Novel naphthoquinone derivatives and evaluation of their trypanocidal and leishmanicidal activities (English)
- New search for: Naujorks, Aline Alves dos Santos
- New search for: Naujorks, Aline Alves dos Santos
- New search for: da Silva, Adriano Olímpio
- New search for: Lopes, Rosangela da Silva
- New search for: de Albuquerque, Sérgio
- New search for: Beatriz, Adilson
- New search for: Marques, Maria Rita
- New search for: de Lima, Dênis Pires
In:
Organic & biomolecular chemistry
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13
, 2
; 428-437
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2015
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ISSN:
- Article (Journal) / Print
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Title:Novel naphthoquinone derivatives and evaluation of their trypanocidal and leishmanicidal activities
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Contributors:
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Published in:Organic & biomolecular chemistry ; 13, 2 ; 428-437
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Publisher:
- New search for: RSC
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Place of publication:Cambridge
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Publication date:2015
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 35.70 / 35.50 / 35.50
- Further information on Basic classification
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Keywords:
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Source:
Table of contents – Volume 13, Issue 2
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 330
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Cucurbituril-based supramolecular engineered nanostructured materialsGürbüz, Sinem / Idris, Muazzam / Tuncel, Dönü et al. | 2014
- 317
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Front cover| 2014
- 319
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Contents list| 2014
- 348
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A peptide topological template for the dispersion of [60]fullerene in waterBartocci, S. / Mazzier, D. / Moretto, A. / Mba, M. et al. | 2014
- 353
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Pd(ii)-catalyzed C–H arylation of aryl and benzyl Weinreb amidesWang, Yan / Zhou, Kai / Lan, Quan / Wang, Xi-Sheng et al. | 2014
- 357
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Artificial metalloenzymes for the diastereoselective reduction of NAD+ to NAD2HQuinto, Tommaso / Häussinger, Daniel / Köhler, Valentin / Ward, Thomas R. et al. | 2014
- 361
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Fe-promoted radical cyanomethylation/arylation of arylacrylamides to access oxindoles via cleavage of the sp3 C–H of acetonitrile and the sp2 C–H of the phenyl groupPan, Changduo / Zhang, Honglin / Zhu, Chengjian et al. | 2014
- 365
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The direct electrophilic cyanation of β-keto esters and amides with cyano benziodoxoleWang, Yao-Feng / Qiu, Jiashen / Kong, Dejie / Gao, Yongtao / Lu, Feipeng / Karmaker, Pran Gopal / Chen, Fu-Xue et al. | 2014
- 365
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The direct electrophilic cyanation of b-keto esters and amides with cyano benziodoxoleWang, Y. F. / Qiu, J. / Kong, D. / Gao, Y. / Lu, F. / Karmaker, P. / Chen, F. X. et al. | 2015
- 369
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Anion binding by biotin[6]uril in waterLisbjerg, Micke / Nielsen, Bjarne E. / Milhøj, Birgitte O. / Sauer, Stephan P. A. / Pittelkow, Michael et al. | 2014
- 374
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Bioorthogonal labelling of 3-nitrotyrosine in peptides and proteins through diazotisation mediated azidationNg, John Y. / Wong, Jason W. H. et al. | 2014
- 379
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Indium-catalyzed intramolecular hydroarylation of aryl propargyl ethersAlonso-Marañón, Lorena / Martínez, M. Montserrat / Sarandeses, Luis A. / Sestelo, José Pérez et al. | 2014
- 388
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PEGylation enhances the tumor selectivity of melanoma-targeted conjugatesAndré, Mathieu / Besse, Sophie / Chezal, Jean-Michel / Mounetou, Emmanuelle et al. | 2014
- 398
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Construction of dispirocyclohexanes via amine-catalyzed [2 + 2 + 2] annulations of Morita–Baylis–Hillman acetates with exocyclic alkenesChen, Rongshun / Xu, Silong / Fan, Xia / Li, Hanyuan / Tang, Yuhai / He, Zhengjie et al. | 2014
- 409
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Microwave-assisted preparation of 4-amino-3-cyano-5-methoxycarbonyl-N-arylpyrazoles as building blocks for the diversity-oriented synthesis of pyrazole-based polycyclic scaffoldsCorre, Laurent Le / Tak-Tak, Lotfi / Guillard, Arthur / Prestat, Guillaume / Gravier-Pelletier, Christine / Busca, Patricia et al. | 2014
- 424
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Preparation of asymmetrical polyynes by a solid-supported Glaser–Hay reactionLampkowski, Jessica S. / Durham, Corinn E. / Padilla, Marshall S. / Young, Douglas D. et al. | 2014
- 428
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Novel naphthoquinone derivatives and evaluation of their trypanocidal and leishmanicidal activitiesNaujorks, Aline Alves dos Santo / da Silva, Adriano Olímpio / Lopes, Rosangela da Silva / de Albuquerque, Sérgio / Beatriz, Adilson / Marques, Maria Rita / de Lima, Dênis Pire et al. | 2014
- 438
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Bidirectional macrocyclization of peptides by double multicomponent reactionsRicardo, Manuel G. / Morales, Fidel E. / Garay, Hilda / Reyes, Osvaldo / Vasilev, Dimitar / Wessjohann, Ludger A. / Rivera, Daniel G. et al. | 2014
- 447
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Efficient merging of copper and photoredox catalysis for the asymmetric cross-dehydrogenative-coupling of alkynes and tetrahydroisoquinolinesPerepichka, Inna / Kundu, Soumen / Hearne, Zoë / Li, Chao-Jun et al. | 2014
- 452
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Ametantrone-based compounds as potential regulators of Tau pre-mRNA alternative splicingArtigas, Gerard / López-Senín, Paula / González, Carlo / Escaja, Núria / Marchán, Vicente et al. | 2014
- 465
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The synthesis of 3-hydroxy-2,4,8-trimethyldec-8-enolides and an approach to 3,4-dihydroxy-2,4,6,8-tetramethyldec-8-enolideBotubol-Ares, J. M. / Durán-Peña, M. J. / Macías-Sánchez, A. J. / Hanson, J. R. / Collado, I. G. / Hernández-Galán, R. et al. | 2014
- 477
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Synthesis and antifungal activity of 1,2,3-triazole phenylhydrazone derivativesDai, Zhi-Cheng / Chen, Yong-Fei / Zhang, Mao / Li, Sheng-Kun / Yang, Ting-Ting / Shen, Li / Wang, Jian-Xin / Qian, Shao-Song / Zhu, Hai-Liang / Ye, Yong-Hao et al. | 2014
- 487
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Mixed non-covalent assemblies of ethynyl nile red and ethynyl pyrene along oligonucleotide templatesEnsslen, Philipp / Fritz, Yannic / Wagenknecht, Hans-Achim et al. | 2014
- 493
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Chiral recognition with a benzofuran receptor that mimics an oxyanion holeFuentes de Arriba, Ángel L. / Herrero, Ángel Gómez / Rubio, Omayra H. / Monleón, Laura M. / Simón Rubio, Lui / Alcázar, Victoria / Sanz, Francisca / Morán, Joaquín R. et al. | 2014
- 502
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Developing a targeting system for bacterial membranes: measuring receptor-phosphatidylglycerol interactions with 1H NMR, ITC and fluorescence correlation spectroscopyAlliband, Amanda / Wang, Zifan / Thacker, Christopher / English, Douglas S. / Burns, Dennis H. et al. | 2014
- 513
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Sc(OTf)3-mediated 1,3-dipolar cycloaddition–ring cleavage–rearrangement: a highly stereoselective access to Z-β-enaminonitrilesWang, Ying-chun / Xie, Yu-yang / Tan, Xian-chun / Wang, Heng-shan / Pan, Ying-ming et al. | 2014
- 513
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Sc(OTf)3-mediated 1,3-dipolar cycloaddition-ring cleavage-rearrangement: a highly stereoselective access to Z-b-enaminonitrilesWang, Y. c. / Xie, Y. y. / Tan, X. c. / Wang, H. s. / Pan, Y. m. et al. | 2015
- 520
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Trifluoromethanesulfonyloxy-group-directed regioselective (3 + 2) cycloadditions of benzynes for the synthesis of functionalized benzo-fused heterocyclesIkawa, Takashi / Kaneko, Hideki / Masuda, Shigeaki / Ishitsubo, Erika / Tokiwa, Hiroaki / Akai, Shuji et al. | 2014
- 527
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Targeting DNA with small molecules: a comparative study of a library of azonia aromatic chromophoresSuárez, Rosa M. / Bosch, Pedro / Sucunza, David / Cuadro, Ana M. / Domingo, Alberto / Mendicuti, Francisco / Vaquero, Juan J. et al. | 2014
- 539
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Late-stage diversification of biologically active pyridazinones via a direct C–H functionalization strategyLi, Wei / Fan, Zhoulong / Geng, Kaijun / Xu, Youjun / Zhang, Ao et al. | 2014
- 549
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Synthesis and evaluation of protein arginine N-methyltransferase inhibitors designed to simultaneously occupy both substrate binding sitesvan Haren, Matthij / van Ufford, Linda Quarle / Moret, Ed E. / Martin, Nathaniel I. et al. | 2014
- 556
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Inside front cover| 2015
- 557
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The tale of RNA G-quadruplexAgarwala, Prachi et al. | 2015
- 561
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pH response and molecular recognition in a low molecular weight peptide hydrogelLange, Stefanie C. / Unsleber, Jan / Drücker, Patrick / Galla, Hans-Joachim / Waller, Mark P. / Ravoo, Bart Jan et al. | 2014
- 562
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Copper-catalyzed aerobic oxidative amination of C(sp3)-H bonds: synthesis of imidazo[1,5-a]pyridinesElectronic supplementary information (ESI) available: 1H and 13C NMR spectra for all compounds and HRMS spectra for new compounds. CCDC 1017738 (3a). For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob00381dRavi, Chitrakar et al. | 2015
- 568
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Heteroatom-substituted tetra(3,4-pyrido)porphyrazines: a stride toward near-infrared-absorbing macrocyclesElectronic supplementary information (ESI) available: Experimental procedures and NMR, MS, absorption and fluorescence spectra. See DOI: 10.1039/c5ob00651aSimunek, Tomas et al. | 2015
- 569
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Galacto configured N-aminoaziridines: a new type of irreversible inhibitor of β-galactosidasesElectronic supplementary information (ESI) available: Scheme S1, Fig. S1, copies of NMR spectra, and HPLC methods and chromatograms. See DOI: 10.1039/c5ob00532aTrapero, Ana et al. | 2015
- 570
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Naphthalene diimides as red fluorescent pH sensors for functional cell imagingDoria, Filippo / Folini, Marco / Grande, Vincenzo / Cimino-Reale, Graziella / Zaffaroni, Nadia / Freccero, Mauro et al. | 2014
- 571
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Indium-catalyzed oxidative cross-dehydrogenative coupling of chromenes with 1,3-dicarbonyls and aryl ringsElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ob00277jLi, Fanmei et al. | 2015
- 577
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l-Valine derived chiral N-sulfinamides as effective organocatalysts for the asymmetric hydrosilylation of N-alkyl and N-aryl protected ketiminesWang, Chao / Wu, Xinjun / Zhou, Li / Sun, Jian et al. | 2014
- 583
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Novel synthesis of 5-methyl-5,10-dihydroindolo[3,2-b]indoles by Pd-catalyzed C–C and two-fold C–N coupling reactionsHung, Tran Quang / Hancker, Sören / Villinger, Alexander / Lochbrunner, Stefan / Dang, Tuan Thanh / Friedrich, Aleksej / Breitsprecher, Wolfgang / Langer, Peter et al. | 2014
- 584
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Tri- and tetra-substituted cyclen based lanthanide(iii) ion complexes as ribonuclease mimics: a study into the effect of log Ka, hydration and hydrophobicity on phosphodiester hydrolysis of the RNA-model 2-hydroxypropyl-4-nitrophenyl phosphate (HPNP)Electronic supplementary information (ESI) available: Fig. S1-7. See DOI: 10.1039/c4ob02384fPlush, Sally. E et al. | 2015
- 592
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Structural insight into the aggregation of l-prolyl dipeptides and its effect on organocatalytic performanceBerdugo, Cristina / Escuder, Beatriu / Miravet, Juan F. et al. | 2014
- 601
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A highly efficient and eco-friendly method for the synthesis of 1,3-indandione ring-fused 3-oxindoles bearing two contiguous quaternary stereocenters via an aldol reaction in aqueous mediaLiu, Xiong-Li / Pan, Bo-Wen / Zhang, Wen-Hui / Yang, Chao / Yang, Jun / Shi, Yang / Feng, Ting-Ting / Zhou, Ying / Yuan, Wei-Cheng et al. | 2014
- 612
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Rhodium(ii)-catalyzed intramolecular formal [4 + 3] cycloadditions of dienyltriazoles: rapid access to fused 2,5-dihydroazepinesTian, Yu / Wang, Yuanhao / Shang, Hai / Xu, Xudong / Tang, Yefeng et al. | 2014
- 620
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Cyclen-based cationic lipids containing a pH-sensitive moiety as gene delivery vectorsHuang, Zheng / Liu, Yan-Hong / Zhang, Yi-Mei / Zhang, Ji / Liu, Qiang / Yu, Xiao-Qi et al. | 2014
- 631
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Back cover| 2014
- 5591
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Stereoselective reaction of 2-carboxythioesters-1,3-dithiane with nitroalkenes: an organocatalytic strategy for the asymmetric addition of a glyoxylate anion equivalentElectronic supplementary information (ESI) available: Experimental details for nitrostyrene derivatives synthesis, catalysts preparation and organocatalytic reactions. Characterization details for Michael addition products and Baclofen synthesis. Determination of absolute configuration of the reaction products. 1H-NMR, 13C-NMR and 19F-NMR spectra and HPLC chromatograms on the chiral stationary phase of addition products. See DOI: 10.1039/c5ob00492fBenaglia, Maurizio et al. | 2015
- 5613
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Direct conversion of allyl arenes to aryl ethylketones via a TBHP-mediated palladium-catalyzed tandem isomerization-Wacker oxidation of terminal alkenesElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ob00586hLiu, Qiang et al. | 2015
- 5621
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Fluorine containing amino acids: synthesis and peptide coupling of amino acids containing the all-cis tetrafluorocyclohexyl motifElectronic supplementary information (ESI) available. CCDC 1057152. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob00650cAyoup, Mohammed Salah et al. | 2015
- 5625
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Simultaneous introduction of trifluoromethyl and λ6-pentafluorosulfanyl substituents using F5S-C&z.tbd;C-CF3 as a dienophileElectronic supplementary information (ESI) available: The experimental details and copy of 1H, 13C and 19F NMR spectra. CCDC 1020179 and 1020180. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob00610dLentz, Dieter et al. | 2015
- 5629
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Maleimide as an efficient nucleophilic partner in the aza-Morita-Baylis-Hillman reaction: synthesis of chiral 3-substituted-3-aminooxindolesElectronic supplementary information (ESI) available. CCDC 1037308. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob00182jKumar, Akshay et al. | 2015
- 5636
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Enantioselective synthesis of chiral heterocycles containing both chroman and pyrazolone derivatives catalysed by a chiral squaramideElectronic supplementary information (ESI) available: Copies of 1H and 13C NMR spectra of new compounds, and HPLC chromatograms. CCDC 1040622. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c4ob02653eLi, Jun-Hua et al. | 2015
- 5646
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Regulation of telomeric i-motif stability by 5-methylcytosine and 5-hydroxymethylcytosine modificationElectronic supplementary information (ESI) available: methods and materials, pH dependent CD spectra of DNA i-motifs, spectra for Tm and pKa determination for molecular crowding studies, physical and electronic properties of substituents at the C5 position of cytosine, HPLC and ESI-MS of DNAs. See DOI: 10.1039/c4ob02646bXu, Baochang et al. | 2015
- 5652
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Carbonic anhydrase II as host protein for the creation of a biocompatible artificial metathesaseElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ob00428dKajetanowicz, Anna et al. | 2015
- 5656
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Discovery, stereospecific characterization and peripheral modification of 1-(pyrrolidin-1-ylmethyl)-2-[(6-chloro-3-oxo-indan)-formyl]-1,2,3,4-tetrahydroisoquinolines as novel selective κ opioid receptor agonistsGan, Zong-Jie et al. | 2015
- 5674
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Colchicine derivatives with potent anticancer activity and reduced P-glycoprotein induction liabilityIIIM Publication number IIIM/1616/2013Electronic supplementary information (ESI) available: Spectra of all compounds. See DOI: 10.1039/c5ob00406cMondhe, Dilip M et al. | 2015
- 5716
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Synthetic studies toward the brasilinolides: controlled assembly of a protected C1-C38 polyol based on fragment union by complex aldol reactionsElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ob00498e. All data accompanying this publication are directly available within the publication and the ESIPaterson, Ian et al. | 2015
- 5734
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Effect of preorganization on the affinity of synthetic DNA binding motifs for nucleotide ligandsElectronic supplementary information (ESI) available: MALDI-TOF mass spectra of modified oligonucleotides, additional UV/VIS-spectra from filtration assays, HPLC traces, UV-melting points, and additional UV-melting curves. See DOI: 10.1039/c5ob00508fRichert, C et al. | 2015
- 5743
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Binaphthyl-1,2,3-triazole peptidomimetics with activity against Clostridium difficile and other pathogenic bacteriaElectronic supplementary information (ESI) available: Experimental procedures, compound characterization data, antibacterial testing methods, hemolysis data and NMR spectra. See DOI: 10.1039/c5ob00576kKing, Amy M et al. | 2015
- 5757
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Resveratrol-based benzoselenophenes with an enhanced antioxidant and chain breaking capacityElectronic supplementary information (ESI) available: NMR spectra of 1-3; optimized stoichiometry ratios for the isolation of 1-3; computational data. See DOI: 10.1039/c5ob00193eNapolitano, Alessandra et al. | 2015
- 5765
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Synthesis of new carolacton derivatives and their activity against biofilms of oral bacteriaElectronic supplementary information (ESI) available: Analytical and spectroscopic data including copies of NMR spectra of synthetic intermediates and new carolacton derivatives as well as copies of NMR spectra of all new compounds can be found with this article online. Additionally it contains live/dead measurements and fluorescence microscopic analyses of carolacton against S. oralis and S. gordonii, MS spectra of reextractions and the quantification of streptococci biofilms after active compound treatment using crystal violet staining. See DOI: 10.1039/c5ob00460hSchmidt, T et al. | 2015
- 5775
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High solid-state luminescence in propeller-shaped AIE-active pyridine-ketoiminate-boron complexesElectronic supplementary information (ESI) available: 1H, 13C NMR and luminescence spectra of compounds 2 and 3. CCDC 1031745 and 1031746. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob00607dHe, Weijiang et al. | 2015
- 5783
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Direct synthesis of a geminal zwitterionic phosphonium/hydridoborate system - developing an alternative tool for generating frustrated Lewis pair hydrogen activation systemsElectronic supplementary information (ESI) available: Details of the experiments, characterization of all compounds and crystal structure data as CIF files. CCDC 1034881-1034888 and 1045775. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob00634aDaniliuc, Constantin G et al. | 2015
- 5817
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BINOL-Al catalysed asymmetric cyclization and amplification: preparation of optically active menthol analogsElectronic supplementary information (ESI) available: Experimental details. See DOI: 10.1039/c5ob00433kYamada, Shinya et al. | 2015
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A preorganized β-amino acid bearing a guanidinium side chain and its use in cell-penetrating peptidesElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ob00389jDemizu, Yosuke et al. | 2015
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Organocatalytic regioselective asymmetric Michael addition of azlactones to o-hydroxy chalcone derivativesElectronic supplementary information (ESI) available: Characterization data and HPLC chromatograms for all compounds. CCDC 1032990. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob00121hLi, Nai-Kai et al. | 2015
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Grignard-mediated reduction of 2,2,2-trichloro-1-arylethanonesElectronic supplementary information (ESI) available: Experimental procedures and spectral information for compounds 1d, 1e and 1f, crystal data and structure refinement tables for 1e, 1f, 2a, 2f, 2h, 2j, 2k, 2o, 2t, 3a, 3b, 6a, 6f and 6h and 1H and 13C spectra for all new compounds. CCDC 1020127 (1e), 1020128 (1f), 1020129 (2a), 1020130 (2f), 1020131 (2h), 1020132 (2j), 1020133 (2k), 1020134 (2o), 1020135 (2t), 1020136 (3a), 1020137 (3b), 1020138 (6a), 1020139 (6f) and 1037684 (6h). For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob00541hLerrick, Reinner I et al. | 2015
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Stereoselective construction of functionalized tetracyclic and pentacyclic coumarinopyranpyrazole/pyrimidinedione/coumarin scaffolds using a solid-state melt reactionElectronic supplementary information (ESI) available: Representative experimental procedures with all spectral data of 5a-h, 8a-b, 10a-b, 13a-f and 16a-b. See DOI: 10.1039/c5ob00442jManikandan, Vasudevan et al. | 2015
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An interactive database to explore herbicide physicochemical propertiesElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ob00469aGandy, Michael N et al. | 2015
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Palladium-catalyzed asymmetric allylic amination of racemic butadiene monoxide with isatin derivativesElectronic supplementary information (ESI) available: Procedure for the synthesis of isatin derivatives, characterization of the products along with the NMR spectra. CCDC 1037747. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob00663eDu, Haifeng et al. | 2015