Synthesis and structure-activity relationships of novel hybrid ferrocenyl compounds based on a bicyclic core skeleton for breast cancer therapy (English)
- New search for: Li, Changhao
- New search for: Li, Changhao
- New search for: Tang, Chu
- New search for: Hu, Zhiye
- New search for: Zhao, Chenxi
- New search for: Li, Chenlu
- New search for: Zhang, Silong
- New search for: Dong, Chune
- New search for: Zhou, Hai-Bing
- New search for: Huang, Jian
In:
Bioorganic & medicinal chemistry
;
24
, 13
; 3062-3074
;
2016
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ISSN:
- Article (Journal) / Print
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Title:Synthesis and structure-activity relationships of novel hybrid ferrocenyl compounds based on a bicyclic core skeleton for breast cancer therapy
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Contributors:Li, Changhao ( author ) / Tang, Chu / Hu, Zhiye / Zhao, Chenxi / Li, Chenlu / Zhang, Silong / Dong, Chune / Zhou, Hai-Bing / Huang, Jian
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Published in:Bioorganic & medicinal chemistry ; 24, 13 ; 3062-3074
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2016
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ISSN:
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
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Keywords:
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Source:
Table of contents – Volume 24, Issue 13
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 2871
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Discovery of new [1,4]dioxino[2,3-f]quinazoline-based inhibitors of EGFR including the T790M/L858R mutantQin, Xuemei / Li, Zhipeng / Yang, Leifu / Liu, Peng / Hu, Liming / Zeng, Chengchu / Pan, Zhiyong et al. | 2016
- 2882
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Novel sulfonamide bearing coumarin scaffolds as selective inhibitors of tumor associated carbonic anhydrase isoforms IX and XIIChandak, Navneet / Ceruso, Mariangela / Supuran, Claudiu T. / Sharma, Pawan K. et al. | 2016
- 2887
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Dihydrochelerythrine and its derivatives: Synthesis and their application as potential G-quadruplex DNA stabilizing agentsMalhotra, Rajesh / Rarhi, Chhanda / Diveshkumar, K.V. / Barik, Rajib / D’cunha, Ruhee / Dhar, Pranab / Kundu, Mrinalkanti / Chattopadhyay, Subrata / Roy, Subho / Basu, Sourav et al. | 2016
- 2897
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Optimization of the phenylurea moiety in a phosphoinositide 3-kinase (PI3K) inhibitor to improve water solubility and the PK profile by introducing a solubilizing group and ortho substituentsKawada, Hatsuo / Ebiike, Hirosato / Tsukazaki, Masao / Yamamoto, Shun / Koyama, Kohei / Nakamura, Mitsuaki / Morikami, Kenji / Yoshinari, Kiyoshi / Yoshida, Miyuki / Ogawa, Kotaro et al. | 2016
- 2907
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Pyrazolylbenzo[d]imidazoles as new potent and selective inhibitors of carbonic anhydrase isoforms hCA IX and XIIKumar, Satish / Ceruso, Mariangela / Tuccinardi, Tiziano / Supuran, Claudiu T. / Sharma, Pawan K. et al. | 2016
- 2914
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Synthesis and evaluation of raloxifene derivatives as a selective estrogen receptor down-regulatorShoda, Takuji / Kato, Masashi / Fujisato, Takuma / Misawa, Takashi / Demizu, Yosuke / Inoue, Hideshi / Naito, Mikihiko / Kurihara, Masaaki et al. | 2016
- 2920
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2-(Thienothiazolylimino)-1,3-thiazolidin-4-ones inhibit cell division cycle 25 A phosphataseHuber-Villaume, Sophie / Revelant, Germain / Sibille, Estelle / Philippot, Stéphanie / Morabito, Angelica / Dunand, Sandrine / Chaimbault, Patrick / Bagrel, Denyse / Kirsch, Gilbert / Hesse, Stéphanie et al. | 2016
- 2929
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New trans dichloro (triphenylphosphine)platinum(II) complexes containing N-(butyl),N-(arylmethyl)amino ligands: Synthesis, cytotoxicity and mechanism of actionDalla Via, Lisa / García-Argáez, Aída Nelly / Agostinelli, Enzo / Belli Dell’Amico, Daniela / Labella, Luca / Samaritani, Simona et al. | 2016
- 2938
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Design, synthesis and anticonvulsant activity of new hybrid compounds derived from N-phenyl-2-(2,5-dioxopyrrolidin-1-yl)-propanamides and -butanamidesKamiński, Krzysztof / Rapacz, Anna / Filipek, Barbara / Obniska, Jolanta et al. | 2016
- 2947
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Discovery of a novel covalent non-β-lactam inhibitor of the metallo-β-lactamase NDM-1Christopeit, Tony / Albert, Anastasia / Leiros, Hanna-Kirsti S. et al. | 2016
- 2954
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Novel free fatty acid receptor 1 (GPR40) agonists based on 1,3,4-thiadiazole-2-carboxamide scaffoldKrasavin, Mikhail / Lukin, Alexey / Zhurilo, Nikolay / Kovalenko, Alexey / Zahanich, Ihor / Zozulya, Sergey / Moore, Daniel / Tikhonova, Irina G. et al. | 2016
- 2964
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Design, synthesis and biological evaluation of novel tetrahydroisoquinoline quaternary derivatives as peripheral κ-opioid receptor agonistsGuo, Ting / Gan, Zongjie / Chen, Jie / Wang, Dechuan / He, Ling / Song, Qiao / Xu, Yungen et al. | 2016
- 2971
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Antiproliferative activity and apoptosis inducing effects of nitric oxide donating derivatives of evodiamineZhao, Nan / Tian, Kang-tao / Cheng, Ke-guang / Han, Tong / Hu, Xu / Li, Da-hong / Li, Zhan-lin / Hua, Hui-ming et al. | 2016
- 2979
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Stable and biocompatible cystine knot peptides from the marine sponge Asteropus sp.Su, Mingzhi / Li, Huayue / Wang, Haibo / Kim, Eun La / Kim, Hyung Sik / Kim, Eun-Hee / Lee, Jaewon / Jung, Jee H. et al. | 2016
- 2988
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Bismuth(III) complexes with 2-acetylpyridine- and 2-benzoylpyridine-derived hydrazones: Antimicrobial and cytotoxic activities and effects on the clonogenic survival of human solid tumor cellsFerreira, Isabella P. / Piló, Elisa D.L. / Recio-Despaigne, Angel A. / Da Silva, Jeferson G. / Ramos, Jonas P. / Marques, Lucas B. / Prazeres, Pedro H.D.M. / Takahashi, Jacqueline A. / Souza-Fagundes, Elaine M. / Rocha, Willian et al. | 2016
- 2999
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Triterpene sapogenin–polyarginine conjugates exhibit promising antibacterial activity against Gram-positive strainsNa, Heiya / Li, Xiangpeng / Zou, Cunbin / Wang, Chenhong / Wang, Chao / Liu, Keliang et al. | 2016
- 3006
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Systematic evaluation of methyl ester bioisosteres in the context of developing alkenyldiarylmethanes (ADAMs) as non-nucleoside reverse transcriptase inhibitors (NNRTIs) for anti-HIV-1 chemotherapyHoshi, Ayako / Sakamoto, Takeshi / Takayama, Jun / Xuan, Meiyan / Okazaki, Mari / Hartman, Tracy L. / Buckheit, Robert W. Jr. / Pannecouque, Christophe / Cushman, Mark et al. | 2016
- 3023
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Comparing the efficacy of photodynamic and sonodynamic therapy in non-melanoma and melanoma skin cancerMcEwan, Conor / Nesbitt, Heather / Nicholas, Dean / Kavanagh, Oisin N. / McKenna, Kevin / Loan, Philip / Jack, Iain G. / McHale, Anthony P. / Callan, John F. et al. | 2016
- 3029
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Inhibitors of secreted phospholipase A2 suppress the release of PGE2 in renal mesangial cellsVasilakaki, Sofia / Barbayianni, Efrosini / Magrioti, Victoria / Pastukhov, Oleksandr / Constantinou-Kokotou, Violetta / Huwiler, Andrea / Kokotos, George et al. | 2016
- 3035
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Identification, synthesis and evaluation of SARS-CoV and MERS-CoV 3C-like protease inhibitorsKumar, Vathan / Tan, Kian-Pin / Wang, Ying-Ming / Lin, Sheng-Wei / Liang, Po-Huang et al. | 2016
- 3043
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Synthesis of 4-(thiazol-2-ylamino)-benzenesulfonamides with carbonic anhydrase I, II and IX inhibitory activity and cytotoxic effects against breast cancer cell linesAbdel Gawad, Nagwa M. / Amin, Noha H. / Elsaadi, Mohammed T. / Mohamed, Fatma M.M. / Angeli, Andrea / De Luca, Viviana / Capasso, Clemente / Supuran, Claudiu T. et al. | 2016
- 3052
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Design, biological evaluation and 3D QSAR studies of novel dioxin-containing triaryl pyrazoline derivatives as potential B-Raf inhibitorsYang, Yu-Shun / Yang, Bing / Zou, Yan / Li, Guigen / Zhu, Hai-Liang et al. | 2016
- 3062
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Synthesis and structure–activity relationships of novel hybrid ferrocenyl compounds based on a bicyclic core skeleton for breast cancer therapyLi, Changhao / Tang, Chu / Hu, Zhiye / Zhao, Chenxi / Li, Chenlu / Zhang, Silong / Dong, Chune / Zhou, Hai-Bing / Huang, Jian et al. | 2016
- 3075
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Antiplasmodial activities of gold(I) complexes involving functionalized N-heterocyclic carbenesHemmert, Catherine / Ramadani, Arba Pramundita / Boselli, Luca / Fernández Álvarez, Álvaro / Paloque, Lucie / Augereau, Jean-Michel / Gornitzka, Heinz / Benoit-Vical, Françoise et al. | 2016
- 3083
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Synthesis, biological evaluation, and physicochemical property assessment of 4-substituted 2-phenylaminoquinazolines as Mer tyrosine kinase inhibitorsWang, Sheng-Biao / Cui, Mu-Tian / Wang, Xiao-Feng / Ohkoshi, Emika / Goto, Masuo / Yang, De-Xuan / Li, Linna / Yuan, Shoujun / Morris-Natschke, Susan L. / Lee, Kuo-Hsiung et al. | 2016
- 3093
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Corrigendum to “Purinylpyridinylamino-based DFG-in/αC-helix-out B-Raf inhibitors: Applying mutant versus wild-type B-Raf selectivity indices for compound profiling” [Bioorg. Med. Chem. 24 (2016) 2215–2234]Liu, Longbin / Lee, Matthew R. / Kim, Joseph L. / Whittington, Douglas A. / Bregman, Howard / Hua, Zihao / Lewis, Richard T. / Martin, Matthew W. / Nishimura, Nobuko / Potashman, Michele et al. | 2016
- IFC
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Editorial board| 2016