Specific inhibitors of Plasmodium falciparum thioredoxin reductase as potential antimalarial agents (English)
- New search for: Andricopulo, A.D.
- New search for: Andricopulo, A.D.
- New search for: Akoachere, M.B.
- New search for: Krogh, R.
- New search for: Nickel, C.
- New search for: Mcleish, M.J.
- New search for: Kenyon, G.L.
- New search for: Arscott, L.D.
- New search for: Williams, C.H.
- New search for: Davioud-Charvet, E.
In:
Bioorganic & medicinal chemistry letters
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16
, 8
; 2283-2292
;
2006
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ISSN:
- Article (Journal) / Print
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Title:Specific inhibitors of Plasmodium falciparum thioredoxin reductase as potential antimalarial agents
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Contributors:Andricopulo, A.D. ( author ) / Akoachere, M.B. / Krogh, R. / Nickel, C. / Mcleish, M.J. / Kenyon, G.L. / Arscott, L.D. / Williams, C.H. / Davioud-Charvet, E.
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Published in:Bioorganic & medicinal chemistry letters ; 16, 8 ; 2283-2292
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2006
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.42
- Further information on Basic classification
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Keywords:
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Source:
Table of contents – Volume 16, Issue 8
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
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Graphical contents list| 2006
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Fluorescent glycosidase inhibiting 1,5-dideoxy-1,5-iminoalditolsGreimel, Peter / Häusler, Herwig / Lundt, Inge / Rupitz, Karen / Stütz, Arnold E. / Tarling, Chris A. / Withers, Stephen G. / Wrodnigg, Tanja M. et al. | 2006
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A new class of bradykinin 1 receptor antagonists containing the piperidine acetic acid tetralin coreFotsch, Christopher / Biddlecome, Gloria / Biswas, Kaustav / Chen, Jian Jeff / D’Amico, Derin C. / Groneberg, Robert D. / Han, Nianhe Bruce / Hsieh, Feng-Yin / Kamassah, Augustus / Kumar, Gondi et al. | 2006
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Synthesis and SAR of heteroaryl-phenyl-substituted pyrazole derivatives as highly selective and potent canine COX-2 inhibitorsCheng, Hengmiao / Lundy DeMello, Kristin M. / Li, Jin / Sakya, Subas M. / Ando, Kazuo / Kawamura, K. / Kato, Tomoki / Rafka, Robert J. / Jaynes, Burton H. / Ziegler, Carl B. et al. | 2006
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N-thiolated 2-oxazolidinones: A new family of antibacterial agents for methicillin-resistant Staphylococcus aureus and Bacillus anthracisMishra, Rajesh Kumar / Revell, Kevin D. / Coates, Cristina M. / Turos, Edward / Dickey, Sonja / Lim, Daniel V. et al. | 2006
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N-Thiolated β-lactams: A new family of anti-Bacillus agentsTuros, Edward / Long, Timothy E. / Heldreth, Bart / Leslie, J. Michelle / Reddy, G. Suresh Kumar / Wang, Yang / Coates, Cristina / Konaklieva, Monika / Dickey, Sonja / Lim, Daniel V. et al. | 2006
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N-Thiolated b-lactams: A new family of anti-Bacillus agentsTuros, Edward et al. | 2006
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Synthesis and evaluation of novel heterocyclic inhibitors of GSK-3Smalley, Terrence L. Jr. / Peat, Andrew J. / Boucheron, Joyce A. / Dickerson, Scott / Garrido, Dulce / Preugschat, Frank / Schweiker, Stephanie L. / Thomson, Stephen A. / Wang, Tony Y. et al. | 2006
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Inhibitors of human mitotic kinesin Eg5: Characterization of the 4-phenyl-tetrahydroisoquinoline lead seriesTarby, Christine M. / Kaltenbach, Robert F. III / Huynh, Tram / Pudzianowski, Andrew / Shen, Henry / Ortega-Nanos, Marie / Sheriff, Steven / Newitt, John A. / McDonnell, Patricia A. / Burford, Neil et al. | 2006
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Synthesis, in vitro and in vivo evaluation of [O-methyl-11C] 2-{4-[4-(3-methoxyphenyl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]-triazine-3,5-dione: A novel agonist 5-HT1A receptor PET ligandPrabhakaran, Jaya / Parsey, Ramin V. / Majo, Vattoly J. / Hsiung, Shu-Chi / Milak, Matthew S. / Tamir, Hadassah / Simpson, Norman R. / Van Heertum, Ronald L. / Mann, J. John / Dileep Kumar, J.S. et al. | 2006
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Design, synthesis and biological evaluations of novel oxindoles as HIV-1 non-nucleoside reverse transcriptase inhibitors. Part IJiang, Tao / Kuhen, Kelli L. / Wolff, Karen / Yin, Hong / Bieza, Kimberly / Caldwell, Jeremy / Bursulaya, Badry / Wu, Tom Yao-Hsing / He, Yun et al. | 2006
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Design, synthesis, and biological evaluations of novel oxindoles as HIV-1 non-nucleoside reverse transcriptase inhibitors. Part 2Jiang, Tao / Kuhen, Kelli L. / Wolff, Karen / Yin, Hong / Bieza, Kimberly / Caldwell, Jeremy / Bursulaya, Badry / Tuntland, Tove / Zhang, Kanyin / Karanewsky, Donald et al. | 2006
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Synthesis of pyrazinamide Mannich bases and its antitubercular propertiesSriram, Dharmarajan / Yogeeswari, Perumal / Reddy, Sushma Pobba et al. | 2006
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Structure–activity relationship study between Ornithyl-Proline and Lysyl-Proline based tripeptidomimics as angiotensin-converting enzyme inhibitorsPavar, Mahesh Chand / Hanif, Kashif / Azam, Amir / lata, Sneh / Qadar Pasha, M.A. / Pasha, Santosh et al. | 2006
- 2122
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Cytotoxic activities of water-soluble chitosan derivatives with different degree of deacetylationJe, Jae-Young / Cho, Young-Sook / Kim, Se-Kwon et al. | 2006
- 2127
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Abacavir prodrugs: Microwave-assisted synthesis and their evaluation of anti-HIV activitiesSriram, Dharmarajan / Yogeeswari, Perumal / Myneedu, Naga Sirisha / Saraswat, Vivek et al. | 2006
- 2130
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Synthesis of Pseudomonas quorum-sensing autoinducer analogs and structural entities required for induction of apoptosis in macrophagesHorikawa, Manabu / Tateda, Kazuhiro / Tuzuki, Etsu / Ishii, Yoshikazu / Ueda, Chihiro / Takabatake, Tohru / Miyairi, Shinichi / Yamaguchi, Keizou / Ishiguro, Masaji et al. | 2006
- 2134
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Quaternary salts of 4,3′ and 4,4′ bis-pyridinium monooximes. Part 2: Synthesis and biological activitySrinivas Rao, Chennamaneni / Venkateswarlu, Vobalaboina / Achaiah, Garlapati et al. | 2006
- 2139
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Synthesis of novel benzofuran isoxazolines as protein tyrosine phosphatase 1B inhibitorsAhmad, Ghufran / Mishra, Pushpesh K. / Gupta, Prasoon / Yadav, Prem P. / Tiwari, Priti / Tamrakar, Akhilesh K. / Srivastava, Arvind K. / Maurya, Rakesh et al. | 2006
- 2144
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Synthesis and ocular effects of imidazole nitrolic acid and amidoxime estersOresmaa, Larisa / Kotikoski, Hanna / Haukka, Matti / Oksala, Olli / Pohjala, Esko / Vapaatalo, Heikki / Vainiotalo, Pirjo / Aulaskari, Paula et al. | 2006
- 2148
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Matrix compare analysis discriminates subtle structural differences in a family of novel antiproliferative agents, diaryl-3-hydroxy-2,3,3a,10a-tetrahydrobenzo[b]cycylopenta[e]azepine-4,10(1H,5H)-dionesKunick, Conrad / Bleeker, Carola / Prühs, Christian / Totzke, Frank / Schächtele, Christoph / Kubbutat, Michael H.G. / Link, Andreas et al. | 2006
- 2154
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Methylated β-cyclodextrin as P-gp modulators for deliverance of doxorubicin across an in vitro model of blood–brain barrierTilloy, Sébastien / Monnaert, Véronique / Fenart, Laurence / Bricout, Hervé / Cecchelli, Roméo / Monflier, Eric et al. | 2006
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Methylated b-cyclodextrin as P-gp modulators for deliverance of doxorubicin across an in vitro model of blood–brain barrierTilloy, Sébastien et al. | 2006
- 2158
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Structure-guided identification of novel VEGFR-2 kinase inhibitors via solution phase parallel synthesisTripathy, Rabindranath / Reiboldt, Alyssa / Messina, Patricia A. / Iqbal, Mohamed / Singh, Jasbir / Bacon, Edward R. / Angeles, Thelma S. / Yang, Shi X. / Albom, Mark S. / Robinson, Candy et al. | 2006
- 2163
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Synthesis and biological activity of diaryl ether inhibitors of malarial enoyl acyl carrier protein reductase. Part 2: 2′-Substituted triclosan derivativesFreundlich, Joel S. / Yu, Min / Lucumi, Edinson / Kuo, Mack / Tsai, Han-Chun / Valderramos, Juan-Carlos / Karagyozov, Luchezar / Jacobs, William R. Jr. / Schiehser, Guy A. / Fidock, David A. et al. | 2006
- 2170
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Isoquinoline derivatives as potential acetylcholinesterase inhibitorsMarkmee, Sutthatip / Ruchirawat, Somsak / Prachyawarakorn, Vilailak / Ingkaninan, Kornkanok / Khorana, Nantaka et al. | 2006
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Design and synthesis of 7H-pyrrolo[2,3-d]pyrimidines as focal adhesion kinase inhibitors. Part 1Choi, Ha-Soon / Wang, Zhicheng / Richmond, Wendy / He, Xiaohui / Yang, Kunyong / Jiang, Tao / Sim, Taebo / Karanewsky, Donald / Gu, Xiang-ju / Zhou, Vicki et al. | 2006
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Synthesis and antibacterial activities of chiral 1,3-oxazinan-2-one derivativesWang, Guijun / Ella-Menye, Jean-Rene / Sharma, Vibha et al. | 2006
- 2182
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Carbonic anhydrase inhibitors: Cloning and sulfonamide inhibition studies of a carboxyterminal truncated α-carbonic anhydrase from Helicobacter pyloriNishimori, Isao / Vullo, Daniela / Minakuchi, Tomoko / Morimoto, Kaori / Onishi, Saburo / Scozzafava, Andrea / Supuran, Claudiu T. et al. | 2006
- 2182
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Carbonic anhydrase inhibitors: Cloning and sulfonamide inhibition studies of a carboxyterminal truncated a-carbonic anhydrase from Helicobacter pyloriNishimori, Isao et al. | 2006
- 2189
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Design, synthesis, and biological evaluation of a scaffold for iGluR ligands based on the structure of (−)-dysiherbaineCohen, Jamie L. / Limon, Agenor / Miledi, Ricardo / Chamberlin, A. Richard et al. | 2006
- 2195
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- 2195
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Synthesis and biological evaluation of a-galactosylceramide (KRN7000) and isoglobotrihexosylceramide (iGb3)Xia, Chengfeng et al. | 2006
- 2200
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- 2205
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Factor VIIa inhibitors: A prodrug strategy to improve oral bioavailabilityRiggs, Jennifer R. / Kolesnikov, Aleksandr / Hendrix, John / Young, Wendy B. / Shrader, William D. / Vijaykumar, Dange / Stephens, Robin / Liu, Liang / Pan, Lin / Mordenti, Joyce et al. | 2006
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Evaluation of anti-inflammatory and antioxidant activities of mixed-ligand Cu(II) complexes of dien and its Schiff dibases with heterocyclic aldehydes and 2-amino-2-thiazolinePontiki, E. / Hadjipavlou-Litina, D. / Chaviara, A.T. / Bolos, C.A. et al. | 2006
- 2238
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The catecholic antioxidant piceatannol is an effective nitrosation inhibitor via an unusual double bond nitrationDe Lucia, Maria / Panzella, Lucia / Crescenzi, Orlando / Napolitano, Alessandra / Barone, Vincenzo / d’Ischia, Marco et al. | 2006
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Factor VIIa inhibitors: Improved pharmacokinetic parametersKolesnikov, Aleksandr / Rai, Roopa / Young, Wendy B. / Mordenti, Joyce / Liu, Liang / Torkelson, Steven / Shrader, William D. / Leahy, Ellen M. / Hu, Huiyong / Gjerstad, Erik et al. | 2006
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Design and structure–activity relationship of heterocyclic analogs of 4-amino-3-benzimidazol-2-ylhydroquinolin-2-ones as inhibitors of receptor tyrosine kinasesFrazier, Kelly / Jazan, Elisa / McBride, Christopher M. / Pecchi, Sabina / Renhowe, Paul A. / Shafer, Cynthia M. / Taylor, Clarke / Bussiere, Dirksen / He, Molly Min / Jansen, Johanna M. et al. | 2006
- 2252
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Analogues of N-hydroxycinnamoylphenalkylamides as inhibitors of human melanocyte-tyrosinaseOkombi, Sabrina / Rival, Delphine / Bonnet, Sébastien / Mariotte, Anne-Marie / Perrier, Eric / Boumendjel, Ahcène et al. | 2006
- 2256
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Pyridone derivatives as potent and selective VLA-4 integrin antagonistsWitherington, Jason / Bordas, Vincent / Gaiba, Alessandra / Green, Phil M. / Naylor, Antoinette / Parr, Nigel / Smith, David G. / Takle, Andrew K. / Ward, Robert W. et al. | 2006
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Potent blockers of the monocarboxylate transporter MCT1: Novel immunomodulatory compoundsGuile, S.D. / Bantick, J.R. / Cheshire, D.R. / Cooper, M.E. / Davis, A.M. / Donald, D.K. / Evans, R. / Eyssade, C. / Ferguson, D.D. / Hill, S. et al. | 2006
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Specific inhibitors of Plasmodium falciparum thioredoxin reductase as potential antimalarial agentsAndricopulo, A.D. / Akoachere, M.B. / Krogh, R. / Nickel, C. / McLeish, M.J. / Kenyon, G.L. / Arscott, L.D. / Williams, C.H. Jr. / Davioud-Charvet, E. / Becker, K. et al. | 2006
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Editorial Board| 2006
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Instructions to contributors| 2006