Thiadiazole derivatives as New Class of (English)
- New search for: Salar, Uzma
- New search for: Salar, Uzma
- New search for: Taha, Muhammad
- New search for: Ismail, Nor Hadiani
- New search for: Khan, Khalid Mohammed
- New search for: Imran, Syahrul
- New search for: Perveen, Shahnaz
- New search for: Wadood, Abdul
- New search for: Riaz, Muhammad
In:
Bioorganic & medicinal chemistry
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24
, 8
; 1909-1918
;
2016
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ISSN:
- Article (Journal) / Print
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Title:Thiadiazole derivatives as New Class of
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Contributors:Salar, Uzma ( author ) / Taha, Muhammad / Ismail, Nor Hadiani / Khan, Khalid Mohammed / Imran, Syahrul / Perveen, Shahnaz / Wadood, Abdul / Riaz, Muhammad
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Published in:Bioorganic & medicinal chemistry ; 24, 8 ; 1909-1918
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2016
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ISSN:
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
- Further information on Basic classification
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Keywords:
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Classification:
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Source:
Table of contents – Volume 24, Issue 8
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1589
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Design, synthesis and biological evaluation of N,N-3-phenyl-3-benzylaminopropanamide derivatives as novel cholesteryl ester transfer protein inhibitorZhao, Dongmei / Xie, Honglei / Bai, Changlin / Liu, Chunchi / Hao, Chenzhou / Zhao, Shizhen / Yuan, Hongli / Luo, Changqun / Wang, Jian / Lin, Bin et al. | 2015
- 1589
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Design, synthesis and biological evaluation ofZhao, Shizhen et al. | 2016
- 1598
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Synthesis, and anticonvulsant activity of new amides derived from 3-methyl- or 3-ethyl-3-methyl-2,5-dioxo-pyrrolidin-1-yl-acetic acidsObniska, Jolanta / Rapacz, Anna / Rybka, Sabina / Góra, Małgorzata / Kamiński, Krzysztof / Sałat, Kinga / Żmudzki, Paweł et al. | 2016
- 1608
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Compound profiling and 3D-QSAR studies of hydrazone derivatives with activity against intracellular Trypanosoma cruziCosta, Lívia Bandeira / Cardoso, Marcos Veríssimo de Oliveira / de Oliveira Filho, Gevanio Bezerra / de Moraes Gomes, Paulo André Teixeira / Espíndola, José Wanderlan Pontes / de Jesus Silva, Thays Gabrielle / Torres, Pedro Henrique Monteiro / Silva, Floriano Paes Junior / Martin, Julio / de Figueiredo, Regina Célia Bressan Queiroz et al. | 2016
- 1608
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Compound profiling and 3D-QSAR studies of hydrazone derivatives with activity against intracellularCosta, Lívia Bandeira et al. | 2016
- 1619
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1,2,4-Triazolyl octahydropyrrolo[2,3-b]pyrroles: A new series of potent and selective dopamine D3 receptor antagonistsMicheli, Fabrizio / Bernardelli, Andrea / Bianchi, Federica / Braggio, Simone / Castelletti, Laura / Cavallini, Palmina / Cavanni, Paolo / Cremonesi, Susanna / Cin, Michele Dal / Feriani, Aldo et al. | 2016
- 1619
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1,2,4-Triazolyl octahydropyrrolo[2,3Micheli, Fabrizio et al. | 2016
- 1637
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Novel nicotine analogues with potential anti-mycobacterial activityGandhi, Paresh T. / Athmaram, Thimmasandra Narayanappa / Arunkumar, Gundaiah Ramesh et al. | 2016
- 1648
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Isatin analogs as novel inhibitors of Candida spp. β-carbonic anhydrase enzymesAkdemir, Atilla / Güzel-Akdemir, Özlen / Karalı, Nilgün / Supuran, Claudiu T. et al. | 2016
- 1648
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Isatin analogs as novel inhibitors ofAkdemir, Atilla et al. | 2016
- 1653
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Antiretroviral (HIV-1) activity of azulene derivativesPeet, Julia / Selyutina, Anastasia / Bredihhin, Aleksei et al. | 2016
- 1658
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Novel indole-based melatonin analogues: Evaluation of antioxidant activity and protective effect against amyloid β-induced damageGurer-Orhan, Hande / Karaaslan, Cigdem / Ozcan, Senem / Firuzi, Omidreza / Tavakkoli, Marjan / Saso, Luciano / Suzen, Sibel et al. | 2016
- 1665
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In vivo phase II-enzymes inducers, as potential chemopreventive agents, based on the chalcone and furoxan skeletonsCabrera, Mauricio / Mastandrea, Ignacio / Otero, Gabriel / Cerecetto, Hugo / González, Mercedes et al. | 2016
- 1675
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A concise synthesis and evaluation of new malonamide derivatives as potential α-glucosidase inhibitorsIslam, Mohammad Shahidul / Barakat, Assem / Al-Majid, Abdullah M. / Ghabbour, Hazem A. / Rahman, A.F.M. Motiur / Javaid, Kulsoom / Imad, Rehan / Yousuf, Sammer / Choudhary, M. Iqbal et al. | 2016
- 1683
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Development of a potent 2-oxoamide inhibitor of secreted phospholipase A2 guided by molecular docking calculations and molecular dynamics simulationsVasilakaki, Sofia / Barbayianni, Efrosini / Leonis, Georgios / Papadopoulos, Manthos G. / Mavromoustakos, Thomas / Gelb, Michael H. / Kokotos, George et al. | 2016
- 1696
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Donor substrate promiscuity of bacterial β1–3-N-acetylglucosaminyltransferases and acceptor substrate flexibility of β1–4-galactosyltransferasesLi, Yanhong / Xue, Mengyang / Sheng, Xue / Yu, Hai / Zeng, Jie / Thon, Vireak / Chen, Yi / Muthana, Musleh M. / Wang, Peng G. / Chen, Xi et al. | 2016
- 1696
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Donor substrate promiscuity of bacterial β1–3Li, Yanhong et al. | 2016
- 1706
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Development of a fluorescent cardiomyocyte specific binding probePes, Lara / Kim, Young / Tung, Ching-Hsuan et al. | 2016
- 1718
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Design and synthesis of small molecule-sulfotyrosine mimetics that inhibit HIV-1 entryDogo-Isonagie, Cajetan / Lee, Su-Lin / Lohith, Katheryn / Liu, Hongbing / Mandadapu, Sivakoteswara R. / Lusvarghi, Sabrina / O’Connor, Robert D. / Bewley, Carole A. et al. | 2016
- 1729
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Design, synthesis of phenstatin/isocombretastatin-oxindole conjugates as antimitotic agentsKumar, G. Bharath / Nayak, V. Lakshma / Sayeed, Ibrahim Bin / Reddy, Vangala Santhosh / Shaik, Anver Basha / Mahesh, Rasala / Baig, Mirza Feroz / Shareef, Mohd Adil / Ravikumar, A. / Kamal, Ahmed et al. | 2016
- 1741
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Novel tricyclic pyrazolo[1,5-d][1,4]benzoxazepin-5(6H)-one: Design, synthesis, model and use as hMAO-B inhibitorsChen, Rui / Xiao, Jie / Ni, Yong / Xu, Han-Fei / Zheng, Min / Tong, Xu / Zhang, Tong-Tian / Liao, Chenzhong / Tang, Wen-Jian et al. | 2016
- 1741
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Novel tricyclic pyrazolo[1,5Chen, Rui et al. | 2016
- 1749
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Synthesis, and docking studies of phenylpyrimidine-carboxamide derivatives bearing 1H-pyrrolo[2,3-b]pyridine moiety as c-Met inhibitorsZhu, Wufu / Wang, Wenhui / Xu, Shan / Wang, Jianqiang / Tang, Qidong / Wu, Chunjiang / Zhao, Yanfang / Zheng, Pengwu et al. | 2016
- 1757
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C-3 benzoic acid derivatives of C-3 deoxybetulinic acid and deoxybetulin as HIV-1 maturation inhibitorsLiu, Zheng / Swidorski, Jacob J. / Nowicka-Sans, Beata / Terry, Brian / Protack, Tricia / Lin, Zeyu / Samanta, Himadri / Zhang, Sharon / Li, Zhufang / Parker, Dawn D. et al. | 2016
- 1771
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Investigation of 4-amino-5-alkynylpyrimidine-2(1Garg, Gaurav et al. | 2016
- 1771
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Investigation of 4-amino-5-alkynylpyrimidine-2(1H)-ones as anti-mycobacterial agentsGarg, Gaurav / Pande, Milind / Agrawal, Ambika / Li, Jie / Kumar, Rakesh et al. | 2016
- 1778
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Molecular simulation of cyclohexanyl nucleic acid (CNA) duplexes with CNA, DNA and RNA and CNA triloop and tetraloop hairpin structuresFroeyen, Matheus / Abu el Asrar, Rania / Abramov, Mikhail / Herdewijn, Piet et al. | 2016
- 1786
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Novel squaramides with in vitro liver stage antiplasmodial activityRibeiro, Carlos J.A. / Espadinha, Margarida / Machado, Marta / Gut, Jiri / Gonçalves, Lídia M. / Rosenthal, Philip J. / Prudêncio, Miguel / Moreira, Rui / Santos, Maria M.M. et al. | 2016
- 1793
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Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agentsWaszkielewicz, A.M. / Gunia-Krzyżak, A. / Powroźnik, B. / Słoczyńska, K. / Pękala, E. / Walczak, M. / Bednarski, M. / Żesławska, E. / Nitek, W. / Marona, H. et al. | 2016
- 1811
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Discovery of novelXie, Honglei et al. | 2016
- 1811
-
Discovery of novel N,N-3-phenyl-3-benzylaminopropionanilides as potent inhibitors of cholesteryl ester transfer protein in vivoXie, Honglei / Li, Yiqun / Bai, Changlin / Wang, Ruifeng / Liu, Chunchi / Hao, Chenzhou / Lin, Bin / Cheng, Maosheng / Zhao, Dongmei et al. | 2016
- 1819
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Design and evaluation of novel glutaminase inhibitorsMcDermott, Lee A. / Iyer, Prema / Vernetti, Larry / Rimer, Shawn / Sun, Jingran / Boby, Melissa / Yang, Tianyi / Fioravanti, Michael / O’Neill, Jason / Wang, Liwei et al. | 2016
- 1840
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Quinoxalinone (Part II). Discovery ofShi, Leilei et al. | 2016
- 1840
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Quinoxalinone (Part II). Discovery of (Z)-3-(2-(pyridin-4-yl)vinyl)quinoxalinone derivates as potent VEGFR-2 kinase inhibitorsShi, Leilei / Zhou, Jianfeng / Wu, Jifeng / Cao, Junya / Shen, Yuemao / Zhou, Hua / Li, Xun et al. | 2016
- 1853
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Design, synthesis, and evaluation of 2-piperidone derivatives for the inhibition of β-amyloid aggregation and inflammation mediated neurotoxicityLi, Lei / Chen, Ming / Jiang, Feng-Chao et al. | 2016
- 1866
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Design and synthesis of thiourea derivatives with sulfur-containing heterocyclic scaffolds as potential tyrosinase inhibitorsLiu, Pingping / Shu, Chen / Liu, Lujie / Huang, Qingchun / Peng, Yanqing et al. | 2016
- 1872
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Exploration of 2-benzylbenzimidazole scaffold as novel inhibitor of NF-κBBoggu, PullaReddy / Venkateswararao, Eeda / Manickam, Manoj / Kwak, Dajin / Kim, Youngsoo / Jung, Sang-Hun et al. | 2016
- 1879
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Rational design, synthesis and biological evaluation of 1,3,4-oxadiazole pyrimidine derivatives as novel pyruvate dehydrogenase complex E1 inhibitorsHe, Haifeng / Wang, Wei / Zhou, Yuan / Xia, Qin / Ren, Yanliang / Feng, Jiangtao / Peng, Hao / He, Hongwu / Feng, Lingling et al. | 2016
- 1889
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Synthesis and biological evaluation of quinoline derivatives as potential anti-prostate cancer agents and Pim-1 kinase inhibitorsLi, Kun / Li, Ying / Zhou, Di / Fan, Yinbo / Guo, Hongye / Ma, Tianyi / Wen, Jiachen / Liu, Dan / Zhao, Linxiang et al. | 2016
- 1898
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Design, synthesis, topoisomerase I & II inhibitory activity, antiproliferative activity, and structure–activity relationship study of pyrazoline derivatives: An ATP-competitive human topoisomerase IIα catalytic inhibitorAhmad, Pervez / Woo, Hyunjung / Jun, Kyu-Yeon / Kadi, Adnan A. / Abdel-Aziz, Hatem A. / Kwon, Youngjoo / Rahman, A.F.M. Motiur et al. | 2016
- 1909
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Thiadiazole derivatives as New Class of β-glucuronidase inhibitorsSalar, Uzma / Taha, Muhammad / Ismail, Nor Hadiani / Khan, Khalid Mohammed / Imran, Syahrul / Perveen, Shahnaz / Wadood, Abdul / Riaz, Muhammad et al. | 2016
- 1909
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Thiadiazole derivatives as New Class ofSalar, Uzma et al. | 2016
- 1919
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Discovery of new low-molecular-weight p53–Mdmx disruptors and their anti-cancer activitiesUesato, Shinichi / Matsuura, Yoshihiro / Matsue, Saki / Sumiyoshi, Takaaki / Hirata, Yoshiyuki / Takemoto, Suzuho / Kawaratani, Yasuyuki / Yamai, Yusuke / Ishida, Kyoji / Sasaki, Tsutomu et al. | 2016
- 1927
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Evaluation of the anti-inflammatory action of curcumin analog (DM1): Effect on iNOS and COX-2 gene expression and autophagy pathwaysPaulino, Niraldo / Paulino, Amarilis Scremin / Diniz, Susana N. / de Mendonça, Sergio / Gonçalves, Ivair D. / Faião Flores, Fernanda / Santos, Reginaldo Pereira / Rodrigues, Carina / Pardi, Paulo Celso / Quincoces Suarez, José Agustin et al. | 2016
- IFC
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Editorial board| 2016