Carbonic Anhydrase Inhibitors. A General Approach for the Preparation of Water-Soluble Sulfonamides Incorporating Polyamino-Polycarboxylate Tails and of Their Metal Complexes Possessing Long-Lasting, Topical Intraocular Pressure-Lowering Properties (English)
- New search for: Scozzafava, A.
- New search for: Scozzafava, A.
- New search for: Menabuoni, L.
- New search for: Mincione, F.
- New search for: Supuran, C.T.
In:
Journal of medicinal chemistry
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45
, 7
; 1466-1476
;
2002
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ISSN:
- Article (Journal) / Print
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Title:Carbonic Anhydrase Inhibitors. A General Approach for the Preparation of Water-Soluble Sulfonamides Incorporating Polyamino-Polycarboxylate Tails and of Their Metal Complexes Possessing Long-Lasting, Topical Intraocular Pressure-Lowering Properties
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Contributors:
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Published in:Journal of medicinal chemistry ; 45, 7 ; 1466-1476
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Publisher:
- New search for: American Chemical Society
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Place of publication:Easton, Pa.
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Publication date:2002
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 770/4230
- New search for: 44.42 / 44.42
- Further information on Basic classification
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Keywords:
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Source:
Table of contents – Volume 45, Issue 7
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1395
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Design, Synthesis, and Evaluation of Opioid Analogues with Non-Peptidic β-Turn Scaffold: Enkephalin and Endomorphin MimeticsEguchi, Masakatsu / Shen, Richard Y. W. / Shea, J. Paul / Lee, Min S. / Kahn, Michael et al. | 2002
- 1395
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Design, Synthesis, and Evaluation of Opioid Analogues with Non-Peptidic b-Turn Scaffold: Enkephalin and Endomorphin MimeticsEguchi, M. et al. | 2002
- 1399
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Toward Selective ERb Agonists for Central Nervous System Disorders: Synthesis and Characterization of Aryl BenzthiophenesSchopfer, U. et al. | 2002
- 1399
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Toward Selective ERβ Agonists for Central Nervous System Disorders: Synthesis and Characterization of Aryl BenzthiophenesSchopfer, Ulrich / Schoeffter, Philippe / Bischoff, Serge F. / Nozulak, Joachim / Feuerbach, Dominik / Floersheim, Philipp et al. | 2002
- 1402
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Identification of Novel Cyclooxygenase-2 Selective Inhibitors Using Pharmacophore ModelsPalomer, Albert / Cabré, Francesc / Pascual, Jaume / Campos, Joaquín / Trujillo, María A. / Entrena, Antonio / Gallo, Miguel A. / García, Lluïsa / Mauleón, David / Espinosa, Antonio et al. | 2002
- 1412
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Molecular Dynamics and Free Energy Analyses of Cathepsin D−Inhibitor Interactions: Insight into Structure-Based Ligand DesignHuo, Shuanghong / Wang, Junmei / Cieplak, Piotr / Kollman, Peter A. / Kuntz, Irwin D. et al. | 2002
- 1420
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Studies on the Mechanism of Hypoxic Selectivity in Copper Bis(Thiosemicarbazone) RadiopharmaceuticalsMaurer, Richard I. / Blower, Philip J. / Dilworth, Jonathan R. / Reynolds, Christopher A. / Zheng, Yifan / Mullen, Gregory E. D. et al. | 2002
- 1432
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Hydroxyethylamine Isostere of an HIV-1 Protease Inhibitor Prefers Its Amine to the Hydroxy Group in Binding to Catalytic Aspartates. A Synchrotron Study of HIV-1 Protease in Complex with a Peptidomimetic InhibitorDohnálek, Jan / Hašek, Jindřich / Dušková, Jarmila / Petroková, Hana / Hradilek, Martin / Souček, Milan / Konvalinka, Jan / Brynda, Jiří / Sedláček, Juraj / Fábry, Milan et al. | 2002
- 1439
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Structural Basis for the Glucocorticoid Response in a Mutant Human Androgen Receptor (ARccr) Derived from an Androgen-Independent Prostate CancerMatias, Pedro M. / Carrondo, Maria Arménia / Coelho, Ricardo / Thomaz, Monica / Zhao, Xiao-Yan / Wegg, Anja / Crusius, Kerstin / Egner, Ursula / Donner, Peter et al. | 2002
- 1447
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Molecular Interaction of the Antagonist N-(Piperidin-1-yl)-5-(4-chlorophenyl)-1- (2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide with the CB1 Cannabinoid ReceptorShim, Joong-Youn / Welsh, William J. / Cartier, Etienne / Edwards, James L. / Howlett, Allyn C. et al. | 2002
- 1460
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Modeling of Binding Modes and Inhibition Mechanism of Some Natural Ligands of Farnesyl Transferase Using Molecular DockingPedretti, Alessandro / Villa, Luigi / Vistoli, Giulio et al. | 2002
- 1466
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Carbonic Anhydrase Inhibitors. A General Approach for the Preparation of Water-Soluble Sulfonamides Incorporating Polyamino−Polycarboxylate Tails and of Their Metal Complexes Possessing Long-Lasting, Topical Intraocular Pressure-Lowering PropertiesScozzafava, Andrea / Menabuoni, Luca / Mincione, Francesco / Supuran, Claudiu T. et al. | 2002
- 1477
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Toward an Optimal Joint Recognition of the S1‘ Subsites of Endothelin Converting Enzyme-1 (ECE-1), Angiotensin Converting Enzyme (ACE), and Neutral Endopeptidase (NEP)Inguimbert, Nicolas / Coric, Pascale / Poras, Hervé / Meudal, Hervé / Teffot, Franck / Fournié-Zaluski, Marie-Claude / Roques, Bernard P. et al. | 2002
- 1487
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Synthesis and Structure−Activity Relationships of 3-Aryloxindoles: A New Class of Calcium-Dependent, Large Conductance Potassium (Maxi-K) Channel Openers with Neuroprotective PropertiesHewawasam, Piyasena / Erway, Matthew / Moon, Sandra L. / Knipe, Jay / Weiner, Harvey / Boissard, Christopher G. / Post-Munson, Debra J. / Gao, Qi / Huang, Stella / Gribkoff, Valentin K. et al. | 2002
- 1500
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1,8-Disubstituted Xanthine Derivatives: Synthesis of Potent A2B-Selective Adenosine Receptor AntagonistsHayallah, Alaa M. / Sandoval-Ramírez, Jesús / Reith, Ulrike / Schobert, Ulrike / Preiss, Birgit / Schumacher, Britta / Daly, John W. / Müller, Christa E. et al. | 2002
- 1511
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4-(4-Cycloalkyl-aryl-oxazol-5-yl)benzenesulfonamides as Selective Cyclooxygenase-2 Inhibitors: Enhancement of the Selectivity by Introduction of a Fluorine Atom and Identification of a Potent, Highly Selective, and Orally Active COX-2 Inhibitor JTE-5221Hashimoto, H. et al. | 2002
- 1511
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4-(4-Cycloalkyl/aryl-oxazol-5-yl)benzenesulfonamides as Selective Cyclooxygenase-2 Inhibitors: Enhancement of the Selectivity by Introduction of a Fluorine Atom and Identification of a Potent, Highly Selective, and Orally Active COX-2 Inhibitor JTE-522Hashimoto, Hiromasa / Imamura, Katsuaki / Haruta, Jun-ichi / Wakitani, Korekiyo et al. | 2002
- 1518
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Novel 5-Substituted 2,4-Thiazolidinedione and 2,4-Oxazolidinedione Derivatives as Insulin Sensitizers with Antidiabetic ActivitiesMomose, Yu / Maekawa, Tsuyoshi / Yamano, Tohru / Kawada, Mitsuru / Odaka, Hiroyuki / Ikeda, Hitoshi / Sohda, Takashi et al. | 2002
- 1535
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Synthesis and Biological Evaluation of Cycloalkylidene Carboxylic Acids as Novel Effectors of Ras/Raf InteractionFriese, Anke / Hell-Momeni, Katja / Zündorf, Ilse / Winckler, Thomas / Dingermann, Theodor / Dannhardt, Gerd et al. | 2002