`Click chemistry' synthesis of a library of 1,2,3-triazole-substituted galactose derivatives and their evaluation against Trypanosoma cruzi and its cell surface trans-sialidase (English)
- New search for: Carvalho, I.
- New search for: Andrade, P.
- New search for: Campo, V. L.
- New search for: Guedes, P. M.
- New search for: Sesti-Costa, R.
- New search for: Silva, J. S.
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- New search for: Carvalho, I.
- New search for: Andrade, P.
- New search for: Campo, V. L.
- New search for: Guedes, P. M.
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In:
BIOORGANIC AND MEDICINAL CHEMISTRY
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18
, 7
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2412-2427
;
2010
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ISSN:
- Article (Journal) / Print
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Title:`Click chemistry' synthesis of a library of 1,2,3-triazole-substituted galactose derivatives and their evaluation against Trypanosoma cruzi and its cell surface trans-sialidase
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Contributors:Carvalho, I. ( author ) / Andrade, P. ( author ) / Campo, V. L. ( author ) / Guedes, P. M. ( author ) / Sesti-Costa, R. ( author ) / Silva, J. S. ( author ) / Schenkman, S. ( author ) / Dedola, S. ( author ) / Hill, L. ( author ) / Rejzek, M. ( author )
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Published in:BIOORGANIC AND MEDICINAL CHEMISTRY ; 18, 7 ; 2412-2427
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Publisher:
- New search for: Elsevier Science B.V., Amsterdam.
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Publication date:2010-01-01
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Size:16 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 615.19
- Further information on Dewey Decimal Classification
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Classification:
DDC: 615.19 -
Source:
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Table of contents – Volume 18, Issue 7
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 2357
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Graphical contents list| 2010
- 2370
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Synthesis and biological evaluation of 4-(hydroxyimino)arylmethyl diarylpyrimidine analogues as potential non-nucleoside reverse transcriptase inhibitors against HIVFeng, Xiao-Qing / Zeng, Zhao-Sen / Liang, Yong-Hong / Chen, Fen-Er / Pannecouque, Christophe / Balzarini, Jan / Clercq, Erik De et al. | 2010
- 2375
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Pyrazolone-fused combretastatins and their precursors: synthesis, cytotoxicity, antitubulin activity and molecular modeling studiesBurja, Bojan / Čimbora-Zovko, Tamara / Tomić, Sanja / Jelušić, Tihana / Kočevar, Marijan / Polanc, Slovenko / Osmak, Maja et al. | 2010
- 2388
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Synthesis of mono-carbonyl analogues of curcumin and their effects on inhibition of cytokine release in LPS-stimulated RAW 264.7 macrophagesZhao, Chengguang / Yang, Ju / Wang, Yi / Liang, Donglou / Yang, Xuyi / Li, Xiaoxia / Wu, Jianzhang / Wu, Xiaoping / Yang, Shulin / Li, Xiaokun et al. | 2010
- 2394
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18F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imagingZhang, Shuting / Wang, Xiao / He, Yong / Ding, Rui / Liu, Hang / Xu, Jingli / Feng, Man / Li, Guixia / Wang, Ming / Peng, Cheng et al. | 2010
- 2402
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Structural development studies of anti-hepatitis C virus agents with a phenanthridinone skeletonNakamura, Masahiko / Aoyama, Atsushi / Salim, Mohammed T.A. / Okamoto, Mika / Baba, Masanori / Miyachi, Hiroyuki / Hashimoto, Yuichi / Aoyama, Hiroshi et al. | 2010
- 2412
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‘Click chemistry’ synthesis of a library of 1,2,3-triazole-substituted galactose derivatives and their evaluation against Trypanosoma cruzi and its cell surface trans-sialidaseCarvalho, Ivone / Andrade, Peterson / Campo, Vanessa L. / Guedes, Paulo M.M. / Sesti-Costa, Renata / Silva, João S. / Schenkman, Sergio / Dedola, Simone / Hill, Lionel / Rejzek, Martin et al. | 2010
- 2428
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Synthesis and preliminary pharmacological characterisation of a new class of nitrogen-containing bisphosphonates (N-BPs)Lolli, Marco L. / Rolando, Barbara / Tosco, Paolo / Chaurasia, Shilpi / Stilo, Antonella Di / Lazzarato, Loretta / Gorassini, Eva / Ferracini, Riccardo / Oliaro-Bosso, Simonetta / Fruttero, Roberta et al. | 2010
- 2439
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Phosphoramidates of 2prime-b-d-arabinouridine (AraU) as phosphate prodrugs; design, synthesis, in vitro activity and metabolismMehellou, Y. / Valente, R. / Mottram, H. / Walsby, E. / Mills, K. I. / Balzarini, J. / McGuigan, C. et al. | 2010
- 2439
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Phosphoramidates of 2′-β-d-arabinouridine (AraU) as phosphate prodrugs; design, synthesis, in vitro activity and metabolismMehellou, Youcef / Valente, Rocco / Mottram, Huw / Walsby, Elisabeth / Mills, Kenneth I. / Balzarini, Jan / McGuigan, Christopher et al. | 2010
- 2447
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Synthesis, molecular modeling and biological evaluation of PSB as targeted antibioticsCheng, Kui / Zheng, Qing-Zhong / Hou, Jin / Zhou, Yang / Liu, Chang-Hong / Zhao, Jing / Zhu, Hai-Liang et al. | 2010
- 2456
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Discovery of inhibitors of brassinin oxidase based on the scaffolds of the phytoalexins brassilexin and wasalexinPedras, M. Soledade C. / Minic, Zoran / Sarma-Mamillapalle, Vijay K. / Suchy, Mojmir et al. | 2010
- 2464
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Total synthesis, antiprotozoal and cytotoxicity activities of rhuschalcone VI and analogsMihigo, Shetonde O. / Mammo, Wendimagegn / Bezabih, Merhatibeb / Andrae-Marobela, Kerstin / Abegaz, Berhanu M. et al. | 2010
- 2474
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Synthesis of 26-hydroxy-22-oxocholestanic frameworks from diosgenin and hecogenin and their in vitro antiproliferative and apoptotic activity on human cervical cancer CaSki cellsFernández-Herrera, María A. / López-Muñoz, Hugo / Hernández-Vázquez, José M.V. / López-Dávila, Moisés / Escobar-Sánchez, María L. / Sánchez-Sánchez, Luis / Pinto, B. Mario / Sandoval-Ramírez, Jesús et al. | 2010
- 2485
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Chromene-3-carboxamide derivatives discovered from virtual screening as potent inhibitors of the tumour maker, AKR1B10Endo, Satoshi / Matsunaga, Toshiyuki / Kuwata, Kazuo / Zhao, Hai-Tao / El-Kabbani, Ossama / Kitade, Yukio / Hara, Akira et al. | 2010
- 2491
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Novel 8-(furan-2-yl)-3-substituted thiazolo [5,4-e][1,2,4] triazolo[1,5-c] pyrimidine-2(3H)-thione derivatives as potential adenosine A2A receptor antagonistsMishra, Chandra Bhushan / Barodia, Sandeep Kumar / Prakash, Amresh / Senthil Kumar, J.B. / Luthra, Pratibha Mehta et al. | 2010
- 2501
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Conjugates of plumbagin and phenyl-2-amino-1-thioglucoside inhibit MshB, a deacetylase involved in the biosynthesis of mycothiolGammon, David W. / Steenkamp, Daniel J. / Mavumengwana, Vuyo / Marakalala, Mohlopheni J. / Mudzunga, Theophilus T. / Hunter, Roger / Munyololo, Muganza et al. | 2010
- 2515
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Enhancement of antiproliferative activity by molecular simplification of catalpolGarcía, Celina / León, Leticia G. / Pungitore, Carlos R. / Ríos-Luci, Carla / Daranas, Antonio H. / Montero, Juan C. / Pandiella, Atanasio / Tonn, Carlos E. / Martín, Víctor S. / Padrón, José M. et al. | 2010
- 2524
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Synthesis and pharmacological characterization of a new series of 5,7-disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazine derivatives as adenosine receptor antagonists: A preliminary inspection of ligand–receptor recognition processPastorin, Giorgia / Federico, Stephanie / Paoletta, Silvia / Corradino, Marta / Cateni, Francesca / Cacciari, Barbara / Klotz, Karl-Norbert / Gao, Zhan-Guo / Jacobson, Kenneth A. / Spalluto, Giampiero et al. | 2010
- 2537
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Synthesis and anticancer activity evaluation of 2(4-alkoxyphenyl)cyclopropyl hydrazides and triazolo phthalazinesDe, Prithwiraj / Baltas, Michel / Lamoral-Theys, Delphine / Bruyère, Céline / Kiss, Robert / Bedos-Belval, Florence / Saffon, Nathalie et al. | 2010
- 2549
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Synthesis and biological evaluation of antitumor-active γ-butyrolactone substituted betulin derivativesCsuk, René / Barthel, Alexander / Schwarz, Stefan / Kommera, Harish / Paschke, Reinhard et al. | 2010
- 2549
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Synthesis and biological evaluation of antitumor-active g-butyrolactone substituted betulin derivativesCsuk, R. / Barthel, A. / Schwarz, S. / Kommera, H. / Paschke, R. et al. | 2010
- 2559
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Water-soluble polymer–drug conjugates for combination chemotherapy against visceral leishmaniasisNicoletti, Salvatore / Seifert, Karin / Gilbert, Ian H. et al. | 2010
- 2566
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Assessing the trypanocidal potential of natural and semi-synthetic diketopiperazines from two deep water marine-derived fungiWatts, Katharine R. / Ratnam, Joseline / Ang, Kean-Hooi / Tenney, Karen / Compton, Jennifer E. / McKerrow, James / Crews, Phillip et al. | 2010
- 2575
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Novel DNA–peptide interaction networksHuang, Jonathan T.B. / Chen, Yen-Chung / Chang, Jung-Cheng / Jeng, Kee-Ching G. / Kao, Karen K.L. / Yang, Robin C.K. / Kan, Lou-Sing / Wey, Ming-Tsair / Waring, Michael J. / Chen, Chee-Shan et al. | 2010
- 2586
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Design, synthesis and antimalarial/anticancer evaluation of spermidine linked artemisinin conjugates designed to exploit polyamine transporters in Plasmodium falciparum and HL-60 cancer cell linesChadwick, James / Jones, Michael / Mercer, Amy E. / Stocks, Paul A. / Ward, Stephen A. / Park, B. Kevin / O’Neill, Paul M. et al. | 2010
- 2598
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Cu(II) cyclen cleavage agent for human islet amyloid peptideJeong, Keunhong / Chung, Woo Young / Kye, Young-Sik / Kim, Dongwook et al. | 2010
- 2602
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Isolation, structure and biological activities of platencin A2–A4 from Streptomyces platensisZhang, Chaowei / Ondeyka, John / Dietrich, Lisa / Gailliot, Francis P. / Hesse, Michelle / Lester, Michael / Dorso, Karen / Motyl, Mary / Ha, Sookhee N. / Wang, Jun et al. | 2010
- 2611
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Synthesis and antibacterial studies of binaphthyl-based tripeptoids. Part 1Bremner, John B. / Keller, Paul A. / Pyne, Stephen G. / Boyle, Timothy P. / Brkic, Zinka / David, Dorothy M. / Robertson, Mark / Somphol, Kittiya / Baylis, Dean / Coates, Jonathan A. et al. | 2010
- 2621
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Antiproliferative activity of synthetic naphthoquinones related to lapachol. First synthesis of 5-hydroxylapacholBonifazi, Evelyn L. / Ríos-Luci, Carla / León, Leticia G. / Burton, Gerardo / Padrón, José M. / Misico, Rosana I. et al. | 2010
- 2631
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Bioconjugates of curcumin display improved protection against glutathione depletion mediated oxidative stress in a dopaminergic neuronal cell line: Implications for Parkinson’s diseaseHarish, G. / Venkateshappa, C. / Mythri, Rajeswara Babu / Dubey, Shiv Kumar / Mishra, Krishna / Singh, Neetu / Vali, Shireen / Bharath, M.M. Srinivas et al. | 2010
- 2639
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Regioselective one-pot synthesis and anti-proliferative and apoptotic effects of some novel tetrazolo[1,5-a]pyrimidine derivativesHussein, Ahmed M. / Ahmed, Osama M. et al. | 2010
- 2645
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Synthesis of new β-1-C-alkylated imino-l-iditols: A comparative study of their activity as β-glucocerebrosidase inhibitorsSchönemann, Wojciech / Gallienne, Estelle / Compain, Philippe / Ikeda, Kyoko / Asano, Naoki / Martin, Olivier R. et al. | 2010
- 2645
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Synthesis of new b-1-C-alkylated imino-l-iditols: A comparative study of their activity as b-glucocerebrosidase inhibitorsSchonemann, W. / Gallienne, E. / Compain, P. / Ikeda, K. / Asano, N. / Martin, O. R. et al. | 2010
- 2651
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Inhibition of Escherichia coli glycosyltransferase MurG and Mycobacterium tuberculosis Gal transferase by uridine-linked transition state mimicsTrunkfield, Amy E. / Gurcha, Sudagar S. / Besra, Gurdyal S. / Bugg, Timothy D.H. et al. | 2010
- 2664
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Investigating the anti-proliferative activity of styrylazanaphthalenes and azanaphthalenedionesMrozek-Wilczkiewicz, Anna / Kalinowski, Danuta S. / Musiol, Robert / Finster, Jacek / Szurko, Agnieszka / Serafin, Katarzyna / Knas, Magdalena / Kamalapuram, Sishir K. / Kovacevic, Zaklina / Jampilek, Josef et al. | 2010
- 2672
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Preparation and in vitro photodynamic activity of amphiphilic zinc(II) phthalocyanines substituted with 2-(dimethylamino)ethylthio moieties and their N-alkylated derivativesDuan, Wubiao / Lo, Pui-Chi / Duan, Lei / Fong, Wing-Ping / Ng, Dennis K.P. et al. | 2010
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Zinc(II) complexes of the second-generation quinolone antibacterial drug enrofloxacin: Structure and DNA or albumin interactionTarushi, Alketa / Raptopoulou, Catherine P. / Psycharis, Vassilis / Terzis, Aris / Psomas, George / Kessissoglou, Dimitris P. et al. | 2010
- 2686
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Statistical molecular design of a focused salicylidene acylhydrazide library and multivariate QSAR of inhibition of type III secretion in the Gram-negative bacterium YersiniaDahlgren, Markus K. / Zetterström, Caroline E. / Gylfe, Åsa / Linusson, Anna / Elofsson, Mikael et al. | 2010
- 2704
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Synthesis, X-ray crystal structure study and antitumoral evaluations of 5,6-disubstituted pyrimidine derivativesKraljević, Tatjana Gazivoda / Krištafor, Svjetlana / Šuman, Lidija / Kralj, Marijeta / Ametamey, Simon M. / Cetina, Mario / Raić-Malić, Silvana et al. | 2010
- 2713
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New 3-methylquinoxaline-2-carboxamide 1,4-di-N-oxide derivatives as anti-Mycobacterium tuberculosis agentsAncizu, Saioa / Moreno, Elsa / Solano, Beatriz / Villar, Raquel / Burguete, Asunción / Torres, Enrique / Pérez-Silanes, Silvia / Aldana, Ignacio / Monge, Antonio et al. | 2010
- 2720
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Evaluation of retro-inverso modifications of HTLV-1 protease inhibitors containing a hydroxyethylamine isosterTatsumi, Tadashi / Awahara, Chiyuki / Naka, Hiromi / Aimoto, Saburo / Konno, Hiroyuki / Nosaka, Kazuto / Akaji, Kenichi et al. | 2010
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Structure–activity relationship of novel DAPK inhibitors identified by structure-based virtual screeningOkamoto, Masako / Takayama, Kiyoshi / Shimizu, Tomoko / Muroya, Ayumu / Furuya, Toshio et al. | 2010
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Novel azalides derived from 16-membered macrolides. III. Azalides modified at the C-15 and 4″ positions: Improved antibacterial activitiesMiura, Tomoaki / Natsume, Satomi / Kanemoto, Kenichi / Shitara, Eiki / Fushimi, Hideki / Yoshida, Takuji / Ajito, Keiichi et al. | 2010
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Novel azalides derived from 16-membered macrolides. III. Azalides modified at the C-15 and 4Prime positions: Improved antibacterial activitiesMiura, T. / Natsume, S. / Kanemoto, K. / Shitara, E. / Fushimi, H. / Yoshida, T. / Ajito, K. et al. | 2010
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Application of the phosphoramidate ProTide approach to the antiviral drug ribavirinDerudas, Marco / Brancale, Andrea / Naesens, Lieve / Neyts, Johan / Balzarini, Jan / McGuigan, Christopher et al. | 2010
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Synthesis and structure–activity relationships of antimalarial 4-oxo-3-carboxyl quinolonesZhang, Yiqun / Guiguemde, W. Armand / Sigal, Martina / Zhu, Fangyi / Connelly, Michele C. / Nwaka, Solomon / Guy, R. Kiplin et al. | 2010
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Polysubstituted pyrazoles, part 6. Synthesis of some 1-(4-chlorophenyl)-4-hydroxy-1H-pyrazol-3-carbonyl derivatives linked to nitrogenous heterocyclic ring systems as potential antitumor agentsRostom, Sherif A.F. et al. | 2010
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- IFC
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Editorial board| 2010