Optimization of the aromatase inhibitory activities of pyridylthiazole analogues of resveratrol (English)
- New search for: Mayhoub, Abdelrahman S.
- New search for: Mayhoub, Abdelrahman S.
- New search for: Marler, Laura
- New search for: Kondratyuk, Tamara P.
- New search for: Park, Eun-Jung
- New search for: Pezzuto, John M.
- New search for: Cushman, Mark
In:
Bioorganic & medicinal chemistry
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20
, 7
; 2427-2435
;
2012
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ISSN:
- Article (Journal) / Print
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Title:Optimization of the aromatase inhibitory activities of pyridylthiazole analogues of resveratrol
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Contributors:Mayhoub, Abdelrahman S. ( author ) / Marler, Laura / Kondratyuk, Tamara P. / Park, Eun-Jung / Pezzuto, John M. / Cushman, Mark
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Published in:Bioorganic & medicinal chemistry ; 20, 7 ; 2427-2435
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2012
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
- Further information on Basic classification
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Keywords:
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Classification:
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Source:
Table of contents – Volume 20, Issue 7
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 2191
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Graphical contents list| 2012
- 2199
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C–C bond formation at C-2 of a quinoline ring: Synthesis of 2-(1H-indol-3-yl)quinoline-3-carbonitrile derivatives as a new class of PDE4 inhibitorsKumar, K. Shiva / Kiran Kumar, S. / Yogi Sreenivas, B. / Gorja, Dhilli Rao / Kapavarapu, Ravikumar / Rambabu, D. / Rama Krishna, G. / Reddy, C. Malla / Basaveswara Rao, M.V. / Parsa, Kishore V.L. et al. | 2012
- 2208
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Mutation of active site residues Asn67 to Ile, Gln92 to Val and Leu204 to Ser in human carbonic anhydrase II: Influences on the catalytic activity and affinity for inhibitorsTurkoglu, Sumeyye / Maresca, Alfonso / Alper, Meltem / Kockar, Feray / Işık, Semra / Sinan, Selma / Ozensoy, Ozen / Arslan, Oktay / Supuran, Claudiu T. et al. | 2012
- 2214
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Generation and exploration of new classes of antitubercular agents: The optimization of oxazolines, oxazoles, thiazolines, thiazoles to imidazo[1,2-a]pyridines and isomeric 5,6-fused scaffoldsMoraski, Garrett C. / Markley, Lowell D. / Chang, Mayland / Cho, Sanghyun / Franzblau, Scott G. / Hwang, Chang Hwa / Boshoff, Helena / Miller, Marvin J. et al. | 2012
- 2221
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Synthesis and evaluation of fluorobenzoylated di- and tripeptides as inhibitors of cyclooxygenase-2 (COX-2)Sharma, Sai Kiran / Al-Hourani, Baker Jawabrah / Wuest, Melinda / Mane, Jonathan Y. / Tuszynski, Jack / Baracos, Vickie / Suresh, Mavanur / Wuest, Frank et al. | 2012
- 2227
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Perturbing pro-survival proteins using quinoxaline derivatives: A structure–activity relationship studyRajule, Rajkumar / Bryant, Vashti C. / Lopez, Hernando / Luo, Xu / Natarajan, Amarnath et al. | 2012
- 2235
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Discovery of novel prostaglandin analogs as potent and selective EP2/EP4 dual agonistsKambe, Tohru / Maruyama, Toru / Nakai, Yoshihiko / Yoshida, Hideyuki / Oida, Hiroji / Maruyama, Takayuki / Abe, Nobutaka / Nishiura, Akio / Nakai, Hisao / Toda, Masaaki et al. | 2012
- 2252
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Synthesis, antimicrobial and anticancer activities of a novel series of diphenyl 1-(pyridin-3-yl)ethylphosphonatesAbdel-Megeed, Mohamed F. / Badr, Badr E. / Azaam, Mohamed M. / El-Hiti, Gamal A. et al. | 2012
- 2259
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Favourable involvement of a2A-adrenoreceptor antagonism in the I2-imidazoline binding sites-mediated morphine analgesia enhancementMammoli, V. / Bonifazi, A. / Del Bello, F. / Diamanti, E. / Giannella, M. / Hudson, A. L. / Mattioli, L. / Perfumi, M. / Piergentili, A. / Quaglia, W. et al. | 2012
- 2259
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Favourable involvement of α2A-adrenoreceptor antagonism in the I2-imidazoline binding sites-mediated morphine analgesia enhancementMammoli, Valerio / Bonifazi, Alessandro / Del Bello, Fabio / Diamanti, Eleonora / Giannella, Mario / Hudson, Alan L. / Mattioli, Laura / Perfumi, Marina / Piergentili, Alessandro / Quaglia, Wilma et al. | 2012
- 2266
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Novel coumarins and 2-thioxo-coumarins as inhibitors of the tumor-associated carbonic anhydrases IX and XIICarta, Fabrizio / Maresca, Alfonso / Scozzafava, Andrea / Supuran, Claudiu T. et al. | 2012
- 2274
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Impact of stereochemistry on the biological activity of novel oleandomycin derivativesBauer, Jurica / Vine, Mark / Čorić, Ilija / Bosnar, Martina / Pašalić, Ivanka / Turkalj, Gordana / Lazarevski, Gorjana / Čulić, Ognjen / Kragol, Goran et al. | 2012
- 2282
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Indeno[1,2-b]indole derivatives as a novel class of potent human protein kinase CK2 inhibitorsHundsdörfer, Claas / Hemmerling, Hans-Jörg / Götz, Claudia / Totzke, Frank / Bednarski, Patrick / Le Borgne, Marc / Jose, Joachim et al. | 2012
- 2290
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Antiarrhythmic properties of phenylpiperazine derivatives of phenytoin with α1-adrenoceptor affinitiesHandzlik, Jadwiga / Bajda, Marek / Zygmunt, Małgorzata / Maciąg, Dorota / Dybała, Małgorzata / Bednarski, Marek / Filipek, Barbara / Malawska, Barbara / Kieć-Kononowicz, Katarzyna et al. | 2012
- 2290
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Antiarrhythmic properties of phenylpiperazine derivatives of phenytoin with a1-adrenoceptor affinitiesHandzlik, J. / Bajda, M. / Zygmunt, M. / Maciag, D. / Dybala, M. / Bednarski, M. / Filipek, B. / Malawska, B. / Kiec-Kononowicz, K. et al. | 2012
- 2304
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Synthesis and P2Y2 receptor agonist activities of uridine 5prime-phosphonate analoguesVan Poecke, S. / Barrett, M. O. / Santhosh Kumar, T. / Sinnaeve, D. / Martins, J. C. / Jacobson, K. A. / Kendall Harden, T. / Van Calenbergh, S. et al. | 2012
- 2304
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Synthesis and P2Y2 receptor agonist activities of uridine 5′-phosphonate analoguesVan Poecke, Sara / Barrett, Matthew O. / Santhosh Kumar, T. / Sinnaeve, Davy / Martins, José C. / Jacobson, Kenneth A. / Kendall Harden, T. / Van Calenbergh, Serge et al. | 2012
- 2316
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The synthesis of ethacrynic acid thiazole derivatives as glutathione S-transferase pi inhibitorsLi, Ting / Liu, Guyue / Li, Hongcai / Yang, Xinmei / Jing, Yongkui / Zhao, Guisen et al. | 2012
- 2323
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In silico scaffold evaluation and solid phase approach to identify new gelatinase inhibitorsTopai, Alessandra / Breccia, Perla / Minissi, Franco / Padova, Alessandro / Marini, Stefano / Cerbara, Ilaria et al. | 2012
- 2338
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Design, synthesis, and biological evaluation of 4-arylmethyl-1-phenylpyrazole and 4-aryloxy-1-phenylpyrazole derivatives as novel androgen receptor antagonistsYamamoto, Satoshi / Tomita, Naoki / Suzuki, Yuri / Suzaki, Tomohiko / Kaku, Tomohiro / Hara, Takahito / Yamaoka, Masuo / Kanzaki, Naoyuki / Hasuoka, Atsushi / Baba, Atsuo et al. | 2012
- 2353
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2-Morpholinoisoflav-3-enes as flexible intermediates in the synthesis of phenoxodiol, isophenoxodiol, equol and analogues: Vasorelaxant properties, estrogen receptor binding and Rho/RhoA kinase pathway inhibitionTilley, Andrew J. / Zanatta, Shannon D. / Qin, Cheng Xue / Kim, In-Kyeom / Seok, Young-Mi / Stewart, Alastair / Woodman, Owen L. / Williams, Spencer J. et al. | 2012
- 2362
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Proteasome inhibitors for cancer therapyIqbal, Mohamed / Messina McLaughlin, Patricia A. / Dunn, Derek / Mallya, Satish / Husten, Jean / Ator, Mark A. / Chatterjee, Sankar et al. | 2012
- 2369
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Synthesis and structure–activity relationship of 4-amino-2-phenylpyrimidine derivatives as a series of novel GPR119 agonistsNegoro, Kenji / Yonetoku, Yasuhiro / Maruyama, Tatsuya / Yoshida, Shigeru / Takeuchi, Makoto / Ohta, Mitsuaki et al. | 2012
- 2376
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Tea catechins and flavonoids from the leaves of Camellia sinensis inhibit yeast alcohol dehydrogenaseManir, Md. Maniruzzaman / Kim, Jeong Kee / Lee, Byeong-Gon / Moon, Surk-Sik et al. | 2012
- 2382
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Synthesis of macrocyclic bisbibenzyl derivatives and their anticancer effects as anti-tubulin agentsJiang, Juan / Sun, Bin / Wang, Yan-yan / Cui, Min / Zhang, Li / Cui, Chang-zhi / Wang, Yan-feng / Liu, Xi-gong / Lou, Hong-xiang et al. | 2012
- 2392
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Design and synthesis of thiourea compounds that inhibit transmembrane anchored carbonic anhydrasesMoeker, Janina / Teruya, Kanae / Rossit, Sabine / Wilkinson, Brendan L. / Lopez, Marie / Bornaghi, Laurent F. / Innocenti, Alessio / Supuran, Claudiu T. / Poulsen, Sally-Ann et al. | 2012
- 2405
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New retinoid derivatives as back-ups of AdaroteneGiannini, Giuseppe / Brunetti, Tiziana / Battistuzzi, Gianfranco / Alloatti, Domenico / Quattrociocchi, Gianandrea / Cima, Maria Grazia / Merlini, Lucio / Dallavalle, Sabrina / Cincinelli, Raffaella / Nannei, Raffaella et al. | 2012
- 2416
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The synthesis of 2prime-methylseleno adenosine and guanosine 5prime-triphosphatesSantner, T. / Siegmund, V. / Marx, A. / Micura, R. et al. | 2012
- 2416
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The synthesis of 2′-methylseleno adenosine and guanosine 5′-triphosphatesSantner, Tobias / Siegmund, Vanessa / Marx, Andreas / Micura, Ronald et al. | 2012
- 2419
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1,3-Phenylene bis(ketoacid) derivatives as inhibitors of Escherichia coli dihydrodipicolinate synthaseBoughton, Berin A. / Hor, Lilian / Gerrard, Juliet A. / Hutton, Craig A. et al. | 2012
- 2427
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Optimization of the aromatase inhibitory activities of pyridylthiazole analogues of resveratrolMayhoub, Abdelrahman S. / Marler, Laura / Kondratyuk, Tamara P. / Park, Eun-Jung / Pezzuto, John M. / Cushman, Mark et al. | 2012
- 2435
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Intramolecular hydrogen bonding: A potential strategy for more bioavailable inhibitors of neuronal nitric oxide synthaseLabby, Kristin Jansen / Xue, Fengtian / Kraus, James M. / Ji, Haitao / Mataka, Jan / Li, Huiying / Martásek, Pavel / Roman, Linda J. / Poulos, Thomas L. / Silverman, Richard B. et al. | 2012
- 2444
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N 4-(3-Bromophenyl)-7-(substituted benzyl) pyrrolo[2,3-d]pyrimidines as potent multiple receptor tyrosine kinase inhibitors: Design, synthesis, and in vivo evaluationGangjee, Aleem / Zaware, Nilesh / Raghavan, Sudhir / Yang, Jie / Thorpe, Jessica E. / Ihnat, Michael A. et al. | 2012
- 2455
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Integrated structure-based activity prediction model of benzothiadiazines on various genotypes of HCV NS5b polymerase (1a, 1b and 4) and its application in the discovery of new derivativesIsmail, Mohamed A.H. / Abou El Ella, Dalal A. / Abouzid, Khaled A.M. / Mahmoud, Amr H. et al. | 2012
- 2479
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Corrigendum to “Generation of ‘Unnatural Natural Product’ library and identification of a small molecule inhibitor of XIAP” [Bioorg. Med. Chem. 19 (2011) 4377–4385]Kawamura, Tatsuro / Matsubara, Kohei / Otaka, Hitomi / Tashiro, Etsu / Shindo, Kazutoshi / Yanagita, Ryo C. / Irie, Kazuhiro / Imoto, Masaya et al. | 2012
- IFC
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Editorial board| 2012