Identification of Allosteric PIF‐Pocket Ligands for PDK1 using NMR‐Based Fragment Screening and 1H‐15N TROSY Experiments (English)
- New search for: Stockman, Brian J.
- New search for: Kothe, Michael
- New search for: Kohls, Darcy
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- New search for: Connolly, Brendan J.
- New search for: Sheils, Alissa L.
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- New search for: Cheng, Alan C.
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- New search for: Charlton, Maura E.
- New search for: Stockman, Brian J.
- New search for: Kothe, Michael
- New search for: Kohls, Darcy
- New search for: Weibley, Laura
- New search for: Connolly, Brendan J.
- New search for: Sheils, Alissa L.
- New search for: Cao, Qing
- New search for: Cheng, Alan C.
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In:
Chemical Biology & Drug Design
;
73
, 2
;
179-188
;
2009
- Article (Journal) / Electronic Resource
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Title:Identification of Allosteric PIF‐Pocket Ligands for PDK1 using NMR‐Based Fragment Screening and 1H‐15N TROSY Experiments
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Contributors:Stockman, Brian J. ( author ) / Kothe, Michael ( author ) / Kohls, Darcy ( author ) / Weibley, Laura ( author ) / Connolly, Brendan J. ( author ) / Sheils, Alissa L. ( author ) / Cao, Qing ( author ) / Cheng, Alan C. ( author ) / Yang, Lily ( author ) / Kamath, Ajith V. ( author )
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Published in:Chemical Biology & Drug Design ; 73, 2 ; 179-188
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Publisher:
- New search for: Blackwell Publishing Ltd
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Publication date:2009-02-01
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Size:10 pages
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ISSN:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Keywords:
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Source:
Table of contents – Volume 73, Issue 2
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 157
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CREDO: A Protein–Ligand Interaction Database for Drug DiscoverySchreyer, Adrian / Blundell, Tom et al. | 2009
- 168
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AutoGrow: A Novel Algorithm for Protein Inhibitor DesignDurrant, Jacob D. / Amaro, Rommie E. / McCammon, J. Andrew et al. | 2009
- 179
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Identification of Allosteric PIF‐Pocket Ligands for PDK1 using NMR‐Based Fragment Screening and 1H‐15N TROSY ExperimentsStockman, Brian J. / Kothe, Michael / Kohls, Darcy / Weibley, Laura / Connolly, Brendan J. / Sheils, Alissa L. / Cao, Qing / Cheng, Alan C. / Yang, Lily / Kamath, Ajith V. et al. | 2009
- 189
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A Potent Gelatinase Inhibitor with Anti‐Tumor‐Invasive Activity and its Metabolic DispositionLee, Mijoon / Celenza, Giuseppe / Boggess, Bill / Blase, Jennifer / Shi, Qicun / Toth, Marta / Bernardo, M. Margarida / Wolter, William R. / Suckow, Mark A. / Hesek, Dusan et al. | 2009
- 203
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Chiral N‐Phosphonyl Imine Chemistry: Asymmetric Synthesis of α‐Alkyl β‐Amino Ketones by Reacting Phosphonyl Imines with Ketone‐Derived EnolatesAi, Teng / Han, Jianlin / Chen, Zhong‐Xiu / Li, Guigen et al. | 2009
- 203
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Chiral N-Phosphonyl Imine Chemistry: Asymmetric Synthesis of a-Alkyl b-Amino Ketones by Reacting Phosphonyl Imines with Ketone-Derived EnolatesAi, T. / Han, J. / Chen, Z. X. / Li, G. et al. | 2009
- 209
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Antimicrobial and Cytolytic Activities and Plausible Mode of Bactericidal Action of the Cell Penetrating Peptide Penetratin and Its Lys‐linked Two‐Stranded PeptideZhu, Wan Long / Shin, Song Yub et al. | 2009
- 216
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Novel Reticular Cyclen‐Based Polymer as Gene Vector in DNA TransfectionZhou, Li‐Hong / Yang, Mu / Zhou, Hong / Zhang, Ji / Li, Kun / Xiang, Yong‐Zhe / Wang, Na / Tian, Yun‐Fei / Yu, Xiao‐Qi et al. | 2009
- 225
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Synthesis, Evaluation of Pharmacological Activities and Quantitative Structure–Activity Relationship Studies of a Novel Group of bis(4‐Nitroaryl‐1,4‐dihyropyridine)Miri, Ramin / Javidnia, Katayoun / Hemmateenejad, Bahram / Tabarzad, Maryam / Jafarpour, Mehrnaz et al. | 2009
- 236
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On Three‐Dimensional Holographic Vector of Atomic Interaction Field Analysis for Influenza Neuraminidase InhibitorsLi, Zhiliang S. / Sun, Jiaying Y. / Liang, Guizhao Z. / Lu, Fenglin L. / Zhu, Wanping P. / Zhang, Mengjun J. / Zhang, Yonghong / Yang, Shanbin B. / Shu, Mao / Chen, Guohua H. et al. | 2009
- 244
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Improvement of Multivariate Image Analysis Applied to Quantitative Structure–Activity Relationship (QSAR) Analysis by Using Wavelet‐Principal Component Analysis Ranking Variable Selection and Least‐Squares Support Vector Machine Regression: QSAR Study of Checkpoint Kinase WEE1 InhibitorsCormanich, Rodrigo A. / Goodarzi, Mohammad / Freitas, Matheus P. et al. | 2009
- 253
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Novel Side‐Chain Glucosylated and Adamantylated [Asp2/Glu2]Enkephalin Analogs: Synthesis and In Vitro Growth Inhibition of Human Tumor CellsHorvat, Štefica / Kralj, Marijeta / Perc, Milica / Jerić, Ivanka / Varga‐Defterdarović, Lidija / Jakas, Andreja / Roščić, Maja / Šuman, Lidija / Gredičak, Matija et al. | 2009
- 258
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Predicting Anti‐HIV Activity of Dimethylaminopyridin‐2‐ones: Computational Approach using Topochemical DescriptorsDureja, Harish / Madan, Anil Kumar et al. | 2009
- 271
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Calendar of Events – February 2009| 2009