Novel multifunctional dopamine D2/D3 receptors agonists with potential neuroprotection and anti-alpha synuclein protein aggregation properties (English)
- New search for: Luo, Dan
- New search for: Luo, Dan
- New search for: Sharma, Horrick
- New search for: Yedlapudi, Deepthi
- New search for: Antonio, Tamara
- New search for: Reith, Maarten E.A
- New search for: Dutta, Aloke K
In:
Bioorganic & medicinal chemistry
;
24
, 21
; 5088-5102
;
2016
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ISSN:
- Article (Journal) / Print
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Title:Novel multifunctional dopamine D2/D3 receptors agonists with potential neuroprotection and anti-alpha synuclein protein aggregation properties
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Contributors:Luo, Dan ( author ) / Sharma, Horrick / Yedlapudi, Deepthi / Antonio, Tamara / Reith, Maarten E.A / Dutta, Aloke K
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Published in:Bioorganic & medicinal chemistry ; 24, 21 ; 5088-5102
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2016
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ISSN:
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
- Further information on Basic classification
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Keywords:
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Classification:
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Source:
Table of contents – Volume 24, Issue 21
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 5007
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Advances in rationally designed dual inhibitors of HIV-1 reverse transcriptase and integraseGu, Shuang-Xi / Xue, Ping / Ju, Xiu-Lian / Zhu, Yuan-Yuan et al. | 2016
- 5017
-
Tyrosyl-DNA phosphodiesterase inhibitors: Progress and potentialLaev, Sergey S. / Salakhutdinov, Nariman F. / Lavrik, Olga I. et al. | 2016
- 5028
-
Synthesis and evaluation of 6-pyrazoylamido-3N-substituted azabicyclo[3,1,0]hexane derivatives as T-type calcium channel inhibitors for treatment of neuropathic painKim, Jung Hyun / Nam, Ghilsoo et al. | 2016
- 5036
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The discovery of 2,5-isomers of triazole-pyrrolopyrimidine as selective Janus kinase 2 (JAK2) inhibitors versus JAK1 and JAK3Lee, Sun-Mi / Yoon, Kyoung Bin / Lee, Hyo Jeong / Kim, Jiwon / Chung, You Kyoung / Cho, Won-Jea / Mukai, Chisato / Choi, Sun / Kang, Keon Wook / Han, Sun-Young et al. | 2016
- 5047
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Effect of lysine methylation and acetylation on the RNA recognition and cellular uptake of Tat-derived peptidesLiu, Mu-Chun / Chen, Chin-Yih / Chiang, Chang-Hwa / Wang, Wei-Ming / Cheng, Richard P. et al. | 2016
- 5052
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Synthesis and evaluation of 2,5 and 2,6 pyridine-based CXCR4 inhibitorsGaines, Theresa / Camp, Davita / Bai, Renren / Liang, Zhongxing / Yoon, Younghyoun / Shim, Hyunsuk / Mooring, Suazette Reid et al. | 2016
- 5061
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Triterpenoids from Momordica balsamina: Reversal of ABCB1-mediated multidrug resistanceRamalhete, Cátia / Mulhovo, Silva / Molnar, Joseph / Ferreira, Maria-José U. et al. | 2016
- 5068
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Phosphorothioate analogs of P1,P3-di(nucleosid-5′-yl) triphosphates: Synthesis, assignment of the absolute configuration at P-atoms and P-stereodependent recognition by Fhit hydrolaseKaczmarek, Renata / Krakowiak, Agnieszka / Korczyński, Dariusz / Baraniak, Janina / Nawrot, Barbara et al. | 2016
- 5076
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In vitro antileukemic activity of novel adenosine derivatives bearing boron cluster modificationŻołnierczyk, Jolanta D. / Olejniczak, Agnieszka B. / Mieczkowski, Adam / Błoński, Jerzy Z. / Kiliańska, Zofia M. / Robak, Tadeusz / Leśnikowski, Zbigniew J. et al. | 2016
- 5088
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Novel multifunctional dopamine D2/D3 receptors agonists with potential neuroprotection and anti-alpha synuclein protein aggregation propertiesLuo, Dan / Sharma, Horrick / Yedlapudi, Deepthi / Antonio, Tamara / Reith, Maarten E.A. / Dutta, Aloke K. et al. | 2016
- 5103
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Molecular docking studies and synthesis of novel bisbenzimidazole derivatives as inhibitors of α-glucosidaseÖzil, Musa / Emirik, Mustafa / Beldüz, Ali / Ülker, Serdar et al. | 2016
- 5115
-
Synthesis of arylated coumarins by Suzuki–Miyaura cross-coupling. Reactions and anti-HIV activityHamdy, Aws M. / Khaddour, Zien / Al-Masoudi, Najim A. / Rahman, Qamar / Hering-Junghans, Christian / Villinger, Alexander / Langer, Peter et al. | 2016
- 5127
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Focused screening to identify new adenosine kinase inhibitorsKöse, Meryem / Schiedel, Anke C. / Bauer, Alexander Andreas / Poschenrieder, Hermann / Burbiel, Joachim C. / Akkinepally, Raghuram Rao / Stachel, Hans-Dietrich / Müller, Christa E. et al. | 2016
- 5134
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Development, synthesis and structure–activity-relationships of inhibitors of the macrophage infectivity potentiator (Mip) proteins of Legionella pneumophila and Burkholderia pseudomalleiSeufert, Florian / Kuhn, Maximilian / Hein, Michael / Weiwad, Matthias / Vivoli, Mirella / Norville, Isobel H. / Sarkar-Tyson, Mitali / Marshall, Laura E. / Schweimer, Kristian / Bruhn, Heike et al. | 2016
- 5148
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Blood–brain barrier permeability of ginkgolide: Comparison of the behavior of PET probes 7α-[18F]fluoro- and 10-O-p-[11C]methylbenzyl ginkgolide B in monkey and rat brainsDoi, Hisashi / Sato, Kengo / Shindou, Hideo / Sumi, Kengo / Koyama, Hiroko / Hosoya, Takamitsu / Watanabe, Yasuyoshi / Ishii, Satoshi / Tsukada, Hideo / Nakanishi, Koji et al. | 2016
- 5158
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Anti-influenza activity of monoterpene-derived substituted hexahydro-2H-chromenesPatrusheva, Oksana S. / Zarubaev, Vladimir V. / Shtro, Anna A. / Orshanskaya, Yana R. / Boldyrev, Sergey A. / Ilyina, Irina V. / Kurbakova, Svetlana Yu. / Korchagina, Dina V. / Volcho, Konstantin P. / Salakhutdinov, Nariman F. et al. | 2016
- 5162
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Synthesis and biological evaluation of N-cyanoalkyl-, N-aminoalkyl-, and N-guanidinoalkyl-substituted 4-aminoquinoline derivatives as potent, selective, brain permeable antitrypanosomal agentsSola, Irene / Artigas, Albert / Taylor, Martin C. / Pérez-Areales, F. Javier / Viayna, Elisabet / Clos, M. Victòria / Pérez, Belén / Wright, Colin W. / Kelly, John M. / Muñoz-Torrero, Diego et al. | 2016
- 5172
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Elaboration of a proprietary thymidylate kinase inhibitor motif towards anti-tuberculosis agentsSong, Lijun / Risseeuw, Martijn D.P. / Froeyen, Matheus / Karalic, Izet / Goeman, Jan / Cappoen, Davie / Van der Eycken, Johan / Cos, Paul / Munier-Lehmann, Hélène / Van Calenbergh, Serge et al. | 2016
- 5183
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Synthesis and biological evaluation of santacruzamate A analogues for anti-proliferative and immunomodulatory activityGromek, Samantha M. / deMayo, James A. / Maxwell, Andrew T. / West, Ashley M. / Pavlik, Christopher M. / Zhao, Ziyan / Li, Jin / Wiemer, Andrew J. / Zweifach, Adam / Balunas, Marcy J. et al. | 2016
- 5197
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Synthesis and activity evaluation of the cyclic dipeptides arylidene N-alkoxydiketopiperazinesTian, Xia / Feng, Juan / Fan, Shi-ming / zhen, Xiao-li / Han, Jian-rong / Liu, Shou-xin et al. | 2016
- 5206
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Optimization of pyrimidinol antioxidants as mitochondrial protective agents: ATP production and metabolic stabilityChevalier, Arnaud / Alam, Mohammad Parvez / Khdour, Omar M. / Schmierer, Margaret / Arce, Pablo M. / Cripe, Cameron D. / Hecht, Sidney M. et al. | 2016
- 5221
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Identification of indole scaffold-based dual inhibitors of NOD1 and NOD2Keček Plešec, Kaja / Urbančič, Dunja / Gobec, Martina / Pekošak, Aleksandra / Tomašič, Tihomir / Anderluh, Marko / Mlinarič-Raščan, Irena / Jakopin, Žiga et al. | 2016
- 5235
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Sterol-dependent membrane association of the marine sponge-derived bicyclic peptide Theonellamide A as examined by 1H NMRCornelio, Kimberly / Espiritu, Rafael Atillo / Todokoro, Yasuto / Hanashima, Shinya / Kinoshita, Masanao / Matsumori, Nobuaki / Murata, Michio / Nishimura, Shinichi / Kakeya, Hideaki / Yoshida, Minoru et al. | 2016
- 5243
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Thermodynamic properties of leukotriene A4 hydrolase inhibitorsWittmann, Sandra K. / Kalinowsky, Lena / Kramer, Jan S. / Bloecher, René / Knapp, Stefan / Steinhilber, Dieter / Pogoryelov, Denys / Proschak, Ewgenij / Heering, Jan et al. | 2016
- 5249
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Expedient synthesis of an atypical oxazolidinone compound libraryCully, Sarah J. / Storr, Thomas E. / Rawling, Michael J. / Abeysena, Induka R. / Hamza, Daniel / Jones, Geraint / Pearce, Christopher A. / Quddus, Abdul / Lewis, William / Stockman, Robert A. et al. | 2016
- 5258
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Discovery of N-(1-(3-(4-phenoxyphenyl)-1,2,4-oxadiazol-5-yl)ethyl)acetamides as novel acetyl-CoA carboxylase 2 (ACC2) inhibitors with peroxisome proliferator-activated receptor α/δ (PPARα/δ) dual agonistic activityOkazaki, Shogo / Noguchi-Yachide, Tomomi / Sakai, Taki / Ishikawa, Minoru / Makishima, Makoto / Hashimoto, Yuichi / Yamaguchi, Takao et al. | 2016
- 5270
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Development of acetophenone ligands as potential neuroimaging agents for cholinesterasesJollymore-Hughes, Courtney T. / Pottie, Ian R. / Martin, Earl / Rosenberry, Terrone L. / Darvesh, Sultan et al. | 2016
- 5280
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An LP1 analogue, selective MOR agonist with a peculiar pharmacological profile, used to scrutiny the ligand binding domainRonsisvalle, Simone / Aricò, Giuseppina / Panarello, Federica / Spadaro, Angelo / Pasquinucci, Lorella / Pappalardo, Maria S. / Parenti, Carmela / Ronsisvalle, Nicole et al. | 2016
- 5291
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Synthesis, molecular modeling and SAR study of novel pyrazolo[5,1-f][1,6]naphthyridines as CB2 receptor antagonists/inverse agonistsDore, Antonio / Asproni, Battistina / Scampuddu, Alessia / Gessi, Stefania / Murineddu, Gabriele / Cichero, Elena / Fossa, Paola / Merighi, Stefania / Bencivenni, Serena / Pinna, Gérard A. et al. | 2016
- 5302
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Molecular docking studies, biological and toxicity evaluation of dihydroisoquinoline derivatives as potential anticancer agentsZiemska, Joanna / Guśpiel, Adam / Jarosz, Joanna / Nasulewicz-Goldeman, Anna / Wietrzyk, Joanna / Kawęcki, Robert / Pypowski, Krzysztof / Jarończyk, Małgorzata / Solecka, Jolanta et al. | 2016
- 5315
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Carbohydrate-based peptidomimetics targeting neuropilin-1: Synthesis, molecular docking study and in vitro biological activitiesRichard, Mylène / Chateau, Alicia / Jelsch, Christian / Didierjean, Claude / Manival, Xavier / Charron, Christophe / Maigret, Bernard / Barberi-Heyob, Muriel / Chapleur, Yves / Boura, Cédric et al. | 2016
- 5326
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Synthesis and preclinical characterization of 1-(6′-deoxy-6′-[18F]fluoro-β-d-allofuranosyl)-2-nitroimidazole (β-6′-[18F]FAZAL) as a positron emission tomography radiotracer to assess tumor hypoxiaWanek, Thomas / Kreis, Katharina / Križková, Petra / Schweifer, Anna / Denk, Christoph / Stanek, Johann / Mairinger, Severin / Filip, Thomas / Sauberer, Michael / Edelhofer, Patricia et al. | 2016
- 5340
-
Phosphonate-based irreversible inhibitors of human γ-glutamyl transpeptidase (GGT). GGsTop is a non-toxic and highly selective inhibitor with critical electrostatic interaction with an active-site residue Lys562 for enhanced inhibitory activityKamiyama, Akane / Nakajima, Mado / Han, Liyou / Wada, Kei / Mizutani, Masaharu / Tabuchi, Yukiko / Kojima-Yuasa, Akiko / Matsui-Yuasa, Isao / Suzuki, Hideyuki / Fukuyama, Keiichi et al. | 2016
- 5353
-
Convergent 18F-labeling and evaluation of N-benzyl-phenethylamines as 5-HT2A receptor PET ligandsPetersen, Ida Nymann / Villadsen, Jonas / Hansen, Hanne Demant / Jensen, Anders A. / Lehel, Szabolcs / Gillings, Nic / Herth, Matthias M. / Knudsen, Gitte M. / Kristensen, Jesper L. et al. | 2016
- 5357
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Discovery and structure–activity relationship studies of quinolinone derivatives as potent IL-2 suppressive agentsKwak, Seung-Hwa / Kang, Jung-Ah / Kim, Minjeong / Lee, So-Deok / Park, Jin-Hee / Park, Sung-Gyoo / Ko, Hyojin / Kim, Yong-Chul et al. | 2016
- 5368
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Synthesis and biological evaluation of novel hydrogen sulfide releasing nicotinic acid derivativesSun, Yinxing / Zhang, Yusuo / Li, Yuyao / Cheng, Jian / Chen, Shiyu / Xiao, Yunqi / Ao, Guizhen et al. | 2016
- 5374
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Synthesis, biological evaluation and molecular docking study of N-arylbenzo[d]oxazol-2-amines as potential α-glucosidase inhibitorsWang, Guangcheng / Peng, Zhiyun / Wang, Jing / Li, Juan / Li, Xin et al. | 2016
- 5380
-
Human 15-LOX-1 active site mutations alter inhibitor binding and decrease potencyArmstrong, Michelle / van Hoorebeke, Christopher / Horn, Thomas / Deschamps, Joshua / Freedman, J. Cody / Kalyanaraman, Chakrapani / Jacobson, Matthew P. / Holman, Theodore et al. | 2016
- 5388
-
In silico and in vitro methods to identify ebola virus VP35-dsRNA inhibitorsGlanzer, Jason G. / Byrne, Brendan M. / McCoy, Aaron M. / James, Ben J. / Frank, Joshua D. / Oakley, Greg G. et al. | 2016
- 5393
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Design, synthesis, and biological characterization of novel PEG-linked dimeric modulators for CXCR4Yang, Yilei / Gao, Mei / Zhang, Qinghao / Zhang, Chaozai / Yang, Xiaohong / Huang, Ziwei / An, Jing et al. | 2016
- 5400
-
A new Suzuki synthesis of triphenylethylenes that inhibit aromatase and bind to estrogen receptors α and βZhao, Li-Ming / Jin, Hai-Shan / Liu, Jinzhong / Skaar, Todd C. / Ipe, Joseph / Lv, Wei / Flockhart, David A. / Cushman, Mark et al. | 2016
- 5410
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1,2,3-Triazole-based inhibitors of Porphyromonas gingivalis adherence to oral streptococci and biofilm formationPatil, Pravin C. / Tan, Jinlian / Demuth, Donald R. / Luzzio, Frederick A. et al. | 2016
- 5418
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New potently bioactive alkaloids from Crinum erubescensPresley, Christopher C. / Krai, Priscilla / Dalal, Seema / Su, Qingxi / Cassera, Maria / Goetz, Michael / Kingston, David G.I. et al. | 2016
- 5423
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Synthesis of (benzimidazol-2-yl)aniline derivatives as glycogen phosphorylase inhibitorsGalal, Shadia A. / Khattab, Muhammad / Andreadaki, Fotini / Chrysina, Evangelia D. / Praly, Jean-Pierre / Ragab, Fatma A.F. / El Diwani, Hoda I. et al. | 2016
- 5431
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Optimization and biological evaluation of celastrol derivatives as Hsp90–Cdc37 interaction disruptors with improved druglike propertiesJiang, Fen / Wang, Hui-Jie / Bao, Qi-Chao / Wang, Lei / Jin, Yu-Hui / Zhang, Qiong / Jiang, Di / You, Qi-Dong / Xu, Xiao-Li et al. | 2016
- 5440
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Synthesis and bioactivity of novel isoxazole chalcone derivatives on tyrosinase and melanin synthesis in murine B16 cells for the treatment of vitiligoNiu, Chao / Yin, Li / Nie, Li Fei / Dou, Jun / Zhao, Jiang Yu / Li, Gen / Aisa, Haji Akber et al. | 2016
- 5449
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Discovery of novel free fatty acid receptor 1 agonists bearing triazole core via click chemistryLi, Zheng / Yang, Jianyong / Wang, Xuekun / Li, Huilan / Liu, Chunxia / Wang, Nasi / Huang, Wenlong / Qian, Hai et al. | 2016
- 5455
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Structure–activity relationship studies of non-carboxylic acid peroxisome proliferator-activated receptor α/δ (PPARα/δ) dual agonistsOkazaki, Shogo / Shioi, Ryuta / Noguchi-Yachide, Tomomi / Ishikawa, Minoru / Makishima, Makoto / Hashimoto, Yuichi / Yamaguchi, Takao et al. | 2016
- 5462
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8-Substituted 1,3-dimethyltetrahydropyrazino[2,1-f]purinediones: Water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitorsBrunschweiger, Andreas / Koch, Pierre / Schlenk, Miriam / Rafehi, Muhammad / Radjainia, Hamid / Küppers, Petra / Hinz, Sonja / Pineda, Felipe / Wiese, Michael / Hockemeyer, Jörg et al. | 2016
- 5481
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Free fatty acid receptor 1 (GPR40) agonists containing spirocyclic periphery inspired by LY2881835Krasavin, Mikhail / Lukin, Alexey / Bagnyukova, Daria / Zhurilo, Nikolay / Zahanich, Ihor / Zozulya, Sergey / Ihalainen, Jouni / Forsberg, Markus M. / Lehtonen, Marko / Rautio, Jarkko et al. | 2016
- 5495
-
Design and synthesis of triarylacrylonitrile analogues of tamoxifen with improved binding selectivity to protein kinase CCarpenter, Colleen / Sorenson, Roderick J. / Jin, Yafei / Klossowski, Szymon / Cierpicki, Tomasz / Gnegy, Margaret / Showalter, Hollis D. et al. | 2016
- 5505
-
Synthesis and biological evaluation of azole-diphenylpyrimidine derivatives (AzDPPYs) as potent T790M mutant form of epidermal growth factor receptor inhibitorsSong, Zhendong / Jin, Yue / Ge, Yang / Wang, Changyuan / Zhang, Jianbin / Tang, Zeyao / Peng, Jinyong / Liu, Kexin / Li, Yanxia / Ma, Xiaodong et al. | 2016
- 5513
-
Thioflavones as novel neuroprotective agentsRavishankar, Divyashree / Corona, Giulia / Hogan, Stephanie M. / Spencer, Jeremy P.E. / Greco, Francesca / Osborn, Helen M.I. et al. | 2016
- 5521
-
Investigation of C-5 alkynyl (alkynyloxy or hydroxymethyl) and/or N-3 propynyl substituted pyrimidine nucleoside analogs as a new class of antimicrobial agentsGarg, Saurabh / Shakya, Neeraj / Srivastav, Naveen C. / Agrawal, Babita / Kunimoto, Dennis Y. / Kumar, Rakesh et al. | 2016
- 5534
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Scaffold-hopping from xanthines to tricyclic guanines: A case study of dipeptidyl peptidase 4 (DPP4) inhibitorsPissarnitski, Dmitri A. / Zhao, Zhiqiang / Cole, David / Wu, Wen-Lian / Domalski, Martin / Clader, John W. / Scapin, Giovanna / Voigt, Johannes / Soriano, Aileen / Kelly, Theresa et al. | 2016
- 5546
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Exploration of substituted arylpiperazine–tetrazoles as promising dual norepinephrine and dopamine reuptake inhibitorsPaudel, Suresh / Acharya, Srijan / Yoon, Goo / Kim, Kyeong-Man / Cheon, Seung Hoon et al. | 2016
- 5556
-
Anti-tubercular activities of 5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidin-4-amine analogues endowed with high activity toward non-replicative Mycobacterium tuberculosisSamala, Ganesh / Brindha Devi, Parthiban / Saxena, Shalini / Gunda, Saritha / Yogeeswari, Perumal / Sriram, Dharmarajan et al. | 2016
- 5565
-
Design, synthesis, crystal structure, biological evaluation and molecular docking studies of carbazole-arylpiperazine derivativesXu, Wei / Huang, Junjun / Shao, Binhao / Xu, Xingjie / Jiang, Renwang / Yuan, Mu et al. | 2016
- 5573
-
New inhibitors of tyrosyl-DNA phosphodiesterase I (Tdp 1) combining 7-hydroxycoumarin and monoterpenoid moietiesKhomenko, Tatyana / Zakharenko, Alexandra / Odarchenko, Tatyana / Arabshahi, Homayon John / Sannikova, Victoriya / Zakharova, Olga / Korchagina, Dina / Reynisson, Jóhannes / Volcho, Konstantin / Salakhutdinov, Nariman et al. | 2016
- 5582
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Arylsulfonamide derivatives of (aryloxy)ethyl pyrrolidines and piperidines as α1-adrenergic receptor antagonist with uro-selective activityRak, Aleksandra / Canale, Vittorio / Marciniec, Krzysztof / Żmudzki, Paweł / Kotańska, Magdalena / Knutelska, Joanna / Siwek, Agata / Stachowicz, Gabriela / Bednarski, Marek / Nowiński, Leszek et al. | 2016
- 5592
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Synthesis, characterization, and evaluation of (E)-methyl 2-((2-oxonaphthalen-1(2H)-ylidene)methylamino)acetate as a biological agent and an anion sensorZeyrek, Celal Tuğrul / Boyacioğlu, Bahadir / Yıldız, Mustafa / Ünver, Hüseyin / Yolal, Devrim / Demir, Neslihan / Elmali, Ayhan / Tadesse, Solomon / Aslan, Kadir et al. | 2016
- 5602
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Development of 6-arylcoumarins as nonsteroidal progesterone antagonists. Structure–activity relationships and fluorescence propertiesKinoshita, Marie / Negishi, Mai / Sakai, Haruka / Hirano, Tomoya / Mori, Shuichi / Fujii, Shinya / Kagechika, Hiroyuki / Tanatani, Aya et al. | 2016
- 5611
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Design and synthesis of novel HDAC8 inhibitory 2,5-disubstituted-1,3,4-oxadiazoles containing glycine and alanine hybrids with anti cancer activityPidugu, Vijaya Rao / Yarla, Nagendra Sastry / Pedada, Srinivasa Rao / Kalle, Arunasree M. / Satya, A. Krishna et al. | 2016
- 5618
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Analysis of quinolinequinone reactivity, cytotoxicity, and anti-HIV-1 propertiesAlfadhli, Ayna / Mack, Andrew / Harper, Logan / Berk, Sam / Ritchie, Christopher / Barklis, Eric et al. | 2016
- 5626
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Synthesis of phenylpiperazine derivatives of 1,4-benzodioxan as selective COX-2 inhibitors and anti-inflammatory agentsSun, Juan / Wang, Su / Sheng, Gui-Hua / Lian, Zhi-Min / Liu, Han-Yu / Zhu, Hai-Liang et al. | 2016
- 5633
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Identification of 5,6-dihydroimidazo[2,1-b]thiazoles as a new class of antimicrobial agentsLi, Yangmei / Bionda, Nina / Fleeman, Renee / Wang, Hongjie / Ozawa, Akihiko / Houghten, Richard A. / Shaw, Lindsey et al. | 2016
- 5639
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Discovery of O 6-benzyl glaziovianin A, a potent cytotoxic substance and a potent inhibitor of α,β-tubulin polymerizationHayakawa, Ichiro / Shioda, Shuya / Chinen, Takumi / Hatanaka, Taisei / Ebisu, Haruna / Sakakura, Akira / Usui, Takeo / Kigoshi, Hideo et al. | 2016
- 5646
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Design, synthesis, and structure–activity relationship of novel and effective apixaban derivatives as FXa inhibitors containing 1,2,4-triazole/pyrrole derivatives as P2 binding elementWang, Yong / Sun, Xiaoqing / Yang, Di / Guo, Zhuang / Fan, Xuxu / Nie, Minhua / Zhang, Feng / Liu, Yue / Li, Yue / Wang, Yulin et al. | 2016
- IFC
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Editorial board| 2016