2-(3-Aryl-2-propenoyl)-3-methylquinoxaline-1,4-dioxides: A novel cluster of tumor-specific cytotoxins which reverse multidrug resistance (English)
- New search for: Das, U.
- New search for: Pati, H. N.
- New search for: Panda, A. K.
- New search for: Clercq, E. D.
- New search for: Balzarini, J.
- New search for: Molnar, J.
- New search for: Barath, Z.
- New search for: Ocsovszki, I.
- New search for: Kawase, M.
- New search for: Zhou, L.
- New search for: Das, U.
- New search for: Pati, H. N.
- New search for: Panda, A. K.
- New search for: Clercq, E. D.
- New search for: Balzarini, J.
- New search for: Molnar, J.
- New search for: Barath, Z.
- New search for: Ocsovszki, I.
- New search for: Kawase, M.
- New search for: Zhou, L.
In:
BIOORGANIC AND MEDICINAL CHEMISTRY
;
17
, 11
;
3909-3915
;
2009
-
ISSN:
- Article (Journal) / Print
-
Title:2-(3-Aryl-2-propenoyl)-3-methylquinoxaline-1,4-dioxides: A novel cluster of tumor-specific cytotoxins which reverse multidrug resistance
-
Contributors:Das, U. ( author ) / Pati, H. N. ( author ) / Panda, A. K. ( author ) / Clercq, E. D. ( author ) / Balzarini, J. ( author ) / Molnar, J. ( author ) / Barath, Z. ( author ) / Ocsovszki, I. ( author ) / Kawase, M. ( author ) / Zhou, L. ( author )
-
Published in:BIOORGANIC AND MEDICINAL CHEMISTRY ; 17, 11 ; 3909-3915
-
Publisher:
- New search for: Elsevier Science B.V., Amsterdam.
-
Publication date:2009-01-01
-
Size:7 pages
-
ISSN:
-
Type of media:Article (Journal)
-
Type of material:Print
-
Language:English
- New search for: 615.19
- Further information on Dewey Decimal Classification
-
Classification:
DDC: 615.19 -
Source:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Table of contents – Volume 17, Issue 11
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 3747
-
Graphical contents list| 2009
- 3756
-
Synthesis and antiviral activity evaluation of acyclic 2′-azanucleosides bearing a phosphonomethoxy function in the side chainKoszytkowska-Stawińska, Mariola / Clercq, Erik De / Balzarini, Jan et al. | 2009
- 3756
-
Synthesis and antiviral activity evaluation of acyclic 2prime-azanucleosides bearing a phosphonomethoxy function in the side chainKoszytkowska-Stawinska, M. / Clercq, E. D. / Balzarini, J. et al. | 2009
- 3763
-
Anti-inflammatory cembranolides from the soft coral Lobophytum durumCheng, Shi-Yie / Wen, Zhi-Hong / Wang, Shang-Kwei / Chiou, Shu-Fen / Hsu, Chi-Hsin / Dai, Chang-Feng / Duh, Chang-Yih et al. | 2009
- 3770
-
A novel photoaffinity ligand for the dopamine transporter based on pyrovaleroneLapinsky, David J. / Aggarwal, Shaili / Huang, Yurong / Surratt, Christopher K. / Lever, John R. / Foster, James D. / Vaughan, Roxanne A. et al. | 2009
- 3775
-
Preparation and fluorescence properties of fluorophore-labeled avidin–biotin system immobilized on Fe3O4 nanoparticles through functional indolequinone linkerHirata, Nao / Tanabe, Kazuhito / Narita, Asako / Tanaka, Kazuo / Naka, Kensuke / Chujo, Yoshiki / Nishimoto, Sei-ichi et al. | 2009
- 3782
-
Transcription and reverse transcription of artificial nucleic acids involving backbone modification by template-directed DNA polymerase reactionsKuwahara, Masayasu / Takeshima, Hidetoshi / Nagashima, Jun-ichi / Minezaki, Satoshi / Ozaki, Hiroaki / Sawai, Hiroaki et al. | 2009
- 3789
-
Biological activity of endomorphin and [Dmt1]endomorphin analogs with six-membered proline surrogates in position 2Perlikowska, Renata / Gach, Katarzyna / Fichna, Jakub / Toth, Geza / Walkowiak, Bogdan / do-Rego, Jean-Claude / Janecka, Anna et al. | 2009
- 3795
-
Synthesis and in vitro anti Mycobacterium tuberculosis activity of a series of phthalimide derivativesSantos, Jean L. / Yamasaki, Paulo R. / Chin, Chung Man / Takashi, Célio H. / Pavan, Fernando R. / Leite, Clarice Q.F. et al. | 2009
- 3800
-
Structure–activity relationships of 3,5-disubstituted benzamides as glucokinase activators with potent in vivo efficacyIino, Tomoharu / Hashimoto, Noriaki / Sasaki, Kaori / Ohyama, Sumika / Yoshimoto, Riki / Hosaka, Hideka / Hasegawa, Takuro / Chiba, Masato / Nagata, Yasufumi / Eiki, Jun-ichi et al. | 2009
- 3810
-
Design and synthesis of novel chloramphenicol amine derivatives as potent aminopeptidase N (APN/CD13) inhibitorsYang, Kanghui / Wang, Qiang / Su, Li / Fang, Hao / Wang, Xuejian / Gong, Jianzhi / Wang, Binghe / Xu, Wenfang et al. | 2009
- 3818
-
Reversible signal regulation system of 19F NMR by redox reactions using a metal complex as a switching moduleTanaka, Kazuo / Kitamura, Narufumi / Takahashi, Yuichi / Chujo, Yoshiki et al. | 2009
- 3824
-
Cyclobutane-containing peptides: Evaluation as novel metallocarboxypeptidase inhibitors and modelling of their mode of actionFernández, Daniel / Torres, Elisabeth / Avilés, Francesc X. / Ortuño, Rosa M. / Vendrell, Josep et al. | 2009
- 3829
-
Design, synthesis and biological investigation of certain pyrazole-3-carboxylic acid derivatives as novel carriers for nitric oxideAbdel-Hafez, El-Shimaa M.N. / Abuo-Rahma, Gamal El-Din A.A. / Abdel-Aziz, Mohamed / Radwan, Mohamed F. / Farag, Hassan H. et al. | 2009
- 3838
-
Bulky 1,4-benzoxazine derivatives with antifungal activityFringuelli, Renata / Giacchè, Nicola / Milanese, Lara / Cenci, Elio / Macchiarulo, Antonio / Vecchiarelli, Anna / Costantino, Gabriele / Schiaffella, Fausto et al. | 2009
- 3847
-
Synthesis and biological evaluation of 3,4,6-triaryl-2-pyranones as a potential new class of anti-breast cancer agentsShankar, Ravi / Chakravarti, Bandana / Singh, Uma Sharan / Ansari, Mohd. Imran / Deshpande, Shreekant / Dwivedi, Shailendra Kumar Dhar / Bid, Hemant Kumar / Konwar, Rituraj / Kharkwal, Geetika / Chandra, Vishal et al. | 2009
- 3857
-
Synthesis and activity of tryptophan sulfonamide derivatives as novel non-hydroxamate TNF-α converting enzyme (TACE) inhibitorsPark, Kaapjoo / Gopalsamy, Ariamala / Aplasca, Alexis / Ellingboe, John W. / Xu, Weixin / Zhang, Yuhua / Levin, Jeremy I. et al. | 2009
- 3857
-
Synthesis and activity of tryptophan sulfonamide derivatives as novel non-hydroxamate TNF-a converting enzyme (TACE) inhibitorsPark, K. / Gopalsamy, A. / Aplasca, A. / Ellingboe, J. W. / Xu, W. / Zhang, Y. / Levin, J. I. et al. | 2009
- 3866
-
Antibacterial activity of berberine-NorA pump inhibitor hybrids with a methylene ether linking groupSamosorn, Siritron / Tanwirat, Bongkot / Muhamad, Nussara / Casadei, Gabriele / Tomkiewicz, Danuta / Lewis, Kim / Suksamrarn, Apichart / Prammananan, Therdsak / Gornall, Karina C. / Beck, Jennifer L. et al. | 2009
- 3873
-
Synthesis and activity evaluation of phenylurea derivatives as potent antitumor agentsSong, Dan-Qing / Du, Na-Na / Wang, Yue-Ming / He, Wei-Ying / Jiang, En-Zhu / Cheng, Shi-Xiang / Wang, Yan-Xiang / Li, Ying-Hong / Wang, Yu-Ping / Li, Xin et al. | 2009
- 3879
-
Design, synthesis, antibacterial activity and physicochemical parameters of novel N-4-piperazinyl derivatives of norfloxacinAbuo-Rahma, Gamal El-Din A.A. / Sarhan, Hatem. A. / Gad, Gamal F.M. et al. | 2009
- 3887
-
Convenient and highly effective fluorescence sensing for Hg2+ in aqueous solution and thin filmLiu, Yu / Yu, Miao / Chen, Yong / Zhang, Ning et al. | 2009
- 3892
-
Phosphonate analogues of cyclopropavir phosphates and their E-isomers. Synthesis and antiviral activityMhaske, Santosh B. / Ksebati, Bashar / Prichard, Mark N. / Drach, John C. / Zemlicka, Jiri et al. | 2009
- 3900
-
Design and synthesis of enediyne–peptide conjugates and their inhibiting activity against chymotrypsinDutta, Sansa / Basak, Amit / Dasgupta, Swagata et al. | 2009
- 3909
-
2-(3-Aryl-2-propenoyl)-3-methylquinoxaline-1,4-dioxides: A novel cluster of tumor-specific cytotoxins which reverse multidrug resistanceDas, Umashankar / Pati, Hari N. / Panda, Atulya K. / Clercq, Erik De / Balzarini, Jan / Molnár, Joseph / Baráth, Zoltán / Ocsovszki, Imre / Kawase, Masami / Zhou, Li et al. | 2009
- 3916
-
A library of novel allosteric inhibitors against fructose 1,6-bisphosphataseHeng, Sabrina / Gryncel, Kimberly R. / Kantrowitz, Evan R. et al. | 2009
- 3923
-
Investigation of various N-heterocyclic substituted piperazine versions of 5/7-{[2-(4-aryl-piperazin-1-yl)-ethyl]-propyl-amino}-5,6,7,8-tetrahydro-naphthalen-2-ol: Effect on affinity and selectivity for dopamine D3 receptorBrown, Dennis A. / Mishra, Manoj / Zhang, Suhong / Biswas, Swati / Parrington, Ingrid / Antonio, Tamara / Reith, Maarten E.A. / Dutta, Aloke K. et al. | 2009
- 3934
-
Design, parallel synthesis, and crystal structures of biphenyl antithrombotics as selective inhibitors of tissue factor FVIIa complex. Part 1: Exploration of S2 pocket pharmacophoresKotian, Pravin L. / Krishnan, Raman / Rowland, Scott / El-Kattan, Yahya / Saini, Surendra K. / Upshaw, Ramanda / Bantia, Shanta / Arnold, Shane / Sudhakar Babu, Y. / Chand, Pooran et al. | 2009
- 3959
-
Preparation of novel (Z)-4-ylidenebenzo[b]furo[3,2-d][1,3]oxazines and their biological activityTabuchi, Yukako / Ando, Yuko / Kanemura, Hidemi / Kawasaki, Ikuo / Ohishi, Takahiro / Koida, Masao / Fukuyama, Ryo / Nakamuta, Hiromichi / Ohta, Shunsaku / Nishide, Kiyoharu et al. | 2009
- 3968
-
Dysideamine, a new sesquiterpene aminoquinone, protects hippocampal neuronal cells against iodoacetic acid-induced cell deathSuna, Hideaki / Arai, Masayoshi / Tsubotani, Yoshie / Hayashi, Asami / Setiawan, Andi / Kobayashi, Motomasa et al. | 2009
- 3973
-
Design, synthesis and evaluations of acridone derivatives using Candida albicans—Search for MDR modulators led to the identification of an anti-candidiasis agentSingh, Palwinder / Kaur, Jatinder / Yadav, Bhawna / Komath, Sneha Sudha et al. | 2009
- 3980
-
Design, microwave-assisted synthesis and HIV-RT inhibitory activity of 2-(2,6-dihalophenyl)-3-(4,6-dimethyl-5-(un)substituted-pyrimidin-2-yl)thiazolidin-4-onesChen, Hua / Bai, Jie / Jiao, Lingling / Guo, Zaihong / Yin, Qingmei / Li, Xiaoliu et al. | 2009
- 3987
-
Clobenpropit analogs as dual activity ligands for the histamine H3 and H4 receptors: Synthesis, pharmacological evaluation, and cross-target QSAR studiesLim, Herman D. / Istyastono, Enade P. / van de Stolpe, Andrea / Romeo, Giuseppe / Gobbi, Silvia / Schepers, Marjo / Lahaye, Roger / Menge, Wiro M.B.P. / Zuiderveld, Obbe P. / Jongejan, Aldo et al. | 2009
- 3995
-
N-tert-Butyl and N-methyl nitrones derived from aromatic aldehydes inhibit macromolecular permeability increase induced by ischemia/reperfusion in hamstersDias, Ayres G. / Santos, Carlos E.V. / Cyrino, Fatima Z.G.A. / Bouskela, Eliete / Costa, Paulo R.R. et al. | 2009
- 3999
-
3D-QSAR studies of 2,2-diphenylpropionates to aid discovery of novel potent muscarinic antagonistsBhattacharjee, Apurba K. / Gordon, Jonathan A. / Marek, Elizabeth / Campbell, Amy / Gordon, Richard K. et al. | 2009
- I
-
Instructions to contributors| 2009
- IFC
-
Editorial board| 2009