Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 2687
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Graphical contents list| 2010
- 2705
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Synthesis and biological evaluation of 1,4-diazepane derivatives as T-type calcium channel blockersGu, Su Jin / Lee, Jae Kyun / Pae, Ae Nim et al. | 2010
- 2709
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Chromone-2- and -3-carboxylic acids inhibit differently monoamine oxidases A and BAlcaro, Stefano / Gaspar, Alexandra / Ortuso, Francesco et al. | 2010
- 2713
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Click reaction synthesis of carbohydrate derivatives from ristocetin aglycon with antibacterial and antiviral activityPintér, Gábor / Bereczki, Ilona / Batta, Gyula et al. | 2010
- 2718
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Gold nanoparticles capped with sulfate-ended ligands as anti-HIV agentsDi Gianvincenzo, Paolo / Marradi, Marco / Martínez-Ávila, Olga María et al. | 2010
- 2722
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Synthesis and evaluation of a series of C5prime-substituted duocarmycin SA analogsRobertson, W. M. / Kastrinsky, D. B. / Hwang, I. et al. | 2010
- 2722
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Synthesis and evaluation of a series of C5′-substituted duocarmycin SA analogsRobertson, William M. / Kastrinsky, David B. / Hwang, Inkyu et al. | 2010
- 2726
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Transkarbams as transdermal permeation enhancers: Effects of ester position and ammonium carbamate formationNovotný, Michal / Hrabálek, Alexandr / Janůšová, Barbora et al. | 2010
- 2729
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(−)-Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channelsOrtar, Giorgio / Petrocellis, Luciano De / Morera, Ludovica et al. | 2010
- 2733
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Symmetrical α-bromoacryloylamido diaryldienone derivatives as a novel series of antiproliferative agents. Design, synthesis and biological evaluationRomagnoli, Romeo / Baraldi, Pier Giovanni / Cruz-Lopez, Olga et al. | 2010
- 2733
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Symmetrical a-bromoacryloylamido diaryldienone derivatives as a novel series of antiproliferative agents. Design, synthesis and biological evaluationRomagnoli, R. / Baraldi, P. G. / Cruz-Lopez, O. et al. | 2010
- 2740
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Exploration of secondary and tertiary pharmacophores in unsymmetrical N,N′-diaryl urea inhibitors of soluble epoxide hydrolaseAnandan, Sampath-Kumar / Gless, Richard D. et al. | 2010
- 2740
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Exploration of secondary and tertiary pharmacophores in unsymmetrical N,Nprime-diaryl urea inhibitors of soluble epoxide hydrolaseAnandan, S. K. / Gless, R. D. et al. | 2010
- 2745
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Identification of a novel series of potent RON receptor tyrosine kinase inhibitorsRaeppel, Stéphane / Gaudette, Frédéric / Mannion, Michael et al. | 2010
- 2750
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Synthesis and biological evaluation of modified pentapeptides as potent proteinase K inhibitorsKore, Anilkumar R. / Shanmugasundaram, Muthian / Charles, Irudaya et al. | 2010
- 2755
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Novel substituted pyrrolidines are high affinity histamine H3 receptor antagonistsStocking, Emily M. / Aluisio, Leah / Atack, John R. et al. | 2010
- 2761
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Squalenoyl nucleoside monophosphate nanoassemblies: New prodrug strategy for the delivery of nucleotide analoguesCaron, Joachim / Reddy, L. Harivardhan / Lepêtre-Mouelhi, Sinda et al. | 2010
- 2765
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Synthesis and biological activity of 2H-quinolizin-2-one based p38α MAP kinase inhibitorsTynebor, Robert M. / Chen, Meng-Hsin / Natarajan, Swaminathan R. et al. | 2010
- 2765
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Synthesis and biological activity of 2H-quinolizin-2-one based p38a MAP kinase inhibitorsTynebor, R. M. / Chen, M. H. / Natarajan, S. R. et al. | 2010
- 2770
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Probing the cannabinoid CB1/CB2 receptor subtype selectivity limits of 1,2-diarylimidazole-4-carboxamides by fine-tuning their 5-substitution patternLange, Jos H.M. / van der Neut, Martina A.W. / Borst, Alice J.M. et al. | 2010
- 2776
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Expression and characterization of Mycobacterium tuberculosis methionine aminopeptidase type 1aLu, Jing-Ping / Ye, Qi-Zhuang et al. | 2010
- 2780
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Synthesis and biological evaluation of combretastatin analogs as cell cycle inhibitors of the G1 to S transition in Saccharomyces cerevisiaeCoccetti, Paola / Montano, Giuseppe / Lombardo, Alessandro et al. | 2010
- 2785
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Synthesis of 7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-ylamine and its analogs as bombesin receptor subtype-3 agonistsGuo, Cheng / Guzzo, Peter R. / Hadden, Mark et al. | 2010
- 2790
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Cytotoxicity and inhibition of DNA topoisomerase I of polyhydroxylated triterpenoids and triterpenoid glycosidesWang, Ping / Ownby, Stacy / Zhang, Zhizhen et al. | 2010
- 2797
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Potent tricyclic pyrazole tetrazole agonists of the nicotinic acid receptor (GPR109a)Boatman, P. Douglas / Schrader, Thomas O. / Kasem, Michelle et al. | 2010
- 2801
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Identification and structure–activity relationship of 8-hydroxy-quinoline-7-carboxylic acid derivatives as inhibitors of Pim-1 kinaseSliman, Faten / Blairvacq, Mélina / Durieu, Emilie et al. | 2010
- 2806
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2-C-Methyluridine modified hammerhead ribozyme against the estrogen receptorPontiggia, Rodrigo / Pontiggia, Osvaldo / Simian, Marina et al. | 2010
- 2809
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Heterocyclic cycloalkanol ethylamines as norepinephrine reuptake inhibitorsSabatucci, Joseph P. / Mahaney, Paige E. / Leiter, Jennifer et al. | 2010
- 2813
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A rapid oxime linker-based library approach to identification of bivalent inhibitors of the Yersinia pestis protein-tyrosine phosphatase, YopHLiu, Fa / Hakami, Ramin Mollaaghababa / Dyas, Beverly et al. | 2010
- 2817
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Design of environmentally sensitive fluorescent 2′-deoxyguanosine containing arylethynyl moieties: Distinction of thymine base by base-discriminating fluorescent (BDF) probeShinohara, Yuta / Matsumoto, Katsuhiko / Kugenuma, Kenji et al. | 2010
- 2817
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Design of environmentally sensitive fluorescent 2prime-deoxyguanosine containing arylethynyl moieties: Distinction of thymine base by base-discriminating fluorescent (BDF) probeShinohara, Y. / Matsumoto, K. / Kugenuma, K. et al. | 2010
- 2821
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Cytotoxicity against KB and NCI-H187 cell lines of modified flavonoids from Kaempferia parvifloraYenjai, Chavi / Wanich, Suchana et al. | 2010
- 2824
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Inhibition of antigen-induced degranulation by aryl compounds isolated from the bark of Betula platyphylla in RBL-2H3 cellsKim, Seung Hyun / Park, Jung Hyun / Kim, Tae Bum et al. | 2010
- 2828
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Discovery of pyrazolthiazoles as novel and potent inhibitors of bacterial gyraseRonkin, Steven M. / Badia, Michael / Bellon, Steve et al. | 2010
- 2832
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Imidazoacridin-6-ones as novel inhibitors of the quinone oxidoreductase NQO2Nolan, K.A. / Humphries, M.P. / Bryce, R.A. et al. | 2010
- 2837
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Piperazine sulfonamide BACE1 inhibitors: Design, synthesis, and in vivo characterizationCumming, Jared / Babu, Suresh / Huang, Ying et al. | 2010
- 2843
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The cytotoxic styryl lactone goniothalamin is an inhibitor of nucleocytoplasmic transportWach, Jean-Yves / Güttinger, Stephan / Kutay, Ulrike et al. | 2010
- 2847
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New diterpenoids from Caesalpinia species and their cytotoxic activityDas, Biswanath / Srinivas, Yallamalla / Sudhakar, Chithaluri et al. | 2010
- 2851
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Discovery of novel leukotriene A4 hydrolase inhibitors based on piperidine and piperazine scaffoldsSandanayaka, Vincent / Mamat, Bjorn / Bhagat, Nikhil et al. | 2010
- 2855
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Synthesis and anti-tumor activities of methyl 2-O-aryl-6-O-arylprime-d-glucopyranosidesShi, H. / Zhou, B. / Li, W. et al. | 2010
- 2855
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Synthesis and anti-tumor activities of methyl 2-O-aryl-6-O-aryl′-d-glucopyranosidesShi, Hefang / Zhou, Bingcheng / Li, Wenwen et al. | 2010
- 2859
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4-Substituted 4-(1H-1,2,3-triazol-1-yl)piperidine: Novel C7 moieties of fluoroquinolones as antibacterial agentsHuang, Xiaoguang / Zhang, Aiqin / Chen, Dongliang et al. | 2010
- 2864
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Methylene amine substituted arylindenopyrimidines as potent adenosine A2A/A1 antagonistsShook, Brian C. / Rassnick, Stefanie / Hall, Daniel et al. | 2010
- 2868
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Optimization of arylindenopyrimidines as potent adenosine A2A/A1 antagonistsShook, Brian C. / Rassnick, Stefanie / Chakravarty, Devraj et al. | 2010
- 2872
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Chlorin e6–cholesterol conjugate and its copper complex. Simple synthesis and entrapping in phospholipid vesiclesNikolaeva, Irina A. / Misharin, Alexander Yu. / Ponomarev, Gelii V. et al. | 2010
- 2876
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Discovery and structural optimization of pyrazole derivatives as novel inhibitors of Cdc25BChen, Hai-Jun / Liu, Yong / Wang, Li-Na et al. | 2010
- 2880
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Synthesis and antibacterial activities of a novel alkylide: 3-O-(3-aryl-2-propargyl) and 3-O-(3-aryl-2-propenyl)clarithromycin derivativesLiang, Jian-Hua / Wang, Yue-Ying / Wang, He et al. | 2010
- 2884
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Design and an efficient synthesis of new thiorotenone derivativesYao, Changsheng / Wang, Cuihua / Jiang, Bei et al. | 2010
- 2888
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Design of new dopamine D2 receptor ligands: Biosynthesis and pharmacological evaluation of the hydroxylated metabolite of LASSBio-581Pazini, Francine / Menegatti, Ricardo / Sabino, José R. et al. | 2010
- 2892
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Identification of benzimidazole-based inhibitors of the mitogen activated kinase-5 signaling pathwayFlaherty, Patrick T. / Chopra, Ishveen / Jain, Prashi et al. | 2010
- 2897
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The development and SAR of pyrrolidine carboxamide 11b-HSD1 inhibitorsCheng, H. / Hoffman, J. / Le, P. et al. | 2010
- 2897
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The development and SAR of pyrrolidine carboxamide 11β-HSD1 inhibitorsCheng, Hengmiao / Hoffman, Jacqui / Le, Phuong et al. | 2010
- 2903
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Synthesis of 4-(3-biaryl)quinoline sulfones as potent liver X receptor agonistsUllrich, John W. / Morris, Robert / Bernotas, Ronald C. et al. | 2010
- 2908
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Selective targeting of 2prime-deoxy-5-fluorouridine to urokinase positive malignant cells in vitroVine, K. L. / Locke, J. M. / Bremner, J. B. et al. | 2010
- 2908
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Selective targeting of 2′-deoxy-5-fluorouridine to urokinase positive malignant cells in vitroVine, Kara L. / Locke, Julie M. / Bremner, John B. et al. | 2010
- 2912
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Synthesis and SAR of heterocyclic carboxylic acid isosteres based on 2-biarylethylimidazole as bombesin receptor subtype-3 (BRS-3) agonists for the treatment of obesityHadden, Mark / Goodman, Allan / Guo, Cheng et al. | 2010
- 2916
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The discovery and structure–activity relationships of 2-(piperidin-3-yl)-1H-benzimidazoles as selective, CNS penetrating H1-antihistamines for insomniaLavrador-Erb, Karine / Ravula, Satheesh Babu / Yu, Jinghua et al. | 2010
- 2920
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Truxillic acid derivatives act as peroxisome proliferator-activated receptor γ activatorsSteri, Ramona / Rupp, Matthias / Proschak, Ewgenij et al. | 2010
- 2920
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Truxillic acid derivatives act as peroxisome proliferator-activated receptor g activatorsSteri, R. / Rupp, M. / Proschak, E. et al. | 2010
- 2924
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Optimization of 7-alkene-3-quinolinecarbonitriles as Src kinase inhibitorsBoschelli, Diane H. / Wang, Daniel / Wang, Yan et al. | 2010
- 2928
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Water-soluble PDE4 inhibitors for the treatment of dry eyeGovek, Steven P. / Oshiro, Guy / Anzola, John V. et al. | 2010
- 2933
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Synthesis and structure-activity relationships of 2-aryl-4-oxazolylmethoxy benzylglycines and 2-aryl-4-thiazolylmethoxy benzylglycines as novel, potent PPARa selective activators- PPARa and PPARg selectivity modulationYe, X. Y. / Chen, S. / Zhang, H. et al. | 2010
- 2933
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Synthesis and structure–activity relationships of 2-aryl-4-oxazolylmethoxy benzylglycines and 2-aryl-4-thiazolylmethoxy benzylglycines as novel, potent PPARα selective activators- PPARα and PPARγ selectivity modulationYe, Xiang-Yang / Chen, Stephanie / Zhang, Hao et al. | 2010
- 2938
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A prodrug approach towards the development of tricyclic-based FBPase inhibitorsTsukada, Tomoharu / Tamaki, Kazuhiko / Tanaka, Jun et al. | 2010
- 2942
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Structure-based rational design, synthesis and antifungal activity of oxime-containing azole derivativesXu, Yulan / Sheng, Chunquan / Wang, Wenya et al. | 2010
- 2946
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Bivalent 5,8,9,13b-tetrahydro-6H-isoquino[1,2-a]isoquinolines and -isoquinolinium salts: Novel heterocyclic templates for butyrylcholinesterase inhibitorsSchulze, Maria / Siol, Oliver / Decker, Michael et al. | 2010
- 2950
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Molecular modelling, synthesis and acetylcholinesterase inhibition of ethyl 5-amino-2-methyl-6,7,8,9-tetrahydrobenzo[b][1,8]naphthyridine-3-carboxylateSoriano, Elena / Samadi, Abdelouahid / Chioua, Mourad et al. | 2010
- 2954
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A 3D-pharmacophore model for σ2 receptors based on a series of substituted benzo[d]oxazol-2(3H)-one derivativesLaurini, Erik / Zampieri, Daniele / Mamolo, Maria Grazia et al. | 2010
- 2958
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Inhibition of γ-secretase by the CK1 inhibitor IC261 does not depend on CK1δHöttecke, Nicole / Liebeck, Miriam / Baumann, Karlheinz et al. | 2010
- 2958
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Inhibition of g-secretase by the CK1 inhibitor IC261 does not depend on CK1dHottecke, N. / Liebeck, M. / Baumann, K. et al. | 2010
- 2964
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In vitro selection of a photoresponsive RNA aptamer to heminLiu, Mingzhe / Jinmei, Hiroshi / Abe, Hiroshi et al. | 2010
- 2968
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The discovery and structure–activity relationships of pyrano[3,4-b]indole based inhibitors of hepatitis C virus NS5B polymeraseLaPorte, Matthew G. / Draper, Tandy L. / Miller, Lori E. et al. | 2010
- 2974
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Bioactivity-guided isolation of mosquitocidal constituents from the rhizomes of Plumbago capensis ThunbSreelatha, T. / Hymavathi, A. / Murthy, J. Madhusudhana et al. | 2010
- 2978
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New 5-HT1A receptor ligands containing a Nprime-cyanoisonicotinamidine nucleus: Synthesis and in vitro pharmacological evaluationFiorino, F. / Severino, B. / De Angelis, F. et al. | 2010
- 2978
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New 5-HT1A receptor ligands containing a N′-cyanoisonicotinamidine nucleus: Synthesis and in vitro pharmacological evaluationFiorino, Ferdinando / Severino, Beatrice / De Angelis, Francesca et al. | 2010
- 2983
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Potent dihydroquinolinone dopamine D2 partial agonist/serotonin reuptake inhibitors for the treatment of schizophreniaYan, Yinfa / Zhou, Ping / Rotella, David P. et al. | 2010
- 2987
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Peripheral site acetylcholinesterase inhibitors targeting both inflammation and cholinergic dysfunctionYoung, Sherri / Fabio, Karine / Guillon, Christophe et al. | 2010
- 2991
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Structural requirement(s) of N-phenylthioureas and benzaldehyde thiosemicarbazones as inhibitors of melanogenesis in melanoma B 16 cellsThanigaimalai, P. / Le Hoang, Tuan Anh / Lee, Ki-Cheul et al. | 2010
- 2994
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Cucurbitacin E as a new inhibitor of cofilin phosphorylation in human leukemia U937 cellsNakashima, Souichi / Matsuda, Hisashi / Kurume, Ai et al. | 2010
- 2998
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Design, synthesis and structure–activity relationships of novel biarylamine-based Met kinase inhibitorsWilliams, David K. / Chen, Xiao-Tao / Tarby, Christine et al. | 2010
- 3003
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Synthesis and biological evaluation of novel 2-arylalkylthio-4-amino-6-benzyl pyrimidines as potent HIV-1 non-nucleoside reverse transcriptase inhibitorsQin, Hua / Liu, Chang / Zhang, Jianfang et al. | 2009
- IFC
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Editorial board| 2010