Further characterization of a putative serine protease contributing to the γ-secretase cleavage of β-amyloid precursor protein (English)
- New search for: Peuchmaur, Marine
- New search for: Lacour, Marie-Agnès
- New search for: Sévalle, Jean
- New search for: Lisowski, Vincent
- New search for: Touati-Jallabe, Youness
- New search for: Rodier, Fabien
- New search for: Martinez, Jean
- New search for: Checler, Frédéric
- New search for: Hernandez, Jean-François
- New search for: Peuchmaur, Marine
- New search for: Lacour, Marie-Agnès
- New search for: Sévalle, Jean
- New search for: Lisowski, Vincent
- New search for: Touati-Jallabe, Youness
- New search for: Rodier, Fabien
- New search for: Martinez, Jean
- New search for: Checler, Frédéric
- New search for: Hernandez, Jean-François
In:
Bioorganic and Medicinal Chemistry
;
21
, 4
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1018-1029
;
2012
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ISSN:
- Article (Journal) / Electronic Resource
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Title:Further characterization of a putative serine protease contributing to the γ-secretase cleavage of β-amyloid precursor protein
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Contributors:Peuchmaur, Marine ( author ) / Lacour, Marie-Agnès ( author ) / Sévalle, Jean ( author ) / Lisowski, Vincent ( author ) / Touati-Jallabe, Youness ( author ) / Rodier, Fabien ( author ) / Martinez, Jean ( author ) / Checler, Frédéric ( author ) / Hernandez, Jean-François ( author )
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Published in:Bioorganic and Medicinal Chemistry ; 21, 4 ; 1018-1029
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Publisher:
- New search for: Elsevier Ltd
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Publication date:2012-11-15
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Size:12 pages
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ISSN:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Keywords:Aβ , Amyloid β-peptide , AICD , APP intracellular domain , APP , Amyloid-β Precursor Protein , BACE , beta-site APP cleaving enzyme , DCM , dichloromethane , DMSO , dimethylsulfoxide , ESI , electrospray ionization , EtOAc , ethyl acetate , FBS , fetal bovine serum , GSAP , γ-secretase activating protein , GSI , γ-secretase inhibitor , GSM , γ-secretase modulator , HEK , Human Embryonic Kidney , Hex , hexane , HRMS , high resolution mass spectrometry , LC/MS , liquid chromatography coupled to mass spectrometry , LDH , lactate dehydrogenase , NICD , Notch intracellular domain , PBS , phosphate buffered saline , PS , presenilin , RIPA , radio-immunoprecipitation assay , SDS–PAGE , sodium dodecylsulfate–polyacrylamide gel electrophoresis , TFA , trifluoroacetic acid , THF , tetrahydrofurane , Isocoumarin , Amyloid β peptide , Alzheimer’s disease , γ-Secretase , Serine proteases
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Source:
Table of contents – Volume 21, Issue 4
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 835
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Graphical contents list| 2013
- 841
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Synthesis and anticonvulsant activity of bioisosteres of trimethadione, N-derivative-1,2,3-oxathiazolidine-4-one-2,2-dioxides from α-hydroxyamidesPastore, Valentina / Sabatier, Laureano / Enrique, Andrea / Marder, Mariel / Bruno-Blanch, Luis E. et al. | 2012
- 841
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Synthesis and anticonvulsant activity of bioisosteres of trimethadione, N-derivative-1,2,3-oxathiazolidine-4-one-2,2-dioxides from a-hydroxyamidesPastore, V. / Sabatier, L. / Enrique, A. / Marder, M. / Bruno-Blanch, L. E. et al. | 2013
- 847
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N-(Phenoxyalkyl)amides as MT1 and MT2 ligands: Antioxidant properties and inhibition of Ca2+/CaM-dependent kinase IICarocci, Alessia / Catalano, Alessia / Bruno, Claudio / Lovece, Angelo / Roselli, Maria Grazia / Cavalluzzi, Maria Maddalena / De Santis, Francesco / De Palma, Annalisa / Rusciano, Maria Rosaria / Illario, Maddalena et al. | 2012
- 852
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Design of a new fluorescent probe: Pyrrole/imidazole hairpin polyamides with pyrene conjugation at their γ-turnVaijayanthi, Thangavel / Bando, Toshikazu / Hashiya, Kaori / Pandian, Ganesh N. / Sugiyama, Hiroshi et al. | 2012
- 852
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Design of a new fluorescent probe: Pyrrole/imidazole hairpin polyamides with pyrene conjugation at their g-turnVaijayanthi, T. / Bando, T. / Hashiya, K. / Pandian, G. N. / Sugiyama, H. et al. | 2013
- 856
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Asymmetric total synthesis and identification of tetrahydroprotoberberine derivatives as new antipsychotic agents possessing a dopamine D1, D2 and serotonin 5-HT1A multi-action profileSun, Haifeng / Zhu, Liyuan / Yang, Huicui / Qian, Wangke / Guo, Lin / Zhou, Shengbin / Gao, Bo / Li, Zeng / Zhou, Yu / Jiang, Hualiang et al. | 2012
- 869
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Synthesis of derivatives of the keto-pyrrolyl-difluorophenol scaffold: Some structural aspects for aldose reductase inhibitory activity and selectivityKotsampasakou, Eleni / Demopoulos, Vassilis J. et al. | 2012
- 874
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Effective inhibition of acid and neutral ceramidases by novel B-13 and LCL-464 analoguesBhabak, Krishna P. / Kleuser, Burkhard / Huwiler, Andrea / Arenz, Christoph et al. | 2012
- 883
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Telomere shortening and cell senescence induced by perylene derivatives in A549 human lung cancer cellsTaka, Thanachai / Huang, Liming / Wongnoppavich, Ariyaphong / Tam-Chang, Suk-Wah / Lee, T. Randall / Tuntiwechapikul, Wirote et al. | 2012
- 891
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Synthesis of N 4-(substituted phenyl)-N 4-alkyl/desalkyl-9H-pyrimido[4,5-b]indole-2,4-diamines and identification of new microtubule disrupting compounds that are effective against multidrug resistant cellsGangjee, Aleem / Zaware, Nilesh / Devambatla, Ravi Kumar Vyas / Raghavan, Sudhir / Westbrook, Cara D. / Dybdal-Hargreaves, Nicholas F. / Hamel, Ernest / Mooberry, Susan L. et al. | 2012
- 903
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Probing the steric requirements of the γ-aminobutyric acid aminotransferase active site with fluorinated analogues of vigabatrinJuncosa, Jose I. Jr. / Groves, Andrew P. / Xia, Guoyao / Silverman, Richard B. et al. | 2012
- 903
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Probing the steric requirements of the g-aminobutyric acid aminotransferase active site with fluorinated analogues of vigabatrinJuncosa, J. I. / Groves, A. P. / Xia, G. / Silverman, R. B. et al. | 2013
- 912
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18F-FBHGal for asialoglycoprotein receptor imaging in a hepatic fibrosis mouse modelKao, Hao-Wen / Chen, Chuan-Lin / Chang, Wen-Yi / Chen, Jenn-Tzong / Lin, Wuu-Jyh / Liu, Ren-Shyan / Wang, Hsin-Ell et al. | 2012
- 922
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Development, validation and pilot screening of an in vitro multi-cellular three-dimensional cancer spheroid assay for anti-cancer drug testingLama, Rati / Zhang, Lin / Naim, Janine M. / Williams, Jennifer / Zhou, Aimin / Su, Bin et al. | 2012
- 932
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Binding partners for curcumin in human schwannoma cells: Biologic ImplicationsAngelo, Laura S. / Maxwell, David S. / Wu, Ji Yuan / Sun, Duoli / Hawke, David H. / McCutcheon, Ian E. / Slopis, John M. / Peng, Zhenghong / Bornmann, William G. / Kurzrock, Razelle et al. | 2012
- 940
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Larvicidal isoxazoles: Synthesis and their effective susceptibility towards Aedes aegypti larvaeda Silva-Alves, Diana C.B. / dos Anjos, Janaína V. / Cavalcante, Nery N.M. / Santos, Geanne K.N. / Navarro, Daniela M.do A.F. / Srivastava, Rajendra M. et al. | 2012
- 948
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Synthesis of gatifloxacin derivatives and their biological activities against Mycobacterium leprae and Mycobacterium tuberculosisGomez, Catherine / Ponien, Prishila / Serradji, Nawal / Lamouri, Aazdine / Pantel, Alix / Capton, Estelle / Jarlier, Vincent / Anquetin, Guillaume / Aubry, Alexandra et al. | 2012
- 957
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Discovery of novel inhibitors of LEDGF/p75-IN protein–protein interactionsSanchez, Tino Wilson / Debnath, Bikash / Christ, Frauke / Otake, Hiroyuki / Debyser, Zeger / Neamati, Nouri et al. | 2012
- 964
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Photoprotective activity of resveratrol analoguesPolonini, Hudson Caetano / Lima, Larissa Lavorato / Gonçalves, Karla Mara / do Carmo, Antônio Márcio Resende / da Silva, Adilson David / Raposo, Nádia Rezende Barbosa et al. | 2012
- 969
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Effects of cytoprotective antioxidants on lymphocytes from representative mitochondrial neurodegenerative diseasesGoldschmidt, Ruth / Arce, Pablo M. / Khdour, Omar M. / Collin, Valérie C. / Dey, Sriloy / Jaruvangsanti, Jennifer / Fash, David M. / Hecht, Sidney M. et al. | 2012
- 979
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Discovery of INT131: A selective PPARg modulator that enhances insulin sensitivityTaygerly, J. P. / McGee, L. R. / Rubenstein, S. M. / Houze, J. B. / Cushing, T. D. / Li, Y. / Motani, A. / Chen, J. L. / Frankmoelle, W. / Ye, G. et al. | 2013
- 979
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Discovery of INT131: A selective PPARγ modulator that enhances insulin sensitivityTaygerly, Joshua P. / McGee, Lawrence R. / Rubenstein, Steven M. / Houze, Jonathan B. / Cushing, Timothy D. / Li, Yang / Motani, Alykhan / Chen, Jin-Long / Frankmoelle, Walter / Ye, Guosen et al. | 2012
- 993
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Structure–activity relationship of benzodiazepine derivatives as LXXLL peptide mimetics that inhibit the interaction of vitamin D receptor with coactivatorsMita, Yusuke / Dodo, Kosuke / Noguchi-Yachide, Tomomi / Hashimoto, Yuichi / Ishikawa, Minoru et al. | 2012
- 1006
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Design, synthesis, and evaluation of a water-soluble antofine analogue with high antiproliferative and antitumor activityKwon, Yongseok / Song, Jayoung / Lee, Boeun / In, Jinkyung / Song, Hohyun / Chung, Hwa-Jin / Lee, Sang Kook / Kim, Sanghee et al. | 2012
- 1018
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Further characterization of a putative serine protease contributing to the g-secretase cleavage of b-amyloid precursor proteinPeuchmaur, M. / Lacour, M. A. / Sevalle, J. / Lisowski, V. / Touati-Jallabe, Y. / Rodier, F. / Martinez, J. / Checler, F. / Hernandez, J. F. et al. | 2013
- 1018
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Further characterization of a putative serine protease contributing to the γ-secretase cleavage of β-amyloid precursor proteinPeuchmaur, Marine / Lacour, Marie-Agnès / Sévalle, Jean / Lisowski, Vincent / Touati-Jallabe, Youness / Rodier, Fabien / Martinez, Jean / Checler, Frédéric / Hernandez, Jean-François et al. | 2012
- IFC
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Editorial board| 2013