Structure-Activity Profiles of Complex Biantennary Glycans with Core Fucosylation and with-without Additional a2,3-a2,6 Sialylation: Synthesis of Neoglycoproteins and Their Properties in Lectin Assays, Cell Binding, and Organ Uptake (English)
- New search for: Unverzagt, C.
- New search for: Unverzagt, C.
- New search for: Andre, S.
- New search for: Seifert, J.
- New search for: Kojima, S.
- New search for: Fink, C.
- New search for: Srikrishna, G.
- New search for: Freeze, H.
- New search for: Kayser, K.
- New search for: Gabius, H.-J.
In:
Journal of medicinal chemistry
;
45
, 2
; 478-491
;
2002
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ISSN:
- Article (Journal) / Print
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Title:Structure-Activity Profiles of Complex Biantennary Glycans with Core Fucosylation and with-without Additional a2,3-a2,6 Sialylation: Synthesis of Neoglycoproteins and Their Properties in Lectin Assays, Cell Binding, and Organ Uptake
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Contributors:Unverzagt, C. ( author ) / Andre, S. / Seifert, J. / Kojima, S. / Fink, C. / Srikrishna, G. / Freeze, H. / Kayser, K. / Gabius, H.-J.
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Published in:Journal of medicinal chemistry ; 45, 2 ; 478-491
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Publisher:
- New search for: American Chemical Society
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Place of publication:Easton, Pa.
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Publication date:2002
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 770/4230
- New search for: 44.42 / 44.42
- Further information on Basic classification
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Keywords:
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Source:
Table of contents – Volume 45, Issue 2
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 251
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Looking for Selectivity among Cytochrome P450s InhibitorsCavalli, Andrea / Recanatini, Maurizio et al. | 2002
- 255
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Bacteriopurpurinimides: Highly Stable and Potent Photosensitizers for Photodynamic TherapyChen, Yihui / Graham, Andrew / Potter, William / Morgan, Janet / Vaughan, Lurine / Bellnier, David A. / Henderson, Barbara W. / Oseroff, Allan / Dougherty, Thomas J. / Pandey, Ravindra K. et al. | 2002
- 259
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Design of Substrate-Based Inhibitors of Human β-SecretaseTung, Jay S. / Davis, David L. / Anderson, John P. / Walker, Don E. / Mamo, Shumeye / Jewett, Nancy / Hom, Roy K. / Sinha, Sukanto / Thorsett, Eugene D. / John, Varghese et al. | 2002
- 259
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Design of Substrate-Based Inhibitors of Human b-SecretaseTung, J.S. et al. | 2002
- 263
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Inhibition of nNOS Activity in Rat Brain by Synthetic Kynurenines: Structure−Activity DependenceCamacho, Encarnación / León, Josefa / Carrión, Adoración / Entrena, Antonio / Escames, Germaine / Khaldy, Huda / Acuña-Castroviejo, Darío / Gallo, Miguel A. / Espinosa, Antonio et al. | 2002
- 275
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Antagonistic Effects of Human Cyclic MBP87-99 Altered Peptide Ligands in Experimental Allergic Encephalomyelitis and Human T-Cell ProliferationTselios, Theodore / Apostolopoulos, Vasso / Daliani, Ioanna / Deraos, Spyros / Grdadolnik, Simona / Mavromoustakos, Thomas / Melachrinou, Maria / Thymianou, Sotiria / Probert, Lesley / Mouzaki, Athanasia et al. | 2002
- 284
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Carbonic Anhydrase Activators: High Affinity Isozymes I, II, and IV Activators, Incorporating a b-Alanyl-histidine ScaffoldScozzafava, A. et al. | 2002
- 284
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Carbonic Anhydrase Activators: High Affinity Isozymes I, II, and IV Activators, Incorporating a β-Alanyl-histidine ScaffoldScozzafava, Andrea / Supuran, Claudiu T. et al. | 2002
- 292
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Structure−Activity Relationships of the Antimalarial Agent Artemisinin. 6. The Development of Predictive In Vitro Potency Models Using CoMFA and HQSAR MethodologiesAvery, Mitchell A. / Alvim-Gaston, Maria / Rodrigues, Carlos R. / Barreiro, Eliezer J. / Cohen, Fred E. / Sabnis, Yogesh A. / Woolfrey, John R. et al. | 2002
- 304
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Graphical Model for Estimating Oral Bioavailability of Drugs in Humans and Other Species from Their Caco-2 Permeability and in Vitro Liver Enzyme Metabolic Stability RatesMandagere, Arun K. / Thompson, Thomas N. / Hwang, Kin-Kai et al. | 2002
- 312
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Carbonic Anhydrase Inhibitors: Anticonvulsant Sulfonamides Incorporating Valproyl and Other Lipophilic MoietiesMasereel, Bernard / Rolin, Stéphanie / Abbate, Francesco / Scozzafava, Andrea / Supuran, Claudiu T. et al. | 2002
- 321
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Synthesis, Structure, and Activity of Diclofenac Analogues as Transthyretin Amyloid Fibril Formation InhibitorsOza, Vibha B. / Smith, Craig / Raman, Prakash / Koepf, Edward K. / Lashuel, Hilal A. / Petrassi, H. Mike / Chiang, Kyle P. / Powers, Evan T. / Sachettinni, James / Kelly, Jeffery W. et al. | 2002
- 333
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Elucidating the Inhibiting Mode of AHPBA Derivatives against HIV-1 Protease and Building Predictive 3D-QSAR ModelsHuang, Xaioqin / Xu, Liaosa / Luo, Xiaomin / Fan, Kangnian / Ji, Ruyun / Pei, Gang / Chen, Kaixian / Jiang, Hualiang et al. | 2002
- 344
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Pyrrolo[1,3]benzothiazepine-Based Atypical Antipsychotic Agents. Synthesis, Structure−Activity Relationship, Molecular Modeling, and Biological StudiesCampiani, Giuseppe / Butini, Stefania / Gemma, Sandra / Nacci, Vito / Fattorusso, Caterina / Catalanotti, Bruno / Giorgi, Gianluca / Cagnotto, Alfredo / Goegan, Mara / Mennini, Tiziana et al. | 2002
- 360
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Design, Synthesis, and Preliminary Pharmacological Evaluation of N-Acyl-3-aminoglutarimides as Broad-Spectrum Chemokine Inhibitors in Vitro and Anti-inflammatory Agents in VivoFox, David J. / Reckless, Jill / Warren, Stuart G. / Grainger, David J. et al. | 2002
- 371
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b-Strand Mimicking Macrocyclic Amino Acids: Templates for Protease Inhibitors with Antiviral ActivityGlenn, M.P. et al. | 2002
- 371
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β-Strand Mimicking Macrocyclic Amino Acids: Templates for Protease Inhibitors with Antiviral ActivityGlenn, Matthew P. / Pattenden, Leonard K. / Reid, Robert C. / Tyssen, David P. / Tyndall, Joel D. A. / Birch, Christopher J. / Fairlie, David P. et al. | 2002
- 382
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2-Amino-3-aroyl-4,5-alkylthiophenes: Agonist Allosteric Enhancers at Human A1 Adenosine ReceptorsTranberg, C. Elisabet / Zickgraf, Andrea / Giunta, Brian N. / Luetjens, Henning / Figler, Heidi / Murphree, Lauren J. / Falke, Ruediger / Fleischer, Holger / Linden, Joel / Scammells, Peter J. et al. | 2002
- 390
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C-7 Analogues of Progesterone as Potent Inhibitors of the P-Glycoprotein Efflux PumpLeonessa, Fabio / Kim, Ji-Hyun / Ghiorghis, Alem / Kulawiec, Robert J. / Hammer, Charles / Talebian, Abdelhossein / Clarke, Robert et al. | 2002
- 399
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New Approach to Pharmacophore Mapping and QSAR Analysis Using Inductive Logic Programming. Application to Thermolysin Inhibitors and Glycogen Phosphorylase b InhibitorsMarchand-Geneste, Nathalie / Watson, Kimberly A. / Alsberg, Bjørn K. / King, Ross D. et al. | 2002
- 410
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Synthesis, Biological Evaluation, and Quantitative Structure−Activity Relationship Analysis of New Schiff Bases of Hydroxysemicarbazide as Potential Antitumor Agents †Ren, Shijun / Wang, Rubin / Komatsu, Kenichi / Bonaz-Krause, Patricia / Zyrianov, Yegor / McKenna, Charles E. / Csipke, Csaba / Tokes, Zoltan A. / Lien, Eric J. et al. | 2002
- 420
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2,5‘-Disubstituted Adenosine Derivatives: Evaluation of Selectivity and Efficacy for the Adenosine A1, A2A, and A3 Receptorvan Tilburg, Erica W. / von Frijtag Drabbe Künzel, Jacobien / de Groote, Miriam / IJzerman, Ad P. et al. | 2002
- 430
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A New Type of Mixed Anhydride and Its Applications to the Synthesis of 7-Substituted 8-Chloro-5,5-dioxoimidazo[1,2-b][1,4,2]benzodithiazines with in Vitro Antitumor ActivityBrzozowski, Zdzisław / Sa̧czewski, Franciszek et al. | 2002
- 438
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Novel Spiropiperidines as Highly Potent and Subtype Selective s-Receptor Ligands. Part 1Maier, C.A. et al. | 2002
- 438
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Novel Spiropiperidines as Highly Potent and Subtype Selective σ-Receptor Ligands. Part 1Maier, Christoph A. / Wünsch, Bernhard et al. | 2002
- 449
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Water-Soluble, Core-Modified Porphyrins as Novel, Longer-Wavelength-Absorbing Sensitizers for Photodynamic Therapy. II. Effects of Core Heteroatoms and Meso-Substituents on Biological ActivityHilmey, David G. / Abe, Masako / Nelen, Marina I. / Stilts, Corey E. / Baker, Gary A. / Baker, Sheila N. / Bright, Frank V. / Davies, Sherry R. / Gollnick, Sandra O. / Oseroff, Allan R. et al. | 2002
- 462
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Synthesis and Characterization of a Series of Novel Monoacylated Ascorbic Acid Derivatives, 6-O-Acyl-2-O-a-d-glucopyranosyl-l-ascorbic Acids, as Skin AntioxidantsYamamoto, I. et al. | 2002
- 462
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Synthesis and Characterization of a Series of Novel Monoacylated Ascorbic Acid Derivatives, 6-O-Acyl-2-O-α-d-glucopyranosyl-l-ascorbic Acids, as Skin AntioxidantsYamamoto, Itaru / Tai, Akihiro / Fujinami, Yoshihito / Sasaki, Kenji / Okazaki, Shino et al. | 2002
- 469
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Radiolabeling and In Vivo Behavior of Copper-64-Labeled Cross-Bridged Cyclam LigandsSun, Xiankai / Wuest, Melinda / Weisman, Gary R. / Wong, Edward H. / Reed, David P. / Boswell, C. Andrew / Motekaitis, Ramunas / Martell, Arthur E. / Welch, Michael J. / Anderson, Carolyn J. et al. | 2002
- 478
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Structure-Activity Profiles of Complex Biantennary Glycans with Core Fucosylation and with-without Additional a2,3-a2,6 Sialylation: Synthesis of Neoglycoproteins and Their Properties in Lectin Assays, Cell Binding, and Organ UptakeUnverzagt, C. et al. | 2002
- 478
-
Structure−Activity Profiles of Complex Biantennary Glycans with Core Fucosylation and with/without Additional α2,3/α2,6 Sialylation: Synthesis of Neoglycoproteins and Their Properties in Lectin Assays, Cell Binding, and Organ Uptake †Unverzagt, Carlo / André, Sabine / Seifert, Joachim / Kojima, Shuji / Fink, Christian / Srikrishna, Geetha / Freeze, Hudson / Kayser, Klaus / Gabius, Hans-Joachim et al. | 2002
- 492
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4-(Phenylsulfonyl)piperidines: Novel, Selective, and Bioavailable 5-HT2A Receptor AntagonistsFletcher, Stephen R. / Burkamp, Frank / Blurton, Peter / Cheng, Susan K. F. / Clarkson, Robert / O'Connor, Desmond / Spinks, Daniel / Tudge, Matthew / van Niel, Monique B. / Patel, Smita et al. | 2002
- 504
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Carbonic Anhydrase Activators: Design of High Affinity Isozymes I, II, and IV Activators, Incorporating Tri-/Tetrasubstituted-pyridinium-azole MoietiesIlies, Monica / Banciu, Mircea D. / Ilies, Marc A. / Scozzafava, Andrea / Caproiu, Miron T. / Supuran, Claudiu T. et al. | 2002
- 511
-
Orally-Effective, Long-Acting Sorbitol Dehydrogenase Inhibitors: Synthesis, Structure−Activity Relationships, and in Vivo Evaluations of Novel Heterocycle-Substituted Piperazino-PyrimidinesChu-Moyer, Margaret Y. / Ballinger, William E. / Beebe, David A. / Berger, Richard / Coutcher, James B. / Day, Wesley W. / Li, Jiancheng / Mylari, Banavara L. / Oates, Peter J. / Weekly, R. Matthew et al. | 2002
- 529
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Aldisine Alkaloids from the Philippine Sponge Stylissa m assa Are Potent Inhibitors of Mitogen-Activated Protein Kinase Kinase-1 (MEK-1)Tasdemir, Deniz / Mallon, Robert / Greenstein, Michael / Feldberg, Larry R. / Kim, Steven C. / Collins, Karen / Wojciechowicz, Donald / Mangalindan, Gina C. / Concepción, Gisela P. / Harper, Mary Kay et al. | 2002
- 533
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Design, Synthesis, and Pharmacological Evaluation of New Farnesyl Protein Transferase InhibitorsHoussin, Raymond / Pommery, Jean / Salaün, Marie-Catherine / Deweer, Sophie / Goossens, Jean-François / Chavatte, Philippe / Hénichart, Jean-Pierre et al. | 2002
- 537
-
4‘-Arylpyrrolomorphinans: Effect of a Pyrrolo-N-benzyl Substituent in Enhancing δ-Opioid Antagonist ActivitySrivastava, Sanjay K. / Husbands, Stephen M. / Aceto, Mario D. / Miller, Carl N. / Traynor, John R. / Lewis, John W. et al. | 2002
- 537
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4'-Arylpyrrolomorphinans: Effect of a Pyrrolo-N-benzyl Substituent in Enhancing d-Opioid Antagonist ActivitySrivastava, S.K. et al. | 2002