Synthesis and glycosidase inhibitory activity of novel (2-phenyl-4H-benzopyrimedo[2,1-b]-thiazol-4-yliden)acetonitrile derivatives (English)
- New search for: Patil, Vijay S.
- New search for: Nandre, Kamalakar P.
- New search for: Ghosh, Sougata
- New search for: Rao, Vaidya Jayathirtha
- New search for: Chopade, Balu A.
- New search for: Bhosale, Sheshanath V.
- New search for: Bhosale, Sidhanath V.
- New search for: Patil, Vijay S.
- New search for: Nandre, Kamalakar P.
- New search for: Ghosh, Sougata
- New search for: Rao, Vaidya Jayathirtha
- New search for: Chopade, Balu A.
- New search for: Bhosale, Sheshanath V.
- New search for: Bhosale, Sidhanath V.
In:
Bioorganic and Medicinal Chemistry Letters
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22
, 23
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7011-7014
;
2012
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ISSN:
- Article (Journal) / Electronic Resource
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Title:Synthesis and glycosidase inhibitory activity of novel (2-phenyl-4H-benzopyrimedo[2,1-b]-thiazol-4-yliden)acetonitrile derivatives
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Contributors:Patil, Vijay S. ( author ) / Nandre, Kamalakar P. ( author ) / Ghosh, Sougata ( author ) / Rao, Vaidya Jayathirtha ( author ) / Chopade, Balu A. ( author ) / Bhosale, Sheshanath V. ( author ) / Bhosale, Sidhanath V. ( author )
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Published in:Bioorganic and Medicinal Chemistry Letters ; 22, 23 ; 7011-7014
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Publisher:
- New search for: Elsevier Ltd
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Publication date:2012-10-04
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Size:4 pages
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ISSN:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Keywords:
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Source:
Table of contents – Volume 22, Issue 23
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 6987
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Graphical contents list| 2012
- 7002
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Polyether ionophores—promising bioactive molecules for cancer therapyHuczyński, Adam et al. | 2012
- 7011
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Synthesis and glycosidase inhibitory activity of novel (2-phenyl-4H-benzopyrimedo[2,1-b]-thiazol-4-yliden)acetonitrile derivativesPatil, Vijay S. / Nandre, Kamalakar P. / Ghosh, Sougata / Rao, Vaidya Jayathirtha / Chopade, Balu A. / Bhosale, Sheshanath V. / Bhosale, Sidhanath V. et al. | 2012
- 7015
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Prohormone-substrate peptide sequence recognition by peptidylglycine α-amidating monooxygenase and its reflection in increased glycolate inhibitor potencyMorris, Kelly M. / Cao, Feihua / Onagi, Hideki / Altamore, Timothy M. / Gamble, Allan B. / Easton, Christopher J. et al. | 2012
- 7015
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Prohormone-substrate peptide sequence recognition by peptidylglycine a-amidating monooxygenase and its reflection in increased glycolate inhibitor potencyMorris, K. M. / Cao, F. / Onagi, H. / Altamore, T. M. / Gamble, A. B. / Easton, C. J. et al. | 2012
- 7019
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Inhibitors of the acetyltransferase domain of N-acetylglucosamine-1-phosphate-uridylyltransferase/glucosamine-1-phosphate-acetyltransferase (GlmU). Part 2: Optimization of physical properties leading to antibacterial aryl sulfonamidesStokes, Suzanne S. / Albert, Robert / Buurman, Ed T. / Andrews, Beth / Shapiro, Adam B. / Green, Oluyinka M. / McKenzie, Andrew R. / Otterbein, Ludovic R. et al. | 2012
- 7024
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Synthesis and biological evaluation of 5-aryloxypyrazole derivatives bearing a rhodanine-3-aromatic acid as potential antimicrobial agentsZheng, Chang-Ji / Song, Ming-Xia / Sun, Liang-Peng / Wu, Yan / Hong, Lan / Piao, Hu-Ri et al. | 2012
- 7029
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POMA analyses as new efficient bioinformatics’ platform to predict and optimise bioactivity of synthesized 3a,4-dihydro-3H-indeno[1,2-c]pyrazole-2-carboxamide/carbothioamide analoguesAhsan, Mohamed Jawed / Govindasamy, Jeyabalan / Khalilullah, Habibullah / Mohan, Govind / Stables, James P. / Pannecouque, Christophe / Clercq, Eric De et al. | 2012
- 7036
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Novel series of 3-amino-N-(4-aryl-1,1-dioxothian-4-yl)butanamides as potent and selective dipeptidyl peptidase IV inhibitorsNitta, Aiko / Fujii, Hideaki / Sakami, Satoshi / Satoh, Mikiya / Nakaki, Junko / Satoh, Shiho / Kumagai, Hiroki / Kawai, Hideki et al. | 2012
- 7041
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Synthetic bicyclic iminosugar derivatives fused thiazolidin-4-one as new potential HIV-RT inhibitorsChen, Hua / Yang, Tianyu / Wei, Sinan / Zhang, Hongzhi / Li, Rui / Qin, Zhanbin / Li, Xiaoliu et al. | 2012
- 7045
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Aggregate formation and radiolytic degradation of amphiphilic DNA block copolymer possessing disulfide bondTanabe, Kazuhito / Asada, Takumi / Nishimoto, Sei-ichi et al. | 2012
- 7048
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Linear and cyclic dipeptides with antimalarial activityPérez-Picaso, Lemuel / Olivo, Horacio F. / Argotte-Ramos, Rocío / Rodríguez-Gutiérrez, María / Rios, María Yolanda et al. | 2012
- 7052
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Specific interactions between adenosine and streptavidin/avidinBing, Tao / Chang, Tianjun / Qi, Cui / Zhang, Nan / Liu, Xiangjun / Shangguan, Dihua et al. | 2012
- 7056
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Synthesis, characterization and potent DNA-cleaving activity of copper(II)-complexed berberine carboxylateChen, Jin-Xiang / Lin, Wei-Er / Chen, Ming-Zhen / Zhou, Chun-Qiong / Lin, Yan-Ling / Chen, Ming / Jiang, Zhi-Hong / Chen, Wen-Hua et al. | 2012
- 7060
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Anti-viral activity of (−)- and (+)-usnic acids and their derivatives against influenza virus A(H1N1)2009Sokolov, Dmitriy N. / Zarubaev, Vladimir V. / Shtro, Anna A. / Polovinka, Marina P. / Luzina, Olga A. / Komarova, Nina I. / Salakhutdinov, Nariman F. / Kiselev, Oleg I. et al. | 2012
- 7065
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Synthesis, characterization, antidepressant and antioxidant activity of novel piperamides bearing piperidine and piperazine analoguesPrashanth, M.K. / Revanasiddappa, Hosakere D. / Lokanatha Rai, K.M. / Veeresh, B. et al. | 2012
- 7071
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Synthesis and antitrypanosomal activity of new 6,6,7-trisubstituted thiopyrano[2,3-d][1,3]thiazolesZelisko, Nataliya / Atamanyuk, Dmytro / Vasylenko, Olexandr / Grellier, Philippe / Lesyk, Roman et al. | 2012
- 7075
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Design, synthesis and evaluation of novel zwitterionic compounds as PPARa/g dual agonists (1)Shibata, Y. / Kagechika, K. / Yamaguchi, M. / Kubo, H. / Usui, H. et al. | 2012
- 7075
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Design, synthesis and evaluation of novel zwitterionic compounds as PPARα/γ dual agonists (1)Shibata, Yoshihiro / Kagechika, Katsuji / Yamaguchi, Mitsuhiro / Kubo, Hideo / Usui, Hiroyuki et al. | 2012
- 7080
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Antibacterial activity of substituted 5-methylbenzo[c]phenanthridinium derivativesParhi, Ajit / Kelley, Cody / Kaul, Malvika / Pilch, Daniel S. / LaVoie, Edmond J. et al. | 2012
- 7084
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The structural requirements of histone deacetylase inhibitors: Suberoylanilide hydroxamic acid analogs modified at the C6 positionChoi, Sun Ea / Pflum, Mary Kay H. et al. | 2012
- 7087
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Tyrosine urea muscarinic acetylcholine receptor antagonists: Achiral quaternary ammonium groupsJin, Qi / Davis, Roderick S. / Bullion, Ann M. / Jin, Jian / Wang, Yonghui / Widdowson, Katherine L. / Palovich, Michael R. / Foley, James J. / Schmidt, Dulcie B. / Buckley, Peter T. et al. | 2012
- 7092
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Synthesis of isoindole and benzoisoindole derivatives of teicoplanin pseudoaglycon with remarkable antibacterial and antiviral activitiesSipos, Attila / Török, Zsolt / Rőth, Erzsébet / Kiss-Szikszai, Attila / Batta, Gyula / Bereczki, Ilona / Fejes, Zsolt / Borbás, Anikó / Ostorházi, Eszter / Rozgonyi, Ferenc et al. | 2012
- 7097
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Synthesis of enantiomerically pure perhydro-1,4-diazepine-2,5-dione and 1,4-piperazine-2,5-dione derivatives exhibiting potent activity as apoptosis inhibitorsMoure, Alejandra / Orzáez, Mar / Sancho, Mónica / Messeguer, Angel et al. | 2012
- 7100
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The design and synthesis of indazole and pyrazolopyridine based glucokinase activators for the treatment of Type 2 diabetes mellitusPfefferkorn, Jeffrey A. / Tu, Meihua / Filipski, Kevin J. / Guzman-Perez, Angel / Bian, Jianwei / Aspnes, Gary E. / Sammons, Matthew F. / Song, Wei / Li, Jian-Cheng / Jones, Christopher S. et al. | 2012
- 7106
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Structure–activity relationship exploration of Kv1.3 blockers based on diphenoxylateNguyen, William / Howard, Brittany L. / Jenkins, David P. / Wulff, Heike / Thompson, Philip E. / Manallack, David T. et al. | 2012
- 7110
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Syntheses and structure-activity relationship studies of N-substituted-b-d-glucosaminides as selective cytotoxic agentsWang, B. / Liu, Y. / Wang, Y. / Liu, X. / Cheng, M. S. et al. | 2012
- 7110
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Syntheses and structure–activity relationship studies of N-substituted-β-d-glucosaminides as selective cytotoxic agentsWang, Bo / Liu, Yang / Wang, Yanshi / Liu, Xin / Cheng, Mao-Sheng et al. | 2012
- 7114
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Structural modifications of 5,6-dihydroxypyrimidines with anti-HIV activityGuo, Di-Liang / Zhang, Xing-Jie / Wang, Rui-Rui / Zhou, Yu / Li, Zeng / Xu, Jin-Yi / Chen, Kai-Xian / Zheng, Yong-Tang / Liu, Hong et al. | 2012
- 7119
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Novel progesterone receptor modulators: 4-Aryl-phenylsulfonamidesMcComas, Casey / Cohen, Jeffrey / Huselton, Christine / Marella, Michael / Melenski, Edward / Mugford, Cheryl / Slayden, Ov / Winneker, Richard / Wrobel, Jay / Yudt, Matthew R. et al. | 2012
- 7123
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T-type Ca2+ channel blocker, KYS05047 induces G1 phase cell cycle arrest by decreasing intracellular Ca2+ levels in human lung adenocarcinoma A549 cellsRim, Hong-Kun / Lee, Heon-Woo / Choi, Il Sook / Park, Jin Yeong / Choi, Heung Woo / Choi, Jung-Hye / Cho, Young-Wuk / Lee, Jae Yeol / Lee, Kyung-Tae et al. | 2012
- 7127
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Kibdelomycin A, a congener of kibdelomycin, derivatives and their antibacterial activitiesSingh, Sheo B. / Goetz, Michael A. / Smith, Scott K. / Zink, Deborah L. / Polishook, Jon / Onishi, Russell / Salowe, Scott / Wiltsie, Judyann / Allocco, John / Sigmund, Janet et al. | 2012
- 7131
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Synthesis and antibiofilm activity of marine natural product-based 4-thiazolidinones derivativesRane, Rajesh A. / Sahu, Niteshkumar U. / Shah, Chetan P. et al. | 2012
- 7135
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Design, synthesis and SAR analysis of novel potent and selective small molecule antagonists of NPBWR1 (GPR7)Urbano, Mariangela / Guerrero, Miguel / Zhao, Jian / Velaparthi, Subash / Adrian Saldanha, S. / Chase, Peter / Wang, Zhiwei / Civelli, Olivier / Hodder, Peter / Schaeffer, Marie-Therese et al. | 2012
- 7142
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Anion inhibition studies of the fastest carbonic anhydrase (CA) known, the extremo-CA from the bacterium Sulfurihydrogenibium azorenseVullo, Daniela / De Luca, Viviana / Scozzafava, Andrea / Carginale, Vincenzo / Rossi, Mosè / Supuran, Claudiu T. / Capasso, Clemente et al. | 2012
- 7146
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Antiproliferative activity of salinomycin and its derivativesHuczyński, Adam / Janczak, Jan / Antoszczak, Michał / Wietrzyk, Joanna / Maj, Ewa / Brzezinski, Bogumil et al. | 2012
- 7151
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Novel azulene derivatives for the treatment of erectile dysfunctionLöber, Stefan / Hübner, Harald / Buschauer, Armin / Sanna, Fabrizio / Argiolas, Antonio / Melis, Maria Rosaria / Gmeiner, Peter et al. | 2012
- 7155
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Structure-based bioisosterism design, synthesis and biological evaluation of novel 1,2,4-triazin-6-ylthioacetamides as potent HIV-1 NNRTIsZhan, Peng / Li, Xiao / Li, Zhenyu / Chen, Xuwang / Tian, Ye / Chen, Wenmin / Liu, Xinyong / Pannecouque, Christophe / Clercq, Erik De et al. | 2012
- 7163
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Enriching C-terminal peptide from endopeptidase ArgC digest for protein C-terminal analysisKuyama, Hiroki / Nakajima, Chihiro / Tanaka, Koichi et al. | 2012
- 7169
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Synthesis and structure–activity relationships of a novel series of pyrimidines as potent inhibitors of TBK1/IKKε kinasesMcIver, Edward G. / Bryans, Justin / Birchall, Kristian / Chugh, Jasveen / Drake, Thomas / Lewis, Stephen J. / Osborne, Joanne / Smiljanic-Hurley, Ela / Tsang, William / Kamal, Ahmad et al. | 2012
- 7174
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Synthesis, evaluation and structure–activity relationships of triazine dimers as novel antiviral agentsVenkatraj, Muthusamy / Ariën, Kevin K. / Heeres, Jan / Joossens, Jurgen / Messagie, Jonas / Michiels, Johan / Van der Veken, Pieter / Vanham, Guido / Lewi, Paul J. / Augustyns, Koen et al. | 2012
- 7179
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A new boronic acid based fluorescent reporter for catecholWu, Zhongyu / Li, Minyong / Fang, Hao / Wang, Binghe et al. | 2012
- 7183
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Inhibition of monoamine oxidase by derivatives of piperine, an alkaloid from the pepper plant Piper nigrum, for possible use in Parkinson’s diseaseAl-Baghdadi, Osamah B. / Prater, Natalie I. / Van der Schyf, Cornelis J. / Geldenhuys, Werner J. et al. | 2012
- 7189
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Exploration of cathepsin S inhibitors characterized by a triazole P1–P2 amide replacementMoss, Neil / Xiong, Zhaoming / Burke, Mike / Cogan, Derek / Gao, Donghong A. / Haverty, Kathleen / Heim-Riether, Alexander / Hickey, Eugene R. / Nagaraja, Raj / Netherton, Matthew et al. | 2012
- 7194
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Synthesis and anti-hyperglycemic activity of hesperidin derivativesZhang, Baoshun / Chen, Tingting / Chen, Zhu / Wang, Mingxue / Zheng, Dengyu / Wu, Jinfeng / Jiang, Xiaofei / Li, Xuegang et al. | 2012
- 7198
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Synthesis of a major mitomycin C DNA adduct via a triaminomitoseneChampeil, Elise / Paz, Manuel M. / Lukasiewicz, Elaan / Kong, Wan S. / Watson, Stephanie / Sapse, Anne-Marie et al. | 2012
- 7201
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Development of potent macrocyclic inhibitors of genotype 3a HCV NS3/4A proteaseRudd, Michael T. / McCauley, John A. / Romano, Joseph J. / Butcher, John W. / Bush, Kimberly / McIntyre, Charles J. / Nguyen, Kevin T. / Gilbert, Kevin F. / Lyle, Terry A. / Holloway, M. Katharine et al. | 2012
- 7207
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Development of macrocyclic inhibitors of HCV NS3/4A protease with cyclic constrained P2–P4 linkersRudd, Michael T. / McIntyre, Charles J. / Romano, Joseph J. / Butcher, John W. / Holloway, M. Katharine / Bush, Kimberly / Nguyen, Kevin T. / Gilbert, Kevin F. / Lyle, Terry A. / Liverton, Nigel J. et al. | 2012
- 7214
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Investigations into specificity of azepinomycin for inhibition of guanase: Discrimination between the natural heterocyclic inhibitor and its synthetic nucleoside analoguesChakraborty, Saibal / Shah, Niti H. / Fishbein, James C. / Hosmane, Ramachandra S. et al. | 2012
- 7219
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4-Phenyl tetrahydroisoquinolines as dual norepinephrine and dopamine reuptake inhibitorsPechulis, Anthony D. / Beck, James P. / Curry, Matt A. / Wolf, Mark A. / Harms, Arthur E. / Xi, Ning / Opalka, Chet / Sweet, Mark P. / Yang, Zhicai / Vellekoop, A. Samuel et al. | 2012
- 7223
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Synthesis and SAR development of novel mGluR1 antagonists for the treatment of chronic painBrumfield, Stephanie / Korakas, Peter / Silverman, Lisa S. / Tulshian, Deen / Matasi, Julius J. / Qiang, Li / Bennett, Chad E. / Burnett, Duane A. / Greenlee, William J. / Knutson, Chad E. et al. | 2012
- 7227
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Synthesis and biological evaluation of novel heterocyclic derivatives of combretastatin A-4Nguyen, Thi Thanh Binh / Lomberget, Thierry / Tran, Ngoc Chau / Colomb, Evelyne / Nachtergaele, Lore / Thoret, Sylviane / Dubois, Joëlle / Guillaume, Joren / Abdayem, Rawad / Haftek, Marek et al. | 2012
- 7232
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Identification of novel scaffold of benzothiazepinones as non-ATP competitive glycogen synthase kinase-3β inhibitors through virtual screeningZhang, Peng / Hu, Hai-Rong / Huang, Zhao-Hui / Lei, Jia-Yi / Chu, Yong / Ye, De-Yong et al. | 2012
- 7232
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Identification of novel scaffold of benzothiazepinones as non-ATP competitive glycogen synthase kinase-3b inhibitors through virtual screeningZhang, P. / Hu, H. R. / Huang, Z. H. / Lei, J. Y. / Chu, Y. / Ye, D. Y. et al. | 2012
- 7237
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Synthesis and biological evaluation of 4,4-dimethyl lithocholic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1BHe, Hai-Bing / Gao, Li-Xin / Deng, Qi-Feng / Ma, Wei-Ping / Tang, Chun-Lan / Qiu, Wen-Wei / Tang, Jie / Li, Jing-Ya / Li, Jia / Yang, Fan et al. | 2012
- 7243
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New monoterpene glycosides from Paeonia suffruticosa Andrews and their inhibition on NO production in LPS-induced RAW 264.7 cellsDing, Liqin / Zhao, Feng / Chen, Lixia / Jiang, Zhihu / Liu, Yue / Li, Zhuomin / Qiu, Feng / Yao, Xinsheng et al. | 2012
- 7248
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Detection of pre-mRNA splicing in vitro by an RNA-templated fluorogenic reactionTamura, Yasutsugu / Furukawa, Kazuhiro / Yoshimoto, Rei / Kawai, Yuto / Yoshida, Minoru / Tsuneda, Satoshi / Ito, Yoshihiro / Abe, Hiroshi et al. | 2012
- 7252
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In vivo activity of an azole series of CCR2 antagonistsSmethurst, Chris A. / Bevan, Nicola / Brooks, Carl / Emmons, Amanda / Gough, Peter J. / Mookherjee, Claudette / Moores, Kitty / Peace, Simon / Philp, Joanne / Piercy, Val et al. | 2012
- 7256
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Ferrocene labelings as inhibitors and dual electrochemical sensors of human glutathione S-transferase P1-1Martos-Maldonado, Manuel C. / Quesada-Soriano, Indalecio / García-Maroto, Federico / Vargas-Berenguel, Antonio / García-Fuentes, Luís et al. | 2012
- 7261
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Synthesis and cytotoxicity evaluation of highly functionalized pyranochromenes and pyranopyransEmmadi, Narender Reddy / Atmakur, Krishnaiah / Chityal, Ganesh Kumar / Pombala, Sujitha / Nanubolu, Jagadeesh Babu et al. | 2012
- 7265
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Cytotoxic indole diketopiperazines from the deep sea-derived fungus Acrostalagmus luteoalbus SCSIO F457Wang, Fa-Zuo / Huang, Zhi / Shi, Xue-Feng / Chen, Yu-Chan / Zhang, Wei-Min / Tian, Xin-Peng / Li, Jie / Zhang, Si et al. | 2012
- 7268
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Design, synthesis and biological evaluation of N-arylphenyl-2,2-dichloroacetamide analogues as anti-cancer agentsLi, Tianwen / Yang, Yongchong / Cheng, Changmei / Tiwari, Amit K. / Sodani, Kamlesh / Zhao, Yufen / Abraham, Ioana / Chen, Zhe-Sheng et al. | 2012
- 7272
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Corrigendum to “Symmetrical approach of spiro-pyrazolidinediones as acetyl-CoA carboxylase inhibitors” [Bioorg. Med. Chem. Lett. 22 (2012) 4769–4772]Kamata, Makoto / Yamashita, Tohru / Kina, Asato / Tawada, Michiko / Endo, Satoshi / Mizukami, Atsushi / Sasaki, Masako / Tani, Akiyoshi / Nakano, Yoshihide / Watanabe, Yuuki et al. | 2012
- IFC
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Editorial board| 2012