Silicon Analogues of the Nonpeptidic GnRH Antagonist AG-045572: Syntheses, Crystal Structure Analyses, and Pharmacological Characterization (English)
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- New search for: Daiss, J. O.
- New search for: Gray, I. C.
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- New search for: Tam, L. H.
- New search for: Kuehn, D.
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- New search for: Barnes, M. J.
- New search for: Burschka, C.
- New search for: Bttner, M. W.
- New search for: Conroy, R.
- New search for: Daiss, J. O.
- New search for: Gray, I. C.
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In:
CHEMMEDCHEM
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6
, 11
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2070-2080
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2011
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ISSN:
- Article (Journal) / Print
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Title:Silicon Analogues of the Nonpeptidic GnRH Antagonist AG-045572: Syntheses, Crystal Structure Analyses, and Pharmacological Characterization
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Contributors:Barnes, M. J. ( author ) / Burschka, C. ( author ) / Bttner, M. W. ( author ) / Conroy, R. ( author ) / Daiss, J. O. ( author ) / Gray, I. C. ( author ) / Hendrick, A. G. ( author ) / Tam, L. H. ( author ) / Kuehn, D. ( author ) / Miller, D. J. ( author )
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Published in:CHEMMEDCHEM ; 6, 11 ; 2070-2080
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Publisher:
- New search for: JOHN WILEY & SONS LTD
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Publication date:2011-01-01
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Size:11 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 615.19
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Classification:
DDC: 615.19 -
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Table of contents – Volume 6, Issue 11
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1941
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Cover Picture: Structure–Activity Relationship for the First‐in‐Class Clinical Steroid Sulfatase Inhibitor Irosustat (STX64, BN83495) (ChemMedChem 11/2011)Woo, L. W. Lawrence / Ganeshapillai, Dharshini / Thomas, Mark P. / Sutcliffe, Oliver B. / Malini, Bindu / Mahon, Mary F. / Purohit, Atul / Potter, Barry V. L. et al. | 2011
- 1942
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Inside Cover: Inhibition of Aminoglycoside‐Deactivating Enzymes APH(3′)‐IIIa and AAC(6′)‐Ii by Amphiphilic Paromomycin O2′′‐Ether Analogues (ChemMedChem 11/2011)Szychowski, Janek / Kondo, Jiro / Zahr, Omar / Auclair, Karine / Westhof, Eric / Hanessian, Stephen / Keillor, Jeffrey W. et al. | 2011
- 1943
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Graphical Abstract: ChemMedChem 11/2011| 2011
- 1952
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Spotlights on our sister journals: ChemMedChem 11/2011| 2011
- 1955
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H.‐L. Zhu| 2011
- 1957
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Runaway ROS as a Selective Anticancer StrategyParkinson, Elizabeth I. / Hergenrother, Paul J. et al. | 2011
- 1961
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Inhibition of Aminoglycoside‐Deactivating Enzymes APH(3′)‐IIIa and AAC(6′)‐Ii by Amphiphilic Paromomycin O2′′‐Ether AnaloguesSzychowski, Janek / Kondo, Jiro / Zahr, Omar / Auclair, Karine / Westhof, Eric / Hanessian, Stephen / Keillor, Jeffrey W. et al. | 2011
- 1967
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Revisiting the Rule of Five on the Basis of Pharmacokinetic Data from RatRidder, Lars / Wang, Hongwu / de Vlieg, Jacob / Wagener, Markus et al. | 2011
- 1971
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Discovery of α,β‐ and α,γ‐Diamino Acid Scaffolds for the Inhibition of M1 Family AminopeptidasesGumpena, Rajesh / Kishor, Chandan / Ganji, Roopa Jones / Addlagatta, Anthony et al. | 2011
- 1977
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Derivatives of R‐Aminocarnitine without Ammonium Moiety as Liver Carnitine Palmitoyltransferase I (L‐CPT I) InhibitorsTassoni, Emanuela / Conti, Roberto / Gallo, Grazia / Vincenti, Silvia / Mastrofrancesco, Lucilla / Brunetti, Tiziana / Cabri, Walter / Giannessi, Fabio et al. | 2011
- 1981
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Azabicyclo[3.1.0]hexane‐1‐carbohydrazides as Potent and Selective GHSR1a Ligands Presenting a Specific in vivo BehaviorSabbatini, Fabio Maria / Melotto, Sergio / Bernasconi, Giovanni / Bromidge, Steve M. / D'Adamo, Lucilla / Rinaldi, Marilisa / Savoia, Chiara / Mundi, Claudia / Di Francesco, Carla / Zonzini, Laura et al. | 2011
- 1986
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Structure–Activity Relationships of Neuritogenic Gentiside DerivativesLuo, Yan / Sun, Kaiyue / Li, Lin / Gao, Lijuan / Wang, Guangfa / Qu, Yuan / Xiang, Lan / Chen, Ling / Hu, Yongzhou / Qi, Jianhua et al. | 2011
- 1990
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Chemical and Pharmacological Studies on Enantiomerically Pure p‐Methoxytacripyrines, Promising Multi‐Target‐Directed Ligands for the Treatment of Alzheimer’s DiseaseBartolini, Manuela / Pistolozzi, Marco / Andrisano, Vincenza / Egea, Javier / López, Manuela G. / Iriepa, Isabel / Moraleda, Ignacio / Gálvez, Enrique / Marco‐Contelles, José / Samadi, Abdelouahid et al. | 2011
- 1998
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Antiproliferative Effects of Ester‐ and Amide‐Functionalized Rhizoxin DerivativesKusebauch, Björn / Scherlach, Kirstin / Kirchner, Heike / Dahse, Hans‐Martin / Hertweck, Christian et al. | 2011
- 2003
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Encapsulation of Docetaxel into PEGylated Gold Nanoparticles for Vectorization to Cancer CellsFrançois, Alison / Laroche, Audrey / Pinaud, Noël / Salmon, Lionel / Ruiz, Jaime / Robert, Jacques / Astruc, Didier et al. | 2011
- 2009
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N‐[2‐Methyl‐5‐(triazol‐1‐yl)phenyl]pyrimidin‐2‐amine as a Scaffold for the Synthesis of Inhibitors of Bcr‐AblArioli, Federica / Borrelli, Stella / Colombo, Francesco / Falchi, Federico / Filippi, Irene / Crespan, Emmanuele / Naldini, Antonella / Scalia, Giusy / Silvani, Alessandra / Maga, Giovanni et al. | 2011
- 2019
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Structure–Activity Relationship for the First‐in‐Class Clinical Steroid Sulfatase Inhibitor Irosustat (STX64, BN83495)Woo, L. W. Lawrence / Ganeshapillai, Dharshini / Thomas, Mark P. / Sutcliffe, Oliver B. / Malini, Bindu / Mahon, Mary F. / Purohit, Atul / Potter, Barry V. L. et al. | 2011
- 2035
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Asymmetric Synthesis and Conformational Analysis by NMR Spectroscopy and MD of Aba‐ and α‐MeAba‐Containing Dermorphin AnaloguesVandormael, Bart / De Wachter, Rien / Martins, José C. / Hendrickx, Pieter M. S. / Keresztes, Attila / Ballet, Steven / Mallareddy, Jayapal R. / Tóth, Fanni / Tóth, Géza / Tourwé, Dirk et al. | 2011
- 2048
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Halogen Bonding at the Active Sites of Human Cathepsin L and MEK1 Kinase: Efficient Interactions in Different EnvironmentsHardegger, Leo A. / Kuhn, Bernd / Spinnler, Beat / Anselm, Lilli / Ecabert, Robert / Stihle, Martine / Gsell, Bernard / Thoma, Ralf / Diez, Joachim / Benz, Jörg et al. | 2011
- 2055
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Development of 2,3,5‐Triaryl‐1H‐pyrroles as Estrogen Receptor α Selective LigandsSchäfer, Anja / Wellner, Anja / Strauss, Martin / Wolber, Gerhard / Gust, Ronald et al. | 2011
- 2063
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Hydrophobic Oxime Ethers: A Versatile Class of pDNA and siRNA Transfection LipidsBiswas, Souvik / Knipp, Ralph J. / Gordon, Laura E. / Nandula, Seshagiri R. / Gorr, Sven‐Ulrik / Clark, Geoffrey J. / Nantz, Michael H. et al. | 2011
- 2070
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Silicon Analogues of the Nonpeptidic GnRH Antagonist AG‐045572: Syntheses, Crystal Structure Analyses, and Pharmacological CharacterizationBarnes, Matthew J. / Burschka, Christian / Büttner, Matthias W. / Conroy, Richard / Daiss, Jürgen O. / Gray, Ian C. / Hendrick, Alan G. / Tam, L. H. / Kuehn, Diana / Miller, David J. et al. | 2011
- 2081
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Phosphatidyl myo‐Inositol Mannosides Mimics Built on an Acyclic or Heterocyclic Core: Synthesis and Anti‐inflammatory PropertiesFront, Sophie / Court, Nathalie / Bourigault, Marie‐Laure / Rose, Stéphanie / Ryffel, Bernhard / Erard, François / Quesniaux, Valérie F. J. / Martin, Olivier R. et al. | 2011
- 2094
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Synthesis and Antimalarial Activities of a Diverse Set of Triazole‐Containing Furamidine AnaloguesBerger, Olivier / Kaniti, Archana / van Ba, Christophe Tran / Vial, Henri / Ward, Stephen A. / Biagini, Giancarlo A. / Bray, Patrick G. / O'Neill, Paul M. et al. | 2011
- 2109
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Methods and Principles in Medicinal Chemistry, Vol. 48: Virtual Screening: Principles, Challenges, and Practical Guidelines. Edited by Christoph Sotriffer.Dessolin, Jean et al. | 2011
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Biomarkers in Medicine, Drug Discovery and Environmental Health. Edited by Vishal S. Vaidya and Joseph V. Bonventre.Meissner, Axel et al. | 2011
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Preview: ChemMedChem 12/2011| 2011