ENHANCED INHIBITION OF HIV-1 REPLICATION IN MACROPHAGES BY ANTISENSE OLIGONUCLEOTIDES, RIBOZYMES AND ACYCLIC NUCLEOSIDE PHOSPHONATE ANALOGS DELIVERED IN pH-SENSITIVE LIPOSOMES (Unknown)
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In:
Nucleosides, Nucleotides and Nucleic Acids
;
20
, 4-7
;
515-523
;
2001
- Article (Journal) / Electronic Resource
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Title:ENHANCED INHIBITION OF HIV-1 REPLICATION IN MACROPHAGES BY ANTISENSE OLIGONUCLEOTIDES, RIBOZYMES AND ACYCLIC NUCLEOSIDE PHOSPHONATE ANALOGS DELIVERED IN pH-SENSITIVE LIPOSOMES
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Contributors:Düzgünes, N. ( author ) / Simões, S. ( author ) / Slepushkin, V. ( author ) / Pretzer, E. ( author ) / Rossi, J. J. ( author ) / De Clercq, E. ( author ) / Antao, V. P. ( author ) / Collins, M. L. ( author ) / Pedroso de Lima, M. C. ( author )
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Published in:Nucleosides, Nucleotides and Nucleic Acids ; 20, 4-7 ; 515-523
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Publisher:
- New search for: Taylor & Francis Group
-
Publication date:2001-03-31
-
Size:9 pages
-
ISSN:
-
DOI:
-
Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:Unknown
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Source:
Table of contents – Volume 20, Issue 4-7
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 271
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ACYCLIC/CARBOCYCLIC GUANOSINE ANALOGUES AS ANTI-HERPESVIRUS AGENTSDe Clercq, E. / Andrei, G. / Snoeck, R. / De Bolle, L. / Naesens, L. / Degrève, B. / Balzarini, J. / Zhang, Y. / Schols, D. / Leyssen, P. et al. | 2001
- 287
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NOVEL ARYL SUBSTITUTED BICYCLIC FURO NUCLEOSIDES AS EXTREMELY POTENT AND SELECTIVE ANTI-VZV AGENTSMcGuigan, Christopher / Barucki, Hubert / Carangio, Antonella / Blewett, Sally / Srinivasan, Sheila / Andrei, Graciela / Snoeck, Robert / De Clercq, Erik / Balzarini, Jan et al. | 2001
- 297
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ACTIVATION OF ANTI-REVERSE TRANSCRIPTASE NUCLEOTIDE ANALOGS BY NUCLEOSIDE DIPHOSPHATE KINASE: IMPROVEMENT BY α-BORANOPHOSPHATE SUBSTITUTIONSchneider, Benoit / Meyer, Philippe / Sarfati, Simon / Mulard, Laurence / Guerreiro, Catherine / Boretto, Joëlle / Janin, Joël / Véron, Michel / Deville-Bonne, Dominique / Canard, Bruno et al. | 2001
- 297
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Activation of Anti-reverse Transcriptase Nucleotide Analogs by Nucleoside Diphosphate Kinase: Improvement by a-Boranophosphate SubstitutionSchneider, B. et al. | 2001
- 307
-
SYNTHESIS, HYDROLYSIS AND ANTI-EBV ACTIVITY OF A SERIES OF 3′-MODIFIED cycloSal-BVDUMP PRONUCLEOTIDESMeier, C. / Lomp, A. / Meerbach, A. / Wutzler, P. et al. | 2001
- 315
-
DESIGN OF NEW MONONUCLEOTIDE PRODRUGS: ARYL (SATE) PHOSPHOTRIESTER DERIVATIVESPeyrottes, S. / Schlienger, N. / Beltran, T. / Lefebvre, I. / Pompon, A. / Gosselin, G. / Aubertin, A.-M. / Imbach, J.-L. / Périgaud, C. et al. | 2001
- 323
-
Synthesis and Anticancer Activity of 4-Amino-5-oxo-8-(b-D- xylofuranosyl)pyrido(2,3-d)pyrimidinePietrzkowski, Z. et al. | 2001
- 323
-
SYNTHESIS AND ANTICANCER ACTIVITY OF 4-AMINO-5-OXO-8-(β-D-XYLOFURANOSYL) PYRIDO[2,3-d]PYRIMIDINEPietrzkowski, Zbigniew / Girardet, Jean-Luc / Esler, Cathey / Wang, Guangyi et al. | 2001
- 329
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SYNTHESIS AND ANTIVIRAL ACTIVITY OF METHYLENEDIFLUOROCYCLOPROPANE ANALOGUES OF NUCLEOSIDESWang, R. / Ksebati, M. B. / Drach, J. C. / Zemlicka, J. et al. | 2001
- 333
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RIBOSE MODIFIED NUCLEOSIDES AND NUCLEOTIDES AS LIGANDS FOR PURINE RECEPTORSJacobson, K. A. / Ravi, R. G. / Nandanan, E. / Kim, H. S. / Moro, S. / Kim, Y. C. / Lee, K. / Barak, D. / Marquez, V. E. / Ji, X. D. et al. | 2001
- 343
-
2-SUBSTITUTED PI SYSTEM DERIVATIVES OF ADENOSINE THAT ARE CORONARY VASODILATORS ACTING VIA THE A2A ADENOSINE RECEPTORZablocki, J. / Palle, V. / Blackburn, B. / Elzein, E. / Nudelman, G. / Gothe, S. / Gao, Z. / Li, Z. / Meyer, S. / Belardinelli, L. et al. | 2001
- 361
-
FLUORESCENCE RESONANCE ENERGY TRANSFER DYE NUCLEOTIDE TERMINATORS: A NEW SYNTHETIC APPROACH FOR HIGH-THROUGHOUT DNA SEQUENCINGNampalli, Satyam / Khot, Mahesh / Nelson, John R. / Flick, Parke K. / Fuller, Carl W. / Kumar, Shiv et al. | 2001
- 369
-
DESIGN OF MULTIDYE SYSTEMS FOR FRET-BASED APPLICATIONSShchepinov, Mikhail S. / Korshun, Vladimir A. et al. | 2001
- 375
-
ANALYSIS OF ANTI-HIV NUCLEOSIDE INHIBITORS BY CAPILLARY ELECTROPHORESIS-ELECTROSPRAY IONIZATION MASS SPECTROMETRYAgrofoglio, L. A. / Cahours, X. / Tran, T. T. / Dessans, H. / Kieda, C. / Morin, P. et al. | 2001
- 383
-
THE CONFORMATIONAL SPACE OF NASCENT PEPTIDE-ACCEPTING 3′-AMINOACYL RIBONUCLEOS(T)IDES: 1H NMR DATA AND AB INITIO CALCULATIONS OF PUROMYCIN AND SOME SYNTHETIC ANALOGSTrung, Nhat Quang Nguyen / Strazewski, Peter / Olsson, Martin / Ehrenberg, Måns et al. | 2001
- 385
-
UNDERSTANDING THE MODE OF ACTION OF L-NUCLEOSIDES AS ANTIVIRAL AGENTS: A MOLECULAR MODELING APPROACHLee, Kyeong / Chong, Youhoon / Chu, Chung K. et al. | 2001
- 389
-
LNA (Locked Nucleic Acid) and the Diastereoisomeric a-L-LNA: Conformational Tuning and High-Affinity Recognition of DNA-RNA TargetsWengel, J. et al. | 2001
- 389
-
LNA (LOCKED NUCLEIC ACID) AND THE DIASTEREOISOMERIC α-L-LNA: CONFORMATIONAL TUNING AND HIGH-AFFINITY RECOGNITION OF DNA/RNA TARGETSWengel, Jesper / Petersen, Michael / Nielsen, Kathrine E. / Jensen, Gitte A. / Håkansson, Anders E. / Kumar, Ravindra / Sørensen, Mads D. / Rajwanshi, Vivek K. / Bryld, Torsten / Jacobsen, Jens Peter et al. | 2001
- 397
-
THE ROLE OF ANTISENSE OLIGONUCLEOTIDES IN THE WAVE OF GENOMIC INFORMATIONBaker, Brenda F. et al. | 2001
- 401
-
TELOMERASE INHIBITORS – OLIGONUCLEOTIDE PHOSPHORAMIDATES AS POTENTIAL THERAPEUTIC AGENTSGryaznov, S. / Pongracz, K. / Matray, T. / Schultz, R. / Pruzan, R. / Aimi, J. / Chin, A. / Harley, C. / Shea-Herbert, B. / Shay, J. et al. | 2001
- 411
-
DNA TRIPLE-HELIX FORMATION AT PYRIMIDINE-PURINE INVERSION SITESParel, Serge P. / Marfurt, Judith / Leumann, Christian J. et al. | 2001
- 419
-
PNA-RELATED OLIGONUCLEOTIDE MIMICS AND THEIR EVALUATION FOR NUCLEIC ACID HYBRIDIZATION STUDIES AND ANALYSISEfimov, V. / Choob, M. / Buryakova, A. / Phelan, D. / Chakhmakhcheva, O. et al. | 2001
- 429
-
PROPERTIES OF ARABINONUCLEIC ACIDS (ANA & 20′F-ANA): IMPLICATIONS FOR THE DESIGN OF ANTISENSE THERAPEUTICS THAT INVOKE RNASE H CLEAVAGE OF RNADamha, M. J. / Noronha, A. M. / Wilds, C. J. / Trempe, J.-F. / Denisov, A. / Pon, R. T. / Gehring, K. et al. | 2001
- 441
-
RNA AND N3′ → P5′ KISSING APTAMERS TARGETED TO THE TRANS-ACTIVATION RESPONSIVE (TAR) RNA OF THE HUMAN IMMUNODEFICIENCY VIRUS-1Darfeuille, Fabien / Cazenave, Christian / Gryaznov, Sergei / Ducongé, Frédéric / Di Primo, Carmelo / Toulmé, Jean-Jacques et al. | 2001
- 451
-
INHIBITION OF (CYTOSINE C5)-METHYLTRANSFERASE BY OLIGONUCLEOTIDES CONTAINING FLEXIBLE (CYCLOPENTANE) AND CONFORMATIONALLY CONSTRAINED (BICYCLO[3.1.0]HEXANE) ABASIC SITESMarquez, Victor E. / Wang, Peiyuan / Nicklaus, Marc C. / Maier, Martin / Manoharan, Muthiah / Christman, Judith K. / Banavali, Nilesh K. / Mackerell, Alexander D.Jr. et al. | 2001
- 461
-
INTRACELLULAR Ca2+-MOBILIZING ADENINE NUCLEOTIDES. SYNTHESIS AND BIOLOGICAL ACTIVITY OF CYCLIC ADP-CARBOCYCLIC-RIBOSE AND C-GLYCOSIDIC ANALOG OF ADENOPHOSTIN AShuto, Satoshi / Fukuoka, Masayoshi / Abe, Hiroshi / Matsuda, Akira et al. | 2001
- 471
-
OLIGONUCLEOTIDE ANALOGUE INTERFERENCE WITH THE HIV-1 TAT PROTEIN-TAR RNA INTERACTIONArzumanov, Andrey / Walsh, Andrew P. / Liu, Xiaohai / Rajwanshi, Vivek K. / Wengel, Jesper / Gait, Michael J. et al. | 2001
- 481
-
6-OXOCYTIDINE CONTAINING OLIGONUCLEOTIDES INHIBIT THE HIV-1 INTEGRASE IN VITROBrodin, P. / Pinskaya, M. / Parsch, U. / Bischerour, J. / Leh, H. / Romanova, E. / Engels, J. W. / Gottikh, M. / Mouscadet, J. F. et al. | 2001
- 487
-
ZIDOVUDINE (AZT) RESISTANCE IN H9 CELLS DUE TO DECREASED TK EXPRESSION IS ASSOCIATED WITH HYPERMETHYLATION OF TK GENEGröschel, B. / Höver, G. / Doerr, H. W. / Cinatl, J.Jr. et al. | 2001
- 493
-
STRUCTURAL, DYNAMIC, AND ENZYMATIC PROPERTIES OF MIXED α/β-OLIGONUCLEOTIDES CONTAINING POLARITY REVERSALSGermann, M. W. / Aramini, J. M. / Kalisch, B. W. / van de Sande, J. H. et al. | 2001
- 493
-
Structural, Dynamic, and Enzymatic Properties of Mixed a-b-Oligonucleotides Containing Polarity ReversalsGermann, M.W. et al. | 2001
- 501
-
ANALOGS OF GUANINE NUCLEOSIDE TRIPHOSPHATES FOR SEQUENCING APPLICATIONSMcDougall, Mark G. / Sun, Lei / Livshin, Inna / Hosta, Louis P. / McArdle, Bernard F. / Samols, Sui-Bi / Fuller, Carl W. / Kumar, Shiv et al. | 2001
- 507
-
2′-MODIFIED OLIGONUCLEOTIDES FROM METHOXYOXALAMIDO AND SUCCINIMIDO PRECURSORS: SYNTHESIS, PROPERTIES, AND APPLICATIONSPolushin, N. / Malykh, A. / Malykh, O. / Zenkova, M. / Chumakova, N. / Vlassov, V. / Kozyavkin, S. et al. | 2001
- 515
-
ENHANCED INHIBITION OF HIV-1 REPLICATION IN MACROPHAGES BY ANTISENSE OLIGONUCLEOTIDES, RIBOZYMES AND ACYCLIC NUCLEOSIDE PHOSPHONATE ANALOGS DELIVERED IN pH-SENSITIVE LIPOSOMESDüzgünes, N. / Simões, S. / Slepushkin, V. / Pretzer, E. / Rossi, J. J. / De Clercq, E. / Antao, V. P. / Collins, M. L. / Pedroso de Lima, M. C. et al. | 2001
- 525
-
PHOTOLITHOGRAPHIC SYNTHESIS OF HIGH-DENSITY OLIGONUCLEOTIDE PROBE ARRAYSBarone, Anthony D. / Beecher, Jody E. / Bury, Paul A. / Chen, Chuan / Doede, Tina / Fidanza, Jacqueline A. / McGall, Glenn H. et al. | 2001
- 533
-
HIGH CAPACITY SUBSTRATES AS A PLATFORM FOR A DNA PROBE ARRAY GENOTYPING ASSAYFidanza, Jacqueline / Glazer, Marc / Mutnick, Daniel / McGall, Glenn / Frank, Curt et al. | 2001
- 539
-
SYNTHESIS OF PEPTIDE-OLIGONUCLEOTIDE PHOSPHOROTHIOATE CONJUGATES BY CONVERGENT OR STEPWISE SOLID-PHASE STRATEGIESAntopolsky, Maxim / Azhayev, Alex et al. | 2001
- 551
-
NOVEL CLASS OF DNA BINDING MOTIFS BASED ON BISTETRAHYDROFURAN AND BISFURAN SKELETON WITH LONG ALKYL CHAINSSasaki, Shigeki / Shibata, Takayuki / Torigoe, Hidemine / Shibata, Yosinori / Maeda, Minoru et al. | 2001
- 559
-
COVALENT MODIFICATION AND SURFACE IMMOBILIZATION OF NUCLEIC ACIDS VIA THE DIELS-ALDER BIOCONJUGATION METHODHusar, Gregory M. / Anziano, Dominick J. / Leuck, Michael / Sebesta, David P. et al. | 2001
- 567
-
A CASE STUDY: OLIGONUCLEOTIDE PURIFICATION FROM GRAM TO HUNDRED GRAM SCALEDeshmukh, Ranjit R. / Eriksson, Kjell-Ove / Moore, Peter / Cole, Douglas L. / Sanghvi, Yogesh S. et al. | 2001
- 577
-
8-AZA-7-DEAZAADENINE AND 7-DEAZAGUANINE: SYNTHESIS AND PROPERTIES OF NUCLEOSIDES AND OLIGONUCLEOTIDES WITH NUCLEOBASES LINKED AT POSITION-8Seela, F. / Debelak, H. et al. | 2001
- 587
-
SYNTHESIS OF NEW CLASSES OF BORON-CONTAINING NUCLEOTIDESLin, Jinlai / Shaw, Barbara Ramsay et al. | 2001
- 597
-
ANTI-HBV SPECIFIC β-L-2′-DEOXYNUCLEOSIDESBryant, Martin L. / Bridges, Edward G. / Placidi, Laurent / Faraj, Abdesslem / Loi, Anna-Giulia / Pierra, Claire / Dukhan, David / Gosselin, Gilles / Imbach, Jean-Louis / Hernandez, Brenda et al. | 2001
- 597
-
Anti-HBV Specific b-L-2'-DeoxynucleosidesBryant, M.L. et al. | 2001
- 609
-
1-(3-C-ETHYNYL-β-D-RIBO-PENTOFURANOSYL)CYTOSINE (ECYD, TAS-106)1: ANTITUMOR EFFECT AND MECHANISM OF ACTIONAzuma, Atsushi / Matsuda, Akira / Sasaki, Takuma / Fukushima, Masakazu et al. | 2001
- 609
-
1-(3-C-Ethynyl-b-D-ribo-pentofuranosyl)cytosine (ECyd, tas-106)1: Antitumor Effect and Mechanism of ActionAzuma, A. et al. | 2001
- 621
-
PRACTICAL SYNTHESIS, SEPARATION, AND STEREOCHEMICAL ASSIGNMENT OF THE PMPA PRO-DRUG GS-7340Chapman, H. / Kernan, M. / Prisbe, E. / Rohloff, J. / Sparacino, M. / Terhorst, T. / Yu, R. et al. | 2001
- 629
-
AN ASSAY SYSTEM TO DETECT THE SELECTIVE ADVANTAGE OF ANTI-HIV RIBOZYME EXPRESSING CD4+ T-LYMPHOCYTESKlein, Stefan A. / Klebba, Christian / Engels, Joachim W. et al. | 2001
- 635
-
TENOFOVIR (PMPA) IS LESS SUSCEPTIBLE TO PYROPHOSPHOROLYSIS AND NUCLEOTIDE-DEPENDENT CHAIN-TERMINATOR REMOVAL THAN ZIDOVUDINE OR STAVUDINENaeger, Lisa K. / Margot, Nicolas A. / Miller, Michael D. et al. | 2001
- 641
-
HUMAN RENAL ORGANIC ANION TRANSPORTER 1 (hOAT1) AND ITS ROLE IN THE NEPHROTOXICITY OF ANTIVIRAL NUCLEOTIDE ANALOGSCihlar, Tomas / Ho, Edmund S. / Lin, Deborah C. / Mulato, Andrew S. et al. | 2001
- 649
-
SYNTHESIS AND ANTIPROLIFERATIVE ACTIVITY OF SOME 4′-C-HYDROXYMETHYL-α- AND -β-D-ARABINO-PENTOFURANOSYL PYRIMIDINE NUCLEOSIDESGriffon, Jean-François / Montgomery, John A. / Secrist, John A.III et al. | 2001
- 649
-
Synthesis and Antiproliferative Activity of Some 4'-C-Hydroxymethyl-a- and -b-D-arabino-Pentofuranosyl Pyrimidine NucleosidesGriffon, J.-F. et al. | 2001
- 653
-
SYNTHESIS AND IN VITRO EVALUATION OF NOVEL ANTI-VARICELLA-ZOSTER VIRUS (VZV) NUCLEOSIDESCarangio, Antonella / McGuigan, Christopher / Cahard, D. / Andrei, Graciela / Snoeck, Robert / De Clercq, Erik / Balzarini, Jan et al. | 2001
- 657
-
STRUCTURE-ACTIVITY RELATIONSHIPS OF APIO NUCLEOSIDES AS POTENTIAL ANTIVIRAL AGENTSJeong, Lak Shin / Moon, Hyung Ryong / Hong, Jun Hee / Yoo, Su Jeong / Choi, Won Jun / Kim, Hea Ok / Ahn, Hee Sung / Baek, Hye Woo / Chun, Moon Woo / Kim, Hee-Doo et al. | 2001
- 661
-
SYNTHESIS OF CARBOCYCLIC PHOSPHONONUCLEOSIDESLegeret, B. / Sarakauskaite, Z. / Pradaux, F. / Saito, Y. / Tumkevicius, S. / Agrofoglio, L. A. et al. | 2001
- 665
-
SYNTHESIS AND ANTIVIRAL ACTIVITY OF D- AND L-2′-AZIDO-2′,3′-DIDEOXY-4′-THIOPYRIMIDINE AND PURINE NUCLEOSIDESJeong, Lak Shin / Kim, Yun Ha / Kim, Hea Ok / Yoo, Su Jeong / Park, Yong Hee / Yeon, Sook Hee / Chun, Moon Woo / Kim, Hee-Doo et al. | 2001
- 669
-
DNA SEQUENCE RECOGNITION BY NFκB p50 HOMODIMER: STRICT AND OBSCURE RECOGNITION SITES IN THE BINDING SEQUENCEKittaka, Atsushi / Takayama, Hiroaki / Kurihara, Masaaki / Horii, Chikafumi / Tanaka, Hiromichi / Miyasaka, Tadashi / Inoue, Jun-ichiro et al. | 2001
- 669
-
DNA Sequence Recognition by NFkB p50 Homodimer: Strict and Obscure Recognition Sites in the Binding SequenceKittaka, A. et al. | 2001
- 673
-
FOUR COLOR FRET DYE NUCLEOTIDE TERMINATORS FOR DNA SEQUENCINGRao, T. Sudhakar / Nampalli, Satyam / Lavrenov, Kate / Zhang, Weihong / Xiao, Haiguang / Nelson, John / Kumar, Shiv et al. | 2001
- 677
-
Design Synthesis of Novel Fluorocyclopropanoid NucleosidesLee, Y.R. et al. | 2001
- 677
-
DESIGN AND SYNTHESIS OF NOVEL FLUOROCYCLOPROPANOID NUCLEOSIDESLee, Young Rang / Park, Ju-Hyun / Jeon, Raok / Jeong, Lak Shin / Chun, Moon Woo / Kim, Hee-Doo et al. | 2001
- 681
-
NOVEL NUCLEOSIDES WITH VINYL FLUORIDE OR VINYL BROMIDE MOIETY AS OPEN-CHAIN ANALOGS OF NEPLANOCIN AChoi, Myung-Hee / Lee, Chong-Kyo / Jeong, Lak Shin / Chun, Moon Woo / Kim, Hee-Doo et al. | 2001
- 685
-
MECHANISM OF INACTIVATION OF S-ADENOSYL-L-HOMOCYSTEINE HYDROLASE BY 5′-DEOXY-5′-S-ALLENYLTHIOADENOSINE AND 5′-DEOXY-5′-S-PROPYNYLTHIOADENOSINEGuillerm, G. / Guillerm, D. / Witkowski-Vandenplas, C. et al. | 2001
- 689
-
INACTIVATION OF S-ADENOSYL-L-HOMOCYSTEINE HYDROLASE WITH FLUORINATED ANALOGS OF 2′- AND 3′-DEOXY-5′-METHYLTHIOADENOSINEGuillerm, D. / Guillerm, G. / Witkowski-Vandenplas, C. et al. | 2001
- 695
-
SYNTHESIS AND BIOLOGICAL EVALUATION OF BORONATED NUCLEOSIDES FOR BORON NEUTRON CAPTURE THERAPY (BNCT) OF CANCERTjarks, W. / Wang, J. / Chandra, S. / Ji, W. / Zhuo, J. / Lunato, A. J. / Boyer, C. / Li, Q. / Usova, E. V. / Eriksson, S. et al. | 2001
- 699
-
SYNTHESIS OF NOVEL 3′-DEOXY-3′-C-HYDROXYMETHYL NUCLEOSIDES WITH CONFORMATIONALLY RIGID SUGAR MOIETY AS POTENTIAL ANTIVIRAL AGENTSChun, Moon Woo / Kim, Myung Jung / Jo, Un Hee / Kim, Joong Hyup / Kim, Hee-Doo / Jeong, Lak Shin et al. | 2001
- 703
-
SYNTHESIS OF NOVEL D- AND L-3′-DEOXY-3′-C-HYDROXYMETHYL NUCLEOSIDE WITH EXOCYCLIC METHYLENE AS POTENTIAL RIBONUCLEOTIDE REDUCTASE INHIBITORChun, Moon Woo / Kim, Myung Jung / Jo, Un Hee / Kim, Joong Hyup / Kim, Hee-Doo / Jeong, Lak Shin et al. | 2001
- 707
-
“SECOND GENERATION” OF TSAO COMPOUNDS DIRECTED AGAINST HIV-1 TSAO-RESISTANT STRAINSLobatón, E. / Velázquez, S. / Pérez-Pérez, M. J. / Jimeno, M. L. / San-Félix, A. / De Clercq, E. / Balzarini, J. / Camarasa, M. J. et al. | 2001
- 711
-
4″-H-TSAO-T, A NOVEL PROTOTYPE IN THE HIV-1 SPECIFIC TSAO FAMILYLobatón, E. / Velázquez, S. / San-Félix, A. / De Clercq, E. / Balzarini, J. / Camarasa, M. J. et al. | 2001
- 715
-
A NEW CLASS OF ANTI-HIV-1 OLIGONUCLEOTIDE TARGETED TO THE POLYPURINE TRACT OF VIRAL RNAHiratou, Takashi / Miyano-Kurosaki, Naoko / Gushima, Hiroshi / Takaku, Hiroshi et al. | 2001
- 719
-
EFFECTIVE SUPPRESSION OF HIV-1 GENE EXPRESSION BY A MAMMALIAN tRNA 3′ PROCESSING ENDORIBONUCLEASE AND EXTERNAL GUIDE SEQUENCE OLIGOZYMESKitano, Michiko / Barnor, Jaco S. / Miyano-Kurosaki, Naoko / Endo, Yumihiko / Yukita, Masakazu / Takeuchi, Hiroaki / Tamura, Yutaka / Takai, Kazuyuki / Nashimoto, Masayuki / Takaku, Hiroshi et al. | 2001
- 723
-
INHIBITION OF HIV-1 REPLICATION BY THE CRE-LOXP HAMMERHEAD RIBOZYMEHabu, Yuichiro / Miyano-Kurosaki, Naoko / Takeuchi, Hiroaki / Matsumoto, Norihiko / Tamura, Yutaka / Takaku, Hiroshi et al. | 2001
- 727
-
(D)- AND (L)-CYCLOHEXENYL-G, A NEW CLASS OF ANTIVIRAL AGENTS: SYNTHESIS, CONFORMATIONAL ANALYSIS, MOLECULAR MODELING, AND BIOLOGICAL ACTIVITYWang, J. / Froeyen, M. / Hendrix, C. / Andrei, C. / Snoeck, R. / Lescrinier, E. / De Clercq, E. / Herdewijn, P. et al. | 2001
- 731
-
SYNTHESIS AND BIOLOGICAL EVALUATION OF PYRIDIN-2-ONE NUCLEOSIDESHuntley, Caroline M. / Cotterill, Ann S. / Maillard, Jean-Yves / Balzarini, Jan / Simons, Claire et al. | 2001
- 735
-
ISONUCLEOSIDES INCORPORATING UNIVERSAL BASESNair, Vasu / Sosnouski, David S. / Zhu, Qingming et al. | 2001
- 739
-
A NEW PROCEDURE FOR THE PHOSPHORYLATION OF NUCLEOSIDES: APPLICATION TO THE DISCOVERY OF INHIBITORS OF HIV INTEGRASENair, Vasu / Taktakishvili, Michael et al. | 2001
- 743
-
SYNTHESIS AND BIOLOGICAL ACTIVITY OF 4′-THIO-L-XYLOFURANOSYL NUCLEOSIDESTiwari, Kamal N. / Messini, Lea / Montgomery, John A. / Secrist, John A.III et al. | 2001
- 747
-
SYNTHESIS AND BIOLOGICAL ACTIVITY OF 4′-C-HYDROXYMETHYL-2′-FLUORO-D-ARABINOFURANOSYLPURINE NUCLEOSIDESShortnacy-Fowler, A. T. / Tiwari, K. N. / Montgomery, J. A. / Secrist, J. A.III et al. | 2001
- 751
-
SYNTHESIS AND STUDY OF A NEW SERIES OF PHOSPHORAMIDATE DERIVATIVES AS MONONUCLEOTIDE PRODRUGSEgron, David / Périgaud, Christian / Gosselin, Gilles / Aubertin, Anne-Marie / Imbach, Jean-Louis et al. | 2001
- 755
-
SYNTHESIS AND ANTIVIRAL EVALUATION OF 3′-C-TRIFLUOROMETHYL NUCLEOSIDE DERIVATIVES BEARING ADENINE AS THE BASEJeannot, Frédéric / Mathé, Christophe / Gosselin, Gilles et al. | 2001
- 759
-
Synthesis of 5-Chloro-1-(2,3-dideoxy-3-fluoro-b-D-glycero-hex-2- enopyranose-4-ulosyl)uracil as Potential Anticancer-Antiviral AgentKhan, A.R. et al. | 2001
- 759
-
SYNTHESIS OF 5-CHLORO-1-(2,3-DIDEOXY-3-FLUORO-β-D-GLYCERO-HEX-2-ENOPYRANOSE-4-ULOSYL)URACIL AS POTENTIAL ANTICANCER/ANTIVIRAL AGENTKhan, Abdul R. / Mulligan*, Kimberly X. / Ollapally, Abraham P. et al. | 2001
- 763
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BICYCLIC NUCLEOSIDE INHIBITORS OF VARICELLA-ZOSTER VIRUS (VZV): EFFECT OF TERMINAL UNSATURATION IN THE SIDE-CHAINSrinivasan, Sheila / McGuigan, Christopher / Andrei, Graciela / Snoeck, Robert / De Clercq, Erik / Balzarini, Jan et al. | 2001
- 767
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ANTI-HIV ACTIVITY OF NOVEL PHOSPHONATE DERIVATIVES OF AZT, d4T, AND ddAPokrovsky, A. G. / Pronayeva, T. R. / Fedyuk, N. V. / Shirokova, E. A. / Khandazhinskaya, A. L. / Tarusova, N. B. / Karpenko, I. L. / Krayevsky, A. A. et al. | 2001
- 771
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COUPLING OF 2,6-DISUBSTITUTED PURINES TO RIBOSE-MODIFIED SUGARSVittori, S. / Costanzi, S. / Lambertucci, C. / Volpini, R. / Cristalli, G. et al. | 2001
- 775
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SYNTHETIC PROCEDURE FOR THE PREPARATION OF NOVEL POTENT AND SELECTIVE A3 ADENOSINE RECEPTOR RADIOLIGANDSVolpini, R. / Costanzi, S. / Lambertucci, C. / Vittori, S. / Cristalli, G. et al. | 2001
- 781
-
INCREASED RNA AFFINITY OF HNA ANALOGUES BY INTRODUCING ALKOXY SUBSTITUENTS AT THE C-1 OR C-3 POSITIONVan Aerschot, A. / Meldgaard, M. / Volders, F. / Schepers, G. / Rozenski, J. / Herdewijn, P. et al. | 2001
- 785
-
CYCLOHEXENE NUCLEIC ACIDS (CeNA) FORM STABLE DUPLEXES WITH RNA AND INDUCE RNASE H ACTIVITYWang, J. / Verbeure, B. / Luyten, I. / Froeyen, M. / Hendrix, C. / Rosemeyer, H. / Seela, F. / Van Aerschot, A. / Herdewijn, P. et al. | 2001
- 789
-
SYNTHESIS OF OLIGONUCLEOSIDE BORANOPHOSPHATES VIA AN H-PHOSPHONATE METHOD WITHOUT NUCLEOBASE PROTECTIONSergueev, Dmitri S. / Sergueeva, Zinaida A. / Shaw, Barbara Ramsay et al. | 2001
- 797
-
α-OLIGONUCLEOTIDES WITH ANIONIC PHOSPHODIESTER AND CATIONIC PHOSPHORAMIDATE LINKAGES ENHANCED STABILITY OF DNA TRIPLE HELIXEhrenmann, F. / Vasseur, J.-J. / Debart, F. et al. | 2001
- 797
-
a-Oligonucleotides with Anionic Phosphodiester and Cationic Phosphoramidate Linkages Enhanced Stability of DNA Triple HelixEhrenmann, F. et al. | 2001
- 801
-
A NEW “NATIVE LIGATION” PROCEDURE FOR PEPTIDE-OLIGONUCLEOTIDE CONJUGATIONStetsenko, Dmitry A. / Gait, Michael J. et al. | 2001
- 805
-
POLYIMIDAZOLE CONJUGATED OLIGONUCLEOTIDES REACH THE NUCLEUS OF HELA CELLSMorvan, François / Castex, C. / Vivès, E. / Imbach, Jean-Louis et al. | 2001
- 809
-
RECOGNITION OF DNA BY STRAND INVASION WITH OLIGONUCLEOTIDE-SPERMINE CONJUGATESPotier, Pierre F. / Behr, Jean-Paul et al. | 2001
- 815
-
STACKING AND STABILITY OF RNA DUPLEXES CONTAINING FLUOROBENZENE AND FLUOROBENZIMIDAZOLE NUCLEOSIDESParsch, Jörg / Engels, Joachim W. et al. | 2001
- 819
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OLIGONUCLEOTIDES WITH ISOPOLAR PHOSPHONATE INTERNUCLEOTIDE LINKAGE: A NEW PERSPECTIVE FOR ANTISENSE COMPOUNDS?Rejman, D. / Snášel, J. / Liboska, R. / Točík, Z. / Pačes, O. / Králíková, Š. / Rinnová, M. / Koiš, P. / Rosenberg, I. et al. | 2001
- 825
-
Synthesis and Evaluation of a-LNAChristensen, N.K. et al. | 2001
- 825
-
SYNTHESIS AND EVALUATION OF α-LNAChristensen, Nanna K. / Dalskov, Jakob K. / Nielsen, Paul et al. | 2001
- 829
-
ANTISENSE PROPERTIES OF 2′-O-DIMETHYLAMINOOXYETHYL (2′-O-DMAOE) OLIGONUCLEOTIDESPrakash, Thazha P. / Kawasaki, Andrew M. / Johnston, Joseph F. / Graham, Mark J. / Condon, Thomas P. / Manoharan, Muthiah et al. | 2001
- 833
-
RAPID RNA CLEAVAGE USING AN ANTISENSE SYSTEM WITH TWO TERPYRIDINE · Cu(II) COMPLEXESInoue, Hideo / Furukawa, Takako / Tamura, Takashi / Kamada, Akihiro / Ohtsuka, Eiko et al. | 2001
- 837
-
UNNATURAL ENANTIOMERS OF 5-AZACYTIDINE ANALOGUES: SYNTHESES AND ENZYMATIC PROPERTIESGaubert, G. / Gosselin, G. / Eriksson, S. / Vita, A. / Maury, G. et al. | 2001
- 841
-
A CODE RELATING SEQUENCE TO STRUCTURE IN NUCLEIC ACIDSRemin, Mieczysław et al. | 2001
- 847
-
INTERACTION OF LNA OLIGONUCLEOTIDES WITH MDR1 PROMOTERChernolovskaya, E. L. / Koshkin, A. A. / Vlassov, V. V. et al. | 2001
- 851
-
Cu2+-DEPENDENT DNA-CLEAVING ACTIVITY OF ARENESKoval, O. A. / Chernolovskaya, E. L. / Litvak, V. V. / Vlassov, V. V. et al. | 2001
- 855
-
SIMULTANEOUS HPLC ANALYSIS OF HYDROPHOBIC PRODRUGS AND THEIR HYDROPHILIC METABOLITES IN BIOLOGICAL MEDIA WITHOUT SAMPLE PREPARATION. APPLICATION TO THE BIOTRANSFORMATION STUDIES OF PRONUCLEOTIDES DERIVED FROM 5-FLUOROURACILCoussot, G. / Lefebvre-Tournier, I. / Hollecker, L. / Gosselin, G. / Imbach, J.-L. / Pompon, A. et al. | 2001
- 859
-
INTERACTION OF OLIGONUCLEOTIDES WITH CELLULAR PROTEINSLaktionov, P. / Chelobanov, B. / Rykova, E. / Vlassov, V. et al. | 2001
- 863
-
GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE IS RESPONSIBLE FOR INTRANUCLEAR LOCALIZATION OF SOME OLIGONUCLEOTIDESTomasi, V. / Laktionov, P. P. / Bryksin, A. V. / Volod'ko, N. V. / Griffoni, C. / Rykova, E. Y. / Spisni, E. / Kraft, R. / Vlassov, V. V. et al. | 2001
- 869
-
5-PROPYNYLPYRIMIDINE NUCLEOSIDE DERIVATIVES: RATIONALLY DESIGNED MECHANISM-BASED INACTIVATORS OF THYMIDYLATE SYNTHASEKalman, Thomas I. / Nie, Zhe / Kamat, Ashwini et al. | 2001
- 873
-
INHIBITION OF IN VITRO PRE-mRNA SPLICING IN S. CEREVISIAE BY BRANCHED OLIGONUCLEOTIDESCarriero, S. / Braich, R. S. / Hudson, R. H. E. / Anglin, D. / Friesen, J. D. / Damha, M. J. et al. | 2001
- 879
-
SYNTHESIS OF 3′-THIOAMIDO-MODIFIED 3′-DEOXYTHYMIDINE-5′-TRIPHOSPHATES AND THEIR USE AS CHAIN TERMINATORS IN SANGER-DNA SEQUENCINGSchwarzer, K. / Wojczewski, C. / Engels, J. W. et al. | 2001
- 883
-
NOVEL PROPARGYLAMINE-LINKED NUCLEOSIDES FOR HIGH THROUGHPUT SNP GENOTYPING BY MALDI-TOF MSWenzel, Thomas / Fröhlich, Thomas / Strassburger, Kathrin / Richter, Susann / Bimmler, Jacqueline / Franke, Constance / Thomas, Isabell / Kostrzewa, Markus et al. | 2001
- 889
-
LIPOPLEX-MEDIATED STABLE GENE TRANSFER INTO HeLa CELLSSingh, Moganavelli / Balram, Sharda / Ariatti, Mario et al. | 2001
- 893
-
ROLLING CIRCLE AMPLIFICATION FOR SCORING SINGLE NUCLEOTIDE POLYMORPHISMSRösler, A. / Bailey, L. / Jones, S. / Briggs, J. / Cuss, S. / Horsey, I. / Kenrick, M. / Kingsmore, S. / Kent, L. / Pickering, J. et al. | 2001
- 895
-
THE USE OF (OLIGONUCLEOTIDE-MALEIC ANHYDRIDE COPOLYMER) CONJUGATES IN NUCLEIC ACID DIAGNOSTIC ASSAYS: EFFECT OF THE NUMBER OF OLIGONUCLEOTIDES PER POLYMER ON TEST SENSITIVITY IMPROVEMENTMinard-Basquin, C. / Chaix, C. / Pichot, C. et al. | 2001
- 901
-
SECO C-NUCLEOSIDE ANALOGS OF THE 1,2,4-TRIAZOLEEl Ashry, El Sayed H. / Awad, Laila F. et al. | 2001
- 903
-
2′-O-MODIFIED OLIGORIBONUCLEOTIDES WITH TERMINAL 3′-3′-INTERNUCLEOTIDE LINKAGE AND THEIR DERIVATIVESNovopashina, D. / Kuznetsova, M. / Venyaminova, A. et al. | 2001
- 909
-
DESIGN AND SIMPLE ROUTES OF SYNTHESIS OF OLIGONUCLEOTIDE CONJUGATES FOR STUDIES OF DNA TRIPLE HELIX FORMATIONGrimm, G. N. / Boutorine, A. S. / Lincoln, P. / Hélène, C. et al. | 2001
- 915
-
SITE-DIRECTED ALKYLATION TO CYTIDINE WITHIN DUPLEX BY THE OLIGONUCLEOTIDES CONTAINING FUNCTIONAL NUCLEOBASESNagatsugi, Fumi / Kawasaki, Takeshi / Tokuda, Natsuko / Maeda, Minoru / Sasaki, Shigeki et al. | 2001
- 921
-
SYNTHESIS OF SOME 2′- AND 3′-FLUOROALKYL SUBSTITUTED NUCLEOSIDES AND OLIGONUCLEOTIDESSerafinowski, Pawel J. / Brown, Catherine A. / Barnes, Colin L. et al. | 2001
- 927
-
SYNTHESIS AND PHOTOCHEMICAL BEHAVIOUR OF A T-T DIMER CONTAINING AN AMIDE LINKAGEThomas, Martial / Clivio, Pascale / Guillaume, Dominique / Fourrey, Jean-Louis et al. | 2001
- 927
-
Synthesis and Photochemical Behavior of a T-T Dimer Containing an Amide LinkageThomas, M. et al. | 2001
- 931
-
BENZYL-FUNCTIONALIZED cycloSal-d4T MONOPHOSPHATESRenze, J. / Plath, M. / Ducho, C. / Balzarini, J. / De Clercq, E. / Meier, C. et al. | 2001
- 935
-
SYNTHESIS OF N 2-ALKYLGUANOSINE USING MITSUNOBU REACTION AS A KEY STEPMaruyama, Tokumi / Yorikane, Aya / Kozai, Shigetada et al. | 2001
- 937
-
EFFICIENT SYNTHESIS OF D-[1′-13C]-RIBONUCLEOSIDES FOR INCORPORATION INTO OLIGO-RNASaito, Y. / Nyilas, A. / Agrofoglio, L. A. et al. | 2001
- 941
-
BORANE-AMINE COMPLEXES - VERSATILE REAGENTS IN THE CHEMISTRY OF NUCLEIC ACIDS AND THEIR ANALOGSSergueeva, Zinaida A. / Sergueev, Dmitri S. / Shaw, Barbara Ramsay et al. | 2001
- 947
-
PRO-OLIGONUCLEOTIDE SYNTHESIS USING ALLYL AND ALLYLOXYCARBONYL PROTECTIONS: DIRECT MALDI-TOF MS ANALYSIS ON SOLID SUPPORTSpinelli, N. / Vasseur, J.-J. / Hayakawa, Y. / Imbach, J.-L. et al. | 2001
- 951
-
STEP-BY-STEP CONTROL BY MALDI-TOF MS OF AN OLIGONUCLEOTIDE SYNTHESIS ON STANDARD CPG SOLID-SUPPORTMeyer, A. / Debart, F. / Imbach, J.-L. / Vasseur, J.-J. et al. | 2001
- 955
-
Synthesis of Some Acyclonucleosides a-(Pyrazolo(3,4-d)pyrimidin-4-ylthio)alkylamidesTaha, M.L. et al. | 2001
- 955
-
SYNTHESIS OF SOME ACYCLONUCLEOSIDES α-(PYRAZOLO[3,4-d]PYRIMIDIN-4-YLTHIO)-ALKYLAMIDESTaha, M. L. / Moukha-Chafiq, O. / Lazrek, H. B. / Vasseur, J. J. / Imbach, J. L. et al. | 2001
- 959
-
SYNTHESIS OF NEW HOMO AND HETERODINUCLEOSIDES CONTAINING THE 2′,3′-DIDEOXYNUCLEOSIDES AZT AND D4TTaourirte, M. / Lazrek, H. B. / Vasseur, J. J. / Ferrero, M. / Fernandez, S. / Gotor, V. et al. | 2001
- 963
-
DIRECT MALDI-TOF MS ANALYSIS OF OLIGONUCLEOTIDES ON SOLID SUPPORT THROUGH A PHOTOLABILE LINKERMeyer, A. / Spinelli, N. / Brès, J.-C. / Dell'Aquila, C. / Morvan, F. / Lefebvre, I. / Rayner, B. / Imbach, J.-L. / Vasseur, J.-J. et al. | 2001
- 967
-
5-(PHENYLTHIOMETHYL)-2′-DEOXYURIDINE AS AN EFFICIENT PHOTOREACTIVE PRECURSOR TO GENERATE SINGLE AND MULTIPLE LESIONS WITHIN DNA FRAGMENTSBellon, Sophie / Gasparutto, Didier / Romieu, Anthony / Cadet, Jean et al. | 2001
- 973
-
THE MOX/SUC PRECURSOR STRATEGIES: ROBUST WAYS TO CONSTRUCT FUNCTIONALIZED OLIGONUCLEOTIDESPolushin, N. et al. | 2001
- 977
-
RECOMBINANT BACTERIAL CELLS AS EFFICIENT BIOCATALYSTS FOR THE PRODUCTION OF NUCLEOSIDESSpoldi, E. / Ghisotti, D. / Calì, S. / Grisa, M. / Orsini, G. / Tonon, G. / Zuffi, G. et al. | 2001
- 981
-
METHYL 5-O-BENZOYL-2,3-OXAZOLE-D-RIBOFURANOSIDE: A USEFUL INTERMEDIATE FOR THE SYNTHESIS OF CONFORMATIONALLY RESTRAINED NUCLEOSIDESMolina, José / Maslen, Hannah L. / Simons, Claire et al. | 2001
- 985
-
MULTIPLE OLIGONUCLEOTIDE SYNTHESIS IN TANDEM ON SOLID-PHASE SUPPORTS FOR SMALL AND LARGE SCALE SYNTHESISPon, R. T. / Yu, S. / Sanghvi, Y. S. et al. | 2001
- 991
-
STUDIES OF A CHEMICALLY MODIFIED OLIGODEOXYNUCLEOTIDE CONTAINING A 5-ATOM AMIDE BACKBONE WHICH EXHIBITS IMPROVED BINDING TO RNAWilds, Christopher J. / Minasov, George / Natt, François / von Matt, Peter / Altmann, Karl-Heinz / Egli, Martin et al. | 2001
- 995
-
CHIMERIC RNA WITH MODIFIED BACKBONES: ALTERNATING METHYLENE(METHYLIMINO) LINKED PHOSPHODIESTER BACKBONE OLIGONUCLEOTIDES WITH 2′-OH AND 2′-OMe GROUPSPrhavc, Marija / Bhat, Balkrishen / Just, George / Dan Cook, P. / Manoharan, Muthiah et al. | 2001
- 999
-
SYNTHESIS AND STRUCTURAL STUDY OF PYRIMIDYL CARBOCYCLIC ANALOGUES OF NUCLEOSIDES BASED ON CYCLOPENTENE RINGSTerán, C. / Moa, M. J. González / Mosquera, R. / Santana, L. et al. | 2001
- 1003
-
SYNTHESIS OF 6-FORMYLURIDINE 5′-MONOPHOSPHATE: 6-FORMYL-UMPGroziak, Michael P. et al. | 2001
- 1007
-
EFFICIENT SYNTHESIS OF OLIGONUCLEOTIDE-PEPTIDE CONJUGATES ON LARGE SCALEDoronina, Svetlana O. / Guzaev, Andrei P. / Manoharan, Muthiah et al. | 2001
- 1011
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A NOVEL PROTECTING STRATEGY FOR INTERNUCLEOSIDIC PHOSPHATE AND PHOSPHOROTHIOATE GROUPSGuzaev, Andrei P. / Manoharan, Muthiah et al. | 2001
- 1015
-
SYNTHESIS OF CHIMERIC OLIGONUCLEOTIDES CONTAINING INTERNUCLEOSIDIC PHOSPHODIESTER AND S–PIVALOYLTHIOETHYL PHOSPHOTRIESTER RESIDUESGuzaev, Andrei P. / Bhat, Balkrishen / Balow, Guity / Manoharan, Muthiah et al. | 2001
- 1019
-
Synthesis and Properties of Novel Triphosphate Analogues: Ribonucleoside and Deoxyribonucleoside (a-P-BORANO, a-P-Thio)TriphosphatesLin, J. et al. | 2001
- 1019
-
SYNTHESIS AND PROPERTIES OF NOVEL TRIPHOSPHATE ANALOGUES: RIBONUCLEOSIDE AND DEOXYRIBONUCLEOSIDE (α-P-BORANO, α-P-THIO)TRIPHOSPHATESLin, Jinlai / Porter, Kenneth W. / Shaw, Barbara Ramsay et al. | 2001
- 1025
-
ANTIVIRAL ACTIVITY OF TENOFOVIR (PMPA) AGAINST NUCLEOSIDE-RESISTANT CLINICAL HIV SAMPLESMiller, Michael D. / Margot, Nicolas A. / Hertogs, Kurt / Larder, Brendan / Miller, Veronica et al. | 2001
- 1029
-
SYNTHESIS AND ANTIVIRAL EVALUATION OF C-4-HYDRAZIDE DERIVATIVES OF 2′,3′-DIDEOXYCYTIDINEBoudou-Vivet, Valérie / Mathé, Christophe / Gosselin, Gilles et al. | 2001
- 1033
-
MODIFIED DINUCLEOSIDE TETRAPHOSPHONATES, NEW POTENTIAL INHIBITORS OF HIV REVERSE TRANSCRIPTASEShirokova, E. A. / Khandazhinskaya, A. L. / Skoblov, Yu. S. / Goryunova, L. Ye. / Beabealashvilli, R. S. / Krayevsky, A. A. et al. | 2001
- 1037
-
3′-DEOXYRIBOFURANOSE DERIVATIVES OF 1-DEAZA AND 3-DEAZA-ADENOSINE AND THEIR ACTIVITY AS ADENOSINE DEAMINASE INHIBITORSCostanzi, S. / Lambertucci, C. / Volpini, R. / Vittori, S. / Lupidi, G. / Cristalli, G. et al. | 2001
- 1043
-
POTENT IN VITRO ANTICANCER ACTIVITIES OF RING-EXPANDED (“FAT”) NUCLEOSIDES CONTAINING THE IMIDAZO[4,5-E][1,3]DIAZEPINE RING SYSTEMGill, Juliana K. / Wang, Lijuan / Bretner, Maria / Newman, Rachel / Kyprianou, Natasha / Hosmane, Ramachandra S. et al. | 2001
- 1047
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N-PHENYLIMIDAZOLIUM TRIFLATE AS A HIGHLY EFFECTIVE PROMOTER FOR THE INTERRIBONUCLEOTIDE-BOND FORMATION VIA THE PHOSPHORAMIDITE METHODKawai, Rie / Sugimoto, Jun-ichiro / Kataoka, Masanori / Hayakawa, Yoshihiro et al. | 2001
- 1049
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SYNTHESIS AND STUDY OF THE FLUORESCEIN CONJUGATE OF THE NUCLEOTIDE dPTPCummins, W. J. / Hamilton, A. L. / Smith, C. L. / Briggs, M. S. J. et al. | 2001
- 1053
-
Synthesis and In Vitro Antiviral Activity Evaluation of 9-(2-Azido- 2,3-dideoxy-b-D-threo-pentofuranosyl)adenine DerivativesTakamatsu, S. et al. | 2001
- 1053
-
SYNTHESIS AND IN VITRO ANTIVIRAL ACTIVITY EVALUATION OF 9-(2-AZIDO-2,3-DIDEOXY-β-D-THREO-PENTOFURANOSYL)ADENINE DERIVATIVESTakamatsu, Satoshi / Izawa, Kunisuke / Maruyama, Tokumi / Katayama, Satoshi / Hirose, Naoko / De Clercq, Erik et al. | 2001
- 1059
-
SYNTHESIS AND ANTIVIRAL ACTIVITY OF NOVEL EXOMETHYLENE CYCLOPROPYL NUCLEOSIDESChoi, Bo Gil / Kwak, Eun Yee / Hong, Joon Hee / Lee, Chong Kyo et al. | 2001
- 1063
-
BICYCLIC FURO PYRIMIDINE NUCLEOSIDES WITH ARYLOXYPHENYL AND HALOPHENYL SUBSTITUTED SIDE CHAINS AS POTENT AND SELECTIVE VARICELLA-ZOSTER VIRUS INHIBITORSBlewett, Sally / McGuigan, Christopher / Barucki, Hubert / Andrei, Graciela / Snoeck, Robert / De Clercq, Erik / Balzarini, Jan et al. | 2001
- 1067
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THE DESIGN AND SYNTHESIS OF PURINE INHIBITORS OF CDK2. IIIShum, P. W. / Peet, N. P. / Weintraub, P. M. / Le, T. B. / Zhao, Z. / Barbone, F. / Cashman, B. / Tsay, J. / Dwyer, S. / Loos, P. C. et al. | 2001
- 1079
-
CHEMICAL CROSS-LINKING OF PEPTIDES DERIVED FROM RECA WITH SINGLE-STRANDED OLIGONUCLEOTIDES CONTAINING 5-FORMYL-2′-DEOXYURIDINESugiyama, Toru / Kittaka, Atsushi / Takayama, Hiroaki / Tomioka, Mitsugu / Ida, Yoshiteru / Kuroda, Reiko et al. | 2001
- 1085
-
PURIFICATION OF PMPA AMIDATE PRODRUGS BY SMB CHROMATOGRAPHY AND X-RAY CRYSTALLOGRAPHY OF THE DIASTEREOMERICALLY PURE GS-7340Chapman, H. / Kernan, M. / Rohloff, J. / Sparacino, M. / Terhorst, T. et al. | 2001
- 1091
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METABOLISM OF GS-7340, A NOVEL PHENYL MONOPHOSPHORAMIDATE INTRACELLULAR PRODRUG OF PMPA, IN BLOODEisenberg, Eugene J. / He, Gong-Xin / Lee, William A. et al. | 2001
- 1099
-
AN EFFICIENT PROCESS FOR THE SYNTHESIS OF CYCLIC HPMPCLouie, Michael S. / Chapman, Harlan et al. | 2001
- 1103
-
SYNTHESIS OF 8-AMINO AND 8-SUBSTITUTED AMINO DERIVATIVES OF ACYCLIC PURINE NUCLEOSIDE AND NUCLEOTIDE ANALOGS. ALKYLATION OF 8-SUBSTITUTED PURINE BASESJaneba, Z. / Holý, A. et al. | 2001
- 1107
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MESSENGER RNA ISOLATION USING NOVEL PNA ANALOGUESPhelan, D. / Hondorp, K. / Choob, M. / Efimov, V. / Fernandez, J. et al. | 2001
- 1113
-
SYNTHESIS OF MODIFIED NUCLEOSIDE 5′-TRIPHOSPHATES FOR IN VITRO SELECTION OF CATALYTIC NUCLEIC ACIDS [1]Matulic-Adamic, Jasenka / Daniher, Andrew T. / Karpeisky, Alexander / Haeberli, Peter / Sweedler, David / Beigelman, Leonid et al. | 2001
- 1113
-
Synthesis of Modified Nucleoside 5-Triphosphates for In Vitro Selection of Catalytic Nucleic AcidsMatulic-Adamic, J. et al. | 2001
- 1117
-
LIN-BENZOARISTEROMYCINRajappan, Vasanthakumar P. / Schneller, Stewart W. et al. | 2001
- 1123
-
SYNTHESIS AND IN VITRO ACTIVITY OF D- AND L-ENANTIOMERS OF 5-(TRIFLUOROMETHYL)URACIL NUCLEOSIDE DERIVATIVESSalvetti, Raul / Pregnolato, Massimo / Verri, Annalisa / Focher, Federico / Spadari, Silvio / Marchand, Arnaud / Mathé, Christophe / Gosselin, Gilles et al. | 2001
- 1127
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NEW CARBOCYCLIC NUCLEOSIDES DERIVED FROM INDANAbad, F. / Álvarez, F. / Fernández, F. / García-Mera, X. / Rodríguez-Borges, J. E. et al. | 2001
- 1129
-
MODIFIED CYCLOBUTANE CARBONUCLEOSIDES: SYNTHESIS AND EVALUATION OF THEIR ANTIVIRAL ACTIVITYFernández, F. / Hergueta, A. R. / López, C. / De Clercq, E. / Balzarini, J. et al. | 2001
- 1133
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A CYCLOBUTANE CARBONUCLEOSIDE WITH MARKED SELECTIVITY AGAINST TK+ AND TK− VARICELLA ZOSTER VIRUSLópez, C. / Balo, C. / Blanco, J. M. / Fernández, F. / De Clercq, E. / Balzarini, J. et al. | 2001
- 1137
-
SYNTHESIS AND EVALUATION OF ANTIVIRAL ACTIVITY OF HIGHER HOMOLOGUES OF XYLO-CARBOCYCLIC NUCLEOSIDESCaamaño, O. / Figueira, M. J. / Fernández, F. / García, M. D. / Nieto, M. I. / de Clercq, E. / Balzarini, J. et al. | 2001
- 1141
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NOVEL NUCLEOSIDE TRIPHOSPHATE ANALOGS FOR THE ENZYMATIC LABELING OF NUCLEIC ACIDSBarone, A. D. / Chen, C. / McGall, G. H. / Rafii, K. / Buzby, Philip R. / Dimeo, James J. et al. | 2001
- 1147
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6-AZACYTIDINE - COMPOUND WITH WIDE SPECTRUM OF ANTIVIRAL ACTIVITYAlexeeva, I. / Dyachenko, N. / Nosach, L. / Zhovnovataya, V. / Rybalko, S. / Lozitskaya, R. / Fedchuk, A. / Lozitsky, V. / Gridina, T. / Shalamay, A. et al. | 2001
- 1153
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SYNTHESIS AND ADENOSINE RECEPTOR AFFINITY AND POTENCY OF 8-ALKYNYL DERIVATIVES OF ADENOSINELambertucci, C. / Costanzi, S. / Vittori, S. / Volpini, R. / Cristalli, G. et al. | 2001
- 1159
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KINETICS STUDY OF THE BIOTRANSFORMATION OF AN OLIGONUCLEOTIDE PRODRUG IN CELLS EXTRACT BY MATRIX-ASSISTED LASER DESORPTION/IONIZATION TIME-OF-FLIGHT MASS SPECTROMETRYMorvan, François / Brès, Jean-Charles / Lefebvre, Isabelle / Vasseur, Jean-Jacques / Pompon, Alain / Imbach, Jean-Louis et al. | 2001
- 1165
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CELLULAR UPTAKE AND INTRACELLULAR QUANTIFICATION OF FLUORESCENT LABELED T20 ME-SATE PROOLIGONUCLEOTIDESMorvan, François / Bologna, J. C. / Vivès, E. / Imbach, Jean-Louis et al. | 2001
- 1169
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KINETICALLY SELECTIVE BINDING OF SINGLE STRANDED RNA OVER DNA BY A PYRROLIDINE-AMIDE OLIGONUCLEOTIDE MIMIC (POM)Hickman, David T. / King, Paul M. / Slater, Jonathan M. / Cooper, Matthew A. / Micklefield, Jason et al. | 2001
- 1173
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SYNTHESIS AND BIOPHYSICAL STUDIES OF OLIGONUCLEOTIDES CONTAINING HYDROXAMATE LINKAGESRamasamy, Kanda S. / Stoisavljevic, Vesna / Lau, Johnson Y. N. et al. | 2001
- 1177
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LABELING DURING CLEAVAGE (LDC), A NEW LABELING APPROACH FOR RNAMonnot, V. / Tora, C. / Lopez, S. / Menou, L. / Laayoun, A. et al. | 2001
- 1181
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NEW APPROACHES TOWARDS FLUORESCENCE LABELLING OF MESSENGER RNA TRANSCRIPTSGarnier, Arlette / Hüsken, Dieter / Weiler, Jan et al. | 2001
- 1187
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ENGINEERING PREFERENCES OF HAIRPIN PNA BINDING TO COMPLEMENTARY DNA: EFFECT OF N7G IN aeg/aep PNA BACKBONEKumar, V. A. / D'Costa, M. / Ganesh, K. N. et al. | 2001
- 1193
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SYNTHESIS AND EVALUATION OF PROLYL CARBAMATE NUCLEIC ACIDS (PrCNA)Meena / Kumar, V. A. / Ganesh, K. N. et al. | 2001
- 1197
-
CONSTRAINED FLEXIBILITY IN PNA: DNA BINDING STUDIES WITH BRIDGED AMINOPROPYLGLYCYL PNALonkar, P. S. / Kumar, V. A. / Ganesh, K. N. et al. | 2001
- 1201
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EXTRA STABLE 2′,5′-LINKED RNA LOOPSHannoush, Rami N. / Damha, Masad J. et al. | 2001
- 1205
-
EFFECT OF SUBSTITUTING ARABINONUCLEOSIDES FOR DEOXYNUCLEOTIDES IN THE DNA PRIMING STRAND ON THE POLYMERASE ACTION OF HIV-1 RTNoronha, Anne M. / Arion, Dominique / Parniak, Michael A. / Damha, Masad J. et al. | 2001
- 1211
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MOLECULAR MODELLING OF 2′-OH MEDIATED HYDROGEN BONDING IN RIBONUCLEOS(T)IDES BY NMR CONSTRAINED AM1 AND MMX CALCULATIONSAcharya, Parag / Velikian, Irina / Acharya, Sandipta / Chattopadhyaya, Jyoti et al. | 2001
- 1219
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DO THE 16 MER, 5′-GUGGUCUGAUGAGGCC-3′ AND THE 25 MER, 5′-GGCCGAAACUCGUAAGAGUCACCAC-3′, FORM A HAMMERHEAD RIBOZYME STRUCTURE IN PHYSIOLOGICAL CONDITIONS? AN NMR AND UV THERMODYNAMIC STUDYZamaratski, Edouard / Trifonova, Anna / Acharya, Parag / Isaksson, Johan / Maltseva, Tatiana / Chattopadhayaya, Jyoti et al. | 2001
- 1225
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THE NMR CONFORMATION STUDY OF THE COMPLEXES OF DEOXYCYTIDINE KINASE (dCK) AND 2′-DEOXYCYTIDINE/2′-DEOXYADENOSINEMaltseva, T. / Usova, E. / Eriksson, S. / Milecki, J. / Földesi, A. / Chattopadhayaya, J. et al. | 2001
- 1229
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AN ENERGETIC CORRELATION OF AB INITIO AND NMR STUDIES OF THE 3′-GAUCHE EFFECT IN 3′-SUBSTITUTED THYMIDINESAcharya, Parag / Thibaudeau, Christophe / Chattopadhyaya, Jyoti et al. | 2001
- 1235
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PROMOTION OF TRIPLEX FORMATION BY 2′-O,4′-C-METHYLENE BRIDGED NUCLEIC ACID (2′,4′-BNA) MODIFICATION: THERMODYNAMIC AND KINETIC STUDIESTorigoe, Hidetaka / Obika, Satoshi / Imanishi, Takeshi et al. | 2001
- 1239
-
A DNA-BINDING PEPTIDE FROM A PHAGE DISPLAY LIBRARYWölcke, Julian / Weinhold, Elmar et al. | 2001
- 1243
-
INHIBITION OF HUMAN TELOMERASE BY L-ENANTIOMERS OF NATURAL 2′-DEOXYRIBONUCLEOSIDE 5′-TRIPHOSPHATESYamaguchi, Toyofumi / Yamada, Rieko / Tomikawa, Aki / Shudo, Koichi / Saito, Motoki / Ishikawa, Fuyuki / Saneyoshi, Mineo et al. | 2001
- 1247
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MECHANISTIC STUDIES TO UNDERSTAND THE INHIBITION OF WILD TYPE AND MUTANT HIV-1 REVERSE TRANSCRIPTASE BY CARBOVIR-TRIPHOSPHATERay, Adrian S. / Anderson, Karen S. et al. | 2001
- 1251
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ACCELERATION OF NUCLEIC ACID HYBRIDIZATION ON DNA MICROARRAYS DRIVEN BY pH TUNABLE MODIFICATIONSZhang, Peiming / Briones, Natalia / Liu, Chang-Gong / Brush, Charles K. / Powdrill, Tom / Belosludtsev, Yuri / Hogan, Mike et al. | 2001
- 1255
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LABORATORY DIAGNOSIS OF RESPIRATORY DISEASES: PCR VERSUS SEROLOGYHaaheim, H. / Vorland, L. / Gutteberg, T. J. et al. | 2001
- 1259
-
PHOTOSENSITIZED AND CATALYTIC OXIDATION OF DNA BY METALLOPHTHALOCYANINE-OLIGONUCLEOTIDE CONJUGATESKoval, V. V. / Chernonosov, A. A. / Abramova, T. V. / Ivanova, T. M. / Fedorova, O. S. / Derkacheva, V. M. / Lukyanets, E. A. et al. | 2001
- 1263
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SYNTHESIS OF 2′,3′-DIDEOXY-2′,3′-DIDEHYDRO NUCLEOSIDES VIA A SERENDIPITOUS ROUTEGuo, Z. / Sanghvi, Y. S. / Brammer, L. E.Jr. / Hudlicky, T. et al. | 2001
- 1267
-
UNEXPECTED RESULTS AND RECOURSE IN PROCESS OPTIMIZATION OF NUCLEOSIDE 3′-O-SUCCINATESSong, Quanlai / Sanghvi, Yogesh S. et al. | 2001
- 1271
-
A NEW FACILE METHOD FOR SPIN-LABELING OF OLIGONUCLEOTIDESStrube, Thorsten / Schiemann, Olav / MacMillan, Fraser / Prisner, Thomas / Engels, Joachim W. et al. | 2001
- 1275
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PHENYLALKYL BACKBONE MODIFIED OLIGODEOXYNUCLEOTIDES, THEIR SYNTHESIS AND THE INFLUENCE OF THE ALKYL CHAIN LENGTHAmberg, Stefan / Engels, Joachim W. et al. | 2001
- 1279
-
SYNTHESIS AND BASE PAIRING PROPERTIES OF 9-DEAZAPURINE N7-NUCLEOSIDES IN OLIGONUCLEOTIDE DUPLEXES AND TRIPLEXESLeonard, P. / Wiglenda, T. / Seela, F. et al. | 2001
- 1283
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PARALLEL DNA CONTAINING PYRAZOLO[3,4-D]PYRIMIDINE ANALOGUES OF ISOGUANINESeela, F. / Kröschel, R. / He, Y. et al. | 2001
- 1287
-
BRIDGED CYCLIC OLIGORIBONUCLEOTIDES—TOWARDS MODELS FOR CODON-ANTICODON PAIRINGMicura, R. / Pils, W. / Grubmayr, K. / Ebert, M.-O. / Jaun, B. et al. | 2001
- 1291
-
LARGE-SCALE MANUFACTURING OF ALL FOUR 2′-DEOXYNUCLEOSIDES VIA NOVEL STRATEGIES INCLUDING A CHEMO-ENZYMATIC PROCESSKomatsu, Hironori / Awano, Hirokazu / Tanikawa, Hiroharu / Itou, Kiyoshi / Ikeda, Ichirou et al. | 2001
- 1295
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KINETIC STUDIES OF THE DEGRADATION OF OXYCARBONYLOXYMETHYL PRODRUG OF ADEFOVIR AND TENOFOVIR IN SOLUTIONOliyai, Reza / Yuan, Lung-Chi / Dahl, Terry et al. | 2001
- 1299
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DEALKYLATION OF PHOSPHONATE ESTERS WITH CHLOROTRIMETHYLSILANEGutierrez, A. J. / Prisbe, E. J. / Rohloff, J. C. et al. | 2001
- 1303
-
SYNTHESES OF DNA DUPLEXES CONTAINING A C‒C INTERSTRAND CROSS-LINKNoronha, Anne M. / Noll, David M. / Miller, Paul S. et al. | 2001
- 1309
-
SYNTHESIS AND NMR-ANALYSIS OF TRICYCLIC NUCLEOSIDESNielsen, Poul / Petersen, Michael / Jacobsen, Jens Peter et al. | 2001
- 1313
-
SPECIFIC BINDING AND STABILIZATION OF DNA AND PHOSPHOROTHIOATE DNA BY AMPHIPHILIC α-HELICAL PEPTIDESKubo, Takanori / Fujii, Masayuki et al. | 2001
- 1313
-
Specific Binding and Stabilization of DNA and Phosphorothioate DNA by Amphiphilic a-Helical PeptidesKubo, T. et al. | 2001
- 1317
-
Amphiphilic b-Sheet Peptides Can Bind to Double and Triple Stranded DNAYokoyama, K. et al. | 2001
- 1317
-
AMPHIPHILIC β-SHEET PEPTIDES CAN BIND TO DOUBLE AND TRIPLE STRANDED DNAYokoyama, Kinuko / Kubo, Takanori / Fujii, Masayuki et al. | 2001
- 1321
-
A NOVEL APPROACH FOR THE SOLID PHASE SYNTHESIS OF DNA-PEPTIDE CONJUGATESKubo, Takanori / Dubey, Krishna / Fujii, Masayuki et al. | 2001
- 1325
-
SYNTHESIS OF A NOVEL NUCLEIC ACID MIMIC: P-BORANOMETHYLPHOSPHONATELin, Jinlai / Shaw, Barbara Ramsay et al. | 2001
- 1329
-
A NEW SYNTHETIC METHODOLOGY FOR TIAZOFURINRamasamy, Kanda S. / Lau, Johnson Y. N. et al. | 2001
- 1333
-
SYNTHETIC STUDIES TO IMPROVE THE DEUTERIUM LABELLING IN NUCLEOSIDES FOR FACILITATING STRUCTURAL STUDIES OF LARGE RNAS BY HIGH-FIELD NMR SPECTROSCOPYKundu, Mrinal K. / Trifonova, Anna / Dinya, Zoltán / Földesi, András / Chattopadhyaya, Jyoti et al. | 2001
- 1339
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THE SYNTHESIS OF, AND STUDIES ON, 2′-C-MODIFIED NUCLEOTIDESBrennan, Lavinia / Fettes, Kevin J. / O'Neil, Ian A. / Cosstick, Richard et al. | 2001
- 1343
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DESIGN AND PROPERTIES OF HEPATITIS C VIRUS ANTISENSE OLIGONUCLEOTIDES FOR LIVER SPECIFIC DRUG TARGETINGLehmann, Thomas J. / Serwe, Matthias / Caselmann, Wolfgang H. / Engels, Joachim W. et al. | 2001
- 1347
-
NOVEL MACROCYCLES DERIVED FROM NUCLEOSIDESCalcerrada-Muñoz, Noelia / O'Neil, Ian / Cosstick, Richard et al. | 2001
- 1351
-
SOLID-PHASE SYNTHESIS OF OLIGODEOXYNUCLEOTIDES CONTAINING 3′-S-PHOSPHOROTHIOLATE LINKAGESFettes, Kevin J. / O'Neil, Ian / Roberts, Stanley M. / Cosstick, Richard et al. | 2001
- 1355
-
SYNTHESIS AND BIOLOGICAL ACTIVITIES OF CYCLIC ADP-CARBOCYCLIC-RIBOSE AND ITS ANALOGSFukuoka, Masayoshi / Shuto, Satoshi / Minakawa, Noriaki / Ueno, Yoshihito / Matsuda, Akira et al. | 2001
- 1359
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RESOLUTION OF RACEMIC MIXTURES OF CARBOCYCLIC ANALOGUES OF NUCLEOSIDES AND ASSIGNMENT OF THEIR ABSOLUTE CONFIGURATIONBesada, P. / Terán, C. / Quezada, E. / Seco, J. M. / Uriarte, E. et al. | 2001
- 1363
-
1,2-DISUBSTITUTED CYCLOHEXANE CARBOCYCLIC ANALOGUES OF NUCLEOSIDESViña, D. / Santana, L. / Uriarte, E. et al. | 2001
- 1367
-
Asymmetric Synthesis of Carbocyclic Pyrimidine Nucleosides via p-Allylpalladium ComplexShi, J. et al. | 2001
- 1367
-
ASYMMETRIC SYNTHESIS OF CARBOCYCLIC PYRIMIDINE NUCLEOSIDES VIA π-ALLYLPALLADIUM COMPLEXShi, Junxing / Schinazi, Raymond F. et al. | 2001
- 1371
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THE USE AND EVALUATION OF 2+2 PHOTOADDITION IN IMMOBILIZATION OF OLIGONUCLEOTIDES ON A THREE DIMENSIONAL HYDROGEL MATRIXElghanian, R. / Xu, Y. / McGowen, J. / Seithoff, M. / Liu, C. G. / Winick, J. / Fuller, N. / Ramakrishnan, R. / Beuhler, A. / Johnson, T. et al. | 2001
- 1377
-
SYNTHESIS AND HYBRIDIZATION OF NOVEL CHIRAL PYRROLIDINE BASED PNA ANALOGUESlaitas, Andis / Yeheskiely, Esther et al. | 2001
- 1381
-
Evaluation of Several Economical Computational Methods for Geometry Optimization of Phosphorus Acid DerivativesSigurdsson, S. et al. | 2001
- 1381
-
EVALUATION OF SEVERAL ECONOMICAL COMPUTATIONAL METHODS FOR GEOMETRY OPTIMISATION OF PHOSPHORUS ACID DERIVATIVESSigurdsson, Susannah / Strömberg, Roger et al. | 2001
- 1385
-
A METHOD FOR SYNTHESIS OF AN ARTIFICIAL RIBONUCLEASEÅström, Hans / Strömberg, Roger et al. | 2001
- 1389
-
PREPARATION OF 3′-C-BRANCHED URIDINE ANALOGUES, SUITABLE FOR CONVERSION INTO FUNCTIONALISED 3′-C-METHYLENE DERIVATIVESWinqvist, Anna / Strömberg, Roger et al. | 2001
- 1389
-
Preparation of 3'-C-Branched Uridine Analogues, Suitable for Conversion into Functionalized 3'-C-Methylene DerivativesWinqvist, A. et al. | 2001
- 1393
-
SYNTHESIS OF NEW CHIRAL PEPTIDE NUCLEIC ACID (PNA) MONOMERSFalkiewicz, Bogdan / Wiśniowski, Wojciech / Kołodziejczyk, Aleksandra S. / Wiśniewski, Kazimierz et al. | 2001
- 1399
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RESTRICTED ROTATION IN CHIRAL PEPTIDE NUCLEIC ACID (PNA) MONOMERS - INFLUENCE OF SUBSTITUENTS STUDIED BY MEANS OF 1H NMROleszczuk, Marta / Rodziewicz-Motowidło, Sylwia / Falkiewicz, Bogdan et al. | 2001
- 1403
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PREPARATION OF OLIGODEOXYNUCLEOTIDE 5′-TRIPHOSPHATES USING SOLID SUPPORT APPROACHLebedev, A. V. / Koukhareva, I. I. / Beck, T. / Vaghefi, M. M. et al. | 2001
- 1411
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PHARMACOKINETICS OF SALICYLATE ESTER PRODRUGS OF CYCLIC HPMPC IN DOGSOliyai, Reza / Arimilli, Murty N. / Jones, Robert J. / Lee, William A. et al. | 2001
- 1415
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LC/MS DETERMINATION OF THE INTRACELLULAR CONCENTRATION OF TWO NOVEL ARYL PHOSPHORAMIDATE PRODRUGS OF PMPA AND THEIR METABOLITES IN DOG PBMCLynch, Theresa / Eisenberg, Gene / Kernan, Michael et al. | 2001
- 1421
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PHOSPHORAMIDITES AND OLIGONUCLEOTIDES CONTAINING 7-DEAZAPURINES AND PYRIMIDINES CARRYING AMINOPROPARGYL SIDE CHAINSSeela, F. / Ramzaeva, N. / Leonard, P. / Chen, Y. / Debelak, H. / Feiling, E. / Kröschel, R. / Zulauf, M. / Wenzel, T. / Fröhlich, T. et al. | 2001
- 1425
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ANTISENSE OLIGONUCLEOTIDE ISIS 2922 TARGETS IE-EXPRESSION AND PREVENTS HCMV-IE-INDUCED SUPPRESSION OF TSP-1 AND TSP-2 EXPRESSIONMargraf, S. / Bittoova, M. / Vogel, J-U. / Kotchekov, R. / Doerr, H. W. / Cinatl, J.Jr. et al. | 2001
- 1429
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BASE MUTATION ANALYSIS BY A FERROCENYL NAPHTHALENE DIIMIDE DERIVATIVETakenaka, Shigeori / Miyahara, Hiroyoshi / Yamashita, Kenichi / Takagi, Makoto / Kondo, Hiroki et al. | 2001
- 1433
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CYTARABINE TREATMENT OF HUMAN T-LYMPHOID CELLS INDUCES DECREASED HIV-1 RECEPTOR EXPRESSION AND REDUCED HIV-1 SUSCEPTIBILITYGröschel, B. / Kaufmann, A. / Cinatl, J. / Doerr, H. W. et al. | 2001