Synthesis and antimalarial and antituberculosis activities of a series of natural and unnatural 4-methoxy-6-styryl-pyran-2-ones, dihydro analogues and photo-dimers (English)
- New search for: McCracken, Stephen T.
- New search for: Kaiser, Marcel
- New search for: Boshoff, Helena I.
- New search for: Boyd, Peter D.W.
- New search for: Copp, Brent R.
- New search for: McCracken, Stephen T.
- New search for: Kaiser, Marcel
- New search for: Boshoff, Helena I.
- New search for: Boyd, Peter D.W.
- New search for: Copp, Brent R.
In:
Bioorganic and Medicinal Chemistry
;
20
, 4
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1482-1493
;
2011
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ISSN:
- Article (Journal) / Electronic Resource
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Title:Synthesis and antimalarial and antituberculosis activities of a series of natural and unnatural 4-methoxy-6-styryl-pyran-2-ones, dihydro analogues and photo-dimers
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Contributors:McCracken, Stephen T. ( author ) / Kaiser, Marcel ( author ) / Boshoff, Helena I. ( author ) / Boyd, Peter D.W. ( author ) / Copp, Brent R. ( author )
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Published in:Bioorganic and Medicinal Chemistry ; 20, 4 ; 1482-1493
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Publisher:
- New search for: Elsevier Ltd
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Publication date:2011-12-23
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Size:12 pages
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ISSN:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Keywords:WYRDHDIRUVIXLT-UHFFFAOYSA-N , OVXOWIKMOIVICB-UHFFFAOYSA-N , BYHVZDRLSCCTND-UHFFFAOYSA-N , GBJRDULCMRSYSL-GQCTYLIASA-N , DKKJNZYHGRUXBS-BQYQJAHWSA-N , HXQHFAZJCRQKPB-UHFFFAOYSA-N , XRZOOBAREQKOOU-LDTJXHHCSA-N , OVIALWVJQXNHPR-AATRIKPKSA-N , LLUFWUGHFINWQU-QPJJXVBHSA-N , DJDGKNOLKXZSFR-JXMROGBWSA-N , GLWFCJOUIQRVSV-DUXPYHPUSA-N , MRYPIYDPVCUZPN-ZHACJKMWSA-N , OGTRIKSHCZMDDQ-DHZHZOJOSA-N , ORQOZZSYYGWBRL-NXZHAISVSA-N , JWISZNPEUKLOBM-YDFGWWAZSA-N , HRSLPCPLMOACJK-SNAWJCMRSA-N , RYGXLCMLRSWYBS-MDZDMXLPSA-N , VAGMONAMFIQZIK-VQHVLOKHSA-N , QVNXHWCUVXBSNR-FIFLTTCUSA-N , LJHLGAYQRPRZAM-UHFFFAOYSA-N , UACFBTNFAATILJ-UHFFFAOYSA-N , HVTZRXFNQOOCIV-UHFFFAOYSA-N , KDYSXPHDKMPJDB-UHFFFAOYSA-N , MZIHDUKSNXTLMD-UHFFFAOYSA-N , AJVALXXXOAULDB-UHFFFAOYSA-N , DEQIKGZYUVQMOR-UHFFFAOYSA-N , HAIJOOHLJUJNNU-ZBPDXVSDSA-N , TVFKEDHLIOUCTR-UHFFFAOYSA-N , OLSSKGLZSHZYMY-OHBBPIINSA-N , Malaria , Tuberculosis , Natural product , Pyran-2-one , Photochemical dimerisation
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Source:
Table of contents – Volume 20, Issue 4
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1365
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Graphical contents list| 2012
- 1373
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Synthesis, molecular docking and biological evaluation of 1,3,4-oxadiazole derivatives as potential immunosuppressive agentsYan, Ru / Zhang, Zhi-Ming / Fang, Xian-Ying / Hu, Yang / Zhu, Hai-Liang et al. | 2012
- 1380
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Biodegradable cyclen-based linear and cross-linked polymers as non-viral gene vectorsLi, Shuo / Wang, Yu / Wang, Shan / Zhang, Ji / Wu, Shi-Fei / Wang, Bo-Lin / Zhu, Wen / Yu, Xiao-Qi et al. | 2012
- 1388
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QSAR study and synthesis of new phenyltropanes as ligands of the dopamine transporter (DAT)Mavel, Sylvie / Mincheva, Zoya / Méheux, Nathalie / Carcenac, Yvan / Guilloteau, Denis / Abarbri, Mohamed / Emond, Patrick et al. | 2012
- 1396
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A facile ‘click’ approach to novel 15β-triazolyl-5α-androstane derivatives, and an evaluation of their antiproliferative activities in vitroKádár, Zalán / Molnár, Judit / Schneider, Gyula / Zupkó, István / Frank, Éva et al. | 2012
- 1396
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A facile `click' approach to novel 15b-triazolyl-5a-androstane derivatives, and an evaluation of their antiproliferative activities in vitroKadar, Z. / Molnar, J. / Schneider, G. / Zupko, I. / Frank, E. et al. | 2012
- 1403
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Cloning, characterization and sulfonamide inhibition studies of an α-carbonic anhydrase from the living fossil sponge Astrosclera willeyanaOhradanova, Anna / Vullo, Daniela / Pastorekova, Silvia / Pastorek, Jaromir / Jackson, Daniel J. / Wörheide, Gert / Supuran, Claudiu T. et al. | 2012
- 1403
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Cloning, characterization and sulfonamide inhibition studies of an a-carbonic anhydrase from the living fossil sponge Astrosclera willeyanaOhradanova, A. / Vullo, D. / Pastorekova, S. / Pastorek, J. / Jackson, D. J. / Worheide, G. / Supuran, C. T. et al. | 2012
- 1411
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Design, synthesis and biological evaluation of N-phenylsulfonylnicotinamide derivatives as novel antitumor inhibitorsZhang, Hui / Lu, Xiang / Zhang, Li-Rong / Liu, Jia-Jia / Yang, Xian-Hui / Wang, Xiao-Ming / Zhu, Hai-Liang et al. | 2012
- 1417
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Design, synthesis and CoMFA studies of N1-amino acid substituted 2,4,5-triphenyl imidazoline derivatives as p53–MDM2 binding inhibitorsHu, Chunqi / Dou, Xiaoxue / Wu, Yizhe / Zhang, Lei / Hu, Yongzhou et al. | 2012
- 1425
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Polypseudorotaxanes of pegylated α-cyclodextrin/polyamidoamine dendrimer conjugate with cyclodextrins as a sustained release system for DNAMotoyama, Keiichi / Hayashida, Kayoko / Higashi, Taishi / Arima, Hidetoshi et al. | 2011
- 1425
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Polypseudorotaxanes of pegylated a-cyclodextrin/polyamidoamine dendrimer conjugate with cyclodextrins as a sustained release system for DNAMotoyama, K. / Hayashida, K. / Higashi, T. / Arima, H. et al. | 2012
- 1434
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QSAR studies for prediction of cross-β sheet aggregate binding affinity and selectivityCisek, Katryna / Kuret, Jeff et al. | 2011
- 1434
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QSAR studies for prediction of cross-b sheet aggregate binding affinity and selectivityCisek, K. / Kuret, J. et al. | 2012
- 1442
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Angiogenesis inhibitors identified by cell-based high-throughput screening: Synthesis, structure–activity relationships and biological evaluation of 3-[(E)-styryl]benzamides that specifically inhibit endothelial cell proliferationHada, Kihito / Suda, Atsushi / Asoh, Kohsuke / Tsukuda, Takuo / Hasegawa, Masami / Sato, Yasuko / Ogawa, Kotaro / Kuramoto, Shino / Aoki, Yuko / Shimma, Nobuo et al. | 2011
- 1461
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In vitro biological evaluation of platinum(II) complexes with 1-(methoxy substituted benzyl) azetidine-3,3-dicarboxylato ligandsYin, Runting / Gou, Shaohua / Sun, Yanyan / Liu, Xia et al. | 2011
- 1468
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Conjugation of cell-penetrating peptides leads to identification of anti-HIV peptides from matrix proteinsNarumi, Tetsuo / Komoriya, Mao / Hashimoto, Chie / Wu, Honggui / Nomura, Wataru / Suzuki, Shintaro / Tanaka, Tomohiro / Chiba, Joe / Yamamoto, Naoki / Murakami, Tsutomu et al. | 2011
- 1475
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Synthesis and evaluation of debromohymenialdisine-derived Chk2 inhibitorsSaleem, Rahman Shah Zaib / Lansdell, Theresa A. / Tepe, Jetze J. et al. | 2011
- 1482
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Synthesis and antimalarial and antituberculosis activities of a series of natural and unnatural 4-methoxy-6-styryl-pyran-2-ones, dihydro analogues and photo-dimersMcCracken, Stephen T. / Kaiser, Marcel / Boshoff, Helena I. / Boyd, Peter D.W. / Copp, Brent R. et al. | 2011
- 1494
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Chemical reactivity and microbicidal action of bethoxazinChee, Gaik-Lean / Bhattarai, Bharat / Daniel Gietz, R. / Alrushaid, Samaa / Nitiss, John L. / Hasinoff, Brian B. et al. | 2011
- 1502
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Synthesis and in vitro evaluation of 68Ga-DOTA-4-FBn-TN14003, a novel tracer for the imaging of CXCR4 expressionHennrich, Ute / Seyler, Lisa / Schäfer, Martin / Bauder-Wüst, Ulrike / Eisenhut, Michael / Semmler, Wolfhard / Bäuerle, Tobias et al. | 2011
- 1511
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Synthesis and evaluation of malonate-based inhibitors of phosphosugar-metabolizing enzymes: Class II fructose-1,6-bis-phosphate aldolases, type I phosphomannose isomerase, and phosphoglucose isomeraseDesvergnes, Stéphanie / Courtiol-Legourd, Stéphanie / Daher, Racha / Dabrowski, Maciej / Salmon, Laurent / Therisod, Michel et al. | 2011
- 1521
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6-Nitrobenzimidazole derivatives: Potential phosphodiesterase inhibitors: Synthesis and structure–activity relationshipKhan, K.M. / Shah, Zarbad / Ahmad, V.U. / Ambreen, N. / Khan, M. / Taha, M. / Rahim, F. / Noreen, S. / Perveen, S. / Choudhary, M.I. et al. | 2011
- 1527
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Synthesis and antiplasmodial evaluation of novel chromeno[2,3-b]chromene derivativesDevakaram, Ruth / Black, David StC. / Choomuenwai, Vanida / Davis, Rohan A. / Kumar, Naresh et al. | 2011
- 1535
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17β-Arylsulfonamides of 17β-aminoestra-1,3,5(10)-trien-3-ol as highly potent inhibitors of steroid sulfataseMostafa, Yaser A. / Taylor, Scott D. et al. | 2011
- 1535
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17b-Arylsulfonamides of 17b-aminoestra-1,3,5(10)-trien-3-ol as highly potent inhibitors of steroid sulfataseMostafa, Y. A. / Taylor, S. D. et al. | 2012
- 1545
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Quinoline- and isoquinoline-sulfonamide derivatives of LCAP as potent CNS multi-receptor—5-HT1A/5-HT2A/5-HT7 and D2/D3/D4—agents: The synthesis and pharmacological evaluationZajdel, Paweł / Marciniec, Krzysztof / Maślankiewicz, Andrzej / Satała, Grzegorz / Duszyńska, Beata / Bojarski, Andrzej J. / Partyka, Anna / Jastrzębska-Więsek, Magdalena / Wróbel, Dagmara / Wesołowska, Anna et al. | 2011
- 1557
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Synthesis and evaluation of non-basic inhibitors of urokinase-type plasminogen activator (uPA)Venkatraj, Muthusamy / Messagie, Jonas / Joossens, Jurgen / Lambeir, Anne-Marie / Haemers, Achiel / Van der Veken, Pieter / Augustyns, Koen et al. | 2011
- 1569
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Synthesis of novel sulfonamide-1,2,4-triazoles, 1,3,4-thiadiazoles and 1,3,4-oxadiazoles, as potential antibacterial and antifungal agents. Biological evaluation and conformational analysis studiesZoumpoulakis, P. / Camoutsis, Ch. / Pairas, G. / Soković, M. / Glamočlija, J. / Potamitis, C. / Pitsas, A. et al. | 2011
- 1584
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Coumarin polysulfides inhibit cell growth and induce apoptosis in HCT116 colon cancer cellsSaidu, Nathaniel Edward Bennett / Valente, Sergio / Bana, Emilie / Kirsch, Gilbert / Bagrel, Denyse / Montenarh, Mathias et al. | 2011
- 1594
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Synthesis of 2′-O-guanidinopropyl-modified nucleoside phosphoramidites and their incorporation into siRNAs targeting hepatitis B virusBrzezinska, Jolanta / D’Onofrio, Jennifer / Buff, Maximilian C.R. / Hean, Justin / Ely, Abdullah / Marimani, Musa / Arbuthnot, Patrick / Engels, Joachim W. et al. | 2011
- 1594
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Synthesis of 2prime-O-guanidinopropyl-modified nucleoside phosphoramidites and their incorporation into siRNAs targeting hepatitis B virusBrzezinska, J. / D'Onofrio, J. / Buff, M. C. / Hean, J. / Ely, A. / Marimani, M. / Arbuthnot, P. / Engels, J. W. et al. | 2012
- 1607
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Quinol derivatives as potential trypanocidal agentsCapes, Amy / Patterson, Stephen / Wyllie, Susan / Hallyburton, Irene / Collie, Iain T. / McCarroll, Andrew J. / Stevens, Malcolm F.G. / Frearson, Julie A. / Wyatt, Paul G. / Fairlamb, Alan H. et al. | 2011
- 1616
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Tannic acid inhibited norovirus binding to HBGA receptors, a study of 50 Chinese medicinal herbsZhang, Xu-Fu / Dai, Ying-Chun / Zhong, Weiming / Tan, Ming / Lv, Zhi-Ping / Zhou, Ying-Chun / Jiang, Xi et al. | 2011
- 1624
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Substrate specificity of acetoxy derivatives of coumarins and quinolones towards Calreticulin mediated transacetylation: Investigations on antiplatelet functionKathuria, Abha / Priya, Nivedita / Chand, Karam / Singh, Prabhjot / Gupta, Anjali / Jalal, Sarah / Gupta, Shilpi / Raj, Hanumantharao G. / Sharma, Sunil K. et al. | 2011
- IFC
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Editorial board| 2012