ARTICLES - 5-Aryl-1,2,3,4-tetrahydrochromeno(3,4-f)quinolin-3-ones as a Novel Class of Nonsteroidal Progesterone Receptor Agonists: Effect of A-Ring Modification (English)
- New search for: Zhi, Lin
- New search for: Zhi, Lin
- New search for: Tegley, Christopher M.
- New search for: Marschke, Keith B.
- New search for: Mais, Dale E.
- New search for: Jones, Todd K.
In:
Journal of medicinal chemistry
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42
, 8
; 1466-1472
;
1999
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ISSN:
- Article (Journal) / Print
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Title:ARTICLES - 5-Aryl-1,2,3,4-tetrahydrochromeno(3,4-f)quinolin-3-ones as a Novel Class of Nonsteroidal Progesterone Receptor Agonists: Effect of A-Ring Modification
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Contributors:
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Published in:Journal of medicinal chemistry ; 42, 8 ; 1466-1472
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Publisher:
- New search for: American Chemical Society
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Place of publication:Easton, Pa.
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Publication date:1999
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 770/4230
- New search for: 44.42 / 44.42
- Further information on Basic classification
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Keywords:
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Classification:
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Source:
Table of contents – Volume 42, Issue 8
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1329
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ANNOUNCEMENTS - Termination of Page Charges Free Electronic Reprints| 1999
- 1330
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COMMUNICATIONS TO THE EDITOR - Synthesis and Antitumor Activity of Novel Thioester Derivatives of LeinamycinKanda, Yutaka et al. | 1999
- 1330
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Synthesis and Antitumor Activity of Novel Thioester Derivatives of LeinamycinKanda, Yutaka / Ashizawa, Tadashi / Kakita, Shingo / Takahashi, Yuichi / Kono, Motomichi / Yoshida, Mayumi / Saitoh, Yutaka / Okabe, Masami et al. | 1999
- 1333
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Potent, Highly Selective, and Non-Thiol Inhibitors of Protein Geranylgeranyltransferase-IVasudevan, Anil / Qian, Yimin / Vogt, Andreas / Blaskovich, Michelle A. / Ohkanda, Junko / Sebti, Said M. / Hamilton, Andrew D. et al. | 1999
- 1333
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EXPEDITED ARTICLES - Potent, Highly Selective, and Non-Thiol Inhibitors of Protein Geranylgeranyltransferase-IVasudevan, Anil et al. | 1999
- 1341
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Comparison of Four 64Cu-Labeled Somatostatin Analogues in Vitro and in a Tumor-Bearing Rat Model: Evaluation of New Derivatives for Positron Emission Tomography Imaging and Targeted Radiotherapy ‖Lewis, Jason S. / Lewis, Michael R. / Srinivasan, Ananth / Schmidt, Michelle A. / Wang, Jian / Anderson, Carolyn J. et al. | 1999
- 1341
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ARTICLES - Comparison of Four 64Cu-Labeled Somatostatin Analogues in Vitro and in a Tumor-Bearing Rat Model: Evaluation of New Derivatives for Positron Emission Tomography Imaging and Targeted RadiotherapyLewis, Jason S. et al. | 1999
- 1348
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ARTICLES - Identification of Highly Selective Inhibitors of Collagenase-1 from Combinatorial Libraries of DiketopiperazinesSzardenings, Anna Katrin et al. | 1999
- 1348
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Identification of Highly Selective Inhibitors of Collagenase-1 from Combinatorial Libraries of DiketopiperazinesSzardenings, Anna Katrin / Antonenko, Valery / Campbell, David A. / DeFrancisco, Nuria / Ida, Satoru / Shi, Lihong / Sharkov, Nikolai / Tien, David / Wang, Yongwen / Navre, Marc et al. | 1999
- 1358
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ARTICLES - Conformational and Quantitative Structure-Activity Relationship Study of Cytotoxic 2-ArylidenebenzocycloalkanonesDimmock, Jonathan R. et al. | 1999
- 1358
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Conformational and Quantitative Structure−Activity Relationship Study of Cytotoxic 2-ArylidenebenzocycloalkanonesDimmock, Jonathan R. / Kandepu, N. Murthi / Nazarali, Adil J. / Kowalchuk, Travis P. / Motaganahalli, Narasimhan / Quail, J. Wilson / Mykytiuk, Patricia A. / Audette, Gerald F. / Prasad, Lata / Perjési, Pál et al. | 1999
- 1367
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Secondary Structure Peptide Mimetics: Design, Synthesis, and Evaluation of β-Strand Mimetic Thrombin InhibitorsBoatman, P. Douglas / Ogbu, Cyprian O. / Eguchi, Masakatsu / Kim, Hwa-Ok / Nakanishi, Hiroshi / Cao, Bolong / Shea, J. Paul / Kahn, Michael et al. | 1999
- 1367
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ARTICLES - Secondary Structure Peptide Mimetics: Design, Synthesis, and Evaluation of b-Strand Mimetic Thrombin InhibitorsBoatman, P.Douglas et al. | 1999
- 1376
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Bound Structures of Novel P3−P1‘ β-Strand Mimetic Inhibitors of Thrombin †St. Charles, Robert / Matthews, John H. / Zhang, Erli / Tulinsky, A. et al. | 1999
- 1376
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ARTICLES - Bound Structures of Novel P3-P1' b-Strand Mimetic Inhibitors of ThrombinCharles, Robert St et al. | 1999
- 1384
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ARTICLES - 5'-N-Substituted Carboxamidoadenosines as Agonists for Adenosine ReceptorsZwart, Maarten de et al. | 1999
- 1384
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5‘-N-Substituted Carboxamidoadenosines as Agonists for Adenosine Receptorsde Zwart, Maarten / Kourounakis, Angeliki / Kooijman, Huub / Spek, Anthony L. / Link, Regina / von Frijtag Drabbe Künzel, Jacobien K. / IJzerman, Ad P. et al. | 1999
- 1393
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N 6,5‘-Disubstituted Adenosine Derivatives as Partial Agonists for the Human Adenosine A3 Receptorvan Tilburg, Erica W. / von Frijtag Drabbe Künzel, Jacobien / de Groote, Miriam / Vollinga, Roel C. / Lorenzen, Anna / IJzerman, Ad P. et al. | 1999
- 1393
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ARTICLES - N6,5'-Disubstituted Adenosine Derivatives as Partial Agonists for the Human Adenosine A3 ReceptorTilburg, Erica W.van et al. | 1999
- 1401
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ARTICLES - Chicoric Acid Analogues as HIV-1 Integrase InhibitorsLin, Zhaiwei et al. | 1999
- 1401
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Chicoric Acid Analogues as HIV-1 Integrase InhibitorsLin, Zhaiwei / Neamati, Nouri / Zhao, He / Kiryu, Yoshimitsu / Turpin, Jim A. / Aberham, Claudia / Strebel, Klaus / Kohn, Kurt / Witvrouw, Myriam / Pannecouque, Christophe et al. | 1999
- 1415
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1-(N-Alkylamino)-11-(N-ethylamino)-4,8-diazaundecanes: Simple Synthetic Polyamine Analogues That Differentially Alter Tubulin PolymerizationWebb, Heather K. / Wu, Zhiqian / Sirisoma, Nilantha / Ha, Hyo Chol / Casero,, Robert A. / Woster, Patrick M. et al. | 1999
- 1415
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ARTICLES - 1-(N-Alkylamino)-11-(N-ethylamino)-4,8-diazaundecanes: Simple Synthetic Polyamine Analogues That Differentially Alter Tubulin PolymerizationWebb, Heather K. et al. | 1999
- 1422
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Synthesis and Voltage-Clamp Studies of Methyl 1,4-Dihydro-2,6-dimethyl-5-nitro-4-(benzofurazanyl)pyridine-3-carboxylate Racemates and Enantiomers and of Their Benzofuroxanyl AnaloguesVisentin, Sonja / Amiel, Pascale / Fruttero, Roberta / Boschi, Donatella / Roussel, Christian / Giusta, Laura / Carbone, Emilio / Gasco, Alberto et al. | 1999
- 1422
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ARTICLES - Synthesis and Voltage-Clamp Studies of Methyl 1,4-Dihydro-2,6-dimethyl-5-nitro-4-(benzofurazanyl)pyridine- 3-carboxylate Racemates and Enantiomers and of Their Benzofuroxanyl AnaloguesVisentin, Sonja et al. | 1999
- 1428
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ARTICLES - Potent, Low-Molecular-Weight Non-Peptide Inhibitors of Malarial Aspartyl Protease Plasmepsin IIHaque, Tasir S. et al. | 1999
- 1428
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Potent, Low-Molecular-Weight Non-Peptide Inhibitors of Malarial Aspartyl Protease Plasmepsin IIHaque, Tasir S. / Skillman, A. Geoffrey / Lee, Christina E. / Habashita, Hiromu / Gluzman, Ilya Y. / Ewing, Todd J. A. / Goldberg, Daniel E. / Kuntz, Irwin D. / Ellman, Jonathan A. et al. | 1999
- 1441
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Synthesis and Dopamine Receptor Modulating Activity of Novel Peptidomimetics of l-Prolyl-l-leucyl-glycinamide Featuring α,α-Disubstituted Amino AcidsEvans, Margaret C. / Pradhan, Ashish / Venkatraman, Shankar / Ojala, William H. / Gleason, William B. / Mishra, Ram K. / Johnson, Rodney L. et al. | 1999
- 1441
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ARTICLES - Synthesis and Dopamine Receptor Modulating Activity of Novel Peptidomimetics of L-Prolyl-L-leucyl-glycinamide Featuring a,a-Disubstituted Amino AcidsEvans, Margaret C. et al. | 1999
- 1448
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Novel Cyclopropapyrroloindole Derivative (AT-3510) Bearing Methoxycarbonyl and Trifluoromethyl GroupsFukuda, Yasumichi / Furuta, Hirosuke / Kusama, Yoshie / Ebisu, Hiroyuki / Oomori, Yasuo / Terashima, Shiro et al. | 1999
- 1448
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ARTICLES - Novel Cyclopropapyrroloindole Derivative (AT-3510) Bearing Methoxycarbonyl and Trifluoromethyl GroupsFukuda, Yasumichi et al. | 1999
- 1459
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Antineoplastic Agents. 410. Asymmetric Hydroxylation of trans-Combretastatin A-4Pettit, George R. / Toki, Brian E. / Herald, Delbert L. / Boyd, Michael R. / Hamel, Ernest / Pettit, Robin K. / Chapuis, J. Charles et al. | 1999
- 1459
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ARTICLES - Antineoplastic Agents. 410. Asymmetric Hydroxylation of trans-Combretastatin A-4Pettit, George R. et al. | 1999
- 1466
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ARTICLES - 5-Aryl-1,2,3,4-tetrahydrochromeno(3,4-f)quinolin-3-ones as a Novel Class of Nonsteroidal Progesterone Receptor Agonists: Effect of A-Ring ModificationZhi, Lin et al. | 1999
- 1466
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5-Aryl-1,2,3,4-tetrahydrochromeno[3,4-f]quinolin-3-ones as a Novel Class of Nonsteroidal Progesterone Receptor Agonists: Effect of A-Ring ModificationZhi, Lin / Tegley, Christopher M. / Marschke, Keith B. / Mais, Dale E. / Jones, Todd K. et al. | 1999
- 1473
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Bisphosphonate Prodrugs: Synthesis and in Vitro Evaluation of Novel Clodronic Acid Dianhydrides as Bioreversible Prodrugs of ClodronateAhlmark, Marko / Vepsäläinen, Jouko / Taipale, Hannu / Niemi, Riku / Järvinen, Tomi et al. | 1999
- 1473
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BRIEF ARTICLES - Bisphosphonate Prodrugs: Synthesis and in Vitro Evaluation of Novel Clodronic Acid Dianhydrides as Bioreversible Prodrugs of ClodronateAhlmark, Marko et al. | 1999
- 1477
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Synthesis and Antimalarial Activity of 11 Dispiro-1,2,4,5-tetraoxane Analogues of WR 148999. 7,8,15,16-Tetraoxadispiro[5.2.5.2]hexadecanes Substituted at the 1 and 10 Positions with Unsaturated and Polar Functional GroupsDong, Yuxiang / Matile, Hugues / Chollet, Jacques / Kaminsky, Ronald / Wood, James K. / Vennerstrom, Jonathan L. et al. | 1999
- 1477
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BRIEF ARTICLES - Synthesis and Antimalarial Activity of 11 Dispiro-1,2,4,5-tetraoxane Analogues of WR 148999. 7,8,15,16-Tetraoxadispiro(5.2.5.2)hexadecanes Substituted at the 1 and 10 Positions with Unsaturated and Polar Functional GroupsDong, Yuxiang et al. | 1999