Synthesis and structure-activity relationships of novel 9-oxime acylides with improved bactericidal activity (English)
- New search for: Han, Xu
- New search for: Han, Xu
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- New search for: Guo, Si-Yang
- New search for: Cushman, Mark
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In:
Bioorganic & medicinal chemistry
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23
, 19
; 6437-6453
;
2015
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ISSN:
- Article (Journal) / Print
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Title:Synthesis and structure-activity relationships of novel 9-oxime acylides with improved bactericidal activity
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Contributors:
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Published in:Bioorganic & medicinal chemistry ; 23, 19 ; 6437-6453
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2015
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ISSN:
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
- Further information on Basic classification
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Keywords:
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Source:
Table of contents – Volume 23, Issue 19
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 6229
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Graphical contents list| 2015
- 6237
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Synthesis of five and six-membered heterocycles bearing an arylpiperazinylalkyl side chain as orally active antinociceptive agentsVergelli, Claudia / Ciciani, Giovanna / Cilibrizzi, Agostino / Crocetti, Letizia / Di Cesare Mannelli, Lorenzo / Ghelardini, Carla / Guerrini, Gabriella / Iacovone, Antonella / Giovannoni, Maria Paola et al. | 2015
- 6246
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Novel inhibitors targeting PPM1D phosphatase potently suppress cancer cell proliferationOgasawara, Sari / Kiyota, Yuhei / Chuman, Yoshiro / Kowata, Ayano / Yoshimura, Fumihiko / Tanino, Keiji / Kamada, Rui / Sakaguchi, Kazuyasu et al. | 2015
- 6250
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Synthesis and biological evaluation of novel 7-substituted 3-(4-phenoxyphenyl)thieno[3,2-c]pyridin-4-amines as potent Bruton’s tyrosine kinase (BTK) inhibitorsXin, Minhang / Zhao, Xinge / Huang, Wei / Jin, Qiu / Wu, Gang / Wang, Yazhou / Tang, Feng / Xiang, Hua et al. | 2015
- 6258
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Development of N-hydroxybenzamide derivatives with indole-containing cap group as histone deacetylases inhibitorsLi, Xiaoyang / Wu, Jingde / Li, Xiaoguang / Mu, Weiwei / Liu, Xueliang / Jin, Yiming / Xu, Wenfang / Zhang, Yingjie et al. | 2015
- 6271
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Synthesis of new opioid derivatives with a propellane skeleton and their pharmacologies: Part 5, novel pentacyclic propellane derivatives with a 6-amide side chainNakajima, Ryo / Yamamoto, Naoshi / Hirayama, Shigeto / Iwai, Takashi / Saitoh, Akiyoshi / Nagumo, Yasuyuki / Fujii, Hideaki / Nagase, Hiroshi et al. | 2015
- 6280
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Discovery and SAR of novel pyrazolo[1,5-a]pyrimidines as inhibitors of CDK9Phillipson, Louisa J. / Segal, David H. / Nero, Tracy L. / Parker, Michael W. / Wan, Soo San / de Silva, Melanie / Guthridge, Mark A. / Wei, Andrew H. / Burns, Christopher J. et al. | 2015
- 6297
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Biological activity of N(4)-boronated derivatives of 2′-deoxycytidine, potential agents for boron-neutron capture therapyNizioł, Joanna / Uram, Łukasz / Szuster, Magdalena / Sekuła, Justyna / Ruman, Tomasz et al. | 2015
- 6305
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Synthesis, antiproliferative activity and possible mechanism of action of novel 2-acetamidobenzamides bearing the 2-phenoxy functionalityRaffa, Demetrio / Maggio, Benedetta / Plescia, Fabiana / Cascioferro, Stella / Raimondi, Maria Valeria / Cancemi, Gabriella / D’Anneo, Antonella / Lauricella, Marianna / Cusimano, Maria Grazia / Bai, Ruoli et al. | 2015
- 6317
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Synthesis, electronic properties, antioxidant and antibacterial activity of some new benzimidazolesMavrova, Anelia Ts. / Yancheva, Denitsa / Anastassova, Neda / Anichina, Kamelya / Zvezdanovic, Jelena / Djordjevic, Aleksandra / Markovic, Dejan / Smelcerovic, Andrija et al. | 2015
- 6327
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Isolation and anticancer, anthelminthic, and antiviral (HIV) activity of acylphloroglucinols, and regioselective synthesis of empetrifranzinans from Hypericum roeperianumFobofou, Serge Alain Tanemossu / Franke, Katrin / Sanna, Giuseppina / Porzel, Andrea / Bullita, Enrica / La Colla, Paolo / Wessjohann, Ludger A. et al. | 2015
- 6335
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Revisiting 1,3,4-Oxadiazol-2-ones: Utilization in the Development of ABHD6 InhibitorsPatel, Jayendra Z. / van Bruchem, John / Laitinen, Tuomo / Kaczor, Agnieszka A. / Navia-Paldanius, Dina / Parkkari, Teija / Savinainen, Juha R. / Laitinen, Jarmo T. / Nevalainen, Tapio J. et al. | 2015
- 6346
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New carbocyclic N6-substituted adenine and pyrimidine nucleoside analogues with a bicyclo[2.2.1]heptane fragment as sugar moiety; synthesis, antiviral, anticancer activity and X-ray crystallographyTănase, Constantin I. / Drăghici, Constantin / Cojocaru, Ana / Galochkina, Anastasia V. / Orshanskaya, Jana R. / Zarubaev, Vladimir V. / Shova, Sergiu / Enache, Cristian / Maganu, Maria et al. | 2015
- 6355
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Deprotometalation–iodolysis and computed CH acidity of 1,2,3- and 1,2,4-triazoles. Application to the synthesis of resveratrol analoguesNagaradja, Elisabeth / Bentabed-Ababsa, Ghenia / Scalabrini, Mathieu / Chevallier, Floris / Philippot, Stéphanie / Fontanay, Stéphane / Duval, Raphaël E. / Halauko, Yury S. / Ivashkevich, Oleg A. / Matulis, Vadim E. et al. | 2015
- 6364
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Next generation macrocyclic and acyclic cationic lipids for gene transfer: Synthesis and in vitro evaluationJubeli, Emile / Maginty, Amanda B. / Abdul Khalique, Nada / Raju, Liji / Abdulhai, Mohamad / Nicholson, David G. / Larsen, Helge / Pungente, Michael D. / Goldring, William P.D. et al. | 2015
- 6379
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Design, synthesis, and pharmacological evaluation of JDTic analogs to examine the significance of the 3- and 4-methyl substituentsCarroll, F. Ivy / Gichinga, Moses G. / Kormos, Chad M. / Maitra, Rangan / Runyon, Scott P. / Thomas, James B. / Mascarella, S. Wayne / Decker, Ann M. / Navarro, Hernán A. et al. | 2015
- 6389
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Multifunctional novel Diallyl disulfide (DADS) derivatives with β-amyloid-reducing, cholinergic, antioxidant and metal chelating properties for the treatment of Alzheimer’s diseaseManral, Apra / Saini, Vikas / Meena, Poonam / Tiwari, Manisha et al. | 2015
- 6404
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Curcumin-inspired cytotoxic 3,5-bis(arylmethylene)-1-(N-(ortho-substituted aryl)maleamoyl)-4-piperidones: A novel group of topoisomerase II alpha inhibitorsJha, Amitabh / Duffield, Katherine M. / Ness, Matthew R. / Ravoori, Sujatha / Andrews, Gabrielle / Bhullar, Khushwant S. / Rupasinghe, H.P. Vasantha / Balzarini, Jan et al. | 2015
- 6418
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Design and synthesis of 4-benzylpiperidine carboxamides as dual serotonin and norepinephrine reuptake inhibitorsPaudel, Suresh / Cao, Yongkai / Guo, Shuohan / An, Byeongkwan / Kim, Kyeong-Man / Cheon, Seung Hoon et al. | 2015
- 6427
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Discovery and SAR study of 3-(tert-butyl)-4-hydroxyphenyl benzoate and benzamide derivatives as novel farnesoid X receptor (FXR) antagonistsSong, Kebiao / Xu, Xing / Liu, Peng / Chen, Lili / Shen, Xu / Liu, Junhua / Hu, Lihong et al. | 2015
- 6437
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Synthesis and structure–activity relationships of novel 9-oxime acylides with improved bactericidal activityHan, Xu / Lv, Wei / Guo, Si-Yang / Cushman, Mark / Liang, Jian-Hua et al. | 2015
- 6454
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Design and synthesis of conformationally constrained hydroxylated 4-phenyl-2-aryl chromenopyridines as novel and selective topoisomerase II-targeted antiproliferative agentsThapa, Pritam / Jun, Kyu-Yeon / Kadayat, Tara Man / Park, Chanmi / Zheng, Zhi / Thapa Magar, Til Bahadur / Bist, Ganesh / Shrestha, Aarajana / Na, Younghwa / Kwon, Youngjoo et al. | 2015
- 6467
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Discovery of potent nitrotriazole-based antitrypanosomal agents: In vitro and in vivo evaluationPapadopoulou, Maria V. / Bloomer, William D. / Rosenzweig, Howard S. / O’Shea, Ivan P. / Wilkinson, Shane R. / Kaiser, Marcel / Chatelain, Eric / Ioset, Jean-Robert et al. | 2015
- 6477
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Synthesis and anticancer effects evaluation of 1-alkyl-3-(6-(2-methoxy-3-sulfonylaminopyridin-5-yl)benzo[d]thiazol-2-yl)urea as anticancer agents with low toxicityXie, Xiao-Xiao / Li, Huan / Wang, Juan / Mao, Shuai / Xin, Min-Hang / Lu, She-Min / Mei, Qi-Bing / Zhang, San-Qi et al. | 2015
- 6486
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Synthesis of a series of unsaturated ketone derivatives as selective and reversible monoamine oxidase inhibitorsChoi, Ji Won / Jang, Bo Ko / Cho, Nam-chul / Park, Jong-Hyun / Yeon, Seul Ki / Ju, Eun Ji / Lee, Yong Sup / Han, Gyoonhee / Pae, Ae Nim / Kim, Dong Jin et al. | 2015
- 6497
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Synthesis, antiangiogenesis evaluation and molecular docking studies of 1-aryl-3-[(thieno[3,2-b]pyridin-7-ylthio)phenyl]ureas: Discovery of a new substitution pattern for type II VEGFR-2 Tyr kinase inhibitorsMachado, Vera A. / Peixoto, Daniela / Costa, Raquel / Froufe, Hugo J.C. / Calhelha, Ricardo C. / Abreu, Rui M.V. / Ferreira, Isabel C.F.R. / Soares, Raquel / Queiroz, Maria-João R.P. et al. | 2015
- 6510
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Discovery of 4-benzoylamino-N-(prop-2-yn-1-yl)benzamides as novel microRNA-21 inhibitorsJiang, Cong-shan / Wang, Xiao-meng / Zhang, San-qi / Meng, Lie-su / Zhu, Wen-hua / Xu, Jing / Lu, She-min et al. | 2015
- 6520
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Kinase hinge binding scaffolds and their hydrogen bond patternsXing, Li / Klug-Mcleod, Jacquelyn / Rai, Brajesh / Lunney, Elizabeth A. et al. | 2015
- 6528
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Reengineered tricyclic anti-cancer agentsKastrinsky, David B. / Sangodkar, Jaya / Zaware, Nilesh / Izadmehr, Sudeh / Dhawan, Neil S. / Narla, Goutham / Ohlmeyer, Michael et al. | 2015
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Instructions to contributors| 2015
- IFC
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Editorial board| 2015