Peptidomimetic C5a receptor antagonists with hydrophobic substitutions at the C-terminus: Increased receptor specificity and in vivo activity (English)
- New search for: Schnatbaum, K.
- New search for: Locardi, E.
- New search for: Scharn, D.
- New search for: Richter, U.
- New search for: Hawlisch, H.
- New search for: Knolle, J.
- New search for: Polakowski, T.
- New search for: Schnatbaum, K.
- New search for: Locardi, E.
- New search for: Scharn, D.
- New search for: Richter, U.
- New search for: Hawlisch, H.
- New search for: Knolle, J.
- New search for: Polakowski, T.
In:
BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
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16
, 19
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5088-5092
;
2006
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ISSN:
- Article (Journal) / Print
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Title:Peptidomimetic C5a receptor antagonists with hydrophobic substitutions at the C-terminus: Increased receptor specificity and in vivo activity
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Contributors:Schnatbaum, K. ( author ) / Locardi, E. ( author ) / Scharn, D. ( author ) / Richter, U. ( author ) / Hawlisch, H. ( author ) / Knolle, J. ( author ) / Polakowski, T. ( author )
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Published in:BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS ; 16, 19 ; 5088-5092
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Publisher:
- New search for: Elsevier Science B.V., Amsterdam.
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Publication date:2006-01-01
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Size:5 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 572.5
- Further information on Dewey Decimal Classification
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Classification:
DDC: 572.5 -
Source:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Table of contents – Volume 16, Issue 19
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
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Graphical contents list| 2006
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Improved replicon cellular activity of non-nucleoside allosteric inhibitors of HCV NS5B polymerase: From benzimidazole to indole scaffoldsBeaulieu, Pierre L. / Gillard, James / Bykowski, Darren / Brochu, Christian / Dansereau, Nathalie / Duceppe, Jean-Simon / Haché, Bruno / Jakalian, Araz / Lagacé, Lisette / LaPlante, Steven et al. | 2006
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Novel benzimidazole-based MCH R1 antagonistsCarpenter, Andrew J. / Al-Barazanji, Kamal A. / Barvian, Kevin K. / Bishop, Michael J. / Britt, Christy S. / Cooper, Joel P. / Goetz, Aaron S. / Grizzle, Mary K. / Hertzog, Donald L. / Ignar, Diane M. et al. | 2006
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Identification of potent agonists of photoreceptor-specific nuclear receptor (NR2E3) and preparation of a radioligandWolkenberg, Scott E. / Zhao, Zhijian / Kapitskaya, Marianna / Webber, Andrea L. / Petrukhin, Konstantin / Tang, Yui Sing / Dean, Dennis C. / Hartman, George D. / Lindsley, Craig W. et al. | 2006
- 5005
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Antitumour properties of fluorinated benzothiazole-substituted hydroxycyclohexa-2,5-dienones (‘quinols’)Lion, Cedric J. / Matthews, Charles S. / Wells, Geoffrey / Bradshaw, Tracey D. / Stevens, Malcolm F.G. / Westwell, Andrew D. et al. | 2006
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Syntheses of triazole-modified zanamivir analogues via click chemistry and anti-AIV activitiesLi, Jian / Zheng, Mingyue / Tang, Wei / He, Pei-Lan / Zhu, Weiliang / Li, Tianxian / Zuo, Jian-Ping / Liu, Hong / Jiang, Hualiang et al. | 2006
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Growth inhibition of human cancer cells in vitro by T-type calcium channel blockersLee, Jae Yeol / Park, Seong Jun / Park, Sung Jun / Lee, Min Joo / Rhim, Hyewhon / Seo, Seon Hee / Kim, Ki-Sun et al. | 2006
- 5018
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A novel class of AMPA receptor allosteric modulators. Part 1: Design, synthesis, and SAR of 3-aryl-4-cyano-5-substituted-heteroaryl-2-carboxylic acid derivativesFernandez, Maria-Carmen / Castaño, Ana / Dominguez, Esteban / Escribano, Ana / Jiang, Delu / Jimenez, Alma / Hong, Eric / Hornback, William J. / Nisenbaum, Eric S. / Rankl, Nancy et al. | 2006
- 5062
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Selectivity in DNA interstrand-stackingLangenegger, Simon M. / Häner, Robert et al. | 2006
- 5066
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Solid-phase synthesis and structure–activity relationships of novel biarylethers as melanin-concentrating hormone receptor-1 antagonistsMa, Vu / Bannon, Anthony W. / Baumgartner, Jamie / Hale, Clarence / Hsieh, Faye / Hulme, Christopher / Rorrer, Kirk / Salon, John / Staden, Carlo van / Tempest, Paul et al. | 2006
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Pyrrolidine bis-cyclic guanidines with antimicrobial activity against drug-resistant Gram-positive pathogens identified from a mixture-based combinatorial libraryHensler, Mary E. / Bernstein, Gregory / Nizet, Victor / Nefzi, Adel et al. | 2006
- 5080
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Synthesis and neuroprotective effects of serofendic acid analoguesTerauchi, Taro / Doko, Takashi / Yonaga, Masahiro / Kajiwara, Akiharu / Niidome, Tetsuhiro / Taguchi, Ryota / Kume, Toshiaki / Akaike, Akinori / Sugimoto, Hachiro et al. | 2006
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The molecular basis for the selection of captopril cis and trans conformations by angiotensin I converting enzymeTzakos, Andreas G. / Naqvi, Nawazish / Comporozos, Konstantinos / Pierattelli, Roberta / Theodorou, Vassiliki / Husain, Ahsan / Gerothanassis, Ioannis P. et al. | 2006
- 5088
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Peptidomimetic C5a receptor antagonists with hydrophobic substitutions at the C-terminus: Increased receptor specificity and in vivo activitySchnatbaum, Karsten / Locardi, Elsa / Scharn, Dirk / Richter, Uwe / Hawlisch, Heiko / Knolle, Jochen / Polakowski, Thomas et al. | 2006
- 5093
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Design and regioselective synthesis of a new generation of targeted chemotherapeutics. Part 1: EC145, a folic acid conjugate of desacetylvinblastine monohydrazideVlahov, Iontcho R. / Santhapuram, Hari Krishna R. / Kleindl, Paul J. / Howard, Stephen J. / Stanford, Katheryn M. / Leamon, Christopher P. et al. | 2006
- 5097
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- 5097
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Synthesis of 3H-spiro[benzofuran-2,1prime-cyclohexane] derivatives from naturally occurring filifolinol and their classical complement pathway inhibitory activityUseglio, M. / Castellano, P. M. / Operto, M. A. / Torres, R. / Kaufman, T. S. et al. | 2006
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Novel tricyclic azepine derivatives: Biological evaluation of pyrimido[4,5-b]-1,4-benzoxazepines, thiazepines, and diazepines as inhibitors of the epidermal growth factor receptor tyrosine kinaseSmith, Leon II / Wong, Wai C. / Kiselyov, Alexander S. / Burdzovic-Wizemann, Sabina / Mao, Yunyu / Xu, Yongjiang / Duncton, Matthew A.J. / Kim, Ki / Piatnitski, Evgueni L. / Doody, Jacqueline F. et al. | 2006
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Search of antitubercular activities in tetrahydroacridines: Synthesis and biological evaluationTripathi, R.P. / Verma, S.S. / Pandey, Jyoti / Agarwal, K.C. / Chaturvedi, Vinita / Manju, Y.K. / Srivastva, A.K. / Gaikwad, A. / Sinha, S. et al. | 2006
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Synthesis of 16-mercaptohexadecylphosphocholine, a miltefosine analog with leishmanicidal activityHornillos, Valentín / Saugar, José María / de la Torre, Beatriz G. / Andreu, David / Rivas, Luis / Acuña, A. Ulises / Amat-Guerri, Francisco et al. | 2006
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Kinase-mediated trapping of bi-functional conjugates of paclitaxel or vinblastine with thymidine in cancer cellsAspland, Simon E. / Ballatore, Carlo / Castillo, Rosario / Desharnais, Joel / Eustaquio, Trisha / Goelet, Philip / Guo, Zijian / Li, Qing / Nelson, David / Sun, Chengzao et al. | 2006
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Editorial Board| 2006
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Instructions to contributors| 2006