A New Class of Diamine-Based Human Histamine H3 Receptor Antagonists: 4-(Aminoalkoxy)benzylamines (Unknown)
- New search for: Apodaca, Richard
- New search for: Dvorak, Curt A.
- New search for: Xiao, Wei
- New search for: Barbier, Ann J.
- New search for: Boggs, Jamin D.
- New search for: Wilson, Sandy J.
- New search for: Lovenberg, Timothy W.
- New search for: Carruthers, Nicholas I.
- New search for: Apodaca, Richard
- New search for: Dvorak, Curt A.
- New search for: Xiao, Wei
- New search for: Barbier, Ann J.
- New search for: Boggs, Jamin D.
- New search for: Wilson, Sandy J.
- New search for: Lovenberg, Timothy W.
- New search for: Carruthers, Nicholas I.
In:
Journal of Medicinal Chemistry
;
46
, 18
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3938-3944
;
2003
- Article (Journal) / Electronic Resource
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Title:A New Class of Diamine-Based Human Histamine H3 Receptor Antagonists: 4-(Aminoalkoxy)benzylamines
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Additional title:J. Med. Chem.
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Contributors:Apodaca, Richard ( author ) / Dvorak, Curt A. ( author ) / Xiao, Wei ( author ) / Barbier, Ann J. ( author ) / Boggs, Jamin D. ( author ) / Wilson, Sandy J. ( author ) / Lovenberg, Timothy W. ( author ) / Carruthers, Nicholas I. ( author )
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Published in:Journal of Medicinal Chemistry ; 46, 18 ; 3938-3944
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Publisher:
- New search for: American Chemical Society
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Publication date:2003-08-28
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ISSN:
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Coden:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:Unknown
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Source:
Table of contents – Volume 46, Issue 18
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 3771
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Structure-Based Design of a Macrocyclic Inhibitor for Peptide DeformylaseHu, Xubo / Nguyen, Kiet T. / Verlinde, Christophe L. M. J. / Hol, Wim G. J. / Pei, Dehua et al. | 2003
- 3775
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N6-Substituted D-4‘-Thioadenosine-5‘-methyluronamides: Potent and Selective Agonists at the Human A3 Adenosine ReceptorJeong, Lak Shin / Jin, Dong Zhe / Kim, Hea Ok / Shin, Dae Hong / Moon, Hyung Ryong / Gunaga, Prashantha / Chun, Moon Woo / Kim, Yong-Chul / Melman, Neli / Gao, Zhan-Guo et al. | 2003
- 3778
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Fluorine Substitution Can Block CYP3A4 Metabolism-Dependent Inhibition: Identification of (S)-N-[1-(4-Fluoro-3- morpholin-4-ylphenyl)ethyl]-3- (4-fluorophenyl)acrylamide as an Orally Bioavailable KCNQ2 Opener Devoid of CYP3A4 Metabolism-Dependent InhibitionWu, Yong-Jin / Davis, Carl D. / Dworetzky, Steven / Fitzpatrick, William C. / Harden, David / He, Huan / Knox, Ronald J. / Newton, Amy E. / Philip, Thomas / Polson, Craig et al. | 2003
- 3782
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A Novel Approach of Water-Soluble Paclitaxel Prodrug with No Auxiliary and No Byproduct: Design and Synthesis of IsotaxelHayashi, Yoshio / Skwarczynski, Mariusz / Hamada, Yoshio / Sohma, Youhei / Kimura, Tooru / Kiso, Yoshiaki et al. | 2003
- 3785
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Influence of Phenyl Ring Disubstitution on Bisbenzimidazole and Terbenzimidazole Cytotoxicity: Synthesis and Biological Evaluation as RadioprotectorsTawar, Urmila / Jain, Akash K. / Dwarakanath, B. S. / Chandra, Ramesh / Singh, Yogendra / Chaudhury, N. K. / Khaitan, Divya / Tandon, Vibha et al. | 2003
- 3793
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Thalidomide Metabolites and Analogues. 3. Synthesis and Antiangiogenic Activity of the Teratogenic and TNFa-Modulatory Thalidomide Analogue 2-(2,6-Dioxopiperidine-3-yl)phthalimidine1Luzzio, F.A. et al. | 2003
- 3793
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Thalidomide Metabolites and Analogues. 3. Synthesis and Antiangiogenic Activity of the Teratogenic and TNFα-Modulatory Thalidomide Analogue 2-(2,6-Dioxopiperidine-3-yl)phthalimidineLuzzio, Frederick A. / Mayorov, Alexander V. / Ng, Sylvia S. W. / Kruger, Erwin A. / Figg, William D. et al. | 2003
- 3800
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Novel Pyrone Side Tetracyclic Psoralen Derivatives: Synthesis and Photobiological EvaluationDalla Via, Lisa / Uriarte, Eugenio / Quezada, Elias / Dolmella, Alessandro / Ferlin, Maria Grazia / Gia, Ornella et al. | 2003
- 3811
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3‘-C-Branched-Chain-Substituted Nucleosides and Nucleotides as Potent Inhibitors of Mycobacterium t uberculosis Thymidine Monophosphate KinaseVanheusden, Veerle / Munier-Lehmann, Hélène / Froeyen, Matheus / Dugué, Laurence / Heyerick, Arne / De Keukeleire, Denis / Pochet, Sylvie / Busson, Roger / Herdewijn, Piet / Van Calenbergh, Serge et al. | 2003
- 3822
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Synthesis and Pharmacological Evaluation of Potent and Highly Selective D3 Receptor Ligands: Inhibition of Cocaine-Seeking Behavior and the Role of Dopamine D3/D2 Receptors †Campiani, Giuseppe / Butini, Stefania / Trotta, Francesco / Fattorusso, Caterina / Catalanotti, Bruno / Aiello, Francesca / Gemma, Sandra / Nacci, Vito / Novellino, Ettore / Stark, Jennifer Ann et al. | 2003
- 3840
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Stereospecific Synthesis of 5-Substituted 2-Bisarylthiocyclopentane Carboxylic Acids as Specific Matrix Metalloproteinase InhibitorsLe Diguarher, Thierry / Chollet, Anne-Marie / Bertrand, Marc / Hennig, Philippe / Raimbaud, Eric / Sabatini, Massimo / Guilbaud, Nicolas / Pierré, Alain / Tucker, Gordon C. / Casara, Patrick et al. | 2003
- 3853
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Synthesis, Biological Evaluation, and Receptor Docking Simulations of 2-((Acylamino)ethyl)-1,4-benzodiazepines as k-Opioid Receptor Agonists Endowed with Antinociceptive and Antiamnesic ActivityAnzini, M. et al. | 2003
- 3853
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Synthesis, Biological Evaluation, and Receptor Docking Simulations of 2-[(Acylamino)ethyl]-1,4-benzodiazepines as κ-Opioid Receptor Agonists Endowed with Antinociceptive and Antiamnesic ActivityAnzini, Maurizio / Canullo, Laura / Braile, Carlo / Cappelli, Andrea / Gallelli, Andrea / Vomero, Salvatore / Menziani, M. Cristina / De Benedetti, Pier G. / Rizzo, Milena / Collina, Simona et al. | 2003
- 3865
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Potent, Small-Molecule Inhibitors of Human Mast Cell Tryptase. Antiasthmatic Action of a Dipeptide-Based Transition-State Analogue Containing a Benzothiazole KetoneCostanzo, Michael J. / Yabut, Stephen C. / Almond,, Harold R. / Andrade-Gordon, Patricia / Corcoran, Thomas W. / de Garavilla, Lawrence / Kauffman, Jack A. / Abraham, William M. / Recacha, Rosario / Chattopadhyay, Debashish et al. | 2003
- 3877
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Oxindole-Based Compounds Are Selective Inhibitors of Plasmodium f alciparum Cyclin Dependent Protein KinasesWoodard, Cassandra L. / Li, Zhiyu / Kathcart, April K. / Terrell, James / Gerena, Lucia / Lopez-Sanchez, Miriam / Kyle, Dennis E. / Bhattacharjee, Apurba K. / Nichols, Daniel A. / Ellis, William et al. | 2003
- 3883
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N-(w-(4-(2-Methoxyphenyl)piperazin-1-yl)alkyl)carboxamides as Dopamine D2 and D3 Receptor LigandsHackling, A. et al. | 2003
- 3883
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N-(ω-(4-(2-Methoxyphenyl)piperazin-1-yl)alkyl)carboxamides as Dopamine D2 and D3 Receptor LigandsHackling, Anneke / Ghosh, Robin / Perachon, Sylvie / Mann, André / Höltje, Hans-Dieter / Wermuth, Camille G. / Schwartz, Jean-Charles / Sippl, Wolfgang / Sokoloff, Pierre / Stark, Holger et al. | 2003
- 3900
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Synthesis and Biological Evaluation of Novel Flavone-8-acetic Acid Derivatives as Reversible Inhibitors of Aminopeptidase N/CD13Bauvois, Brigitte / Puiffe, Marie-Line / Bongui, Jean-Bernard / Paillat, Sandrine / Monneret, Claude / Dauzonne, Daniel et al. | 2003
- 3914
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DNA Binding Ligands Targeting Drug-Resistant Bacteria: Structure, Activity, and PharmacologyKaizerman, Jacob A. / Gross, Matthew I. / Ge, Yigong / White, Sarah / Hu, Wenhao / Duan, Jian-Xin / Baird, Eldon E. / Johnson, Kirk W. / Tanaka, Richard D. / Moser, Heinz E. et al. | 2003
- 3930
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Binding of Tetrahydrocarboline Derivatives at Human 5-HT5A ReceptorsKhorana, Nantaka / Smith, Carol / Herrick-Davis, Kathy / Purohit, Anil / Teitler, Milt / Grella, Brian / Dukat, Małgorzata / Glennon, Richard A. et al. | 2003
- 3938
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A New Class of Diamine-Based Human Histamine H3 Receptor Antagonists: 4-(Aminoalkoxy)benzylaminesApodaca, Richard / Dvorak, Curt A. / Xiao, Wei / Barbier, Ann J. / Boggs, Jamin D. / Wilson, Sandy J. / Lovenberg, Timothy W. / Carruthers, Nicholas I. et al. | 2003
- 3945
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Pyrazole Derivatives as Partial Agonists for the Nicotinic Acid Receptorvan Herk, T. / Brussee, J. / van den Nieuwendijk, A. M. C. H. / van der Klein, P. A. M. / IJzerman, A. P. / Stannek, C. / Burmeister, A. / Lorenzen, A. et al. | 2003
- 3952
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Books of Interest| 2003