3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase Inhibitors (Unknown)
- New search for: Massa, Silvio
- New search for: Mai, Antonello
- New search for: Sbardella, Gianluca
- New search for: Esposito, Monica
- New search for: Ragno, Rino
- New search for: Loidl, Peter
- New search for: Brosch, Gerald
- New search for: Massa, Silvio
- New search for: Mai, Antonello
- New search for: Sbardella, Gianluca
- New search for: Esposito, Monica
- New search for: Ragno, Rino
- New search for: Loidl, Peter
- New search for: Brosch, Gerald
In:
Journal of Medicinal Chemistry
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44
, 13
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2069-2072
;
2001
- Article (Journal) / Electronic Resource
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Title:3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase Inhibitors
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Additional title:J. Med. Chem.
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Contributors:Massa, Silvio ( author ) / Mai, Antonello ( author ) / Sbardella, Gianluca ( author ) / Esposito, Monica ( author ) / Ragno, Rino ( author ) / Loidl, Peter ( author ) / Brosch, Gerald ( author )
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Published in:Journal of Medicinal Chemistry ; 44, 13 ; 2069-2072
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Publisher:
- New search for: American Chemical Society
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Publication date:2001-06-21
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ISSN:
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Coden:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:Unknown
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Source:
Table of contents – Volume 44, Issue 13
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 2039
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Secretase Targets for Alzheimer's Disease: Identification and Therapeutic Potential †Wolfe, Michael S. et al. | 2001
- 2061
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Design and Synthesis of 2-Methyl-2-{4-[2-(5-methyl-2-aryloxazol- 4-yl)ethoxy]phenoxy}propionic Acids: A New Class of Dual PPARα/γ AgonistsBrooks, Dawn A. / Etgen, Garret J. / Rito, Christopher J. / Shuker, Anthony J. / Dominianni, Samuel J. / Warshawsky, Alan M. / Ardecky, Robert / Paterniti, James R. / Tyhonas, John / Karanewsky, Donald S. et al. | 2001
- 2061
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Letters - Design and Synthesis of 2-Methyl-2-(4-(2-(5-methyl-2-aryloxazol- 4-yl)ethoxy)phenoxy)propionic Acids: A New Class of Dual PPAR a-g AgonistsBrooks, Dawn A. et al. | 2001
- 2065
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Letters - Potential New Antitumor Agents from an Innovative Combination of Demethylcantharidin, a Modified Traditional Chinese Medicine, with a Platinum MoietyHo, Yee-Ping et al. | 2001
- 2065
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Potential New Antitumor Agents from an Innovative Combination of Demethylcantharidin, a Modified Traditional Chinese Medicine, with a Platinum MoietyHo, Yee-Ping / To, Kenneth K. W. / Au-Yeung, Steve C. F. / Wang, Xinning / Lin, Ge / Han, Xiuwen et al. | 2001
- 2069
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Letters - 3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase InhibitorsMassa, Silvio et al. | 2001
- 2069
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3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase InhibitorsMassa, Silvio / Mai, Antonello / Sbardella, Gianluca / Esposito, Monica / Ragno, Rino / Loidl, Peter / Brosch, Gerald et al. | 2001
- 2073
-
Articles - Transformation of a k-Opioid Receptor Antagonist to a k-Agonist by Transfer of a Guanidinium Group from the 5'- to 6'-Position of NaltrindoleSharma, Shiv Kumar et al. | 2001
- 2073
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Transformation of a κ-Opioid Receptor Antagonist to a κ-Agonist by Transfer of a Guanidinium Group from the 5‘- to 6‘-Position of NaltrindoleSharma, Shiv Kumar / Jones, Robert M. / Metzger, Thomas G. / Ferguson, David M. / Portoghese, Philip S. et al. | 2001
- 2080
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Adenosine Analogues as Selective Inhibitors of Glyceraldehyde-3-phosphate Dehydrogenase of Trypanosomatidae via Structure-Based Drug DesignBressi, Jerome C. / Verlinde, Christophe L. M. J. / Aronov, Alex M. / Shaw, My Le / Shin, Sam S. / Nguyen, Lisa N. / Suresh, Stephen / Buckner, Frederick S. / Van Voorhis, Wesley C. / Kuntz, Irwin D. et al. | 2001
- 2080
-
Articles - Adenosine Analogues as Selective Inhibitors of Glyceraldehyde-3-phosphate Dehydrogenase of Trypanosomatidae via Structure-Based Drug DesignBressi, Jerome C. et al. | 2001
- 2094
-
Development of Potent Non-Carbohydrate Imidazole-Based Small Molecule Selectin Inhibitors with Antiinflammatory ActivitySlee, Deborah H. / Romano, Suzanne J. / Yu, Jinghua / Nguyen, Truc N. / John, Judy K. / Raheja, Neil K. / Axe, Frank U. / Jones, Todd K. / Ripka, William C. et al. | 2001
- 2094
-
Articles - Development of Potent Non-Carbohydrate Imidazole-Based Small Molecule Selectin Inhibitors with Antiinflammatory ActivitySlee, Deborah H. et al. | 2001
- 2108
-
Articles - Bicyclic Analogues of D-myo-Inositol 1,4,5-Trisphosphate Related to Adenophostin A: Synthesis and Biological ActivityRiley, Andrew M. et al. | 2001
- 2108
-
Bicyclic Analogues of d-myo-Inositol 1,4,5-Trisphosphate Related to Adenophostin A: Synthesis and Biological ActivityRiley, Andrew M. / Correa, Vanessa / Mahon, Mary F. / Taylor, Colin W. / Potter, Barry V. L. et al. | 2001
- 2118
-
Articles - Synthesis, Biological Evaluation, and Pharmacophore Generation of New Pyridazinone Derivatives with Affinity toward a1- and a2-AdrenoceptorsBarbaro, Roberta et al. | 2001
- 2118
-
Synthesis, Biological Evaluation, and Pharmacophore Generation of New Pyridazinone Derivatives with Affinity toward α1- and α2-AdrenoceptorsBarbaro, Roberta / Betti, Laura / Botta, Maurizio / Corelli, Federico / Giannaccini, Gino / Maccari, Laura / Manetti, Fabrizio / Strappaghetti, Giovannella / Corsano, Stefano et al. | 2001
- 2133
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Discovery of 4-Amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin- 3-yl)pyrido[2,3-d]pyrimidine, an Orally Active, Non-Nucleoside Adenosine Kinase InhibitorLee, Chih-Hung / Jiang, Meiqun / Cowart, Marlon / Gfesser, Greg / Perner, Richard / Kim, Ki Hwan / Gu, Yu Gui / Williams, Michael / Jarvis, Michael F. / Kowaluk, Elizabeth A. et al. | 2001
- 2133
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Articles - Discovery of 4-Amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin- 3-yl)pyrido(2,3-d)-pyrimidine, an Orally Active, Non-Nucleoside Adenosine Kinase InhibitorLee, Chih-Hung et al. | 2001
- 2139
-
Articles - Synthesis and Activities of Pyoverdin-Quinolone Adducts: A Prospective Approach to a Specific Therapy Against Pseudomonas aeruginosaHennard, Christophe et al. | 2001
- 2139
-
Synthesis and Activities of Pyoverdin−Quinolone Adducts: A Prospective Approach to a Specific Therapy Against Pseudomonas a eruginosaHennard, Christophe / Truong, Que Chi / Desnottes, Jean-François / Paris, Jean-Marc / Moreau, Nicole J. / Abdallah, Mohamed A. et al. | 2001
- 2152
-
Articles - Synthesis of Novel g-Aminobutyric Acid (GABA) Uptake Inhibitors. 5. Preparation and Structure-Activity Studies of Tricyclic Analogues of Known GABA Uptake InhibitorsAndersen, Knud Erik et al. | 2001
- 2152
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Synthesis of Novel γ-Aminobutyric Acid (GABA) Uptake Inhibitors. 5. Preparation and Structure−Activity Studies of Tricyclic Analogues of Known GABA Uptake InhibitorsAndersen, Knud Erik / Sørensen, Jan L. / Lau, Jesper / Lundt, Behrend F. / Petersen, Hans / Huusfeldt, Per O. / Suzdak, Peter D. / Swedberg, Michael D. B. et al. | 2001
- 2164
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Synthesis, Cytotoxicity, and Antitumor Activity of Copper(II) and Iron(II) Complexes of 4 N-Azabicyclo[3.2.2]nonane Thiosemicarbazones Derived from Acyl DiazinesEasmon, Johnny / Pürstinger, Gerhard / Heinisch, Gottfried / Roth, Thomas / Fiebig, Heinz H. / Holzer, Wolfgang / Jäger, Walter / Jenny, Marcel / Hofmann, Johann et al. | 2001
- 2164
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Articles - Synthesis, Cytotoxicity, and Antitumor Activity of Copper(II) and Iron(II) Complexes of 4N-Azabicyclo(3.2.2)nonane Thiosemicarbazones Derived from Acyl DiazinesEasmon, Johnny et al. | 2001
- 2172
-
Combinatorial Synthesis of Cholesterol Ester Transfer Protein-mRNA Ligands and Screening by Nondenaturating Gel-ElectrophoresisBaumann, Michael / Bischoff, Hilmar / Schmidt, Delf / Griesinger, Christian et al. | 2001
- 2172
-
Articles - Combinatorial Synthesis of Cholesterol Ester Transfer Protein-mRNA Ligands and Screening by Nondenaturating Gel-ElectrophoresisBaumann, Michael et al. | 2001
- 2178
-
Probing the Interaction of Dengue Virus Envelope Protein with Heparin: Assessment of Glycosaminoglycan-Derived InhibitorsMarks, Rory M. / Lu, Hong / Sundaresan, Renuka / Toida, Toshihiko / Suzuki, Atsushi / Imanari, Toshio / Hernáiz, María J. / Linhardt, Robert J. et al. | 2001
- 2178
-
Articles - Probing the Interaction of Dengue Virus Envelope Protein with Heparin: Assessment of Glycosaminoglycan-Derived InhibitorsMarks, Rory M. et al. | 2001
- 2188
-
Amphiphilic Anionic Analogues of Galactosylceramide: Synthesis, Anti-HIV-1 Activity, and gp120 BindingFaroux-Corlay, Barbara / Greiner, Jacques / Terreux, Raphaël / Cabrol-Bass, Daniel / Aubertin, Anne-Marie / Vierling, Pierre / Fantini, Jacques et al. | 2001
- 2188
-
Articles - Amphiphilic Anionic Analogues of Galactosylceramide: Synthesis, Anti-HIV-1 Activity, and gp120 BindingFaroux-Corlay, Barbara et al. | 2001
- 2204
-
Articles - Novel, Potent, and Selective Phosphodiesterase 5 Inhibitors: Synthesis and Biological Activities of a Series of 4-Aryl-1-isoquinolinone DerivativesUkita, Tatsuzo et al. | 2001
- 2204
-
Novel, Potent, and Selective Phosphodiesterase 5 Inhibitors: Synthesis and Biological Activities of a Series of 4-Aryl-1-isoquinolinone DerivativesUkita, Tatsuzo / Nakamura, Yoshinori / Kubo, Akira / Yamamoto, Yasuo / Moritani, Yasunori / Saruta, Kunio / Higashijima, Takanori / Kotera, Jun / Takagi, Michino / Kikkawa, Kohei et al. | 2001
- 2219
-
5-(Tryptophyl)amino-1,3-dioxoperhydropyrido[1,2-c]pyrimidine-Based Potent and Selective CCK1 Receptor Antagonists: Structure−Activity Relationship Studies on the Substituent at N2-PositionBartolomé-Nebreda, José M. / Patiño-Molina, Rosario / Martín-Martínez, Mercedes / Gómez-Monterrey, Isabel / García-López, M. Teresa / González-Muñiz, Rosario / Cenarruzabeitia, Edurne / Latorre, Miriam / Río, Joaquín Del / Herranz, Rosario et al. | 2001
- 2219
-
Articles - 5-(Tryptophyl)amino-1,3-dioxoperhydropyrido(1,2-c)-pyrimidine-Based Potent and Selective CCK1 Receptor Antagonists: Structure-Activity Relationship Studies on the Substituent at N2-PositionBartolomé-Nebreda, José M. et al. | 2001
- 2229
-
Articles - Synthesis, Nicotinic Acetylcholine Receptor Binding, and Antinociceptive Properties of 2-exo-2-(2'-Substituted 5'-pyridinyl)- 7-azabicyclo(2.2.1)heptanes. Epibatidine AnaloguesCarroll, F.Ivy et al. | 2001
- 2229
-
Synthesis, Nicotinic Acetylcholine Receptor Binding, and Antinociceptive Properties of 2-exo-2-(2‘-Substituted 5‘-pyridinyl)-7-azabicyclo[2.2.1]heptanes. Epibatidine AnaloguesCarroll, F. Ivy / Liang, Feng / Navarro, Hernán A. / Brieaddy, Lawrence E. / Abraham, Philip / Damaj, M. I. / Martin, Billy R. et al. | 2001
- 2238
-
Potent Somatostatin Undecapeptide Agonists Selective for Somatostatin Receptor 1 (sst1)Rivier, Jean E. / Hoeger, Carl / Erchegyi, Judit / Gulyas, Jozsef / DeBoard, Ryan / Craig, A. Grey / Koerber, Steven C. / Wenger, Sandra / Waser, Beatrice / Schaer, Jean-Claude et al. | 2001
- 2238
-
Articles - Potent Somatostatin Undecapeptide Agonists Selective for Somatostatin Receptor 1 (sst1)Rivier, Jean E. et al. | 2001
- 2247
-
Articles - Characterization of Melanocortin NDP-MSH Agonist Peptide Fragments at the Mouse Central and Peripheral Melanocortin ReceptorsHaskell-Luevano, Carrie et al. | 2001
- 2247
-
Characterization of Melanocortin NDP-MSH Agonist Peptide Fragments at the Mouse Central and Peripheral Melanocortin ReceptorsHaskell-Luevano, Carrie / Holder, Jerry Ryan / Monck, Eileen K. / Bauzo, Rayna M. et al. | 2001
- 2253
-
Articles - Protease Inhibitors: Synthesis of a Series of Bacterial Collagenase Inhibitors of the Sulfonyl Amino Acyl Hydroxamate TypeClare, Brian W. et al. | 2001
- 2253
-
Protease Inhibitors: Synthesis of a Series of Bacterial Collagenase Inhibitors of the Sulfonyl Amino Acyl Hydroxamate TypeClare, Brian W. / Scozzafava, Andrea / Supuran, Claudiu T. et al. | 2001