In vitro evolution of an HIV integrase binding protein from a library of C-terminal domain γS-crystallin variants (English)
- New search for: Moody, Issa S.
- New search for: Verde, Shawn C.
- New search for: Overstreet, Cathie M.
- New search for: Edward Robinson, W. Jr.
- New search for: Weiss, Gregory A.
- New search for: Moody, Issa S.
- New search for: Verde, Shawn C.
- New search for: Overstreet, Cathie M.
- New search for: Edward Robinson, W. Jr.
- New search for: Weiss, Gregory A.
In:
Bioorganic and Medicinal Chemistry Letters
;
22
, 17
;
5584-5589
;
2012
-
ISSN:
- Article (Journal) / Electronic Resource
-
Title:In vitro evolution of an HIV integrase binding protein from a library of C-terminal domain γS-crystallin variants
-
Contributors:Moody, Issa S. ( author ) / Verde, Shawn C. ( author ) / Overstreet, Cathie M. ( author ) / Edward Robinson, W. Jr. ( author ) / Weiss, Gregory A. ( author )
-
Published in:Bioorganic and Medicinal Chemistry Letters ; 22, 17 ; 5584-5589
-
Publisher:
- New search for: Elsevier Ltd
-
Publication date:2012-07-03
-
Size:6 pages
-
ISSN:
-
DOI:
-
Type of media:Article (Journal)
-
Type of material:Electronic Resource
-
Language:English
-
Keywords:
-
Source:
Table of contents – Volume 22, Issue 17
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 5331
-
Graphical contents list| 2012
- 5352
-
Modulation of DNA repair by pharmacological inhibitors of the PIKK protein kinase familyFinlay, M. Raymond V. / Griffin, Roger J. et al. | 2012
- 5360
-
Set-up of a new series of HDAC inhibitors: the 5,11-dihydrodibenzo[b,e]azepin-6-ones as privileged structuresBigioni, Mario / Ettorre, Alessandro / Felicetti, Patrizia / Mauro, Sandro / Rossi, Cristina / Maggi, Carlo Alberto / Marastoni, Elena / Binaschi, Monica / Parlani, Massimo / Fattori, Daniela et al. | 2012
- 5363
-
Design, synthesis and evaluation of clinafloxacin triazole hybrids as a new type of antibacterial and antifungal agentsWang, Yan / Damu, Guri L.V. / Lv, Jing-Song / Geng, Rong-Xia / Yang, Da-Cheng / Zhou, Cheng-He et al. | 2012
- 5367
-
DBD dyes as fluorescent probes for sensing lipophilic environmentsWawrzinek, Robert / Wessig, Pablo / Möllnitz, Kristian / Nikolaus, Jörg / Schwarzer, Roland / Müller, Peter / Herrmann, Andreas et al. | 2012
- 5372
-
Design, synthesis, and structure–activity relationships of a series of 2-Ar-8-methyl-5-alkylaminoquinolines as novel CRF1 receptor antagonistsTakeda, Kunitoshi / Terauchi, Taro / Hashizume, Minako / Shin, Kogyoku / Ino, Mitsuhiro / Shibata, Hisashi / Yonaga, Masahiro et al. | 2012
- 5379
-
Fluorescence sensing of caffeine in aqueous solution with carbazole-based probe and imaging application in live cellsMahapatra, Ajit Kumar / Roy, Jagannath / Sahoo, Prithidipa / Mukhopadhyay, Subhra Kanti / Mukhopadhyay, Anindita Roy / Mandal, Debasish et al. | 2012
- 5384
-
Regioselective synthesis of fraxinellone-based hydrazone derivatives as insecticidal agentsGuo, Yong / Yan, Yuan-Yuan / Yang, Chun / Yu, Xiang / Zhi, Xiao-Yan / Xu, Hui et al. | 2012
- 5388
-
Urea/thiourea catalyzed, solvent-free synthesis of 5-arylidenethiazolidine-2,4-diones and 5-arylidene-2-thioxothiazolidin-4-onesShah, Sakshi / Singh, Baldev et al. | 2012
- 5392
-
2-Phenylamino-6-cyano-1H-benzimidazole-based isoform selective casein kinase 1 gamma (CK1γ) inhibitorsHua, Zihao / Huang, Xin / Bregman, Howard / Chakka, Nagasree / DiMauro, Erin F. / Doherty, Elizabeth M. / Goldstein, Jon / Gunaydin, Hakan / Huang, Hongbing / Mercede, Stephanie et al. | 2012
- 5392
-
2-Phenylamino-6-cyano-1H-benzimidazole-based isoform selective casein kinase 1 gamma (CK1g) inhibitorsHua, Z. / Huang, X. / Bregman, H. / Chakka, N. / DiMauro, E. F. / Doherty, E. M. / Goldstein, J. / Gunaydin, H. / Huang, H. / Mercede, S. et al. | 2012
- 5396
-
Discovery of XL888: A novel tropane-derived small molecule inhibitor of HSP90Bussenius, Joerg / Blazey, Charles M. / Aay, Naing / Anand, Neel K. / Arcalas, Arlyn / Baik, TaeGon / Bowles, Owen J. / Buhr, Chris A. / Costanzo, Simona / Curtis, Jeffrey K. et al. | 2012
- 5405
-
Near-infrared fluorescent divalent RGD ligand for integrin αvβ3-targeted optical imagingYe, Yunpeng / Akers, Walter / Xu, Baogang / Bloch, Sharon / Odonkor, Charles / Achilefu, Samuel et al. | 2012
- 5405
-
Near-infrared fluorescent divalent RGD ligand for integrin avb3-targeted optical imagingYe, Y. / Akers, W. / Xu, B. / Bloch, S. / Odonkor, C. / Achilefu, S. et al. | 2012
- 5410
-
Combined receptor-based and ligand-based approach to delineate the mode of binding of guaianolide–endoperoxides to PfATP6Helal, Mohamed A. / Avery, Mitchell A. et al. | 2012
- 5415
-
Homodimeric SV40 NLS peptide formed by disulfide bond as enhancer for gene deliveryKim, Bieong-Kil / Kang, Hyungu / Doh, Kyung-Oh / Lee, Seong-Hye / Park, Jong-Won / Lee, Su-Jin / Lee, Tae-Jin et al. | 2012
- 5419
-
Highly potent aminopyridines as Syk kinase inhibitorsCastillo, Marcos / Forns, Pilar / Erra, Montse / Mir, Marta / López, Manel / Maldonado, Mónica / Orellana, Adelina / Carreño, Cristina / Ramis, Isabel / Miralpeix, Montserrat et al. | 2012
- 5424
-
Synthesis and biological evaluation of novel triazoles and isoxazoles linked 2-phenyl benzothiazole as potential anticancer agentsKumbhare, Ravindra M. / Kosurkar, Umesh B. / Janaki Ramaiah, M. / Dadmal, Tulshiram L. / Pushpavalli, S.N.C.V.L. / Pal-Bhadra, Manika et al. | 2012
- 5428
-
Combining pharmacophore, docking and substructure search approaches to identify and optimize novel B-RafV600E inhibitorsXu, Zhijian / Yan, Guirui / Wang, Gaihong / Li, Bo / Zhu, Jianming / Sun, Peng / Zhang, Xiaodong / Luo, Cheng / Wang, Heyao / Zhu, Weiliang et al. | 2012
- 5438
-
Benzimidazole bearing oxadiazole and triazolo-thiadiazoles nucleus: Design and synthesis as anticancer agentsHusain, Asif / Rashid, Mohd / Mishra, Ravinesh / Parveen, Shama / Shin, Dong-Soo / Kumar, Deepak et al. | 2012
- 5445
-
Development of isoform selective PI3-kinase inhibitors as pharmacological tools for elucidating the PI3K pathwayBruce, Ian / Akhlaq, Mohammed / Bloomfield, Graham C. / Budd, Emma / Cox, Brian / Cuenoud, Bernard / Finan, Peter / Gedeck, Peter / Hatto, Julia / Hayler, Judy F. et al. | 2012
- 5451
-
Synthesis and anti-HIV activities of symmetrical dicarboxylate esters of dinucleoside reverse transcriptase inhibitorsAgarwal, Hitesh K. / Buckheit, Karen W. / Buckheit, Robert W. Jr. / Parang, Keykavous et al. | 2012
- 5455
-
Synthesis and in vitro evaluation of new chloroquine-chalcone hybrids against chloroquine-resistant strain of Plasmodium falciparumSashidhara, Koneni V. / Avula, Srinivasa Rao / Palnati, Gopala Reddy / Singh, Shiv Vardan / Srivastava, Kumkum / Puri, Sunil K. / Saxena, J.K. et al. | 2012
- 5460
-
Structure-based design, synthesis, and biological evaluation of dihydroquinazoline-derived potent b-secretase inhibitorsGhosh, A. K. / Pandey, S. / Gangarajula, S. / Kulkarni, S. / Xu, X. / Rao, K. V. / Huang, X. / Tang, J. et al. | 2012
- 5460
-
Structure-based design, synthesis, and biological evaluation of dihydroquinazoline-derived potent β-secretase inhibitorsGhosh, Arun K. / Pandey, Satyendra / Gangarajula, Sudhakar / Kulkarni, Sarang / Xu, Xiaoming / Rao, Kalapala Venkateswara / Huang, Xiangping / Tang, Jordan et al. | 2012
- 5466
-
2-Amino-1,3,4-thiadiazole derivative (FABT) inhibits the extracellular signal-regulated kinase pathway and induces cell cycle arrest in human non-small lung carcinoma cellsJuszczak, M. / Matysiak, J. / Szeliga, M. / Pożarowski, P. / Niewiadomy, A. / Albrecht, J. / Rzeski, W. et al. | 2012
- 5470
-
Anti-androgen receptor activity of apoptotic CK2 inhibitor CX4945 in human prostate cancer LNCap cellsRyu, Byung Jun / Baek, Seung-hwa / Kim, Jiyeon / Bae, Su Jung / Chang, Sung-Youn / Heo, Jung-Nyoung / Lee, Hyuk / Lee, Sang Yeol / Kim, Seong Hwan et al. | 2012
- 5475
-
Important role of Maillard reaction in the protective effect of heat-processed ginsenoside Re-serine mixture against cisplatin-induced nephrotoxicity in LLC-PK1 cellsLee, Ji Hwan / Lee, Woojung / Lee, Seungyong / Jung, Yujung / Park, Soon-Hye / Choi, Pilju / Kim, Su-Nam / Ham, Jungyeob / Kang, Ki Sung et al. | 2012
- 5480
-
Selected chromone derivatives as inhibitors of monoamine oxidaseLegoabe, Lesetja J. / Petzer, Anél / Petzer, Jacobus P. et al. | 2012
- 5485
-
N-1-Alkyl-2-oxo-2-aryl amides as novel antagonists of the TRPA1 receptorVallin, Karl S.A. / Sterky, Karin J. / Nyman, Eva / Bernström, Jenny / From, Rebecka / Linde, Christian / Minidis, Alexander B.E. / Nolting, Andreas / Närhi, Katja / Santangelo, Ellen M. et al. | 2012
- 5493
-
Exploration of ring size in a series of cyclic vicinal diamines with σ 1 receptor affinityMoussa, Iman A. / Banister, Samuel D. / Manoli, Miral / Doddareddy, Munikumar Reddy / Cui, Jinquan / Mach, Robert H. / Kassiou, Michael et al. | 2012
- 5498
-
Design, synthesis and identification of novel benzimidazole derivatives as highly potent NPY Y5 receptor antagonists with attractive in vitro ADME profilesTamura, Yuusuke / Omori, Naoki / Kouyama, Naoki / Nishiura, Yuji / Hayashi, Kyouhei / Watanabe, Kana / Tanaka, Yukari / Chiba, Takeshi / Yukioka, Hideo / Sato, Hiroki et al. | 2012
- 5503
-
Small molecule modulators of aggregation in synthetic melanin polymerizationsBelitsky, Jason M. / Ellowitz, Micah Z. / Lye, Diane / Kilbo, Alexander L. et al. | 2012
- 5508
-
Identification of selective tubulin inhibitors as potential anti-trypanosomal agentsLama, Rati / Sandhu, Ranjodh / Zhong, Bo / Li, Bibo / Su, Bin et al. | 2012
- 5517
-
Synthesis and characterization of avb3-targeting peptidomimetic chelate conjugates for PET and SPECT imagingKim, Y. S. / Nwe, K. / Milenic, D. E. / Brechbiel, M. W. / Satz, S. / Baidoo, K. E. et al. | 2012
- 5517
-
Synthesis and characterization of αvβ3-targeting peptidomimetic chelate conjugates for PET and SPECT imagingKim, Young-Seung / Nwe, Kido / Milenic, Diane E. / Brechbiel, Martin W. / Satz, Stanley / Baidoo, Kwamena E. et al. | 2012
- 5523
-
Design, synthesis and molecular simulation studies of dihydrostilbene derivatives as potent tyrosinase inhibitorsVontzalidou, Argyro / Zoidis, Grigoris / Chaita, Eliza / Makropoulou, Maria / Aligiannis, Nektarios / Lambrinidis, George / Mikros, Emmanuel / Skaltsounis, Alexios-Leandros et al. | 2012
- 5527
-
Synthesis and characterization of quinoline-based thiosemicarbazones and correlation of cellular iron-binding efficacy to anti-tumor efficacySerda, Maciej / Kalinowski, Danuta S. / Mrozek-Wilczkiewicz, Anna / Musiol, Robert / Szurko, Agnieszka / Ratuszna, Alicja / Pantarat, Namfon / Kovacevic, Zaklina / Merlot, Angelica M. / Richardson, Des R. et al. | 2012
- 5532
-
A fluorescent reporter of ATP binding-competent receptor kinasesSicard, Renaud / Dhuguru, Jyothi / Liu, Wenjun / Patel, Nirav / Landgraf, Ralf / Wilson, James N. et al. | 2012
- 5536
-
4-Substituted boro-proline dipeptides: Synthesis, characterization, and dipeptidyl peptidase IV, 8, and 9 activitiesWu, Wengen / Liu, Yuxin / Milo, Lawrence J. Jr. / Shu, Ying / Zhao, Peng / Li, Youhua / Woznica, Iwona / Yu, Gengli / Sanford, David G. / Zhou, Yuhong et al. | 2012
- 5541
-
Fluorogenic assay of alkaline phosphatase activity based on the modulation of excited-state intramolecular proton transferPark, Jihye / Helal, Aasif / Kim, Hong-Seok / Kim, Youngmi et al. | 2012
- 5545
-
Dipeptidyl peptidase-4 inhibitor with b-amino amide scaffold: Synthesis, SAR and biological evaluationKim, H. J. / Kwak, W. Y. / Min, J. P. / Sung, S. Y. / Kim, H. D. / Kim, M. K. / Kim, H. S. / Park, K. J. / Son, M. H. / Kim, S. H. et al. | 2012
- 5545
-
Dipeptidyl peptidase-4 inhibitor with β-amino amide scaffold: Synthesis, SAR and biological evaluationKim, Heung Jae / Kwak, Woo Young / Min, Jong Pil / Sung, Si Young / Kim, Ha Dong / Kim, Mi Kyung / Kim, Hae Sun / Park, Kyung Jin / Son, Moon Ho / Kim, Soon Hoe et al. | 2012
- 5550
-
Hybrid molecules of carvacrol and benzoyl urea/thiourea with potential applications in agriculture and medicinePete, Umesh D. / Zade, Chetan M. / Bhosale, Jitendra D. / Tupe, Santosh G. / Chaudhary, Preeti M. / Dikundwar, Amol G. / Bendre, Ratnamala S. et al. | 2012
- 5555
-
Two novel bioactive glucosinolates from Broccoli (Brassica oleracea L. var. italica) floretsSurvay, Nazneen Shaik et al. | 2012
- 5559
-
Anti-inflammatory sesquiterpene lactones from the flower of Vernonia cinereaYoun, Ui Joung / Park, Eun-Jung / Kondratyuk, Tamara P. / Simmons, Charles J. / Borris, Robert P. / Tanamatayarat, Patcharawan / Wongwiwatthananukit, Supakit / Toyama, Onoomar / Songsak, Thanapat / Pezzuto, John M. et al. | 2012
- 5563
-
Isosteric replacements for benzothiazoles and optimisation to potent Cathepsin K inhibitors free from hERG channel inhibitionDossetter, Alexander G. / Bowyer, Jonathan / Cook, Calum R. / Crawford, James J. / Finlayson, Jonathan E. / Heron, Nicola M. / Heyes, Christine / Highton, Adrian J. / Hudson, Julian A. / Jestel, Anja et al. | 2012
- 5569
-
Antitrypanosomal and antioxidant properties of 4-hydroxycoumarins derivativesPérez-Cruz, Fernanda / Serra, Silvia / Delogu, Giovanna / Lapier, Michel / Maya, Juan Diego / Olea-Azar, Claudio / Santana, Lourdes / Uriarte, Eugenio et al. | 2012
- 5574
-
The development of first Staphylococcus aureus SplB protease inhibitors: Phosphonic analogues of glutamineEwa, Burchacka / Maciej, Walczak / Marcin, Sieńczyk / Grzegorz, Dubin / Michał, Zdżalik / Jan, Potempa / Józef, Oleksyszyn et al. | 2012
- 5579
-
A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model: From in silico screening to cyclodextrin formulationRadi, Marco / Evensen, Lasse / Dreassi, Elena / Zamperini, Claudio / Caporicci, Marialessandra / Falchi, Federico / Musumeci, Francesca / Schenone, Silvia / Lorens, James B. / Botta, Maurizio et al. | 2012
- 5584
-
In vitro evolution of an HIV integrase binding protein from a library of C-terminal domain gS-crystallin variantsMoody, I. S. / Verde, S. C. / Overstreet, C. M. / Edward Robinson, W. / Weiss, G. A. et al. | 2012
- 5584
-
In vitro evolution of an HIV integrase binding protein from a library of C-terminal domain γS-crystallin variantsMoody, Issa S. / Verde, Shawn C. / Overstreet, Cathie M. / Edward Robinson, W. Jr. / Weiss, Gregory A. et al. | 2012
- 5590
-
Evaluation of siRNAs that contain internal variable-length spacer linkagesEfthymiou, Tim C. / Peel, Brandon / Huynh, Vanthi / Desaulniers, Jean-Paul et al. | 2012
- 5595
-
Novel 2-methoxyacylhydrazones as potent, selective PDE10A inhibitors with activity in animal models of schizophreniaCutshall, Neil S. / Onrust, Rene / Rohde, Alex / Gragerov, Sasha / Hamilton, Lauren / Harbol, Kevin / Shen, Hui-Rong / McKee, Shawn / Zuta, Charles / Gragerova, Galina et al. | 2012
- 5600
-
Design of inhibitors of Helicobacter pylori glutamate racemase as selective antibacterial agents: Incorporation of imidazoles onto a core pyrazolopyrimidinedione scaffold to improve bioavailabiltyBasarab, Gregory S. / Hill, Pamela / Eyermann, Charles J. / Gowravaram, Madhu / Käck, Helena / Osimoni, Ekundayo et al. | 2012
- 5608
-
ortho Substituent effects on the anticonvulsant properties of 4-hydroxy-trifluoroethyl phenolsMishra, Rajesh K. / Baker, Max T. et al. | 2012
- 5612
-
High-affinity and selective dopamine D3 receptor full agonistsChen, Jianyong / Levant, Beth / Wang, Shaomeng et al. | 2012
- 5618
-
Structure and activity relationship in the (S)-N-chroman-3-ylcarboxamide series of voltage-gated sodium channel blockersKers, Inger / Csjernyik, Gabor / Macsari, Istvan / Nylöf, Martin / Sandberg, Lars / Skogholm, Karin / Bueters, Tjerk / Eriksson, Anders B. / Oerther, Sandra / Lund, Per-Eric et al. | 2012
- 5625
-
GSK2578215A; A potent and highly selective 2-arylmethyloxy-5-substitutent-N-arylbenzamide LRRK2 kinase inhibitorReith, Alastair D. / Bamborough, Paul / Jandu, Karamjit / Andreotti, Daniele / Mensah, Lucy / Dossang, Pamela / Choi, Hwan Geun / Deng, Xianming / Zhang, Jinwei / Alessi, Dario R. et al. | 2012
- 5630
-
Anion inhibition studies of an α-carbonic anhydrase from the thermophilic bacterium Sulfurihydrogenibium yellowstonense YO3AOP1De Luca, Viviana / Vullo, Daniela / Scozzafava, Andrea / Carginale, Vincenzo / Rossi, Mosè / Supuran, Claudiu T. / Capasso, Clemente et al. | 2012
- 5630
-
Anion inhibition studies of an a-carbonic anhydrase from the thermophilic bacterium Sulfurihydrogenibium yellowstonense YO3AOP1De Luca, V. / Vullo, D. / Scozzafava, A. / Carginale, V. / Rossi, M. / Supuran, C. T. / Capasso, C. et al. | 2012
- 5635
-
Diaminopropionic acid lipopeptides: Characterization studies of polyplexes aimed at pDNA deliveryViola, Joana R. / Strömberg, Roger / Simonson, Oscar E. / Andaloussi, Samir EL / Edvard Smith, C.I. / Murtola, Merita et al. | 2012
- 5639
-
Pd-mediated functionalization of polysubstituted pyrroles: Their evaluation as potential inhibitors of PDE4Bhaskar Kumar, T. / Sumanth, Ch. / Vaishaly, S. / Srinivasa Rao, M. / Chandra Sekhar, K.B. / Meda, Chandana Lakshmi T. / Kandale, Ajit / Rambabu, D. / Rama Krishna, G. / Malla Reddy, C. et al. | 2012
- 5648
-
Glucose uptake stimulatory effect of 4-hydroxypipecolic acid by increased GLUT 4 translocation in skeletal muscle cellsNaresh, G. / Jaiswal, N. / Sukanya, P. / Srivastava, A.K. / Tamrakar, A.K. / Narender, T. et al. | 2012
- 5652
-
Synthesis and SAR of pyridothiazole substituted pyrimidine derived HCV replication inhibitorsGirijavallabhan, Vinay M. / Alvarez, Carmen / Bennett, Frank / Chen, Lei / Gavalas, Stephen / Huang, Yuhua / Kim, Seong-Heon / Kosinski, Aneta / Pinto, Patrick / Rizvi, Razia et al. | 2012
- 5658
-
N-Aryl pyrrolidinonyl oxadiazoles as potent mGluR5 positive allosteric modulatorsPackiarajan, Mathivanan / Mazza Ferreira, Christine G. / Hong, Sang-Phyo / White, Andrew D. / Chandrasena, Gamini / Pu, Xiaosui / Brodbeck, Robbin M. / Robichaud, Albert J. et al. | 2012
- 5663
-
Design and synthesis of photolabile caged cytokininHayashi, Ken-ichiro / Kusaka, Naoyuki / Ando, Kazuki / Mitsui, Taichi / Aoyama, Takashi / Nozaki, Hiroshi et al. | 2012
- 5668
-
Discovery of potent and selective rhodanine type IKKβ inhibitors by hit-to-lead strategySong, Hyeseung / Lee, Yun Suk / Roh, Eun Joo / Seo, Jae Hong / Oh, Kwang-Seok / Lee, Byung Ho / Han, Hogyu / Shin, Kye Jung et al. | 2012
- 5668
-
Discovery of potent and selective rhodanine type IKKb inhibitors by hit-to-lead strategySong, H. / Lee, Y. S. / Roh, E. J. / Seo, J. H. / Oh, K. S. / Lee, B. H. / Han, H. / Shin, K. J. et al. | 2012
- 5675
-
Identification of a novel serum and glucocorticoid regulated kinase-1 (SGK1) ligand from virtual screeningGeldenhuys, Werner J. / Talasila, Phani K. / Sadana, Prabodh et al. | 2012
- 5679
-
Structural requirements for the antitubercular quaternized triflupromazine pharmacophoreKunciw, Dominique L. / Liechty, Jacob J. / Mitchell, Miguel O. / Wan, Baojie / Franzblau, Scott G. et al. | 2012
- 5681
-
Orally available pyridinylpyrimidine derivatives as novel RANKL-induced osteoclastogenesis inhibitorsMiyata, Junji / Kasahara, Chiyoshi / Asano, Toru / Ito, Shinji / Seki, Norio / Kato, Yasuko / Morikawa, Noriyuki / Nozaki, Kazuyoshi / Nishimura, Kouji / Akamatsu, Hisashi et al. | 2012
- 5685
-
Optimization of tricyclic Nec-3 necroptosis inhibitors for in vitro liver microsomal stabilityChoi, Sungwoon / Keys, Heather / Staples, Richard J. / Yuan, Junying / Degterev, Alexei / Cuny, Gregory D. et al. | 2012
- 5689
-
A Co(III) complex cleaving soluble oligomers of h-IAPP in the presence of polymeric aggregates of h-IAPPLee, Tae Yeon / Chei, Woo Suk / Ju, Heeyeon / Lee, Mi-Sook / Lee, Jung Weon / Suh, Junghun et al. | 2012
- 5694
-
Metronidazole thiosalicylate conjugates: Synthesis, crystal structure, docking studies and antiamoebic activitySalahuddin, Attar / Agarwal, Subhash M. / Avecilla, Fernando / Azam, Amir et al. | 2012
- 5700
-
Synthesis and biological evaluation of novel oxindole derivatives for imaging neurofibrillary tangles in Alzheimer’s diseaseWatanabe, Hiroyuki / Ono, Masahiro / Kimura, Hiroyuki / Matsumura, Kenji / Yoshimura, Masashi / Okamoto, Yoko / Ihara, Masafumi / Takahashi, Ryosuke / Saji, Hideo et al. | 2012
- 5704
-
Synthesis of N-(1-methyl-1H-indol-3-yl)methyleneamines and 3,3-diaryl-4-(1-methyl-1H-indol-3-yl)azetidin-2-ones as potential antileishmanial agentsSingh, Girija S. / Al-kahraman, Yasser M.S.A. / Mpadi, Disah / Yasinzai, Masoom et al. | 2012
- 5707
-
Design and synthesis of Pictet–Spengler condensation products that exhibit oncogenic-RAS synthetic lethality and induce non-apoptotic cell deathSkouta, Rachid / Hayano, Miki / Shimada, Kenichi / Stockwell, Brent R. et al. | 2012
- 5714
-
Synthesis and structure–activity relationships of dual PI3K/mTOR inhibitors based on a 4-amino-6-methyl-1,3,5-triazine sulfonamide scaffoldWurz, Ryan P. / Liu, Longbin / Yang, Kevin / Nishimura, Nobuko / Bo, Yunxin / Pettus, Liping H. / Caenepeel, Sean / Freeman, Daniel J. / McCarter, John D. / Mullady, Erin L. et al. | 2012
- 5721
-
Discovery of triazolopyrimidine-based PDE8B inhibitors: Exceptionally ligand-efficient and lipophilic ligand-efficient compounds for the treatment of diabetesDeNinno, Michael P. / Wright, Stephen W. / Etienne, John B. / Olson, Thanh V. / Rocke, Benjamin N. / Corbett, Jeffrey W. / Kung, Daniel W. / DiRico, Kenneth J. / Andrews, Kim M. / Millham, Michele L. et al. | 2012
- 5727
-
Green synthesis and anti-infective activities of fluorinated pyrazoline derivativesShelke, Sharad N. / Mhaske, Ganesh R. / Bonifácio, Vasco D.B. / Gawande, Manoj B. et al. | 2012
- 5731
-
Design, synthesis and biological evaluation of simplified side chains of the macrolide antibiotic etnangienAltendorfer, Mario / Irschik, Herbert / Menche, Dirk et al. | 2012
- 5735
-
Synthesis of 3-(1-alkyl/aminoalkyl-3-vinyl-piperidin-4-yl)-1-(quinolin-4-yl)-propan-1-ones and their 2-methylene derivatives as potential spermicidal and microbicidal agentsPandey, Rishi Ranjan / Srivastava, Akansha / Malasoni, Richa / Naqvi, Arshi / Jain, Ashish / Maikhuri, Jagdamba Prasad / Paliwal, Sarvesh / Gupta, Gopal / Dwivedi, Anil Kumar et al. | 2012
- 5739
-
Synthesis and antibacterial activity of 6-O-(heteroaryl-isoxazolyl)propynyl 2-fluoro ketolidesSugimoto, Tomohiro / Shimazaki, Yoichi / Manaka, Akira / Tanikawa, Tetsuya / Suzuki, Keiko / Nanaumi, Kayoko / Kaneda, Yoshie / Yamasaki, Yukiko / Sugiyama, Hiroyuki et al. | 2012
- 5744
-
The antioxidant effect of imine resveratrol analoguesLu, Jing / Li, Chang / Chai, Yun-Feng / Yang, De-Yu / Sun, Cui-Rong et al. | 2012
- 5748
-
Synthesis and structure–activity relationship of (1-halo-2-naphthyl) carbamate-based inhibitors of KIAA1363 (NCEH1/AADACL1)Shreder, Kevin R. / Lin, Emme C.K. / Wu, Jiangyue / Cajica, Julia / Amantea, Christopher M. / Hu, Yi / Okerberg, Eric / Brown, Heidi E. / Pham, Lan M. / Chung, De Michael et al. | 2012
- 5752
-
Corrigendum to “Cytotoxic cytochalasins from the endozoic fungus Phoma sp. of the giant jellyfish Nemopilema nomurai” [Bioorg. Med. Chem. Lett. 22 (2012) 3126–3129]Kim, Eun La / Li, Jian Lin / Dang, Hung The / Hong, Jongki / Lee, Chong-Ok / Kim, Dong-Kyoo / Yoon, Won Duk / Kim, Euikyung / Liu, Yonghong / Jung, Jee H. et al. | 2012
- IFC
-
Editorial board| 2012