Synthesis of benzimidazolyl-1,3,4-oxadiazol-2ylthio-N-phenyl (benzothiazolyl) acetamides as antibacterial, antifungal and antituberculosis agents (English)
- New search for: Patel, R. V.
- New search for: Patel, P. K.
- New search for: Kumari, P.
- New search for: Rajani, D. P.
- New search for: Chikhalia, K. H.
- New search for: Patel, R. V.
- New search for: Patel, P. K.
- New search for: Kumari, P.
- New search for: Rajani, D. P.
- New search for: Chikhalia, K. H.
In:
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
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53
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41-51
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2012
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ISSN:
- Article (Journal) / Print
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Title:Synthesis of benzimidazolyl-1,3,4-oxadiazol-2ylthio-N-phenyl (benzothiazolyl) acetamides as antibacterial, antifungal and antituberculosis agents
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Contributors:Patel, R. V. ( author ) / Patel, P. K. ( author ) / Kumari, P. ( author ) / Rajani, D. P. ( author ) / Chikhalia, K. H. ( author )
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Published in:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY ; 53 ; 41-51
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Publisher:
- New search for: Elsevier Science B.V., Amsterdam.
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Publication date:2012-01-01
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Size:11 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 615.1
- Further information on Dewey Decimal Classification
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Classification:
DDC: 615.1 -
Source:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Table of contents – Volume 53
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1
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Synthesis and antitumor activity of lapathoside D and its analogsPanda, P. / Appalashetti, M. / Natarajan, M. / Chan-Park, M. B. / Venkatraman, S. S. / Judeh, Z. M. A. et al. | 2012
- 13
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Synthesis and molecular modelling studies of novel carbapeptide analogs for inhibition of HIV-1 proteasePawar, S. A. / Jabgunde, A. M. / Govender, P. / Maguire, G. E. M. / Kruger, H. G. / Parboosing, R. / Soliman, M. E. S. / Sayed, Y. / Dhavale, D. D. / Govender, T. et al. | 2012
- 22
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Synthesis, antitumor activity and SAR study of novel [1,2,4]triazino[4,5-a]benzimidazole derivativesEl-Nassan, H. B. et al. | 2012
- 28
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Synthesis and antitumor evaluation of novel Benzo[d]pyrrolo[2,1-b]thiazole derivativesChaniyara, R. / Tala, S. / Chen, C. W. / Lee, P. C. / Kakadiya, R. / Dong, H. / Marvania, B. / Chen, C. H. / Chou, T. C. / Lee, T. C. et al. | 2012
- 41
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Synthesis of benzimidazolyl-1,3,4-oxadiazol-2ylthio-N-phenyl (benzothiazolyl) acetamides as antibacterial, antifungal and antituberculosis agentsPatel, R. V. / Patel, P. K. / Kumari, P. / Rajani, D. P. / Chikhalia, K. H. et al. | 2012
- 52
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12-N-Methylated 5,6-dihydrobenzo[c]acridine derivatives: A new class of highly selective ligands for c-myc G-quadruplex DNALiao, S. R. / Zhou, C. X. / Wu, W. B. / Ou, T. M. / Tan, J. H. / Li, D. / Gu, L. Q. / Huang, Z. S. et al. | 2012
- 64
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Isoxazolo(aza)naphthoquinones: A new class of cytotoxic Hsp90 inhibitorsBargiotti, A. / Musso, L. / Dallavalle, S. / Merlini, L. / Gallo, G. / Ciacci, A. / Giannini, G. / Cabri, W. / Penco, S. / Vesci, L. et al. | 2012
- 76
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Self-organizing molecular field analysis of NSAIDs: Assessment of pharmacokinetic and physicochemical properties using 3D-QSPkR approachHoney / Thareja, S. / Kumar, M. / Sinha, V. R. et al. | 2012
- 83
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5-Acetyl-2-arylbenzimidazoles as antiviral agents. Part 4Vitale, G. / Corona, P. / Loriga, M. / Carta, A. / Paglietti, G. / Giliberti, G. / Sanna, G. / Farci, P. / Marongiu, M. E. / La Colla, P. et al. | 2012
- 98
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Investigation on the pharmacological profile of 2,6-diacetylpyridine bis(benzoylhydrazone) derivatives and their antimony(III) and bismuth(III) complexesFerraz, K. S. O. / Silva, N. F. / da Silva, J. G. / de Miranda, L. F. / Romeiro, C. F. D. / Souza-Fagundes, E. M. / Mendes, I. C. / Beraldo, H. et al. | 2012
- 107
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Quinazolino-benzothiazoles: Fused pharmacophores as anticonvulsant agentsUgale, V. G. / Patel, H. M. / Wadodkar, Sudhir.G. / Bari, S. B. / Shirkhedkar, A. A. / Surana, S. J. et al. | 2012
- 114
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Synthesis of N^6-alkyl(aryl)-2-alkyl(aryl)thioadenosines as antiplatelet agentsLiu, G. / Xu, J. / Chen, N. / Zhang, S. / Ding, Z. / Du, H. et al. | 2012
- 124
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Benzothiazoles as probes for the 5HT"1"A receptor and the serotonin transporter (SERT): A search for new dual-acting agents as potential antidepressantsZhu, X. Y. / Etukala, J. R. / Eyunni, S. V. K. / Setola, V. / Roth, B. L. / Ablordeppey, S. Y. et al. | 2012
- 133
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Quinazoline-tyrphostin as a new class of antitumor agents, molecular properties prediction, synthesis and biological testingAlafeefy, A. M. / Alqasoumi, S. I. / Ashour, A. E. / Masand, V. / Al-Jaber, N. A. / Ben Hadda, T. / Mohamed, M. A. et al. | 2012
- 141
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New quinazolinone-pyrimidine hybrids: Synthesis, anti-inflammatory, and ulcerogenicity studiesAbbas, S. E. / Awadallah, F. M. / Ibrahin, N. A. / Said, E. G. / Kamel, G. M. et al. | 2012
- 150
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Structure-based virtual screening of novel inhibitors of the uridyltransferase activity of Xanthomonas oryzae pv. oryzae GlmUMin, J. / Lin, D. / Zhang, Q. / Zhang, J. / Yu, Z. et al. | 2012
- 159
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Synthesis of 4-methylcoumarin derivatives containing 4,5-dihydropyrazole moiety to scavenge radicals and to protect DNAXiao, C. / Luo, X. Y. / Li, D. J. / Lu, H. / Liu, Z. Q. / Song, Z. G. / Jin, Y. H. et al. | 2012
- 168
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Synthesis, characterization and in vitro antitumour activity of a series of novel platinum(II) complexes bearing Schiff base ligandsProetto, M. / Liu, W. / Hagenbach, A. / Abram, U. / Gust, R. et al. | 2012
- 176
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Synthesis, characterization, antimicrobial activities and QSAR studies of some 10a-phenylbenzo[b]indeno[1,2-e][1,4]thiazin-11(10aH)-onesMor, S. / Pahal, P. / Narasimhan, B. et al. | 2012
- 190
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Discovery, design and synthesis of Y-shaped peroxisome proliferator-activated receptor @d agonists as potent anti-obesity agents in vivoHam, J. / Hwang, H. / Kim, E. / Kim, J. a. / Cho, S. J. / Ko, J. / Lee, W. / Lee, J. / Holla, H. / Banerjee, J. et al. | 2012
- 203
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Design, synthesis and biological evaluation of a novel series of 1,3,4-oxadiazole bearing N-methyl-4-(trifluoromethyl)phenyl pyrazole moiety as cytotoxic agentsPuthiyapurayil, P. / Poojary, B. / Chikkanna, C. / Buridipad, S. K. et al. | 2012
- 211
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A variant peptide of buffalo colostrum @b-lactoglobulin inhibits angiotensin I-converting enzyme activityRohit, A. C. / Sathisha, K. / Aparna, H. S. et al. | 2012
- 220
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Synthesis and antiviral evaluation of C5-substituted-(1,3-diyne)-2'-deoxyuridinesSari, O. / Roy, V. / Balzarini, J. / Snoeck, R. / Andrei, G. / Agrofoglio, L. A. et al. | 2012
- 229
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Chiral resolution, absolute configuration assignment and biological activity of racemic diarylpyrimidine CH(OH)-DAPY as potent nonnucleoside HIV-1 reverse transcriptase inhibitorsGu, S. X. / Li, Z. M. / Ma, X. D. / Yang, S. Q. / He, Q. Q. / Chen, F. E. / De Clercq, E. / Balzarini, J. / Pannecouque, C. et al. | 2012
- 235
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Synthesis and evaluation of curcumin-related compounds for anticancer activityWei, X. / Du, Z. Y. / Zheng, X. / Cui, X. X. / Conney, A. H. / Zhang, K. et al. | 2012
- 246
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Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivativesSecci, D. / Bizzarri, B. / Bolasco, A. / Carradori, S. / D'Ascenzio, M. / Rivanera, D. / Mari, E. / Polletta, L. / Zicari, A. et al. | 2012
- 254
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2-Anilino-4-(benzimidazol-2-yl)pyrimidines - A multikinase inhibitor scaffold with antiproliferative activity toward cancer cell linesDetermann, R. / Dreher, J. / Baumann, K. / Preu, L. / Jones, P. G. / Totzke, F. / Schachtele, C. / Kubbutat, M. H. G. / Kunick, C. et al. | 2012
- 264
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@b-Lapachone analogs with enhanced antiproliferative activityRios-Luci, C. / Bonifazi, E. L. / Leon, L. G. / Montero, J. C. / Burton, G. / Pandiella, A. / Misico, R. I. / Padron, J. M. et al. | 2012
- 275
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Design, synthesis and antiviral activity of novel quinazolinonesWang, Z. / Wang, M. / Yao, X. / Li, Y. / Tan, J. / Wang, L. / Qiao, W. / Geng, Y. / Liu, Y. / Wang, Q. et al. | 2012
- 283
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Synthesis and fungicidal activity of novel pimprinine analoguesZhang, M. Z. / Chen, Q. / Mulholland, N. / Beattie, D. / Irwin, D. / Gu, Y. C. / Yang, G. F. / Clough, J. et al. | 2012
- 292
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Design, synthesis and structure-activity relationships of new triazole derivatives containing N-substituted phenoxypropylamino side chainsWang, S. / Jin, G. / Wang, W. / Zhu, L. / Zhang, Y. / Dong, G. / Liu, Y. / Zhuang, C. / Miao, Z. / Yao, J. et al. | 2012
- 300
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Synthesis and antimycobacterial activity of novel 1,3-dimethylisocyanurate derivativesShulaeva, M. M. / Fattakhov, S. G. / Saifina, L. F. / Chestnova, R. V. / Valijev, R.Sh. / Mingaleev, D. N. / Voloshina, A. D. / Reznik, V. S. et al. | 2012
- 308
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Synthesis, hypoglycemic and hypolipidemic activities of novel thiazolidinedione derivatives containing thiazole/triazole/oxadiazole ringMohammed Iqbal, A. K. / Khan, A. Y. / Kalashetti, M. B. / Belavagi, N. S. / Gong, Y. D. / Khazi, I. A. M. et al. | 2012
- 316
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Structure-activity relationships of saponin derivatives: A series of entry inhibitors for highly pathogenic H5N1 influenza virusDing, N. / Chen, Q. / Zhang, W. / Ren, S. / Guo, Y. / Li, Y. et al. | 2012
- 327
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Microwave assisted synthesis of spirocyclic pyrrolidines -@s"1 receptor ligands with modified benzene-N-distanceJasper, A. / Schepmann, D. / Lehmkuhl, K. / Vela, J. M. / Buschmann, H. / Holenz, J. / Wunsch, B. et al. | 2012
- 337
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Alkylidene branched lupane derivatives: Synthesis and antitumor activityCsuk, R. / Stark, S. / Nitsche, C. / Barthel, A. / Siewert, B. et al. | 2012
- 346
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Synthesis, in vitro and in silico screening of ethyl 2-(6-substituted benzo[d]thiazol-2-ylamino)-2-oxoacetates as protein-tyrosine phosphatase 1B inhibitorsNavarrete-Vazquez, G. / Ramirez-Martinez, M. / Estrada-Soto, S. / Nava-Zuazo, C. / Paoli, P. / Camici, G. / Escalante-Garcia, J. / Medina-Franco, J. L. / Lopez-Vallejo, F. / Ortiz-Andrade, R. et al. | 2012
- 356
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Convenient synthesis of novel geiparvarin analogs with potential anti-cancer activity via click chemistryZhang, Y. / Lv, Z. / Zhong, H. / Geng, D. / Zhang, M. / Zhang, T. / Li, Y. / Li, K. et al. | 2012
- 364
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Synthesis, evaluation of anticancer activity and COMPARE analysis of N-bis(trifluoromethyl)alkyl-N'-substituted ureas with pharmacophoric moietiesLuzina, E. L. / Popov, A. V. et al. | 2012
- 374
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The synthesis of 2,5-bis(4-amidinophenyl)thiophene derivatives providing submicromolar-range inhibition of the botulinum neurotoxin serotype A metalloproteaseOpsenica, I. / Filipovic, V. / Nuss, J. E. / Gomba, L. M. / Opsenica, D. / Burnett, J. C. / Gussio, R. / Solaja, B. A. / Bavari, S. et al. | 2012
- 380
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Synthesis and characterization of some new complexes of Cu(II), Ni(II) and V(IV) with Schiff base derived from indole-3-carboxaldehyde. Biological activity on prokaryotes and eukaryotesRosu, T. / Pahontu, E. / Ilies, D. C. / Georgescu, R. / Mocanu, M. / Leabu, M. / Shova, S. / Gulea, A. et al. | 2012
- 390
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Appraisal of GABA and PABA as linker: Design and synthesis of novel benzamide based histone deacetylase inhibitorsRajak, H. / Kumar, P. / Parmar, P. / Thakur, B. S. / Veerasamy, R. / Sharma, P. C. / Sharma, A. K. / Gupta, A. K. / Dangi, J. S. et al. | 2012
- 398
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Synthesis of new 2-galactosylthiazolidine-4-carboxylic acid amides. Antitumor evaluation against melanoma and breast cancer cellsSerra, A. C. / Rocha Gonsalves, A. M.d'A. / Laranjo, M. / Abrantes, A. M. / Goncalves, A. C. / Sarmento-Ribeiro, A. B. / Botelho, M. F. et al. | 2012
- 403
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Anticancer and radiosensitizing evaluation of some new pyranothiazole-Schiff bases bearing the biologically active sulfonamide moietyGhorab, M. M. / Shaaban, M. A. / Refaat, H. M. / Heiba, H. I. / Ibrahim, S. S. et al. | 2012
- 408
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Synthesis and in vitro characterization of trans- and cis-[^1^8F]-4-methylbenzyl 4-[(pyrimidin-2-ylamino)methyl]-3-fluoropiperidine-1-carboxylates as new potential PET radiotracer candidates for the NR2B subtype N-methyl-d-aspartate receptorKoudih, R. / Gilbert, G. / Dhilly, M. / Abbas, A. / Barre, L. / Debruyne, D. / Sobrio, F. et al. | 2012
- 416
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A solvent free, four-component synthesis and 1,3-dipolar cycloaddition of 4(H)-pyrans with nitrile oxides: Synthesis and discovery of antimycobacterial activity of enantiomerically pure 1,2,4-oxadiazolesAlmansour, A. I. / Suresh Kumar, R. / Arumugam, N. / Sriram, D. et al. | 2012