Steric structure-activity relationship studies on a new butyrophenone derivative (English)
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- New search for: Li, J. Pengman
- New search for: Biel, John H.
- New search for: Li, J. Pengman
- New search for: Biel, John H.
In:
Journal of Medicinal Chemistry
;
12
, 5
;
917-919
;
1969
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ISSN:
- Article (Journal) / Electronic Resource
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Title:Steric structure-activity relationship studies on a new butyrophenone derivative
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Additional title:J. Med. Chem.
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Contributors:Li, J. Pengman ( author ) / Biel, John H. ( author )
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Published in:Journal of Medicinal Chemistry ; 12, 5 ; 917-919
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Publisher:
- New search for: American Chemical Society
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Publication date:1969-09-01
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ISSN:
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Coden:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Source:
Table of contents – Volume 12, Issue 5
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 3A
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Masthead| 1969
- 731
-
Synthesis and some pharmacological activities of [2-L-valine]-oxytocin and [2-L-leucine]-oxytocinHruby, Victor J. / Du Vigneaud, Vincent et al. | 1969
- 733
-
Angiotensin II analogs. I. Synthesis and biological evaluation of [Gly1,Gly2,Ile5]-angiotensin II, [Ac-Gly1,Gly2,Ile5]-angiotensin II, and [Gly1,Gly2,Ile5,His(Bzl)6]-angiotensin IIJorgensen, Eugene C. / Windridge, Graham C. / Patton, Walter / Lee, Thomas Choy et al. | 1969
- 737
-
Synthesis and microbiological properties of dipeptides containing cyclopentaneglycine and .beta.-2-thienylalanineHill, Jim Tom / Dunn, Floyd W. et al. | 1969
- 740
-
Kinetics and mechanisms of action of drugs on microorganisms. VIII. Quantification and prediction of the biological activities of meta- and para-substituted N1-phenylsulfanilamides by microbial kineticsGarrett, Edward R. / Mielck, Jobst B. / Seydel, Joachim K. / Kessler, Hans J. et al. | 1969
- 746
-
Homolytic constants in the correlation of chloramphenicol structure with activityHansch, Corwin / Kutter, Eberhard / Leo, A. et al. | 1969
- 749
-
Structure-activity relationships among substrates for a rabbit kidney reductase. Quantum chemical calculation of substituent parametersHermann, Robert B. / Culp, Hilman W. / McMahon, Robert E. / Marsh, Max M. et al. | 1969
- 754
-
Species difference in the competitive binding of 2-(4'-hydroxybenzeneazo)benzoic acid (HBABA) and .alpha.-(4-chlorophenoxy)-.alpha.-methylpropionic acid (CPMPA) to serum albumin. A possible model system for studying allosteric transitionsWitiak, Donald T. / Sokoloski, Theodore D. / Whitehouse, Michael W. / Hermann, Freya et al. | 1969
- 761
-
Molecular orbital calculations on anticonvulsant drugsAndrews, P. R. et al. | 1969
- 764
-
Molecular orbital calculations on a new series of substituted-phenyl choline ethersCrow, James / Wassermann, Otmar / Holland, William C. et al. | 1969
- 766
-
Comparison of parameters currently used in the study of structure-activity relationshipsLeo, A. / Hansch, Corwin / Church, C. et al. | 1969
- 771
-
Potential antitumor agents. II. Effects of modifications in the side chain of 1-formylisoquinoline thiosemicarbazoneAgrawal, Krishna C. / Sartorelli, Alan C. et al. | 1969
- 775
-
Synthesis and relationship between structure and activity of 2-nitroimidazole derivativesLancini, Gian C. / Lazzari, Ettore / Arioli, V. / Bellani, P. et al. | 1969
- 780
-
Lincomycin. VIII. 4'-Alkyl-1'-demethyl-4'-depropylclindamycins, potent antibacterial and antimalarial agentsMagerlein, Barney J. / Kagan, Fred et al. | 1969
- 784
-
Preparation and antimycotic properties of derivatives of 1-phenethylimidazoleGodefroi, Erik F. / Heeres, Jan / Van Cutsem, Jan / Janssen, Paul A. J. et al. | 1969
- 791
-
Imidoylureas. A new class of anthelminticsDiana, Guy D. / Yarinsky, Allen / Zalay, Ethel S. / Berberian, Dicran A. / Schalit, Samuel et al. | 1969
- 794
-
ImidazolylphosphonamidochloridothionatesBudde, Paul B. / Tolkmith, Henry et al. | 1969
- 797
-
Diaminoquinoline antimalarialsHeindel, Ned D. / Bechara, Ibrahim S. / Ohnmacht, Cyrus J. / Molnar, James / Lemke, Thomas F. / Kennewell, Peter D. et al. | 1969
- 801
-
Antimalarials. 4-Proximal hydrazino derivatives of 7-chloroquinolineSingh, Tara / Stein, Robert G. / Biel, John H. et al. | 1969
- 804
-
Imidazolecarbohydrazides. III. Chemistry and biological evaluationNulu, J. R. / Nematollahi, Jay et al. | 1969
- 806
-
Anthelmintic quaternary salts. IV. Aminopentadienylideneammonium saltsGarmaise, David L. / Paris, Gerard Y. / Komlossy, Jacqueline / McCrae, R. C. et al. | 1969
- 810
-
Steroids. LXXXIII. Effects of some steroidal alkylating agents on experimental animal mammary tumor and leukemia systemsWall, Monroe E. / Abernethy, G. Shuford / Carroll, F. I. / Taylor, Dorothy Jane et al. | 1969
- 818
-
Fluorescent alkylating agents. 1-(.beta.-chloroethyl)bisbenzimidazolesTsou, Kwan Chung / Rabiger, Dorothy J. / Sobel, Barbara et al. | 1969
- 822
-
Derivatives of fluorene. XXX. Rearrangement and antitumor activities of some 9-oxofluorene oximes. 6(5H)-phenanthridinones. 1Pan, Hsi-Lung / Fletcher, T. Lloyd et al. | 1969
- 825
-
Potential carcinolytic agents. VII. Substituted bis(2-methanesulfonoxyethyl)anilinesPapanastassiou, Zion B. / Bruni, Robert J. / Estes, Peggy B. / Wodinsky, Isidore et al. | 1969
- 828
-
Charge-spatial models. cis- and trans-3- and -4-Substituted cyclohexyl phosphates as analogs of 2'-deoxyuridine 5'-phosphateMertes, Mathias P. / Coats, Eugene A. et al. | 1969
- 832
-
Physicochemical model for the mechanism of action of antihistaminics and cortisolBotre, Claudio / Marchetti, Marcello / Del Vecchio-Blanco, Camillo / Lionetti, G. / Memoli, Adriana et al. | 1969
- 836
-
Bicyclic homologs of piperazine. IX. Synthesis and pharmacological properties of phenothiazine and of 10,11-dihydrodibenzocycloheptene derivatives of 3,8-diazabicyclo[3.2.1]octanesCignarella, Giorgio / Occelli, Emilio / Maffii, Giulio / Testa, Emilio et al. | 1969
- 839
-
Stereochemical studies on medicinal agents. VII. Absolute stereochemistry of methadol isomers and the role of the 6-methyl group in analgetic activityPortoghese, Philip S. / Williams, David Allen et al. | 1969
- 845
-
1,2,3,4,5,6-Hexahydro-6-phenyl-2,6-methano-3-benzazocines. I. 3-Carboxamido-8-hydroxy derivative as an orally effective analgeticBlock, Fred B. / Clarke, Frank Henderson et al. | 1969
- 848
-
3-Acetoxyquinuclidine methiodide. Resolution, absolute configuration, and stereospecificity of interaction with the acetylcholine binding sitesRobinson, John Barry / Belleau, Bernard / Cox, Barry et al. | 1969
- 851
-
2-(N,N-dialkylamino)ethyl esters of .alpha.-(3-pyridyl)mandelic acids. Synthesis and pharmacological evaluationNovelli, Armando / Barrio, Jorge R. / Huidobro, H. et al. | 1969
- 854
-
Malonamic esters. New class of sedative-tranquilizersLoev, Bernard / Macko, Edward / Fried, Irving M. et al. | 1969
- 860
-
Synthesis and central nervous system depressant activity of new piperazine derivatives and related compounds. IIVadodaria, D. J. / Deliwala, Chimanlal V. / Mandrekar, S. S. / Sheth, U. K. et al. | 1969
- 865
-
Synthesis and central nervous system depressant activity of new piperazine and related derivatives. IIIPetigara, R. B. / Deliwala, Chimanlal / Mandrekar, S. S. / Dadkar, N. K. / Sheth, U. K. et al. | 1969
- 870
-
Synthesis and pharmacological activity of alkylaminoalkyl esters and amides of 2-hydroxy- (or alkoxy-) 3-methoxybenzoic acidTsatsas, Georges / Costakis, E. / Zaroslinski, John F. / Browne, Ronald K. / Possley, Leroy H. et al. | 1969
- 873
-
Synthesis and antialdosterone activity of substituted 2,3,3-triphenylpropylaminesBlank, Benjamin / Zuccarello, William A. / Cohen, Suzanne R. / Frishmuth, Gertrude J. / Scaricaciottoli, Daniel et al. | 1969
- 876
-
Psychosedative agents. N-(4-phenyl-1-piperazinylalkyl)-substituted cyclic imidesWu, Yao-Hua / Smith, Kenneth R. / Rayburn, James W. / Kissel, John W. et al. | 1969
- 881
-
Mammalian antifertility agents. VI. A novel sequence for the preparation of 1,2-disubstituted 3,4-dihydronaphthalenesLednicer, Daniel / Emmert, D. Edward / Lyster, Stanley C. / Duncan, Gordon W. et al. | 1969
- 885
-
3-Deoxy-16-haloestra-1,3,5(10)-trienesJohns, William F. et al. | 1969
- 888
-
Biologically oriented organic sulfur chemistry. III. Formation of mercaptals, mercaptoles, an orthothioformate, and thiazolidines for the latentiation of thiolsSweetman, B. J. / Bellas, Michael / Field, Lamar et al. | 1969
- 891
-
Quaternary thiazolylpyridinium salts. Oral hypoglycemic agentsWiegand, Gretchen E. / Bauer, Victor J. / Safir, Sidney R. / Blickens, D. A. / Riggi, S. J. et al. | 1969
- 894
-
Irreversible enzyme inhibitors. CLIX. Effect of substitution on transport and isozyme specificity of p-(4,6-diamino-1,2-dihydro-2,2-dimethyl-s-triazin-1-yl)-o-chlorophenoxyacetamido-benzenesulfonyl fluoride, an active-site-directed irreversible inhibitor of dihydrofolic reductaseBaker, Bernard Randall / Ashton, Wallace T. et al. | 1969
- 898
-
Irreversible enzyme inhibitors. CLX. Some factors in cell wall transport of active-site-directed irreversible inhibitors of dihydrofolic reductase derived from 4,6-diamino-1,2-dihydro-2,2-dimethyl-1-(phenylalkylphenyl)-s-triazinesBaker, Bernard Randall / Janson, Eunice E. / Vermeulen, Nicolaas M. J. et al. | 1969
- 902
-
Irreversible enzyme inhibitors. CLXI. Proteolytic enzymes. 13. Inhibitors of guinea pig complement derived by quaternization of 3-acylamidopyridines with .alpha.-bromomethylbenzenesulfonyl fluoridesBaker, Bernard Randall / Hurlbut, Jeffrey A. et al. | 1969
- 906
-
Monoquaternary muscle paralyzing agents. III. Synthesis of N-(.omega.-phthalimidoalkyl)trialkylammonium iodidesDonahoe, Hugh B. / Seiwald, Robert J. / Sister Mary Marguerite Neumann / Heitmeier, Donald E. / Kimura, Kazuo K. et al. | 1969
- 907
-
Some organoboron compounds containing a bis(2-chloroethyl)amino group joined to boronShealy, Y. Fulmer / Struck, Robert F. et al. | 1969
- 911
-
Compounds related to insect juvenile hormone. IVWakabayashi, Nobel / Sonnet, Philip E. / Law, M. W. et al. | 1969
- 913
-
Synthesis of some substituted 5H-dibenz[b,f]azepines as potential antimalarialsVarma, Rajendra S. / Whisenant, L. K. / Boykin, David W. et al. | 1969
- 914
-
1,3-Dihydro-1-methyl-5,6- (and 5,7-) diaryl-2H-1,4-diazepin-2-onesHofmann, Corris Mabelle / Safir, Sidney R. et al. | 1969
- 917
-
Steric structure-activity relationship studies on a new butyrophenone derivativeLi, J. Pengman / Biel, John H. et al. | 1969
- 919
-
Synthesis of compounds with potential central nervous system stimulant activity. I. 2-Amino-2-oxazolin-4-one-5-spirocycloalkanes and 2-amino-2-oxazolin-4-one-5-spiro(4'-piperidines)Harnden, Michael R. / Rasmussen, Ray R. et al. | 1969
- 921
-
N-aminonormorphineModiri, Ali / Cannon, Joseph G. / Yeh, S. Y. et al. | 1969
- 922
-
Receptor binding of the analgetic aryl moiety. I. .alpha.-Prodine analogsSabih, Khalid / Wiley, Robert A. et al. | 1969
- 923
-
Biochemorphology of cyclobutanecarboximidesZirvi, Karimullah A. / Jarboe, Charles H. et al. | 1969
- 925
-
Isolation and identification of cephalexin from human urineChou, Ta-Sen et al. | 1969
- 926
-
Diamides of cyclobutane-1,1-dicarboxylic acidZirvi, Karimullah A. / Jarboe, Charles H. et al. | 1969
- 927
-
Substituted chromones as coronary vasodilatorsBariana, Dilbagh S. et al. | 1969
- 928
-
N-[3-(1-alkylpiperidyl)]acetamides and N,N-dimethyl-N'-[3-(1-alkyl-piperidyl)]ureas as cholinesterase inhibitors. IMathison, Ian W. / Beasley, James G. / Fowler, Kathleen C. / Peters, Elizabeth R. et al. | 1969
- 931
-
The cholinergic receptor. IV. Synthesis and muscarinic activity of 3,7-dimethyl-2,4-dioxa-7-azaspiro[3,4]octane methiodideRidley, Horace F. / Chatterjee, Shym S. / Moran, John F. / Triggle, David J. et al. | 1969
- 933
-
Derivatives of 2-azabicyclo[2.2.2]octane. III. Substituted phenylsulfonylureido derivativesVillani, Frank J. / Wefer, Elizabeth A. / Mann, Thomas A. / Ellis, Claire A. et al. | 1969
- 935
-
Angiotensin II analogs. II. Cyclo-(-Val-Tyr-Ile-His-Pro-Phe-)Jorgensen, Eugene C. / Patton, Walter et al. | 1969
- 936
-
Hypotensive, antiadrenergic, and antihistaminic 3-substituted 2-methyl-(or 2-phenyl-) 4(3H)-quinazolonesHayao, Shin / Havera, H. J. / Strycker, W. G. / Hong, Enrique et al. | 1969
- 938
-
meta-Substituted benzenesulfonylureas as hypoglycemic agentsShah, Madhusudan H. / Darnule, T. V. / Ananthanarayanan, Kodaganallur G. / Deliwala, Chimanlal V. et al. | 1969
- 940
-
.beta.-Aminopropionohydroxamic acids and .beta.-aminopropionic esters with hypotensive propertiesCoutts, Ronald T. / Midha, Kamal K. / Prasad, K. et al. | 1969
- 941
-
Hypoglycemic esters of 2-chloroethanolSiggins, James E. / Harding, Homer R. / Potts, Gordon O. et al. | 1969
- 943
-
Quaternary oxazolylpyridinium salts. Oral hypoglycemic agentsWiegand, Gretchen E. / Bauer, Victor J. / Safir, Sidney R. / Blickens, D. A. / Riggi, S. J. et al. | 1969
- 944
-
Hypoglycemic quaternary azolylpyridinium salts. Inactive analogsBauer, Victor J. / Wiegand, Gretchen E. / Fanshawe, William J. / Safir, Sidney R. et al. | 1969
- 945
-
4-Azolylpyridine 1-oxides. Analogs of the hypoglycemic 4-azolylpyridinium saltsBauer, Victor J. / Fanshawe, William J. / Wiegand, Gretchen E. / Safir, Sidney R. et al. | 1969
- 946
-
5,5-Diarylpenta-2,4-dienoic acid amides as potential antimalarial agents. IILange, Judy Hayford / Colwell, William T. / Henry, David W. et al. | 1969
- 948
-
Synthesis and antiinflammatory activity of 5-substituted 2,3-bis(p-methoxyphenyl)indolesYoungdale, Gilbert A. / Glenn, E. Myles / Lednicer, Daniel / Szmuszkovicz, Jacob et al. | 1969
- 949
-
Antimalarials. Chloroquine analogs with the 1,2,3,6-tetrahydropyridyl function in the side chainSingh, Tara / Stein, Robert G. / Biel, John H. et al. | 1969
- 950
-
N-Acyl- and N-sulfonylcysteine derivativesMartin, Tellis A. et al. | 1969
- 953
-
Amides of N-acylcysteines as potential amino acid antagonists in bacteriaZygmunt, Walter A. / Martin, Tellis A. et al. | 1969
- 955
-
Synthetic amebicides. X. Antiamebic, antimalarial, and anthelmintic effects of distal hydrazine analogs of azacrine, quinacrine, and 7-{ [3-(octylamino)propyl]amino}benz[c]acridineElslager, Edward F. / Worth, Donald F. et al. | 1969
- 957
-
Trifluoromethylbenzanilides as anticoccidial agentsWelch, Dean E. / Baron, Robert R. et al. | 1969
- 959
-
Synthesis of 3,5-dihydroxy-4-methoxy-.alpha.-methylphenethanolamine and analogsLee, Fred G. H. / Dickson, Donald E. / Benigni, Joseph D. / Minnis, R. L. / Gannon, Walter F. / Manian, Albert A. et al. | 1969
- 961
-
Stable oxaziridinesChakravarty, Jyotirmoy / Truitt, Price et al. | 1969
- 961
-
Oxidation of fluorenamines and preparation of 2,2'-and 4,4'-azofluoreneYost, Yul et al. | 1969
- 962
-
Possible anticonvulsant thiazolo[3,2-a]benzimidazole Mannich bases. XISingh, Jag Megh et al. | 1969
- 963
-
Progress in Biochemical Pharmacology. Volume 4. Recent Advances in AtherosclerosisBach, Frederick et al. | 1969
- 963
-
Annual Review of Pharmacology. Volume 9Burger, Alfred et al. | 1969
- 963
-
Psychopharmacology. A Review of Progress, 1957-1967Burger, Alfred et al. | 1969
- 963
-
Biogenesis and Action of Steroid HormonesAxelrod, Leonard et al. | 1969
- 964
-
Principles of Radiological HealthBurger, Alfred et al. | 1969