Design and Synthesis of Motilin Antagonists Derived from the (1-4) Fragment of Porcine Motilin (English)
- New search for: Haramura, M.
- New search for: Haramura, M.
- New search for: Okamachi, A.
- New search for: Tsuzuki, K.
- New search for: Yogo, K.
- New search for: Ikuta, M.
- New search for: Kozono, T.
- New search for: Takanashi, H.
- New search for: Murayama, E.
In:
Journal of medicinal chemistry
;
45
, 3
; 670-675
;
2002
-
ISSN:
- Article (Journal) / Print
-
Title:Design and Synthesis of Motilin Antagonists Derived from the (1-4) Fragment of Porcine Motilin
-
Contributors:Haramura, M. ( author ) / Okamachi, A. / Tsuzuki, K. / Yogo, K. / Ikuta, M. / Kozono, T. / Takanashi, H. / Murayama, E.
-
Published in:Journal of medicinal chemistry ; 45, 3 ; 670-675
-
Publisher:
- New search for: American Chemical Society
-
Place of publication:Easton, Pa.
-
Publication date:2002
-
ISSN:
-
ZDBID:
-
Type of media:Article (Journal)
-
Type of material:Print
-
Language:English
- New search for: 770/4230
- New search for: 44.42 / 44.42
- Further information on Basic classification
-
Keywords:
-
Classification:
-
Source:
Table of contents – Volume 45, Issue 3
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 541
-
Designing Non-Peptide Peptidomimetics in the 21st Century: Inhibitors Targeting Conformational EnsemblesBursavich, Matthew G. / Rich, Daniel H. et al. | 2002
- 559
-
Design, Synthesis and Activity of Ascorbic Acid Prodrugs of Nipecotic, Kynurenic and Diclophenamic Acids, Liable to Increase Neurotropic ActivityManfredini, Stefano / Pavan, Barbara / Vertuani, Silvia / Scaglianti, Martina / Compagnone, Donatello / Biondi, Carla / Scatturin, Angelo / Tanganelli, Sergio / Ferraro, Luca / Prasad, Puttur et al. | 2002
- 563
-
Discovery of a 3-Amino-6-phenyl-pyridazine Derivative as a New Synthetic Antineuroinflammatory CompoundMirzoeva, Salida / Sawkar, Anu / Zasadzki, Magdalena / Guo, Ling / Velentza, Anastasia V. / Dunlap, Vincent / Bourguignon, Jean-Jacques / Ramstrom, Helena / Haiech, Jacques / Van Eldik, Linda J. et al. | 2002
- 567
-
Synthesis and Evaluation of Potent and Selective b3 Adrenergic Receptor Agonists Containing Acylsulfonamide, Sulfonylsulfonamide, and Sulfonylurea Carboxylic Acid IsosteresUehling, D.E. et al. | 2002
- 567
-
Synthesis and Evaluation of Potent and Selective β3 Adrenergic Receptor Agonists Containing Acylsulfonamide, Sulfonylsulfonamide, and Sulfonylurea Carboxylic Acid Isosteres †Uehling, David E. / Donaldson, Kelly H. / Deaton, David N. / Hyman, Clifton E. / Sugg, Elizabeth E. / Barrett, David G. / Hughes, Robert G. / Reitter, Barbara / Adkison, Kim K. / Lancaster, Mary E. et al. | 2002
- 584
-
Identification of a Second Binding Site in the Estrogen Receptorvan Hoorn, Willem P. et al. | 2002
- 590
-
Antitumor Polycyclic Acridines. 8.1 Synthesis and Telomerase-Inhibitory Activity of Methylated Pentacyclic Acridinium SaltsHeald, R.A. et al. | 2002
- 590
-
Antitumor Polycyclic Acridines. 8. Synthesis and Telomerase-Inhibitory Activity of Methylated Pentacyclic Acridinium SaltsHeald, Robert A. / Modi, Chetna / Cookson, Jenny C. / Hutchinson, Ian / Laughton, Charles A. / Gowan, Sharon M. / Kelland, Lloyd R. / Stevens, Malcolm F. G. et al. | 2002
- 598
-
Synthesis and Biological Activity of a Novel Class of Small Molecular Weight Peptidomimetic Competitive Inhibitors of Protein Tyrosine Phosphatase 1BLarsen, Scott D. / Barf, Tjeerd / Liljebris, Charlotta / May, Paul D. / Ogg, Derek / O'Sullivan, Theresa J. / Palazuk, Barbara J. / Schostarez, Heinrich J. / Stevens, F. Craig / Bleasdale, John E. et al. | 2002
- 623
-
Synthesis and Preliminary Characterization of a Novel Antiarrhythmic Compound (KB130015) with an Improved Toxicity Profile Compared with AmiodaroneCarlsson, Bo / Singh, B. N. / Temciuc, Marcel / Nilsson, Stefan / Li, Yi-Lin / Mellin, Charlotta / Malm, Johan et al. | 2002
- 631
-
Design, Synthesis, and Evaluation of Novel 2-Substituted 3-Hydroxypyridin-4-ones: Structure−Activity Investigation of Metalloenzyme Inhibition by Iron Chelators §Liu, Zu D. / Kayyali, Reem / Hider, Robert C. / Porter, John B. / Theobald, Anthony E. et al. | 2002
- 640
-
Synthesis and Optimization of a New Family of Type 3 17β-Hydroxysteroid Dehydrogenase Inhibitors by Parallel Liquid-Phase ChemistryMaltais, René / Luu-The, Van / Poirier, Donald et al. | 2002
- 640
-
Synthesis and Optimization of a New Family of Type 3 17b-Hydroxysteroid Dehydrogenase Inhibitors by Parallel Liquid-Phase ChemistryMaltais, R. et al. | 2002
- 654
-
Expansion of Structure−Activity Studies of Piperidine Analogues of 1-[2-(Diphenylmethoxy)ethyl]-4-(3-phenylpropyl)piperazine (GBR 12935) Compounds by Altering Substitutions in the N-Benzyl Moiety and Behavioral Pharmacology of Selected MoleculesDutta, Aloke K. / Davis, Matthew C. / Fei, Xiang-Shu / Beardsley, Patrick M. / Cook, Charles D. / Reith, Maarten. E. A. et al. | 2002
- 663
-
Correlation of the Antibacterial Activities of Cationic Peptide Antibiotics and Cationic Steroid AntibioticsDing, Bangwei / Guan, Qunying / Walsh, Joshua P. / Boswell, J. Scott / Winter, Tim W. / Winter, Erica S. / Boyd, Stephanie S. / Li, Chunhong / Savage, Paul B. et al. | 2002
- 663
-
Correlation of the Antibacterial Activities of Cationic Peptide Antibiotics and Cationic Steroid Antibiotics1Ding, B. et al. | 2002
- 670
-
Design and Synthesis of Motilin Antagonists Derived from the [1−4] Fragment of Porcine MotilinHaramura, Masayuki / Okamachi, Akira / Tsuzuki, Kouichi / Yogo, Kenji / Ikuta, Makoto / Kozono, Toshiro / Takanashi, Hisanori / Murayama, Eigoro et al. | 2002
- 676
-
Identification of Potent and Selective Mechanism-Based Inhibitors of the Cysteine Protease Cruzain Using Solid-Phase Parallel SynthesisHuang, Lily / Lee, Alice / Ellman, Jonathan A. et al. | 2002
- 685
-
Synthesis of 1-(3,4-Dihydroxy-5-nitrophenyl)-2-phenyl-ethanone and Derivatives as Potent and Long-Acting Peripheral Inhibitors of Catechol-O-methyltransferaseLearmonth, David A. / Vieira-Coelho, Maria A. / Benes, Jan / Alves, Paula C. / Borges, Nuno / Freitas, Ana P. / Soares-da-Silva, Patrício et al. | 2002
- 696
-
2,6-Di(ω-aminoalkyl)-2,5,6,7-tetrahydropyrazolo[3,4,5-mn]pyrimido[5,6,1-de]acridine-5,7-diones: Novel, Potent, Cytotoxic, and DNA-Binding AgentsAntonini, Ippolito / Polucci, Paolo / Magnano, Amelia / Gatto, Barbara / Palumbo, Manlio / Menta, Ernesto / Pescalli, Nicoletta / Martelli, Sante et al. | 2002
- 696
-
2,6-Di(w-aminoalkyl)-2,5,6,7-tetrahydropyrazolo(3,4,5-mn)pyrimido(5- ,6,1-de)acridine-5,7-diones: Novel, Potent, Cytotoxic, and DNA-Binding AgentsAntonini, I. et al. | 2002
- 703
-
Novel Mycophenolic Adenine Bis(phosphonate) Analogues As Potential Differentiation Agents against Human Leukemia1Pankiewicz, K.W. et al. | 2002
- 703
-
Novel Mycophenolic Adenine Bis(phosphonate) Analogues As Potential Differentiation Agents against Human LeukemiaPankiewicz, Krzysztof W. / Lesiak-Watanabe, Krystyna B. / Watanabe, Kyoichi A. / Patterson, Steven E. / Jayaram, Hiremagalur N. / Yalowitz, Joel A. / Miller, Michael D. / Seidman, Michael / Majumdar, Alokes / Prehna, Gerd et al. | 2002
- 713
-
Evaluation of the Dmt−Tic Pharmacophore: Conversion of a Potent δ-Opioid Receptor Antagonist into a Potent δ Agonist and Ligands with Mixed PropertiesBalboni, Gianfranco / Guerrini, Remo / Salvadori, Severo / Bianchi, Clementina / Rizzi, Daniela / Bryant, Sharon D. / Lazarus, Lawrence H. et al. | 2002
- 713
-
Evaluation of the Dmt-Tic Pharmacophore: Conversion of a Potent d-Opioid Receptor Antagonist into a Potent d Agonist and Ligands with Mixed PropertiesBalboni, G. et al. | 2002
- 721
-
Novel Angular Benzophenazines: Dual Topoisomerase I and Topoisomerase II Inhibitors as Potential Anticancer AgentsVicker, Nigel / Burgess, Luke / Chuckowree, Irina S. / Dodd, Rory / Folkes, Adrian J. / Hardick, David J. / Hancox, Timothy C. / Miller, Warren / Milton, John / Sohal, Sukhjit et al. | 2002
- 740
-
Structure−Activity Relationships for Pyrido-, Imidazo-, Pyrazolo-, Pyrazino-, and Pyrrolophenazinecarboxamides as Topoisomerase-Targeted Anticancer AgentsGamage, Swarna A. / Spicer, Julie A. / Rewcastle, Gordon W. / Milton, John / Sohal, Sukhjit / Dangerfield, Wendy / Mistry, Prakash / Vicker, Nigel / Charlton, Peter A. / Denny, William A. et al. | 2002
- 744
-
Antitumor Benzothiazoles. 16.1 Synthesis and Pharmaceutical Properties of Antitumor 2-(4-Aminophenyl)benzothiazole Amino Acid ProdrugsHutchinson, I. et al. | 2002
- 744
-
Antitumor Benzothiazoles. 16. Synthesis and Pharmaceutical Properties of Antitumor 2-(4-Aminophenyl)benzothiazole Amino Acid ProdrugsHutchinson, Ian / Jennings, Sharon A. / Vishnuvajjala, B. Rao / Westwell, Andrew D. / Stevens, Malcolm F. G. et al. | 2002
- 748
-
New Neplanocin Analogues. 12. Alternative Synthesis and Antimalarial Effect of (6'R)-6'-C-Methylneplanocin A, a Potent AdoHcy Hydrolase Inhibitor1Shuto, S. et al. | 2002
- 748
-
New Neplanocin Analogues. 12. Alternative Synthesis and Antimalarial Effect of (6‘R)-6‘-C-Methylneplanocin A, a Potent AdoHcy Hydrolase InhibitorShuto, Satoshi / Minakawa, Noriaki / Niizuma, Satoshi / Kim, Hye-Sook / Wataya, Yusuke / Matsuda, Akira et al. | 2002
- 752
-
Synthesis and Comparative Molecular Field Analysis (CoMFA) of Symmetric and Nonsymmetric Cyclic Sulfamide HIV-1 Protease Inhibitors.Schaal, Wesley / Karlsson, Anna / Ahlsén, Göran / Lindberg, Jimmy / Andersson, Hans O. / Danielson, U. Helena / Classon, Björn / Unge, Torsten / Samuelsson, Bertil / Hultén, Johan et al. | 2002