Optimizing thiadiazole analogues of resveratrol versus three chemopreventive targets (English)
- New search for: Mayhoub, Abdelrahman S.
- New search for: Mayhoub, Abdelrahman S.
- New search for: Marler, Laura
- New search for: Kondratyuk, Tamara P.
- New search for: Park, Eun-Jung
- New search for: Pezzuto, John M.
- New search for: Cushman, Mark
In:
Bioorganic & medicinal chemistry
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20
, 1
; 510-521
;
2012
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ISSN:
- Article (Journal) / Print
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Title:Optimizing thiadiazole analogues of resveratrol versus three chemopreventive targets
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Contributors:Mayhoub, Abdelrahman S. ( author ) / Marler, Laura / Kondratyuk, Tamara P. / Park, Eun-Jung / Pezzuto, John M. / Cushman, Mark
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Published in:Bioorganic & medicinal chemistry ; 20, 1 ; 510-521
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2012
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
- Further information on Basic classification
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Source:
Table of contents – Volume 20, Issue 1
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1
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Graphical contents list| 2011
- 16
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Nucleic acid probe containing fluorescent tricyclic base-linked acyclonucleoside for detection of single nucleotide polymorphismsFurukawa, Kinji / Hattori, Mayumi / Ohki, Tokimitsu / Kitamura, Yoshiaki / Kitade, Yukio / Ueno, Yoshihito et al. | 2011
- 25
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Solid-phase synthesis of 2′-hydroxychalcones. Effects on cell growth inhibition, cell cycle and apoptosis of human tumor cell linesNeves, Marta Perro / Cravo, Sara / Lima, Raquel T. / Vasconcelos, M. Helena / Nascimento, M. São José / Silva, Artur M.S. / Pinto, Madalena / Cidade, Honorina / Corrêa, Arlene G. et al. | 2011
- 25
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Solid-phase synthesis of 2prime-hydroxychalcones. Effects on cell growth inhibition, cell cycle and apoptosis of human tumor cell linesNeves, M. P. / Cravo, S. / Lima, R. T. / Vasconcelos, M. H. / Nascimento, M. S. / Silva, A. M. / Pinto, M. / Cidade, H. / Correa, A. G. et al. | 2012
- 34
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Synthesis and biological evaluation of (4H-1,2,4-triazol-4-yl)isoquinoline derivatives as selective glycine transporter 1 inhibitorsSugane, Takashi / Tobe, Takahiko / Hamaguchi, Wataru / Shimada, Itsuro / Maeno, Kyoichi / Miyata, Junji / Suzuki, Takeshi / Kimizuka, Tetsuya / Morita, Takuma / Sakamoto, Shuichi et al. | 2011
- 42
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Formation of ion-selective channel using cyclic tetrapeptidesSuga, Torao / Osada, Satoshi / Kodama, Hiroaki et al. | 2011
- 47
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Bisubstrate analogue inhibitors of 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase: New design with improved propertiesShi, Genbin / Shaw, Gary / Liang, Yu-He / Subburaman, Priadarsini / Li, Yue / Wu, Yan / Yan, Honggao / Ji, Xinhua et al. | 2011
- 58
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Novel pyrazolo[1,5-a]pyridines as p110a-selective PI3 kinase inhibitors: Exploring the benzenesulfonohydrazide SARKendall, J. D. / Giddens, A. C. / Tsang, K. Y. / Frederick, R. / Marshall, E. S. / Singh, R. / Lill, C. L. / Lee, W. J. / Kolekar, S. / Chao, M. et al. | 2012
- 58
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Novel pyrazolo[1,5-a]pyridines as p110α-selective PI3 kinase inhibitors: Exploring the benzenesulfonohydrazide SARKendall, Jackie D. / Giddens, Anna C. / Tsang, Kit Yee / Frédérick, Raphaël / Marshall, Elaine S. / Singh, Ripudaman / Lill, Claire L. / Lee, Woo-Jeong / Kolekar, Sharada / Chao, Mindy et al. | 2011
- 69
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Discovery of pyrazolo[1,5-a]pyridines as p110a-selective PI3 kinase inhibitorsKendall, J. D. / O'Connor, P. D. / Marshall, A. J. / Frederick, R. / Marshall, E. S. / Lill, C. L. / Lee, W. J. / Kolekar, S. / Chao, M. / Malik, A. et al. | 2012
- 69
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Discovery of pyrazolo[1,5-a]pyridines as p110α-selective PI3 kinase inhibitorsKendall, Jackie D. / O’Connor, Patrick D. / Marshall, Andrew J. / Frédérick, Raphaël / Marshall, Elaine S. / Lill, Claire L. / Lee, Woo-Jeong / Kolekar, Sharada / Chao, Mindy / Malik, Alisha et al. | 2011
- 86
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Investigation of substituted 6-aminohexanoates as skin penetration enhancersBrychtova, Katerina / Dvorakova, Lenka / Opatrilova, Radka / Raich, Ivan / Kacerova, Sandra / Placek, Lukas / Kalinowski, Danuta S. / Richardson, Des R. / Jampilek, Josef et al. | 2011
- 96
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Heavy metal-free 19F NMR probes for quantitative measurements of glutathione reductase activity using silica nanoparticles as a signal quencherTanaka, Kazuo / Kitamura, Narufumi / Chujo, Yoshiki et al. | 2011
- 101
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Novel bioactive metabolites of dipyrone (metamizol)Rogosch, Tobias / Sinning, Christian / Podlewski, Agnes / Watzer, Bernhard / Schlosburg, Joel / Lichtman, Aron H. / Cascio, Maria G. / Bisogno, Tiziana / Di Marzo, Vincenzo / Nüsing, Rolf et al. | 2011
- 108
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Synthesis and biological activities of 2-[(heteroaryl)methyl]imidazolinesSaczewski, Jaroslaw / Hudson, Alan / Scheinin, Mika / Rybczynska, Apolonia / Ma, Daqing / Saczewski, Franciszek / Laird, Shayna / Laurila, Jonne M. / Boblewski, Konrad / Lehmann, Artur et al. | 2011
- 117
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Synthesis, antiproliferative activity and genotoxicity of novel anthracene-containing aminophosphonates and a new anthracene-derived Schiff baseKraicheva, I. / Tsacheva, I. / Vodenicharova, E. / Tashev, E. / Tosheva, T. / Kril, A. / Topashka-Ancheva, M. / Iliev, I. / Gerasimova, Ts. / Troev, K. et al. | 2011
- 125
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Novel inhibitors of epidermal growth factor receptor: (4-(Arylamino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl)(1H-indol-2-yl)methanones and (1H-indol-2-yl)(4-(phenylamino)thieno[2,3-d]pyrimidin-6-yl)methanonesBeckers, Thomas / Sellmer, Andreas / Eichhorn, Emerich / Pongratz, Herwig / Schächtele, Christoph / Totzke, Frank / Kelter, Gerhard / Krumbach, Rebekka / Fiebig, Heinz-Herbert / Böhmer, Frank-D. et al. | 2011
- 137
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Synthesis of novel 3-cyclohexylpropanoic acid-derived nitrogen heterocyclic compounds and their evaluation for tuberculostatic activityGobis, Katarzyna / Foks, Henryk / Bojanowski, Krzysztof / Augustynowicz-Kopeć, Ewa / Napiórkowska, Agnieszka et al. | 2011
- 145
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Design, synthesis and the effect of 1,2,3-triazole sialylmimetic neoglycoconjugates on Trypanosoma cruzi and its cell surface trans-sialidaseCampo, Vanessa L. / Sesti-Costa, Renata / Carneiro, Zumira A. / Silva, João S. / Schenkman, Sergio / Carvalho, Ivone et al. | 2011
- 157
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Layer-by-Layer coated tyrosinase: An efficient and selective synthesis of catecholsGuazzaroni, Melissa / Crestini, Claudia / Saladino, Raffaele et al. | 2011
- 167
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Prediction of drug efficacy for cancer treatment based on comparative analysis of chemosensitivity and gene expression dataWan, Peng / Li, Qiyuan / Larsen, Jens Erik Pontoppidan / Eklund, Aron C. / Parlesak, Alexandr / Rigina, Olga / Nielsen, Søren Jensby / Björkling, Fredrik / Jónsdóttir, Svava Ósk et al. | 2011
- 177
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Design and synthesis of novel β-diketo derivatives as HIV-1 integrase inhibitorsHu, Liming / Zhang, Sulei / He, Xianzhuo / Luo, Zaigang / Wang, Xiaoli / Liu, Wei / Qin, Xuemei et al. | 2011
- 177
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Design and synthesis of novel b-diketo derivatives as HIV-1 integrase inhibitorsHu, L. / Zhang, S. / He, X. / Luo, Z. / Wang, X. / Liu, W. / Qin, X. et al. | 2012
- 183
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Design, synthesis and biological activity of sphingosine kinase 2 selective inhibitorsRaje, Mithun R. / Knott, Kenneth / Kharel, Yugesh / Bissel, Philippe / Lynch, Kevin R. / Santos, Webster L. et al. | 2011
- 195
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Synthesis, anti-inflammatory activity and ulcerogenic liability of novel nitric oxide donating/chalcone hybridsAbuo-Rahma, Gamal El-Din A.A. / Abdel-Aziz, Mohamed / Mourad, Mai A.E. / Farag, Hassan H. et al. | 2011
- 207
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Conjugation of a 3-(1H-phenanthro[9,10-d]imidazol-2-yl)-1H-indole intercalator to a triplex oligonucleotide and to a three-way junctionFatthalla, Maha I. / Elkholy, Yehya M. / Abbas, Nermeen S. / Mandour, Adel H. / Jørgensen, Per T. / Bomholt, Niels / Pedersen, Erik B. et al. | 2011
- 215
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N-4-t-Butylbenzyl 2-(4-methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure–activity relationships in the A-regionKim, Yong Soo / Kil, Min-Jung / Kang, Sang-Uk / Ryu, HyungChul / Kim, Myeong Seop / Cho, Yongsung / Bhondwe, Rahul S. / Thorat, Shivaji A. / Sun, Wei / Liu, Keliang et al. | 2011
- 225
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Discovery of inhibitors and substrates of brassinin hydrolase: Probing selectivity with dithiocarbamate bioisosteresPedras, M. Soledade C. / Minic, Zoran / Hossain, Sajjad et al. | 2011
- 234
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Synthesis, biological evaluation and molecular modeling of 1,2,3-triazole analogs of combretastatin A-1Akselsen, Øyvind W. / Odlo, Kristin / Cheng, Jing-Jy / Maccari, Giorgio / Botta, Maurizio / Hansen, Trond Vidar et al. | 2011
- 243
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Mefloquine–oxazolidine derivatives, derived from mefloquine and arenecarbaldehydes: In vitro activity including against the multidrug-resistant tuberculosis strain T113Gonçalves, Raoni S.B. / Kaiser, Carlos R. / Lourenço, Maria C.S. / Bezerra, Flavio A.F.M. / de Souza, Marcus V.N. / Wardell, James L. / Wardell, Solange M.S.V. / Henriques, Maria das Graças M.de O. / Costa, Thadeu et al. | 2011
- 249
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Stereochemical diversity of AI-2 analogs modulates quorum sensing in Vibrio harveyi and Escherichia coliRui, Fabio / Marques, João C. / Miller, Stephen T. / Maycock, Christopher D. / Xavier, Karina B. / Ventura, M. Rita et al. | 2011
- 257
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Synthesis, radiofluorination and pharmacological evaluation of a fluoromethyl spirocyclic PET tracer for central σ1 receptors and comparison with fluoroalkyl homologsMaisonial, Aurélie / Große Maestrup, Eva / Wiese, Christian / Hiller, Achim / Schepmann, Dirk / Fischer, Steffen / Deuther-Conrad, Winnie / Steinbach, Jörg / Brust, Peter / Wünsch, Bernhard et al. | 2011
- 270
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NMR-based conformational analysis of sphingomyelin in bicellesYamaguchi, Toshiyuki / Suzuki, Takashi / Yasuda, Tomokazu / Oishi, Tohru / Matsumori, Nobuaki / Murata, Michio et al. | 2011
- 279
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Marine sponge Hymeniacidon sp. amphilectane metabolites potently inhibit rat brain microglia thromboxane B2 generationMayer, Alejandro M.S. / Avilés, Edward / Rodríguez, Abimael D. et al. | 2011
- 283
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Amide-modified prenylcysteine based Icmt inhibitors: Structure–activity relationships, kinetic analysis and cellular characterizationMajmudar, Jaimeen D. / Hodges-Loaiza, Heather B. / Hahne, Kalub / Donelson, James L. / Song, Jiao / Shrestha, Liza / Harrison, Marietta L. / Hrycyna, Christine A. / Gibbs, Richard A. et al. | 2011
- 296
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Quantitative structure–activity relationships of 1,3,4-thiadiazol-2(3H)-ones and 1,3,4-oxadiazol-2(3H)-ones as human protoporphyrinogen oxidase inhibitorsZuo, Yang / Yang, Sheng-Gang / Jiang, Li-Li / Hao, Ge-Fei / Wang, Zhi-Fang / Wu, Qiong-You / Xi, Zhen / Yang, Guang-Fu et al. | 2011
- 305
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Radiosynthesis of [13N]dantrolene, a positron emission tomography probe for breast cancer resistant protein, using no-carrier-added [13N]ammoniaKumata, Katsushi / Ogawa, Masanao / Takei, Makoto / Fujinaga, Masayuki / Yoshida, Yuichiro / Nengaki, Nobuki / Fukumura, Toshimitsu / Suzuki, Kazutoshi / Zhang, Ming-Rong et al. | 2011
- 311
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Molecular docking studies of a phlorotannin, dieckol isolated from Ecklonia cava with tyrosinase inhibitory activityKang, Sung-Myung / Heo, Soo-Jin / Kim, Kil-Nam / Lee, Seung-Hong / Yang, Hae-Mi / Kim, Areum-Daseul / Jeon, You-Jin et al. | 2011
- 317
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Design and synthesis of 4,6-substituted-(diaphenylamino)quinazolines as potent EGFR inhibitors with antitumor activityLi, Huan-Qiu / Li, Dong-Dong / Lu, Xiang / Xu, Yun-Yun / Zhu, Hai-Liang et al. | 2011
- 324
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A fluorous and click approach for screening potential PET probes: Evaluation of potential hypoxia biomarkersBejot, Romain / Carroll, Laurence / Bhakoo, Kishore / Declerck, Jérôme / Gouverneur, Veronique et al. | 2011
- 330
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Studies of anti-fibrillogenic activity of phthalocyanines of zirconium containing out-of-plane ligandsKovalska, Vladyslava / Losytskyy, Mykhaylo / Chernii, Viktor / Volkova, Kateryna / Tretyakova, Iryna / Cherepanov, Vsevolod / Yarmoluk, Sergiy / Volkov, Sergiy et al. | 2011
- 335
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Persipeptides A and B, two cyclic peptides from Streptomyces sp. UTMC 1154Mohammadipanah, Fatemeh / Matasyoh, Josphat / Hamedi, Javad / Klenk, Hans-Peter / Laatsch, Hartmut et al. | 2011
- 340
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Reactive metabolites of desipramine and clomipramine: The kinetics of formation and reactivity with DNAKorobkova, Ekaterina A. / Nemeth, John / Cadougan, Mikeisha / Venkatratnam, Abhishek / Bassit, Mohanram / Azar, Nikolay et al. | 2011
- 346
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Investigation of chalcones and benzochalcones as inhibitors of breast cancer resistance proteinJuvale, Kapil / Pape, Veronika F.S. / Wiese, Michael et al. | 2011
- 356
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Design, synthesis, and biological evaluation of novel (1-thioxo-1,2,3,4-tetrahydro-b-carbolin-9-yl)acetic acids as selective inhibitors for AKR1B1Minehira, D. / Takeda, D. / Urata, H. / Kato, A. / Adachi, I. / Wang, X. / Matsuya, Y. / Sugimoto, K. / Takemura, M. / Endo, S. et al. | 2012
- 356
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Design, synthesis, and biological evaluation of novel (1-thioxo-1,2,3,4-tetrahydro-β-carbolin-9-yl)acetic acids as selective inhibitors for AKR1B1Minehira, Daisuke / Takeda, Daisuke / Urata, Hirokazu / Kato, Atsushi / Adachi, Isao / Wang, Xu / Matsuya, Yuji / Sugimoto, Kenji / Takemura, Mayuko / Endo, Satoshi et al. | 2011
- 368
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Structure-based redesign of an edema toxin inhibitorChen, Deliang / Ma, Lili / Kanalas, John J. / Gao, Jian / Pawlik, Jennifer / Jimenez, Maria Estrella / Walter, Mary A. / Peterson, Johnny W. / Gilbertson, Scott R. / Schein, Catherine H. et al. | 2011
- 377
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Elaborate ligand-based modeling and subsequent synthetic exploration unveil new nanomolar Ca2+/calmodulin-dependent protein kinase II inhibitory leadsShahin, Rand / Taha, Mutasem O. et al. | 2011
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Modification of HIV-1 reverse transcriptase and integrase activity by gold(III) complexes in direct biochemical assaysMphahlele, Morore / Papathanasopoulos, Maria / Cinellu, Maria Agostina / Coyanis, Mabel / Mosebi, Salerwe / Traut, Telisha / Modise, Refilwe / Coates, Judy / Hewer, Raymond et al. | 2011
- 408
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Prediction of inhibitory activities of Hsp90 inhibitorsSwuec, Paolo / Barlow, David J. et al. | 2011
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Synthesis of 5-aryl-1,4-benzodiazepine derivatives attached in resorcinaren-PAMAM dendrimers and their anti-cancer activityCortez-Maya, Sandra / Hernández-Ortega, Simón / Ramírez-Apan, Teresa / Lijanova, Irina V. / Martínez-García, Marcos et al. | 2011
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Design, synthesis, and biological evaluation of 4-phenylpyrrole derivatives as novel androgen receptor antagonistsYamamoto, Satoshi / Matsunaga, Nobuyuki / Hitaka, Takenori / Yamada, Masami / Hara, Takahito / Miyazaki, Junichi / Santou, Takashi / Kusaka, Masami / Yamaoka, Masuo / Kanzaki, Naoyuki et al. | 2011
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Synthetic studies of bi-fluorescence-labeled maltooligosaccharides as substrates for α-amylase on the basis of fluorescence resonance energy transfer (FRET)Oka, Hiroyuki / Koyama, Tetsuo / Hatano, Ken / Matsuoka, Koji et al. | 2011
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Synthetic studies of bi-fluorescence-labeled maltooligosaccharides as substrates for a-amylase on the basis of fluorescence resonance energy transfer (FRET)Oka, H. / Koyama, T. / Hatano, K. / Matsuoka, K. et al. | 2012
- 446
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Synthesis and biological evaluation of sialic acid derivatives containing a long hydrophobic chain at the anomeric position and their C-5 linked polymers as potent influenza virus inhibitorsSuzuki, Kaori / Koyama, Tetsuo / Yingsakmongkon, Sangchai / Suzuki, Yasuo / Hatano, Ken / Matsuoka, Koji et al. | 2011
- 455
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Bivalent molecular probes for dopamine D 2-like receptorsHuber, Daniela / Löber, Stefan / Hübner, Harald / Gmeiner, Peter et al. | 2011
- 467
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The design, synthesis and biological evaluations of C-6 or C-7 substituted 2-hydroxyisoquinoline-1,3-diones as inhibitors of hepatitis C virusChen, Yue-Lei / Tang, Jing / Kesler, Matthew J. / Sham, Yuk Y. / Vince, Robert / Geraghty, Robert J. / Wang, Zhengqiang et al. | 2011
- 480
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Efficient microwave-assisted synthesis, antibacterial activity and high fluorescence of 5 benzimidazolyl-2prime-deoxyuridinesKrim, J. / Grunewald, C. / Taourirte, M. / Engels, J. W. et al. | 2012
- 480
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Efficient microwave-assisted synthesis, antibacterial activity and high fluorescence of 5 benzimidazolyl-2′-deoxyuridinesKrim, Jamal / Grünewald, Christian / Taourirte, Moha / Engels, Joachim W. et al. | 2011
- 487
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Design, synthesis, and evaluation of novel small molecule inhibitors of the influenza virus protein NS1Jablonski, Joseph J. / Basu, Dipwanita / Engel, Daniel A. / Geysen, H. Mario et al. | 2011
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The discovery of UK-369003, a novel PDE5 inhibitor with the potential for oral bioavailability and dose-proportional pharmacokineticsRawson, David J. / Ballard, Stephen / Barber, Christopher / Barker, Laura / Beaumont, Kevin / Bunnage, Mark / Cole, Susan / Corless, Martin / Denton, Stephen / Ellis, David et al. | 2011
- 510
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Optimizing thiadiazole analogues of resveratrol versus three chemopreventive targetsMayhoub, Abdelrahman S. / Marler, Laura / Kondratyuk, Tamara P. / Park, Eun-Jung / Pezzuto, John M. / Cushman, Mark et al. | 2011
- 521
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Synthesis and evaluation of novel 4-[(3H,3aH,6aH)-3-phenyl)-4,6-dioxo-2-phenyldihydro-2H-pyrrolo[3,4-d]isoxazol-5(3H,6H,6aH)-yl]benzoic acid derivatives as potent acetylcholinesterase inhibitors and anti-amnestic agentsAnand, Preet / Singh, Baldev et al. | 2011
- 531
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Corrigendum to “Chemistry of ecteinascidins. Part 3: Preparation of 2′-N-acyl derivatives of ecteinascidin 770 and evaluation of cytotoxicity” [Bioorg. Med. Chem. 19 (2011) 4421–4436]Saktrakulkla, Panithi / Toriumi, Satoru / Tsujimoto, Mitsuhiro / Patarapanich, Chamnan / Suwanborirux, Khanit / Saito, Naoki et al. | 2011
- 531
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Corrigendum to "Chemistry of ecteinascidins. Part 3: Preparation of 2prime-N-acyl derivatives of ecteinascidin 770 and evaluation of cytotoxicity" [Bioorg. Med. Chem. 19 (2011) 4421-4436]Saktrakulkla, P. / Toriumi, S. / Tsujimoto, M. / Patarapanich, C. / Suwanborirux, K. / Saito, N. et al. | 2012
- IFC
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Editorial board| 2011