Pinocembrin and its linolenoyl ester derivative induce wound healing activity in HaCaT cell line potentially involving a GPR120/FFA4 mediated pathway (English)
- New search for: Mazzotta, Sarah
- New search for: Governa, Paolo
- New search for: Borgonetti, Vittoria
- New search for: Marcolongo, Paola
- New search for: Nanni, Claudio
- New search for: Gamberucci, Alessandra
- New search for: Manetti, Fabrizio
- New search for: Pessina, Federica
- New search for: Carullo, Gabriele
- New search for: Brizzi, Antonella
- New search for: Aiello, Francesca
- New search for: Mazzotta, Sarah
- New search for: Governa, Paolo
- New search for: Borgonetti, Vittoria
- New search for: Marcolongo, Paola
- New search for: Nanni, Claudio
- New search for: Gamberucci, Alessandra
- New search for: Manetti, Fabrizio
- New search for: Pessina, Federica
- New search for: Carullo, Gabriele
- New search for: Brizzi, Antonella
- New search for: Aiello, Francesca
In:
Bioorganic Chemistry
;
108
;
2021
-
ISSN:
- Article (Journal) / Electronic Resource
-
Title:Pinocembrin and its linolenoyl ester derivative induce wound healing activity in HaCaT cell line potentially involving a GPR120/FFA4 mediated pathway
-
Contributors:Mazzotta, Sarah ( author ) / Governa, Paolo ( author ) / Borgonetti, Vittoria ( author ) / Marcolongo, Paola ( author ) / Nanni, Claudio ( author ) / Gamberucci, Alessandra ( author ) / Manetti, Fabrizio ( author ) / Pessina, Federica ( author ) / Carullo, Gabriele ( author ) / Brizzi, Antonella ( author )
-
Published in:Bioorganic Chemistry ; 108
-
Publisher:
- New search for: Elsevier Inc.
-
Publication date:2021-01-12
-
ISSN:
-
DOI:
-
Type of media:Article (Journal)
-
Type of material:Electronic Resource
-
Language:English
-
Keywords:
-
Source:
Table of contents – Volume 108
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
-
Chemical mining of heterotrophic Shewanella algae reveals anti-infective potential of macrocyclic polyketides against multidrug-resistant pathogensChakraborty, Kajal / Kizhakkekalam, Vinaya Kizhakkepatt / Joy, Minju et al. | 2020
-
Design, synthesis, biological evaluation and molecular docking of new 1,3,4-oxadiazole homonucleosides and their double-headed analogs as antitumor agentsEL Mansouri, Az-eddine / Oubella, Ali / Mehdi, Ahmad / AitItto, Moulay Youssef / Zahouily, Mohamed / Morjani, Hamid / Lazrek, Hassan B. et al. | 2020
-
Identification of fenoldopam as a novel LSD1 inhibitor to abrogate the proliferation of renal cell carcinoma using drug repurposing strategyZheng, Yan / Ma, Yuan / Cao, Huixia / Yan, Lei / Gu, Yue / Ren, Xuejing / Jiao, Xiaojing / Wan, Shengfeng / Shao, Fengmin et al. | 2020
-
Investigation of pyrazolo[1,5-a]quinoxalin-4-ones as novel monoamine oxidase inhibitorsPanova, Valeria A. / Filimonov, Sergey I. / Chirkova, Zhanna V. / Kabanova, Mariya V. / Shetnev, Anton A. / Korsakov, Mikhail K. / Petzer, Anél / Petzer, Jacobus P. / Suponitsky, Kyrill Yu et al. | 2020
-
Discovery and SAR studies of 3-amino-4-(phenylsulfonyl)tetrahydrothiophene 1,1-dioxides as non-electrophilic antioxidant response element (ARE) activatorsJo, Jeyun / Ibrahim, Lara / Iaconelli, Jonathan / Kwak, Jinsook / Kumar, Manoj / Jung, Yunjin / Lairson, Luke L. / Chatterjee, Arnab K. / Schultz, Peter G. / Bollong, Michael J. et al. | 2020
-
Minor immunosuppressive spiroorthoester group-containing pregnane glycosides from the root barks of Periploca sepiumShao, Xing-Cheng / Chen, Zhen-Hua / Liu, Shuang-Shuang / Wu, Fei / Mu, Hong-Yan / Wei, Wen-Hui / Feng, Yi / Zuo, Jian-Ping / Zhang, Ji-Quan / He, Shi-Jun et al. | 2021
-
Synthesis of 6-epi-tuberiferin and the biological activities of tuberiferin, dehydrobrabrachylaenolide, 6-epi-tuberiferin, and their synthetic intermediatesLi, Dan / Higuchi, Yohsuke / Kobayashi, Takafumi / Shimoma, Fumito / Bai, Yuhua / Ando, Masayoshi et al. | 2021
-
Synthesis, inhibition properties against xanthine oxidase and molecular docking studies of dimethyl N-benzyl-1H-1,2,3-triazole-4,5-dicarboxylate and (N-benzyl-1H-1,2,3-triazole-4,5-diyl)dimethanol derivativesYagiz, Güler / Noma, Samir Abbas Ali / Altundas, Aliye / Al-khafaji, Khattab / Taskin-Tok, Tugba / Ates, Burhan et al. | 2021
-
QM/MM analysis, synthesis and biological evaluation of epalrestat based mutual-prodrugs for diabetic neuropathy and nephropathyChoudhary, Shalki / Kumar, Manoj / Silakari, Om et al. | 2020
-
Structural insights into the desymmetrization of bulky 1,2-dicarbonyls through enzymatic monoreductionRabuffetti, Marco / Cannazza, Pietro / Contente, Martina Letizia / Pinto, Andrea / Romano, Diego / Hoyos, Pilar / Alcantara, Andres R. / Eberini, Ivano / Laurenzi, Tommaso / Gourlay, Louise et al. | 2021
-
Synthesis of novel sulfonamide derivatives containing pyridin-3-ylmethyl 4-(benzoyl)piperazine-1-carbodithioate moiety as potent PKM2 activatorsLi, Ridong / Ning, Xianling / He, Jianan / Lin, Zhiqiang / Su, Yue / Li, Runtao / Yin, Yuxin et al. | 2021
-
Swertiamarin from Enicostemma littorale, counteracts PD associated neurotoxicity via enhancement α-synuclein suppressive genes and SKN-1/NRF-2 activation through MAPK pathwayPandey, Taruna / Shukla, Aparna / Trivedi, Mashu / Khan, Feroz / Pandey, Rakesh et al. | 2021
-
Antibiotic resistance and drug modification: Synthesis, characterization and bioactivity of newly modified potent ciprofloxacin derivativesAlsughayer, Abdulhakeem / Elassar, Abdel-Zaher A. / Hasan, Abdulaziz A. / Al Sagheer, Fakhreia et al. | 2021
-
Research progress in biological activities of succinimide derivativesZhao, Zefeng / Yue, Jiangxin / Ji, Xiaotong / Nian, Meng / Kang, Kaiwen / Qiao, Haifa / Zheng, Xiaohui et al. | 2020
-
Dimeric guaianes from leaves of Xylopia vielana as snail inhibitors identified by high content screeningXu, Qi-Qi / Zhang, Chao / Zhang, Ya-Long / Lei, Jian-Li / Kong, Ling-Yi / Luo, Jian-Guang et al. | 2021
-
Discovery of andrastones from the deep-sea-derived Penicillium allii-sativi MCCC 3A00580 by OSMAC strategyXie, Chun-Lan / Liu, Qingmei / He, Zhi-Hui / Gai, Ying-Bao / Zou, Zheng-Biao / Shao, Zong-Ze / Liu, Guang-Ming / Chen, Hai-Feng / Yang, Xian-Wen et al. | 2021
-
Design, synthesis and biological evaluation of potential anti-AD hybrids with monoamine oxidase B inhibitory and iron-chelating effectsGuo, Jianan / Mi, Zhisheng / Jiang, Xiaoying / Zhang, Changjun / Guo, Zili / Li, Linzi / Gu, Jinping / Zhou, Tao / Bai, Renren / Xie, Yuanyuan et al. | 2020
-
Anti-hyperlipidemic potential of natural product based labdane-pyrroles via inhibition of cholesterol and triglycerides synthesisJalaja, Renjitha / Leela, Shyni G. / Mohan, Sangeetha / Nair, Mangalam S. / Gopalan, Raghu K. / Somappa, Sasidhar B. et al. | 2021
-
Exploring the potential intracellular targets of vascular normalization based on active candidatesShan, Yuanyuan / Wang, Jin / Si, Ru / Ma, Yuexiang / Li, Jing / Zhang, Qingqing / Lu, Wen / Zhang, Jie et al. | 2020
-
Synthesis, biological evaluation and molecular docking studies of novel quinazolinones as antitubercular and antimicrobial agentsKumar Pandey, Sarvesh / Yadava, Umesh / Upadhyay, Anjali / Sharma, M.L. et al. | 2020
-
Synthesis of indole-based-thiadiazole derivatives as a potent inhibitor of α-glucosidase enzyme along with in silico studyAlomari, Munther / Taha, Muhammad / Rahim, Fazal / Selvaraj, Manikandan / Iqbal, Naveed / Chigurupati, Sridevi / Hussain, Shafqat / Uddin, Nizam / Almandil, Noor Barak / Nawaz, Muhammad et al. | 2021
-
Chalcone and its analogs: Therapeutic and diagnostic applications in Alzheimer’s diseaseThapa, Pritam / Upadhyay, Sunil P. / Suo, William Z. / Singh, Vikas / Gurung, Prajwal / Lee, Eung Seok / Sharma, Ram / Sharma, Mukut et al. | 2021
-
Issue TOC| 2021
-
Editorial Board| 2021
-
Quinoline carboxamide core moiety-based compounds inhibit P. falciparum falcipain-2: Design, synthesis and antimalarial efficacy studiesSingh, Anju / Kalamuddin, Md / Maqbool, Mudasir / Mohmmed, Asif / Malhotra, Pawan / Hoda, Nasimul et al. | 2020
-
Combined in silico and in vitro studies to identify novel antidiabetic flavonoids targeting glycogen phosphorylaseBrás, Natércia F. / Neves, Rui P.P. / Lopes, Filipa A.A. / Correia, Márcia A.S. / Palma, Angelina S. / Sousa, Sérgio F. / Ramos, Maria J. et al. | 2020
-
Bioactive constituents from Thunbergia erecta as potential anticholinesterase and anti-ageing agents: Experimental and in silico studiesRefaey, Mohamed S. / Abdelhamid, Reda A. / Elimam, Hanan / Elshaier, Yaseen A.M.M. / Ali, A.A. / Orabi, Mohamed A.A. et al. | 2021
-
Evaluation of thionolactones as a new type of hydrogen sulfide (H2S) donors for a blood pressure regulationZaorska, Ewelina / Gawryś-Kopczyńska, Marta / Ostaszewski, Ryszard / Ufnal, Marcin / Koszelewski, Dominik et al. | 2021
-
Dehydroepiandrosterone derived imidazolium salts and their antimicrobial efficacyHryniewicka, Agnieszka / Niemirowicz-Laskowska, Katarzyna / Wielgat, Przemysław / Car, Halina / Hauschild, Tomasz / Morzycki, Jacek W. et al. | 2020
-
Corrigendum to “Acylphloroglucinols with acetylcholinesterase inhibitory effects from the fruits of Eucalyptus robusta”. [Bioorg. Chem. 103 (2020) 104127]Liu, Hui / He, Xiao-Zhi / Feng, Mi-Yan / Yuan Zeng / Rauwolf, Tyler J. / Shao, Li-Dong / Ni, Wei / Yan, Hui / Porco, John A. Jr. / Hao, Xiao-Jiang et al. | 2020
-
Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic propertiesJiang, Bo / Luo, Jiao / Guo, Shuju / Wang, Lijun et al. | 2021
-
Pyrazoline analogs as potential anticancer agents and their apoptosis, molecular docking, MD simulation, DNA binding and antioxidant studiesRana, Manish / Arif, Rizwan / Khan, Faez Iqbal / Maurya, Vikas / Singh, Raja / Faizan, Md Imam / Yasmeen, Shama / Dar, Sajad Hussain / Alam, Raquib / Sahu, Ankita et al. | 2021
-
Antiamoebic effects of sesquiterpene lactones isolated from the zoanthid Palythoa aff. clavataRodríguez-Expósito, Rubén L. / Nocchi, Nathália / Reyes-Batlle, María / Sifaoui, Ines / Suárez-Gómez, Blanca / Díaz-Marrero, Ana R. / Souto, Maria L. / Piñero, José E. / Fernández, José J. / Lorenzo-Morales, Jacob et al. | 2021
-
A novel series of benzothiazepine derivatives as tubulin polymerization inhibitors with anti-tumor potencyWang, Bin / Wang, Li-Ren / Liu, Lu-Lu / Wang, Wei / Man, Ruo-Jun / Zheng, Da-Jun / Deng, Yu-Shan / Yang, Yu-Shun / Xu, Chen / Zhu, Hai-Liang et al. | 2020
-
Multivalent butyrylcholinesterase inhibitor discovered by exploiting dynamic combinatorial chemistryZhao, Shuang / Xu, Jintao / Zhang, Shixin / Han, Maochun / Wu, Yao / Li, Yusi / Hu, Lei et al. | 2021
-
Design, synthesis, molecular docking, in silico ADMET profile and anticancer evaluations of sulfonamide endowed with hydrazone-coupled derivatives as VEGFR-2 inhibitorsSayed, Asmaa M / Taher, Fatma A. / Abdel-Samad, Mohammad R.K. / El-Gaby, Mohamed S.A. / El‐Adl, Khaled / Saleh, Nashwa M. et al. | 2021
-
Eco-friendly sequential one-pot synthesis, molecular docking, and anticancer evaluation of arylidene-hydrazinyl-thiazole derivatives as CDK2 inhibitorsEl-Naggar, Abeer M. / El-Hashash, Maher A. / Elkaeed, Eslam B. et al. | 2020
-
Pesimquinolones I–S, eleven new quinolone alkaloids produced by Penicillium simplicissimum and their inhibitory activity on NO productionDai, Chong / Li, Xiaoxin / Zhang, Kailin / Li, Xiao-Nian / Wang, Wenjing / Zang, Yi / Chen, Xia / Li, Qin / Wei, Mengsha / Chen, Chunmei et al. | 2021
-
Scope and limitations of biocatalytic carbonyl reduction with white-rot fungiZhuk, Tatyana S. / Skorobohatko, Oleksandra S. / Albuquerque, Wendell / Zorn, Holger et al. | 2021
-
Pinocembrin and its linolenoyl ester derivative induce wound healing activity in HaCaT cell line potentially involving a GPR120/FFA4 mediated pathwayMazzotta, Sarah / Governa, Paolo / Borgonetti, Vittoria / Marcolongo, Paola / Nanni, Claudio / Gamberucci, Alessandra / Manetti, Fabrizio / Pessina, Federica / Carullo, Gabriele / Brizzi, Antonella et al. | 2021
-
Influence of core extension and side chain nature in targeting G-quadruplex structures with perylene monoimide derivativesBusto, Natalia / García-Calvo, José / Cuevas, José Vicente / Herrera, Antonio / Mergny, Jean-Louis / Pons, Sebastian / Torroba, Tomás / García, Begoña et al. | 2021
-
Target separation and antitumor metastasis activity of sesquiterpene-based lysine-specific demethylase 1 inhibitors from zedoary turmeric oilRen, Chunling / Lin, Yaolan / Liu, Xiaoqin / Yan, Dan / Xu, Xiao / Zhu, Dongrong / Kong, Lingyi / Han, Chao et al. | 2021
-
Combined 3D-QSAR and docking analysis for the design and synthesis of chalcones as potent and selective monoamine oxidase B inhibitorsMellado, Marco / González, César / Mella, Jaime / Aguilar, Luis F. / Viña, Dolores / Uriarte, Eugenio / Cuellar, Mauricio / Matos, Maria J. et al. | 2021
-
Synthesis and biological evaluation of novel withangulatin A derivatives as potential anticancer agentsZhou, Wu-Xi / Chen, Chen / Liu, Xiao-Qin / Li, Ying / Kong, Ling-Yi / Luo, Jian-Guang et al. | 2021
-
Insights of 8-hydroxyquinolines: A novel target in medicinal chemistryGupta, Rohini / Luxami, Vijay / Paul, Kamaldeep et al. | 2021
-
Design, synthesis and antitumor activity evaluation of novel HDAC inhibitors with tetrahydrobenzothiazole as the skeletonSun, Simin / Zhao, Wenwen / Li, Yongliang / Chi, Ziwei / Fang, Xixi / Wang, Qiang / Han, Zhiwu / Luan, Yepeng et al. | 2021
-
Pentacyclic triterpenes with nitric oxide inhibitory activity from Potentilla chinensisHan, Jae Sang / Kim, Jun Gu / Le, Thi Phuong Linh / Cho, Yong Beom / Lee, Mi Kyeong / Hwang, Bang Yeon et al. | 2021
-
Synthesis of imidazole-pyrazole conjugates bearing aryl spacer and exploring their enzyme inhibition potentialsChaudhry, Faryal / Shahid, Wardah / al-Rashida, Mariya / Ashraf, Muhammad / Ali Munawar, Munawar / Ain Khan, Misbahul et al. | 2021
-
Quinazolin-4(3H)-one based agents bearing thiadiazole-urea: Synthesis and evaluation of anti-proliferative and antiangiogenic activityFaraji, Aram / Motahari, Rasoul / Hasanvand, Zaman / Oghabi Bakhshaiesh, Tayebeh / Toolabi, Mahsa / Moghimi, Setareh / Firoozpour, Loghman / Boshagh, Mohammad Amin / Rahmani, Roya / Ketabforoosh, Shima H.M.E. et al. | 2020
-
Design and synthesis of pyrimidine-5-carbonitrile hybrids as COX-2 inhibitors: Anti-inflammatory activity, ulcerogenic liability, histopathological and docking studiesAlfayomy, Abdallah M. / Abdel-Aziz, Salah A. / Marzouk, Adel A. / Shaykoon, Montaser Sh. A. / Narumi, Atsushi / Konno, Hiroyuki / Abou-Seri, Sahar M. / Ragab, Fatma A.F. et al. | 2020
-
Furan-2-carboxamide derivative, a novel microtubule stabilizing agent induces mitotic arrest and potentiates apoptosis in cancer cellsShwetha, B / Sudhanva, M. Srinivasa / Jagadeesha, G.S / Thimmegowda, N.R / Hamse, Vivek K. / Sridhar, B.T / Thimmaiah, K.N / Ananda Kumar, C.S / Shobith, Rangappa / Rangappa, K.S et al. | 2020
-
Novel phenylpyrimidine derivatives containing a hydrazone moiety protect rice seedlings from injury by metolachlorDeng, Xile / Zheng, Wenna / Jin, Can / Zhan, Qingcai / Bai, Lianyang et al. | 2021
-
7-Amine-spiro[chromeno[4,3-b]quinoline-6,1′-cycloalkanes]: Synthesis and cholinesterase inhibitory activity of structurally modified tacrinesSilva, Letícia B. / Nogara, Pablo A. / Halmenschelager, Paula T. / Alvim, Jéssica C. / Silva, Fernanda D'A. / Feitosa, Sarah C. / Rocha, João B.T. / Martins, Marcos A.P. / Zanatta, Nilo / Bonacorso, Helio G. et al. | 2021
-
Antiinflammatory triterpenoids from the fruiting bodies of Fomitopsis pinicolaKuo, Ping-Chung / Tai, Shih-Huang / Hung, Ching-Che / Hwang, Tsong-Long / Kuo, Liang-Mou / Lam, Sio Hong / Cheng, Kun-Ching / Kuo, Daih-Huang / Hung, Hsin-Yi / Wu, Tian-Shung et al. | 2020
-
Discovery of a novel series of indolylchalcone-benzenesulfonamide hybrids acting as selective carbonic anhydrase II inhibitorsSingh, Priti / Purnachander Yadav, Parvatha / Swain, Baijayantimala / Thacker, Pavitra S. / Angeli, Andrea / Supuran, Claudiu T. / Arifuddin, Mohammed et al. | 2021
-
Diarylheptanoid-chalcone hybrids with PTP1B and α-glucosidase dual inhibition from Alpinia katsumadaiHe, Xiao-Feng / Chen, Ji-Jun / Li, Tian-Ze / Hu, Jing / Zhang, Xue-Mei / Geng, Chang-An et al. | 2021