITY OF OPTICALLY ACTIVE Ga(III) AND Co(III) COMPLEXES WITH LINEAR HEXADENTATE N~4O~2^2^-LIGANDSLoganathan, D. / Smith, H. E. / Mathias, C. J. / Green, M. A. et al. | 2005
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P04-68 SYNTHESIS AND RADIOLABELLING OF A NOVEL IMAGING AGENT FOR HYPOXIC TISSUE IN STROKE AND TUMOURSFalzon, C. L. / Ackermann, U. / White, J. M. / Tochon-Danguy, H. J. / Scott, A. M. et al. | 2005
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P05-17 SYNTHESIS, RADIOLABELING, AND IN VITRO CHARACTERIZATION OF SYN AND ANTI ^9^9^mTc ACBC·BAT AS POSSIBLE TUMOR IMAGING AGENTSGiamis, A. M. / Camp, V. M. / Zhang, Z. / DePompei, A. O. / Yu, W. / Voll, R. J. / McConathy, J. E. / Goodman, M. M. et al. | 2005
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P06-14 SYNTHESIS AND EVALUATION OF NOVEL [^1^2^3I]-LABELLED BENZAMIDES FOR IMAGING MELANOMAPham, T. / Katsifis, A. / Mattner, F. / Liu, X. / Berghofer, P. / Greguric, I. / Ballantyne, P. / Chapman, J. / Jackson, T. / Papazian, V. et al. | 2005
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P06-19 PHARMACOKINETICS AND BIODISTRIBUTION OF RADIOLABELED CHOLINE IN HUMAN SUBJECTS: COMPARISON OF [^1^1C]CHOLINE AND [^1^8F]FLUOROCHOLINEVallabhajosula, S. / Kostakoglu, L. / Kothari, P. J. / Hamacher, K. A. / Goldsmith, S. J. et al. | 2005
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P06-18 A NOVEL F-18 LABELED sigma^2 RECEPTOR LIGAND FOR IMAGING BREAST CANCERTu, Z. / Xu, J. / Jones, L. A. / Li, S. / Wheeler, K. T. / Welch, M. J. / Mach, R. H. et al. | 2005
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P06-31 LABELING AND BIODISTRIBUTION OF AN ANGIOGENIN INHIBITOR IDENTIFIED BY HIGH THROUGHPUT SCREENINGMier, W. / Hoffend, J. / Eisenhut, M. / Haberkorn, U. et al. | 2005
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P06-32 EVALUATION OF [F-18]IRESSA AS A PET IMAGING AGENT FOR TUMORS OVEREXPRESSING EPIDERMAL GROWTH FACTOR (EGF) RECEPTORSMurali, D. / Flores, L. G. / Converse, A. K. / Bartlett, R. M. / Barnhart, T. E. / Armstrong, E. A. / Nickles, R. J. / Harari, P. M. / DeJesus, O. T. et al. | 2005
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P07-01 SYNTHESIS AND EVALUATION OF A RADIOIODINATED COXIB AS A SPECT TRACER FOR CYCLOOXYGENASE-2 EXPRESSIONKuge, Y. / Shimonaka, S. / Katada, Y. / Temma, T. / Kimura, H. / Kiyono, Y. / Yokota, C. / Minematsu, K. / Seki, K.-I. / Tamaki, N. et al. | 2005
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P07-02 NO-CARRIER-ADDED RADIOHALOGENATIONS UTILIZING BORONATE ESTERS AND SALTSKabalka, G. W. / Mereddy, A. R. et al. | 2005
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P08-01 FDG IMAGE DERIVED INPUT FUNCTION MEASUREMENT IN RATS AND MICE FROM THE LEFT VENTRICLERowland, D. J. / Laforest, R. et al. | 2005
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P08-07 RADIOSYNTHESIS AND PET MICRODOSING WITH 1,1'[^1^1C]METHYLENE-DI-(2-NAPHTHOL), A POTENTIAL ANTI-ALZHEIMER DRUGLanger, O. / Brunner, M. / Lanzenberger, R. / Bauer, M. / Paul, M. / Minetti, P. / Celona, D. / Joukhadar, C. / Roeda, D. / Dolle, F. et al. | 2005
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P08-16 5'-AMINO NUCLEOSIDES AS MARKERS FOR HSV1-TK GENE EXPRESSIONChacko, A.-M. / Choi, S.-R. / Zhuang, Z.-P. / Kung, H. F. et al. | 2005
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P08-24 PRACTICAL ASPECTS OF NEW LONG-LIVED WASTE STREAMS FROM GA-68 PET SCINTIGRAPHY AND PEPTIDE RECEPTOR RADIONUCLIDE THERAPY (PRRT) WITH LU-177Breeman, W. A. / Bakker, W. H. / de Jong, L. C. / de Blois, E. / van der Wagt, G. A. / Krenning, E. P. et al. | 2005
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PRELIMINARY STUDIES OF CONDUCTING HIGH LEVEL PRODUCTION RADIOSYNTHESES USING MICROFLUIDIC DEVICESLiow, E. / O Brien, A. / Luthra, S. / Brady, F. / Steel, C. et al. | 2005
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MICRO-FLUIDIC RADIOCHEMISTRY FOR PET AND SPECT TRACER DEVELOPMENTGillies, J. M. / Prenant, C. / Zweit, J. et al. | 2005
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RADIOSYNTHESIS OF A N-[^1^1C]METHYL-1,4-DIHYDROQUINOLINE AS CARRIER FOR DRUG DELIVERY TO THE BRAINGourand, F. / Foucout, L. / Levacher, V. / Perrio, C. / Dupas, G. / Barre, L. et al. | 2005
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CARBORANE DERIVATIVES FOR TARGETING ^9^9^mTc TO NEURORECEPTORSLouie, A. S. / Sogbein, O. O. / Schaffer, P. / Valliant, J. F. et al. | 2005
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PN~2S-PEG-BIOMOLECULE DERIVATIVES LABELED WITH TECHNETIUM-99m IN ABSENCE OF AN EXTERNAL REDUCING AGENTVisentin, R. / Morpurgo, M. / Pasut, G. / Riondato, M. / Rosato, A. / Banzato, A. / Veronese, F. M. / Moschini, G. / Mazzi, U. et al. | 2005
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RADIOSYNTHESIS AND PRELIMINARY EVALUATION OF A FOLIC ACID DERIVATIVE LABELED WITH F-18 FOR IMAGING FOLATE RECEPTOR-POSITIVE TUMORSBettio, A. / Ametamey, S. M. / Honer, M. / Mueller, C. / Schibli, R. / Mueller, U. / Groehn, V. / Schubiger, A. P. et al. | 2005
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P01-08 RECENT DEVELOPMENT IN NEW GENERATION RADIOTRACERS FOR PET IMAGING OF THE NOREPINEPHRINE TRANSPORTERDing, Y.-S. / Lin, K.-S. / Logan, J. et al. | 2005
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P01-30 SYNTHESIS AND IN VIVO EVALUATION OF [^1^1C]SIB-1553A, FOR beta-4 SUBTYPE NICOTINIC ACETYLCHOLINE RECEPTOR IMAGING BY POSITRON EMISSION TOMOGRAPHYSobrio, F. / Debruyne, D. / Dhilly, M. / Quentin, T. / Tymciu, S. / Barre, L. et al. | 2005
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P01-31 SYNTHESIS, LABELLING AND EVALUATION OF 4,6-DICHLORO-3-((3-(4-(2-FLUOROETHOXY)PHENYL)2,4-DIOXOIMIDAZOLIDINE)- 1H-INDOLE-2-CARBOXYLIC ACID AS RADIOTRACER FOR IMAGING THE NMDA-RECEPTOR STATUS IN VIVOBauman, A. / Piel, M. / Hoehnemann, S. / Jennewein, M. / Jansen, M. / Krauss, A. / Schmitt, U. / Dannhardt, G. / Roesch, F. et al. | 2005
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P02-05 MEASUREMENT OF CROSS SECTIONS FOR NATW(p,xn)^1^8^1^-^1^8^6Re REACTIONS UP TO 19 MEVLapi, S. / D Auria, J. M. / Ressler, J. J. / Ruth, T. J. et al. | 2005
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P04-20 SYNTHESIS OF [^1^8F]-FLUOROQUINOLINES FOR THE LABELLING OF A TALNETANT ANALOGUE AS NK-3 RECEPTOR LIGANDPerrio, C. / Gourand, F. / Kerverdo, S. / Barre, L. et al. | 2005
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P04-19 MICROPET IMAGING OF THE BRAIN SEROTONIN TRANSPORTER WITH [^1^1C]mZIENTStehouwer, J. S. / Jarkas, N. / Zeng, F. / Voll, R. J. / Williams, L. / Votaw, J. R. / Goodman, M. M. et al. | 2005
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P04-24 RADIOSYNTHESIS OF 1-[^1^1C]-D-AND L-LACTIC ACID AS POTENTIAL MARKERS OF NEURONAL LACTATE METABOLISMDrandarov, K. / Westera, G. / Wyss, M. / Schubiger, P. A. et al. | 2005
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P04-31 [^1^1C]-METHYLATED LY2181308, AN ANTISENSE OLIGONUCLEOTIDE TO SURVIVIN: RADIOCHEMICAL SYNTHESIS AND PRELIMINARY RODENT BIODISTRIBUTION STUDIESDence, C. S. / Sun, X. / Mach, R. H. / Welch, M. J. et al. | 2005
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P04-56 16alpha,17beta-DIOXOLANE BROMINE-AND IODINE-SUBSTITUTED PROGESTIN FOR BREAST TUMOR IMAGING AND RADIOTHERAPY: SYNTHESISZhou, D. / Carlson, K. E. / Mach, R. H. / Katzenellenbogen, J. A. / Welch, M. J. et al. | 2005
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P04-57 RADIOCHEMICAL PURITY AND SPECIFIC ACTIVITY MEASUREMENTS OF [^1^1C]METHYL TRIFLATE USING ONLY A FLAME IONIZATION DETECTORMock, B. H. / Sullivan, M. L. / DeGrado, T. R. et al. | 2005
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P04-77 OPTIMISATION OF THE SEPARATION OF [^1^8F]FLUOROBROMOMETHANE AND DIBROMOMETHANE USING DISTRIBUTION GAS CHROMATOGRAPHYLehel, S. / Madsen, J. / Gillings, N. et al. | 2005
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P04-82 MODIFICATIONS IN SYNTHESIS OF [^1^8F]-PEPTIDES AND APPLICATION TO SUBSTANCE PHorvath, G. M. / Popkov, A. / Elsinga, P. H. et al. | 2005
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P04-86 FLUORINE-18 LABELLED AROMATIC AMINO ACIDS FOR TUMOR IMAGING USING PETChirakal, R. V. / Ashique, R. / Schrobilgen, G. J. / Vasdev, N. / Gulenchyn, K. V. / Farncombe, T. H. et al. | 2005
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P04-101 SYNTHESIS OF [^1^8F]FLUOROMETHYLSPIPERONE ([^1^8F]FMSP) VIA [^1^8F]FLUOROMETHYL TRIFLATE SYNTHESISKim, H. W. / Jeong, J. M. / Lee, H. J. / Chung, K. H. / Oh, C. H. / Cho, J.-H. / Lee, D. S. / Chung, J.-K. / Lee, M. C. et al. | 2005
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P04-100 SYNTHESIS OF N-SUBSTITUTED 9-AZABICYCLO[3.3.1]NONAN-3alpha-YL PHENYLCARBAMATE ANALOGS AS SIGMA-2 RECEPTOR LIGANDSVangveravong, S. / Xu, J. / Wheeler, K. T. / Mach, R. H. et al. | 2005
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P06-02 EVALUATION OF [N-METHYL-^1^1C]PK 11195 FOR DETECTION OF BREAST CANCERShockley, S. E. / Moerlein, S. M. / Adams, S. G. / Welch, M. J. et al. | 2005
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P06-07 TARGETED IMAGING OF PANCREAS beta-CELLACTIVITY WITH ^9^9^mTc-LABELED NATEGLINIDEAzhdarinia, A. / Oh, C. / Kohanim, S. / Chanda, M. / Yu, D.-F. / Ito, M. / Bryant, J. L. / Kim, E. E. / Yang, D. J. et al. | 2005
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P06-16 CHARACTERIZATION OF IN VIVO RAT METABOLITES OF [O-METHYL-^1^1C]RWAY BY LC-MSShetty, H. U. / Zoghbi, S. S. / McCarron, J. A. / Liow, J.-S. / Hong, J. / Pike, V. W. et al. | 2005
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P06-21 PRECLINICAL STUDIES OF 3'-DEOXY-3'-[^1^8F]FLUOROTHYMIDINEOh, S. J. / Chi, D. Y. / Im, K. C. / Kang, S. H. / Ryu, J. S. / Kim, S. Y. / Lim, S. J. / Moon, D. H. et al. | 2005
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P06-26 AN EASY METHOD FOR NO-CARRIER-ADDED ^1^8F-LABELING OF RGD PEPTIDE: HYDRAZONE FORMATION BETWEEN cRGDyK-HYNIC AND 4-[^1^8F]FLUOROBENZALDEHYDE (FBA)Lee, Y.-S. / Jeong, J. M. / Kim, H. W. / Chang, Y. S. / Ganasha, B. R. / Suh, Y.-G. / Chi, D. Y. / Kang, W. J. / Kang, J. H. / Lee, D. S. et al. | 2005
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P06-29 SYNTHESIS AND IN VITRO BINDING AFFINITY OF PEGYLATED MULTIDENTATE cRGDyK PEPTIDELee, Y.-S. / Jeong, J. M. / Hong, M. K. / Chang, Y. S. / Ganesha, B. R. / Kang, W. J. / Kang, J. H. / Lee, D. S. / Chung, J.-K. / Lee, M. C. et al. | 2005
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P07-03 RHODIUM (III) COMPLEXATION WITH TETRADENTATE ACYCLIC N~2S~2 LIGANDSAkgun, Z. / Engelbrecht, H. / Cutler, C. S. / Barnes, C. L. / Jurisson, S. S. / Lever, S. Z. et al. | 2005
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P07-05 A BORON-BASED SYTHESIS OF [^1^2^3^I^]IODOSTYRYLBENZOXAZOLE, A POTENTIAL SPECT AGENT FOR IMAGING AMYLOID PLAQUES IN THE BRAINMereddy, A. R. / Kabalka, G. W. et al. | 2005
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P07-09 ADDITION OF METHIONINE TO RADIOHALOGENATION REACTIONS OF BIOTIN DERIVATIVES DECREASES FORMATION OF BIOTIN SULFOXIDE BY OXIDANTSWilbur, D. S. / Hamlin, D. K. / Chyan, M.-K. et al. | 2005
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DEVELOPMENT OF RADIOTRACERS FOR MEASURING THE FUNCTION OF MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN IN THE BRAIN IN VIVOOkamura, T. / Kikuchi, T. / Fukushi, K. / Arano, Y. / Irie, T. et al. | 2005
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IMPROVEMENT AND QUALITY CONTROL OF ^6^2Zn/^6^2Cu GENERATOR BASED ON CATION EXCHANGE METHODSFukumura, T. / Okada, K. / Nakao, R. / Suzuki, H. / Mukai, K. / Szelecsenyi, F. / Kovacs, Z. / Suzuki, K. et al. | 2005
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NEW METHODS FOR HALOGENATION OF [^1^8F]-FLUORINATED BENZYL DERIVATIVESKech, C. / Lemaire, C. / Brichard, L. / Plenevaux, A. / Luxen, A. et al. | 2005
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SYNTHESIS AND EVALUATION OF ^1^8F-LABELED FIMPYD AS A PET IMAGING AGENT FOR beta-AMYLOID PLAQUESZeng, F. / Southerland, J. A. / Voll, R. J. / Votaw, J. R. / Williams, L. / Ciliax, B. J. / Goodman, M. M. et al. | 2005
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AN IN VITRO ASSAY TO EVALUATE beta-AMYLOID LIGANDS USING ISOLATED HUMAN AMYLOID PLAQUES OF ALZHEIMER'S DISEASE BRAINCai, L. / Nichols, L. / Temme, S. / Park, K. / Herman, M. M. / Pike, V. W. / Innis, R. B. et al. | 2005
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^1^1^1In-Bz-DTPA-Z~H~E~R~2~:~3~4~2, A CANDIDATE FOR IMAGING FOR HER2-EXPRESSION IN MALIGNANT TUMORSOrlova, A. / Nilsson, F. / Magnusson, M. / Gedda, L. / Widstrom, C. / Wennborg, A. / Tolmachev, V. et al. | 2005
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SYNTHESIS OF ^1^2^3I-RADIOPHARMACEUTICALS WITH THE LABEL IN A BRIDGEHEAD POSITIONHerscheid, J. D. M. / Verbeek, J. / Booij, J. et al. | 2005
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P01-21 NORCHLORO-[^1^8F]FLUOROHOMOEPIBATIDIN: PET EVALUATION OF TRACER PROPERTIES IN PIGSPatt, J. T. / Deuther-Conrad, W. / Brust, P. / Patt, M. / Sabri, O. / Steinbach, J. et al. | 2005
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P01-36 SYNTHESIS OF 5-[^1^1C]ETHYL-A85380 ([^1^1C]5EA) AS A BRAIN NICOTINIC ACETYLCHOLINE RECEPTOR IMAGING AGENT FOR POSITRON EMISSION TOMOGRAPHYOgawa, M. / Nishiyama, S. / Tsukada, H. / Iida, Y. / Saji, H. / Magata, Y. et al. | 2005
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P02-09 MINIMIZING ISOTOPICALLY ENRICHED [N-15]NITROGEN GAS USAGE IN THE PRODUCTION OF O-15 LABELLED WATERPowell, J. / Ramsey, C. A. / Miner, R. / O Neil, J. P. et al. | 2005
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P03-09 BIODISTRIBUTION OF [^2^2^7Th]EDTMP: COMPARISON WITH [^2^2^7Th]CITRATE, [^1^5^3Sm]EDTMP, AND [^2^2^3Ra]CHLORIDEWashiyama, K. / Amano, R. / Sasaki, J. / Ogawa, D. / Kinuya, S. / Tonami, N. / Shiokawa, Y. / Mitsugashira, T. et al. | 2005
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P04-07 RADIOSYNTHESIS AND IN VIVO EVALUATION OF N-[^1^1C]-METHYLATED IMIDAZOPYRIDINE DERIVATIVES AS POSITRON EMISSION TOMOGRAPHY TRACER FOR PERIPHERAL BENZODIAZEPINE RECEPTORSSekimata, K. / Hatano, K. / Ogawa, M. / Abe, J. / Magata, Y. / Biggio, G. / Serra, M. / Trapani, G. / Ito, K. et al. | 2005
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P04-28 RADIOSYNTHESES OF 2-[^1^8F]FLUORO-1,3-THIAZOLESSimeon, F. G. / Pike, V. W. et al. | 2005
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P04-53 PREPARATION OF A REVERSIBLE EGFR INHIBITOR, [^1^1C]CIRC, AS A PET RADIOTRACER FOR TUMOR IMAGINGOwino, N. O. / Shao, X. / Papachristou, M. / Snyder, S. E. et al. | 2005
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P04-60 DEVELOPMENT OF [^1^3N]CISPLATIN FOR CHEMOTHERAPY EVALUATIONYang, X. / Wegman, T. D. / Hendrikse, H. / Elsinga, P. H. et al. | 2005
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P04-67 MEASUREMENT OF BRAIN UPTAKE OF 2-[METHYL-^1^1C]METHOXYESTRADIOL BY MICROPETMun, J. / Kang, S.-H. / Shim, H. / Voll, R. / Williams, L. / Votaw, J. R. / Goodman, M. M. et al. | 2005
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P04-84 A PRACTICAL SYNTHESIS OF [^1^1C]ACETYLENENazih, R. / Blauser, J. P. / Mock, B. H. / DeGrado, T. R. et al. | 2005
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P04-87 NO-CARRIER-ADDED SPECIFIC ACTIVITY (NCA-SA) OF IODINE-124 RADIOPHARMACEUTICALSYordanov, A. T. / Ylimaki, R. / Kiselev, M. et al. | 2005
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P04-99 PET IMAGING OF PANCREATIC CANCER USING Cu-64 LABELLED DOTA-PNA-PEPTIDE CHIMERAZhang, K. / Aruva, M. R. / Mathew, B. / Chakrabarti, A. / Cardi, C. / Wickstrom, E. / Thakur, M. et al. | 2005
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P05-05 CYCLOPENTADIENYLTRICARBONYL RHENIUM(I) AND TECHNETIUM(I) COMPLEXES CONTAINING PENDANT GLUCOSE DERIVATIVESAdam, M. J. / Fisher, C. L. / Orvig, C. / Ewart, C. / Patrick, B. O. et al. | 2005
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P05-31 STUDY ON TWO ^9^9^mTc-NITRIDE HETEROCOMPLEXES AS NOVEL POTENTIAL MYOCARDIAL PERFUSION IMAGING AGENTSChu, J. / Li, B. / Kong, D. / Zhang, J. / Wang, X. et al. | 2005
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P06-11 THE NET RADIOLIGAND (S,S)-[^1^1C]MeNER PRODUCES A LIPOPHILIC LABELED METABOLITE MEASURED IN HUMAN PLASMASchou, M. / Pike, V. W. / Andree, B. / Gulyas, B. / Shchukin, E. / Farde, L. / Halldin, C. et al. | 2005
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P07-10 TOWARDS THE VISUALIZATION OF PERIPHERAL BENZODIAZEPINE RECEPTOR BY SPECTBennacef, I. / Haile, C. N. / Koren, A. O. / Staley, J. K. / Bois, F. / Baldwin, R. M. / Tamagnan, G. D. et al. | 2005
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P07-11 HYDRALINK IS SUPERIOR TO EDC IN PRESERVATION OF AFFINITY OF AN ANTI-PSMA ANTIBODY IN THE CONJUGATION WITH MORPHOLINOSLiu, G. / Dou, S. / He, J. / Knoz, R. / Liu, X. / Wang, Y. / Holmes, E. / Rusckowski, M. / Hnatowich, D. J. et al. | 2005
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P08-10 RENAL ACCUMULATION OF 3-[^1^2^5I]IODO-L-ALPHA-METHYL-TYROSINE IN EXPERIMENTAL FANCONI SYNDROMEShikano, N. / Nakajima, S. / Kotani, T. / Itoh, Y. / Fujimoto, S. / Yagi, A. / Nobayshi, Y. / Nishii, R. / Yoshimoto, M. / Kobayashi, M. et al. | 2005
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P08-15 SYNTHESIS OF RADIOIODINE-LABELED CP-118,954 FOR THE IN VIVO STUDIES OF ACETYLCHOLINESTERASERyu, E. K. / Choe, Y. S. / Choi, B. W. / Choi, Y. / Lee, K. H. / Kim, B. T. et al. | 2005
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P08-23 GSK'S AUTOMATED PET RADIOTRACER SYNTHESIS SYSTEMSBonasera, T. A. / Passchier, J. / Martarello, L. / James, P. J. / Lovegrove, J. W. / Plisson, C. / Gee, A. D. et al. | 2005
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P08-22 PHENOMENOLOGICAL BUILDING BLOCKS: CHAINING BACKWARDS FROM METABOLITESO Halloran, R. L. / Corradini, N. A. / Taurisia, R. / Durkee, B. Y. / Dallas, C. B. / Avila-Rodriguez, M. A. / Converse, A. K. / de Jesus, O. T. / Nickles, R. J. et al. | 2005
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P08-25 FULLY AUTOMATIC PREPARATION OF 16alpha-[^1^8F]FLUOROESTRADIOLKang, S. H. / Oh, S. J. / Mosdzianowski, C. / Chi, D. Y. / Ryu, J. S. / Moon, D. H. et al. | 2005
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P08-27 A HIGHLY FLEXIBLE MODULAR RADIOCHEMISTRY SYSTEMGillings, N. / Larsen, P. et al. | 2005
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RADIOLABELED PHENETHYLGUANIDINES: NOVEL MARKERS OF CARDIAC SYMPATHETIC NEURONS AND ADRENERGIC TUMORSRaffel, D. M. / Jung, Y.-W. / Gildersleeve, D. L. / Chen, W. et al. | 2005
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FDA APPROVAL OF NEW DRUG APPLICATION (NDA) FOR FLUDEOXYGLUCOSE F18 INJECTION (FDG)Vallabhajosula, S. / Kothari, P. J. / Goldsmith, S. J. et al. | 2005
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^1^1C-C BOND FORMATION BY PALLADIUM-MEDIATED CROSS COUPLING OF ALKENYLZIRCONOCENES WITH [^1^1C]METHYL IODIDEWuest, F. / Berndt, M. et al. | 2005
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ISO-STRUCTURAL FLUORESCENT AND ^9^9^mTc PROBES FOR LABELING BIOMOLECULESSchaffer, P. / Guenther, K. J. / Banerjee, S. R. / Zubieta, J. / Babich, J. W. / Valliant, J. F. et al. | 2005
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SELECTIVITY OF THE SIGMA RECEPTOR LIGANDS FOR TUMOR VERSUS INFLAMMATION IN A RODENT MODEL: A COMPARISON WITH FLT AND FDGvan Waarde, A. / Elsinga, P. H. et al. | 2005
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P01-06 EX VIVO EVALUATION OF p-[^1^8F]D-MPPF FOR THE STUDY OF 5-HT~1~A RECEPTORSDefraiteur, C. / Lemaire, C. / Luxen, A. / Plenevaux, A. et al. | 2005
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P01-28 NEW FLUORO-DIPHENYL CHALCOGEN DERIVATIVES TO EXPLORE THE SERT BY PETVercouillie, J. / Deuther-Conrad, W. / Scheunemann, M. / Brust, P. / Steinbach, J. et al. | 2005
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P02-10 AN IMPROVED QUALITY CONTROL PROCEDURE FOR [^1^8F]FDG BY HPLC WITH UV DETECTIONNakao, R. / Ito, T. / Suzuki, K. et al. | 2005
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P03-01 ELEVATION OF 3-[^1^2^5I]IODO-alpha-METHYL-L-TYROSINE TISSUE ACCUMULATION BY REGULATION OF RENAL EXCRETION WITH OAT INHIBITORSKawai, K. / Yoshimoto, M. / Nishii, R. / Kobayashi, M. / Nakajima, S. / Shikano, N. / Tokunaga, J. / Nagamachi, S. / Takamura, N. et al. | 2005
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P03-07 DOTA-OLIGOMERS CONJUGATED TO OCTREOTATE: THE INFLUENCE OF THE NUMBER OF CHELATES ON RECEPTOR BINDING AND BIODISTRIBUTIONMier, W. / Graham, K. / Kramer, S. / Eisenhut, M. / Haberkorn, U. et al. | 2005
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P04-23 N.C.A. ^1^8F-FLUORINATION OF VARIOUS ARENES VIA ARYL(2-THIENYL)IODONIUM SALTSRoss, T. / Ermert, J. / Coenen, H. H. et al. | 2005
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P04-25 SYNTHESIS AND IN VIVO CHARACTERIZATION OF ^7^6Br-LABELED FLUTAMIDE AND BICALUTAMIDE ANALOGSParent, E. / Jenks, C. / Sharp, T. / Katzenellenbogen, J. / Welch, M. et al. | 2005
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P04-33 RADIOSYNTHESIS OF NOVEL COPPER (II) BIS(THIOSEMICARBAZONES) PET TRACERSDonnelly, P. S. / Golovko, O. / Heslop, J. M. / Burke, P. / Clark, J. C. / Dilworth, J. R. / Aigbirhio, F. I. et al. | 2005
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P04-90 DETERMINATION OF THE CHEMICAL PURITY OF [C-11]CHOLINEJacobson, M. S. et al. | 2005
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P04-91 NOVEL FLUORINE-18 LABELED ESTROGEN RECEPTOR LIGAND: FLUOROALKYL CYCLOFENILANALOGUESSeo, J. W. / Chi, D. Y. / Dence, C. C. / Sharp, T. L. / Welch, M. J. / Katzenellenbogen, J. A. et al. | 2005
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P05-09 STABILIZATION OF TECHNETIUM-99m RADIOPHARMACEUTICALS USING HYDROPHILIC THIOETHERSCyr, J. E. / Pearson, D. A. / Lister-James, J. / Dinkelborg, L. et al. | 2005
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P05-19 PREPARATION AND EVALUATION OF INDIRECTLY ^9^9^mTc-LABELED ANTI-HUMAN GASTRIC CANCER MONOCLONAL ANTIBODY 3H11Jia, B. / Liu, Z. / Zhao, H. / Yang, Z. / Wang, F. et al. | 2005
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P05-18 A ^9^9^mTc-TRICARBONYL COMPLEX WITH A CONJUGATE OF 2-PICOLYLAMINE-N-ACETIC ACID AND 2-(4-CHLOROPHENYL)TROPANE AS A POTENTIAL DOPAMINE TRANSPORTER TRACER AGENTKieffer, D. / de Groot, T. / Vanbilloen, H. / Cleynhens, B. / Rattat, D. / Bormans, G. / Verbruggen, A. et al. | 2005
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P05-23 PREPARATION, CHARACTERIZATION AND BIODISTRIBUTION OF A NEW TECHNETIUM-99m COMPLEX WITH HYNIC(TRICINE)-AMDPLiu, L. / Guo, H. / Tang, Z. / Lu, J. / Wang, X. et al. | 2005
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P05-26 INFLUENCE OF Aryl SUBSTITUENTS ON THE REACTIVITY OF ^9^9^mTc COMPLEXES OF TETRAFLUORPHENOL -3,5-DIAMINOBENZOATE DERIVATIVESCalderon Sanchez, O. / Bauer, C. / Mohammed, A. / Haberkorn, U. / Mier, W. / Eisenhut, M. et al. | 2005
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P07-12 SYNTHESIS, RADIOIODINATION AND EVALUATION OF NEW MGMT-INHIBITORS AND THEIR GLUCOSE CONJUGATESMuehlhausen, U. / Schirrmacher, R. / Piel, M. / Kaina, B. / Roesch, F. et al. | 2005
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P08-21 METABOLITE STUDY OF 2-[^1^1C]METHYL-6-(2-PHENYLETHYNYL)PYRIDINE, 2-(2-(3-[^1^1C]METHOXYPHENYL)ETHYNYL)-6-METHYLPYRIDINE, AND 2-(2-(5-[^1^1C]METHOXYPYRIDIN-3-YL)ETHYNYL)PYRIDINE, POTENTIAL PET LIGANDS FOR METABOTROPIC GLUTAMATE SUBTYPE 5 RECEPTORSYu, M. / Wang, X. / Zhu, A. / Brownell, A.-L. et al. | 2005
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RADIOSYNTHESIS AND EVALUATION OF (+)[^1^1C]PHNO AS RADIOTRACER FOR IN VIVO IMAGING OF THE DOPAMINE D2 HIGH AFFINITY STATE WITH POSITRON EMISSION TOMOGRAPHY (PET)Wilson, A. A. / Kapur, S. / McCormick, P. / Garcia, A. / Hussey, D. / Willeit, M. / Houle, S. / Ginovart, N. et al. | 2005
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AN INDIUM-LABELED DO3A CONJUGATE OF NALTRINDOLE HIGH WITH AFFINITY AND SELECTIVITY FOR DELTA OPIOID RECEPTORS: SYNTHESIS, BINDING STUDIES AND BIODISTRIBUTIONDuval, R. A. / Allmon, R. L. / Gustafson, J. L. / Carmack, T. L. / Watkinson, L. D. / Lever, J. R. et al. | 2005
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EXPERIENCE WITH DOUBLE-GRID NIOBIUM [^1^8O]H~2O TARGET FOR HIGH YIELD OF [^1^8F]FLUORIDE PRODUCTION WITH CYCLONE-30Hur, M. G. / Kim, S. W. / Hong, B. H. / Chai, J. S. / Park, J. H. / Yang, S. D. / Yu, K. H. / Oh, H. S. et al. | 2005
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SYNTHESIS OF [^1^1C]OXAZOLIDONE IN AN ISOCYANATE INTERMEDIATE RHODIUM-MEDIATED CARBONYLATION REACTION USING [^1^1C]CARBON MONOXIDEBarletta, J. / Karimi, F. / Doi, H. / Langstrom, B. et al. | 2005
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A NEW CARBON-11 LABELLING METHOD USING [^1^1C]-MONOORGANOTIN REAGENTHuiban, M. / Sobrio, F. / Fouqout, E. / Barre, L. / Perrio, C. et al. | 2005
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FLUORINE-18-LABELING OF PEPTIDES AND PROTEINS USING [^1^8F]FPyME, A [^1^8F]FLUOROPYRIDINE-BASED MALEIMIDE REAGENTKuhnast, B. / de Bruin, B. / Hinnen, F. / Boisgard, R. / Johannes, L. / Samson, A. / Tavitian, B. / Dolle, F. et al. | 2005
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P01-14 SYNTHESIS AND IN VIVO EVALUATION OF ARYLALKYL 4-BENZYL PIPERAZINES AS RADIOLIGAND SIGMA RECEPTORSKassiou, M. / Pham, T. / Fulton, R. / Mattner, F. / Henderson, D. / Katsifis, A. / Liu, X. / Eberl, S. / Greguric, I. / Fulham, M. et al. | 2005
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P01-32 FLUORINE-18 LABELED BENZAZEPINES FOR IMAGING DOPAMINE D1 RECEPTORSWang, C. S. / Collins, D. / Mukherjee, J. et al. | 2005
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P02-02 EVALUATION OF POLYOXOMETALATES TO EXTRACT LANTHANIDESFrancesconi, L. / Howell, R. / Jones, I. R. / Cutler, C. S. et al. | 2005
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P03-02 Ho-166 LABELED DTPA DERIVATIVE FOR INTRAVASCULAR RADIATION THERAPY WITH LIQUID BALLOONS: DUAL-FUNCTIONAL COMPLEX FOR RESTENOSIS PREVENTION AND CT IMAGINGHong, Y.-D. / Choi, O.-J. / Choi, S.-M. / Choi, S.-J. et al. | 2005
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P03-04 PREPARATION AND EVALUATION OF ^1^7^7Lu-CHX-A"-DTPA-ABD-(Z~H~E~R~2~:~3~4~2)~2 AFFIBODY MOLECULE FOR RADIONUCLIDE THERAPY OF DISSEMINATED HER2-EXPRESSING TUMORSTolmachev, V. / Orlova, A. / Magnusson, M. / Lundqvist, H. / Johansson, K. / Baastrup, B. / Wennborg, A. / Nilsson, F. et al. | 2005
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P03-06 TUMOR RESPONSE AND SIDE EFFECTS AFTER [^1^7^7Lu-DOTA,Tyr^3]OCTREOTATE THERAPY IN RATSDe Jong, M. / Bernard, B. / Breeman, W. / Krenning, E. et al. | 2005
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P03-12 MORPHOLINO OLIGOMERS CAN BE RADIOLABELED WITH ^1^8^8Re AT HIGH SPECIFIC ACTIVITY USING MAG~3Liu, G. / Dou, S. / He, J. / Zhang, S. / Wang, Y. / Rusckowski, M. / Hnatowich, D. et al. | 2005
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P04-01 SYNTHESIS, RADIOLABELLING AND BIOLOGICAL EVALUATION OF SYN-[^1^8F]FACBC AS A POTENTIAL TUMOR IMAGING AGENTYu, W. / Camp, V. M. / Zhang, Z. / Kurosaki, F. / Goodman, M. M. et al. | 2005
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P04-21 STRUCTURE-ACTIVITY RELATIONSHIP STUDY OF IMPY DERIVATIVES AS CANDIDATE RADIOLIGANDS FOR beta-AMYLOIDCai, L. / Nichols, L. / Cuevas, J. / Temme, S. / Herman, M. M. / Innis, R. B. / Pike, V. W. et al. | 2005
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P04-45 PREPARATION OF N.C.A. [^1^8F]FLUOROPHENYLUREASOlma, S. / Ermert, J. / Coenen, H. H. et al. | 2005
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P04-51 A NEW MILD METHOD FOR THE ONE-POT SYNTHESIS OF [2-^1^1C]THYMINE USING [^1^1C]PHOSGENESeki, K.-I. / Sanoki, K. / Nishijima, K.-I. / Kuge, Y. / Tamaki, N. / Ohkura, K. et al. | 2005
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P04-58 PROCESSING OF ^6^8Ge/^6^8Ga GENERATOR ELUATES FOR LABELING OF BIOMOLECULES VIA BIFUNCTIONAL CHELATORSZhernosekov, K. P. / Filosofov, D. V. / Jahn, M. / Jennewein, M. / Roesch, F. et al. | 2005
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P04-65 PRODUCTION OF [^1^8F]SPA-RQ AS A PET RADIOLIGAND FOR IMAGING HUMAN BRAIN NK~1 RECEPTORSChin, F. T. / Morse, C. L. / Pike, V. W. et al. | 2005
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P04-92 SYNTHESIS AND IN VIVO CHARACTERIZATION OF ^1^8F LABELED NON-STEROIDALANDROGENSParent, E. / Dence, C. / Seo, J. W. / Sharp, T. / Chi, D. Y. / Katzenellenbogen, J. / Welch, M. et al. | 2005
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P04-93 THE TRACERLAB MAXIMUM (Mx) IS ALSO A FLEXIBLE (Fx) TOOLTadino, V. / Kothari, P. / Le Bars, D. / Villeret, G. / Tesoriere, G. / Ignace, G. / Vallabhajosula, S. / Buono, S. et al. | 2005
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P04-96 EVALUATION OF COMMERCIALAUTOMATED [^1^1C]METHYL IODIDE (MEI-PLUS) SYNTHESIS MODULEKothari, P. J. / Suehiro, M. / Vallabhajosula, S. / Finn, R. et al. | 2005
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P05-12 CYCLOPENTADIENYL RHENIUM (TECHNETIUM) TRICARBONYL COMPLEXES INTEGRATED IN ESTROGEN RECEPTOR (ER) LIGANDS FOR ER+ TUMOR IMAGINGAckroyd, N. C. / Katzenellenbogen, J. A. et al. | 2005
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P05-27 DEVELOPMENT OF BIFUNCTINAL CHELATES WITH ALIPHATIC AMINE DONORS FOR THE COMPLEXATION WITH THE {M(CO)~3}^+ CORE (M = Re, ^9^9^mTc)Lipowska, M. / He, H. / Xu, X. / Marzilli, L. G. / Taylor, A. et al. | 2005
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P06-05 A CANDIDATE HIGH AFFINITY beta~1-ADRENOCEPTOR-SELECTIVE PET RADIOLIGAND: (S)-[METHOXY-^1^1C]-N-[2-[3-(2-CYANO-PHENOXY)-2 -HYDROXY-PROPYLAMINO]-ETHYL]-N'-(4-METHOXY-PHENYL)-UREA (S)-[^1^1C]ICI-OMe)Kopka, K. / Law, M. P. / Engelhardt, S. / Riemann, B. / Pike, V. W. / Schober, O. / Schaefers, M. / Wagner, S. et al. | 2005
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P06-04 EVALUATION OF ^6^4Cu- AND ^8^6Y-LABELED DOTA-(Pro^1, Tyr^4)-BOMBESIN(1-14) A BOMBESIN ANALOGUE FOR TARGETING GRP RECEPTORSBiddlecombe, G. B. / de Visser, M. / de Jong, M. / Rogers, B. E. / Lewis, J. S. et al. | 2005
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P06-10 POST MORTEM AUTORADIOGRAPHY OF THE HUMAN BRAIN NOREPINEPHRINE TRANSPORTER WITH (S,S)-[^1^8F]FMeNER-D~2Schou, M. / Halldin, C. / Pike, V. W. / Mozley, P. D. / Dobson, D. / Innis, R. B. / Farde, L. / Hall, H. et al. | 2005
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P06-24 SYNTHESIS AND IN VITRO EVALUATION OF ^1^1^1In-DOTA-anti-bcl-2-PNA-Tyr^3-OCTREOTATE IN CHRONIC LYMPHOCYTIC LEUKEMIA CELLSJia, F. / Gallazzi, F. / Lever, S. Z. / Hannink, M. / Lewis, M. R. et al. | 2005
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P07-06 SYNTHESIS AND RADIOIODINATION OF A PNA CONTAINING AN [^1^2^5I]IODOURACIL MOIETYWilbur, D. S. / Chyan, M.-K. / Hamlin, D. K. / Hobbs, J. et al. | 2005
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P07-14 111-INDIUM LABELED POLYMERIC MICELLES AS NOVEL DRUG DELIVERY SYSTEM FOR MICRO-SPECT/CT IMAGINGTian, H. / Shuai, X. / Gao, J. / Lee, Z. et al. | 2005
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P08-02 MONITORING IN-VIVO GENE TRANSFER: PET OR BIOLUMINESCENCE?Buursma, A. R. / van Waarde, A. / Beerens, A. M. J. / Vaalburg, W. / Haisma, H. J. / Hospers, G. A. P. / Mulder, N. H. / de Vries, E. F. J. et al. | 2005
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P08-20 SYNTHESES OF [^1^8F] LABELED (2S, 3S, 4R)-2-(N-6-[^1^8F]FLUOROHEXANOYLAMINO)-AND 8-[^1^8F]FLUOROOCTANOYLAMINO)OCTADECANE-1,3,4-TRIOLMoon, B. S. / Lee, K. C. / An, G. I. / Yang, S. D. / Chun, K. S. et al. | 2005
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P08-28 INTERNAL CYCLOTRON TARGETS FOR CLINICAL PRODUCTION OF BROMINE RADIONUCLIDESSzajek, L. P. / Plascjak, P. / Eckelman, W. et al. | 2005
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PREPARATION OF CYCLOTRON Re-186 AND COMPARISON WITH REACTOR Re-186 AND GENERATOR Re-188 FOR THE LABELING OF BOMBESINEhrhardt, G. J. / Moustapha, M. E. / Smith, C. J. / Szajek, L. / Eckelmann, W. C. / Jurisson, S. S. et al. | 2005
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LABELLING VIA FREE RADICAL CARBONYLATION USING ^1^1COItsenko, O. / Langstrom, B. et al. | 2005
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EVALUATION OF NOVEL SELENOLTHIOL AND DITHIOL SEL-TAG VARIANTS FOR PURIFICATION AND ^1^1C-LABELING OF RECOMBINANT PROTEINS PRODUCED IN E. COLICheng, Q. / Johansson, L. / Fredriksson, A. / Thorell, J.-O. / Stone-Elander, S. / Arner, E. S. J. et al. | 2005
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DIFFERENTIAL BRAIN UPTAKE OF THE D/L-ISOMERS OF ALANINE, SERINE, PROLINE AND CIS-4-[^1^8F]FLUOROPROLINE AS POTENTIAL TRACERS FOR PETBauer, D. / Hamacher, K. / Langen, K. J. / Pauleit, D. / Herzog, H. / Coenen, H. H. et al. | 2005
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A NEW STRATEGY FOR LABELING BIOMOLECULES THAT CONTAIN DISULFIDE BONDS WITH RHENIUM AND TECHNETIUMGuenther, K. J. / Schaffer, P. / Yoganathan, S. / Chirakal, R. V. / Dolovich, M. / Zubieta, J. / Banerjee, S. R. / Babich, J. W. / Valliant, J. F. et al. | 2005
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NUCLEAR IMAGING OF NANOPARTICLES IN XENOGRAFT TUMOR MODELSCho, Y. W. / Park, S. A. / Lee, M. / Park, J. S. / Son, D. H. / Oh, S. J. / Moon, D. H. / Kim, S. Y. / Kwon, I. C. / Kim, I.-S. et al. | 2005
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P01-05 EVALUATION OF [^1^8F]FPWAY AND [^1^8F]FBWAY, 5-HT~1~A RECEPTOR PET LIGANDS, FOR SENSITIVITY TO ENDOGENOUS 5-HT IN RATJagoda, E. M. / Lang, L. / Tokugawa, J. / Ma, Y. / Contoreggi, C. / Eckelman, W. C. et al. | 2005
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P01-16 TOWARDS A METABOLICALLY STABLE FLUORINE-18 PET RADIOTRACER FOR SEROTONIN 5HT~1~A RECEPTORSSaigal, N. / Collins, D. / Pichika, R. / Mukherjee, J. et al. | 2005
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P01-19 EVALUATION OF CLINDE, A RADIOLABELLED PERIPHERAL BENZODIAZEPINE RECEPTOR LIGAND IN A MURINE MODEL OF NEURO-INFLAMMATION: POTENTIAL PROBE FOR ASSESSING NEURODEGENERATIONKatsifis, A. / Mattner, F. / Mana, P. / Linares, D. / Ballantyne, P. / Berghofer, P. / Pham, T. / Willenborg, D. et al. | 2005
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P02-01 NEW PRODUCTION ROUTES FOR SOME THERAPEUTIC RADIONUCLIDESSpahn, I. / Hilgers, K. / Tarkanyi, F. / Coenen, H. H. / Qaim, S. M. et al. | 2005
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P02-07 NEW NUCLEAR DATA FOR PRODUCTION OF ^1^2^4I VIA ^3He AND alpha-PARTICLE INDUCED REACTIONS ON ^n^a^tSb AND ^1^2^1SbHassan, K. F. / Qaim, S. M. / Saleh, Z. A. / Coenen, H. H. et al. | 2005
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P02-08 SEPARATION OF ^1^4^3Pr AND ^1^4^3Ce USING HEXAGONAL TUNGSTEN BRONZE INORGANIC SORBENTSFuchs, A. / Smith, S. V. / Hollis, J. / Thorogood, G. / Griffth, C. et al. | 2005
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P03-08 IMPROVEMENT OF N-ISOPROPYL-p-[^1^2^3I]IODOAMPHETAMINE CEREBRALACCUMULATION BY COMPETITIVE DISPLACEMENT OF SERUM PROTEIN BINDING WITH AMINO-ACID INFUSIONKawai, K. / Kuga, N. / Yoshimoto, M. / Kobayashi, M. / Nishii, R. / Yamazsaki, K. / Shigaki, S. / Nagamachi, S. / Takamura, N. / Tamura, S. et al. | 2005
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P04-04 A NOVEL, HIGHLY EFFICIENT WAY TO PREPARE [^1^8F]FLUOROMETHYL BROMIDEZhao, Y. / Luthra, S. / Brady, F. et al. | 2005
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P04-30 SYNTHESIS AND EVALUATION OF CANDIDATE RADIOLIGANDS FOR THE BRAIN CANNABINOID TYPE-1 (CB~1) RECEPTOR BASED ON 1,5-DIARYLPYRAZOLESDonohue, S. / Halldin, C. / Finnema, S. / Gulyas, B. / Schou, M. / Innis, R. B. / Pike, V. W. et al. | 2005
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P04-37 SYNTHESIS AND STRUCTURE ACTIVITY RELATIONSHIP OF 2,5-DISUBSTITUTED THIOPHENE DERIVATIVES FOR ss-AMYLOID PLAQUE IMAGINGChandra, R. / Kung, M.-P. / Kung, H. F. et al. | 2005
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P04-47 FAST AND MILD AQUEOUS-PHASE REDUCTION OF [^1^1C]FORMIC ACID WITH SAMARIUM DIIODIDE TO [^1^1C]METHANOLRoeda, D. / Dolle, F. et al. | 2005
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P04-66 METABOLISM OF CORTICOTROPIN RELEASING HORMONE TYPE 1 RECEPTOR (CRHR1) PET LIGAND - [^7^6Br]MJL-1-109-2Ma, Y. / Lang, L. / Jagoda, E. M. / Kiesewetter, D. O. / Szajek, L. P. / Kim, B. M. / Greiner, E. / Rice, K. C. / Eckelman, W. C. et al. | 2005
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P04-69 ROUTINE RADIOSYNTHESIS OF [^1^1C]METHYLPHENIDATE: CAN IT BE IMPROVED?Studenov, A. R. / Jivan, S. / Lu, J. / Adam, M. J. / Jensen, S. B. / Ding, Y.-S. et al. | 2005
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P04-72 REGIO- AND STEREOSELECTIVE ELECTROPHILIC FLUORINATION OF 3,4,6-TRI-O-ACETYL-D-GLUCAL (TAG) IN ACIDIC MEDIUMChirakal, R. V. / Ashique, R. / Schrobilgen, G. J. / Hughes, D. W. / Gulenchyn, K. V. et al. | 2005
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P04-89 AUTOMATED SYNTHESIS OF [^1^8F]FLUOROMETHYLCHOLINE (FCH)Morandeau, L. M. / DeGrado, T. R. / McKinney, C. J. / Chan, S. Y. / Meyrick, D. P. / Jones, C. G. / Price, R. I. / Lenzo, N. et al. | 2005
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P05-21 MULTIMERIC FORMS OF P-160, A PEPTIDE IDENTIFIED BY PHAGE DISPLAYKraemer, S. / Askoxylakis, V. / Zhang, J. / Zitzmann, S. / Eisenhut, M. / Haberkorn, U. / Mier, W. et al. | 2005
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P05-25 THE STUDY OF ^9^9^mTc MOEDP AS A NEW BONE IMAGING AGENTLiu, L. / Wang, X. et al. | 2005
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P05-29 ^9^9^mTc-LABELLED BIGUANIDE DERIVATIVES: CHEMICAL SPECIATION MODELLING OF AND EVALUATION IN VERVETSWagener, J. M. / Zeevaart, J. R. / Neves, M. / Costa, M. C. / Rodrigues, C. / Dithebe, M. K. / Knoesen, O. / Louw, W. K. et al. | 2005
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P05-30 A NEW RADIO-TLC METHOD FOR THE QUANTIFICATION OF [^1^8F]ALTANSERIN IN HUMAN PLASMABier, D. / Holschbach, M. H. / Lang, M. / Coenen, H. H. et al. | 2005
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P07-08 SYNTHESIS AND BIOLOGICAL EVALUATION OF [^1^2^3I]QUINONOIDS FOR BRAIN TUMOR IMAGINGPark, J. H. / Kim, S. W. / Lee, H. J. / Yang, S. D. / Chun, K. S. / Yu, K. H. et al. | 2005
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P07-07 SYNTHESIS OF A N-3 SUBSTITUTED THYMIDINE DERIVATIVE FOR LABELING WITH TRIVALENT RADIONUCLIDESSchmid, M. / Vogg, A. T. J. / Neumaier, B. / Reske, S. N. et al. | 2005
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P07-13 RADIOIODINATION OF TALNETANT ANALOGUES FOR SPECT IMAGING STUDIES OF NK-3 RECEPTORBennacef, I. / Perrio, C. / Staley, J. K. / Haile, C. N. / Koren, A. O. / Tamagnan, G. D. / Barre, L. et al. | 2005
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P08-09 PENTABODIES AS NOVEL SCAFFOLDS OF PEPTIDES IDENTIFIED BY PHAGE DISPLAY SCREENING: LABELING AND BIODISTRIBUTIONMier, W. / Zhang, J. / Zitzmann, S. / Askoxylakis, V. / Bell, A. / McKenzie, R. / Eisenhut, M. / Haberkorn, U. et al. | 2005
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P04-29 SYNTHESIS AND BIODISTRIBUTION OF 2-[^3^4^mCl]CHLORO-2-DEOXY-GLUCOSE IN RATFukumura, T. / Takei, M. / Maeda, J. / Suzuki, K. et al. | 2005
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P04-35 SYNTHESIS AND RADIOSYNTHESIS OF [^1^8F]FPhEP AND [^1^8F]F~2PhEP, TWO NOVEL HIGH-AFFINITY AND alpha-4-beta-2-SELECTIVE, EPIBATIDINE-BASED RADIOLIGANDS FOR PET IMAGING OF NICOTINIC ACETYLCHOLINE RECEPTORSRoger, G. / Valette, H. / Hinnen, F. / Saba, W. / Coulon, C. / Ottaviani, M. / Bottlaender, M. / Dolle, F. et al. | 2005
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P04-44 RADIOSYNTHESIS OF 2-[^1^1C]METHOXY-3-METHOXY-5-(2'-PROPENYL)-N-[[(2S)-1- (2-PROPENYL)-2-PYRROLIDINYL]METHYL]BENZAMIDE AS A NEW RADIOTRACER FOR DOPAMINE D-2/D-3 RECEPTORSShi, B. / Narayanan, T. K. / Christian, B. T. / Mukherjee, J. et al. | 2005
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P04-49 RADIOSYNTHESIS OF (E)-N-(2-[^1^1C]METHOXYBENZYL)-3-PHENYL-ACRYLAMIDINE, A NOVEL SUBNANOMOLAR NR2B-SUBTYPE SELECTIVE NMDA RECEPTOR LIGANDThominiaux, C. / de Bruin, B. / Bramoulle, Y. / Hinnen, F. / Demphel, S. / Besret, L. / Bottlaender, M. / Valette, H. / Kassiou, M. / Dolle, F. et al. | 2005
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P04-54 SELECTIVE SYNTHESIS OF [2-^1^1C]PROPYLIODIDE AND [1-^1^1C]ETHYL IODIDE USING GRIGNARD REACTION FROM METHYLMAGNESIUM BROMIDEZhang, M.-R. / Ogawa, M. / Yoshida, Y. / Suzuki, K. et al. | 2005
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P04-62 [^1^8F] FESB: AUTOMATED RADIOSYNTHESIS, IMAGING AND beta-AMYLOID PLAQUE STUDIES OF A NOVEL ^1^8F-LABELED PET TRACER IN TRANSGENIC MICE WITH ALZHEIMER'S DISEASEKumar, P. / Zheng, W. / McQuarrie, S. A. / Jhamandas, J. H. / Wiebe, L. I. et al. | 2005
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P04-76 EFFICIENT O-[^1^1C]METHYLATION WITH [^1^1C]METHYL TRIFLATE: SYNTHESIS OF ^1^1C-LABELED DIARYL SUBSTITUTED PYRAZOLE AND IMIDAZOLE CYCLOOXYGENASE INHIBITORSKawamura, K. / Fujisaki, Y. / Ishiwata, K. / Yamamoto, F. / Maeda, M. et al. | 2005
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P05-11 S-TRITYL PROTECTED MERCAPTOACETYL-GLYCYL-GLYCINE-A USEFUL PURIFICATION HANDLE FOR OLIGONUCLEOTIDE-CHELATOR CONJUGATES AS PRECURSORS FOR RADIOLABELING OF APTAMERS WITH Tc(V) AND Re(V)Friebe, M. / Hecht, M. / Graham, K. / Stephens, A. W. / Hilger, C. S. / Johannsen, B. / Dinkelborg, L. M. et al. | 2005
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P05-22 PRELIMINARY STUDY ON THE ^9^9^mTc(CO)~3-PNP5 COMPLEXChu, J. / Kong, D. / Li, B. / Wang, X. et al. | 2005
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P06-08 THE USE OF A BETA PLATE READER FOR RECEPTOR BINDING STUDIES USING ^6^4Cu, ^1^7^7Lu, AND ^1^4^9PmSherman, C. D. / Li, W. P. / Anderson, C. J. et al. | 2005
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P06-12 RADIONUCLIDE THERAPY USING ^1^1^1In-LABELED SOMATOSTATIN ANALOGS; SOMATOSTATIN RECEPTOR EXPRESSION IN A RAT TUMOR MODEL BEFORE AND AFTER THERAPYDe Jong, M. / Capello, A. / Bernard, B. / Breeman, W. / Krenning, E. et al. | 2005
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P06-20 EFFICIENT RADIOSYNTHESIS OF 5-[^1^3^1I]IODO-2'-FLUORODEOXYURIDINES AND BIODISTRIBUTION IN SCID MICE BEARING LYMPHOMAWczasek, K. / Vogg, A. T. J. / Cudek, G. J. / Neumaier, B. / Reske, S. N. et al. | 2005
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P06-22 THE CASPASE INHIBITOR (S)-[1-METHYL-^1^1C]-1-(METHYL)-5-[1-(2-PHENOXYMETHYLPY RROLIDINYL) SULFONYL]ISATIN: A PUTATIVE NONPEPTIDYL CASPASE BINDING RADIOLIGANDFaust, A. / Wagner, S. / Keul, P. / Schober, O. / Levkau, B. / Schaefers, M. / Kopka, K. et al. | 2005
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P08-08 RADIOSYNTHESIS AND EVALUATION OF ^1^8F-AGC393 AS A BIOLOGICAL MARKER OF BETA-AMYLOID DEPOSITSBlagoev, M. / Ametamey, S. M. / Bettio, A. / Mu, L. / Keller, C. / Westera, G. / Wyss, M. / Buck, A. / Treyer, V. / Streffer, J. et al. | 2005
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SYNTHESIS AND EVALUATION OF A NEW ^1^8F-LABELED LIGAND FOR PET IMAGING OF BRAIN PERIPHERAL BENZODIAZEPINE RECEPTORSBriard, E. / Shah, J. / Musachio, J. L. / Zoghbi, S. S. / Fujita, M. / Imaizumi, M. / Cropley, V. / Innis, R. B. / Pike, V. W. et al. | 2005
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A SERIES OF HYDRATED HEXAGONAL TUNGSTEN BRONZE SORBENTS FOR USE IN THE SEPARATION OF RADIOMETALIONSSmith, S. V. / Kennedy, S. J. / Fuchs, A. et al. | 2005
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A CHIEVEING HIGH (APPARENT) SPECIFIC ACTIVITY FORMULATIONS USING FLUOROUS-PHASE CHEMISTRYDonovan, A. C. / Forbes, J. / Babich, J. W. / Valliant, J. F. et al. | 2005
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DEVELOPMENT OF ^1^1^1In-LABELED TUMOR ASSOCIATED ANTIGEN PEPTIDES FOR NON-INVASIVE MONITORING OF DENDRITIC CELL BASED IMMUNOTHERAPYLaverman, P. / de Vries, J. M. / Adema, G. J. / Boerman, O. C. et al. | 2005
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FUTURE QUALITY ASSURANCE STRATEGIES FOR PET RADIOPHARMACEUTICALS AT SUNY BUFFALOHaka, M. S. / Toorongian, S. A. / Lapham, J. M. / Church, S. P. et al. | 2005
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P01-13 C-11 LABELED 6-CHLORO-5-(PYRIDIN-3-YL) ANALOGS OF AZETIDINYLAND PYRROLIDINYL 3-PYRIDYL ETHERS: SYNTHESIS AND EVALUATION AS IN VIVO TRACERS OF NICOTINIC ACETYLCHOLINE RECEPTORFan, H. / Horti, A. G. / Ravert, H. T. / Scheffel, U. A. / Holt, D. P. / Rauseo, P. A. / Xiao, Y. / Kellar, K. J. / Wong, D. F. / Dannals, R. F. et al. | 2005
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P01-18 SYNTHESIS AND RADIOIODINATION OF HALOGENATED BENZAMIDE DERIVATIVES FOR THE NON-INVASIVE VISUALIZATION OF D2-LIKE DOPAMINE RECEPTORSStark, D. / Piel, M. / Bier, D. / Holschbach, M. / Schmitt, U. / Huebner, H. / Gmeiner, P. / Lueddens, H. / Roesch, F. et al. | 2005
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P01-26 N-[^1^8F]FLUOROETHYLPIPERIDIN-4-YLMETHYLACETATE, A ^1^8F-LABELLED PROBE ANALOGOUS WITH [^1^1C]MP4A FOR MEASURING CEREBRALACETYLCHOLINESTERASE ACTIVITYKikuchi, T. / Obayashi, S. / Nagai, Y. / Ming-rong, Z. / Okamura, T. / Suzuki, K. / Tanada, S. / Fukushi, K. / Irie, T. et al. | 2005
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P02-04 SELF-SUFFICIENCY AND OPPORTUNITY COST: NAVIGATING TOWARD EXPANDED DISTRIBUTION OF PET FEEDSTOCKSNye, J. A. / Avila-Rodriguez, M. A. / Dallas, C. B. / Vandehey, N. T. / Weichert, J. P. / Converse, A. K. / Nickles, R. J. et al. | 2005
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P03-03 TUMOR TARGETING USING ^1^7^7Lu-CHX-A"-DTPA-PERTUZUMABPersson, M. / Tolmachev, V. / Andersson, K. / Gedda, L. / Sandstrom, M. / Carlsson, J. et al. | 2005
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P03-15 IMPROVED METHOD FOR LABELING OF ANTI-CEA HUMANIZED CHIMERIC ANTIBODY RCH24 WITH ^1^3^1IYang, Z. / Rang, Y. / Xu, B. / Wang, X. et al. | 2005
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P03-14 PREPARATION OF ^1^8^8Re-HEDP AND ITS PRE-CLINICAL STUDYYin, D. / Zhou, W. / Guo, Z. / Min, X. / Wang, Y. et al. | 2005
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P04-02 C-11 LABELLING AND BIODISTRIBUTION OF AG1478Ackermann, U. / Ardipradja, K. / Lee, F. T. / Tochon-Danguy, H. J. / Young, K. / Scott, A. M. et al. | 2005
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SYNTHESIS AND IN VIVO EVALUATION OF A NOVEL PET RADIOLIGAND FOR IMAGING THE PERIPHERAL BENZODIAZEPINE RECEPTORJames, M. / Fulton, R. / Henderson, D. / Eberl, S. / Fulham, M. / Allan, R. / Thompson, S. / Dolle, F. / Kassiou, M. et al. | 2005
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ACCESS TO REMOTELY CONTROLLED PRODUCTION OF ^8^6Y USING A QUEOUS TARGET MATRICES AS ALTERNATIVE TO SOLID STATE TARGETRYVogg, A. T. J. / Neumaier, B. / Scheel, W. / Reske, S. N. et al. | 2005
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SYNTHESIS, RADIOLABELING AND IN VIVO EVALUATION OF S- AND R- N-Me[^1^8F]FAMP AS PET TUMOR IMAGING CANDIDATESYu, W. / Williams, L. / Malveaux, E. / Camp, V. M. / Zhang, Z. / Goodman, M. M. et al. | 2005
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IN SILICO, IN VITRO AND IN VIVO EVALUATION OF TECHNETIUM-99m AND RHENIUM THYMIDINE COMPLEXES FOR POTENTIAL USE IN SUICIDE GENE THERAPY AND CANCER DIAGNOSISDesbouis, D. / Stichelberger, M. / Spiwok, V. / Scapozza, L. / Schibli, R. et al. | 2005
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CORRELATION OF [1-^1^1C] ACETATE UPTAKE TO FATTY ACID SYNTHASE EXPRESSION IN PROSTATE TUMORSVavere, A. L. / Lewis, J. S. et al. | 2005
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P01-01 mu-OPIOID RECEPTOR TARGETING WITH ^1^8F-LABELED 4-ANILIDOPIPERIDINESHenriksen, G. / Platzer, S. / Berthele, A. / Hauser, A. / Schwaiger, M. / Wester, H.-J. et al. | 2005
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P01-09 DESIGN OF HALOGENATED PIPERIDINES AS SELECTIVE PROBES FOR IMAGING OF MONOAMINE TRANSPORTERSSmith, M. P. / Keith, D. F. / Femia, F. J. / Babich, J. W. et al. | 2005
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P01-17 SYNTHESIS AND EVALUATION OF THIONAPHTHENE DERIVATIVES AS LIGANDS FOR IMAGING beta-AMYLOID PLAQUES IN THE BRAINChang, Y. S. / Jeong, J. M. / Lee, Y.-S. / Cho, J. H. / Oh, C. H. / Lee, D. S. / Chung, J.-K. / Lee, M. C. et al. | 2005
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P03-10 SURFACE MODIFICATION OF THE MAGNETITE NANOPARTICLE AND ITS APPLICATION IN RADIOIMMUNOTHERAPYWang, Y. / Yin, D. / Li, G. / Dong, M. / Cao, J. et al. | 2005
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P04-14 NOVEL F-18 LABELLED AMINOALKYLINDOLE WITH POTENTIAL FOR IMAGING NEURONAL CANNABINOID RECEPTOR BY POSITRON EMISSION TOMOGRAPHYWillis, P. G. / Pavlova, O. A. / Chefer, S. I. / Vaupel, D. B. / Mukhin, A. G. / Horti, A. G. et al. | 2005
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P04-17 SYNTHESIS AND REACTIVITY OF NOVEL ^1^8F-LABELED ARYLSULFONATE ESTERS OF 2-FLUOROETHANOLMusachio, J. L. / Shah, J. / Pike, V. W. et al. | 2005
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P04-22 SYNTHESIS AND IN VIVO EVALUATION OF C-11 LABELED MAZINDOLANALOGS FOR IMAGING THE NOREPINEPHRINE TRANSPORTER WITH PETLin, K.-S. / Ding, Y.-S. / Betzel, T. / Quandt, G. et al. | 2005
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P04-36 SYNTHESIS AND RADIOLABELING OF N-[4-[4-(2-[^1^1C]METHOXYPHENYL)PIPERAZIN-1-YL]BUTYL] BENZO[b]THIOPHENE-2-CARBOXAMIDE, A POTENTIAL RADIOTRACER FOR D3 RECEPTOR IMAGING WITH PETKuhnast, B. / Demphel, S. / Besret, L. / Coulon, C. / Ottaviani, M. / Guillermier, M. / Valette, H. / Bottlaender, M. / Dolle, F. et al. | 2005
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P04-43 TETRA- OR MONO- ORGANOTIN REAGENTS IN THE STILLE REACTION FOR THE LABELLING OF POTENTIAL RADIOTRACERS WITH CARBON-11: A COMPARATIVE STUDYBourdier, T. / Huiban, M. / Sobrio, F. / Perrio, C. / Barre, L. et al. | 2005
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P04-63 IODONIUM CHEMISTRY: SCOPE AND SELECTIVITY IN AROMATIC NUCLEOPHILIC LABELLING REACTIONSConway, L. K. / Manning, C. O. / Lawrie, K. W. / Plisson, C. / Gee, A. D. / Passchier, J. et al. | 2005
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P04-78 A FULLY AUTOMATED ONE-POT SYNTHESIS OF [CARBONYL-11C]WAY-100635: VALIDATION IN ROUTINE PET STUDIESShchukin, E. V. / Krasikova, R. N. / Andersson, J. / Truong, P. / Christer, H. et al. | 2005