Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 5725
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Graphical contents list| 2007
- 5740
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Discovery of potent T-type calcium channel blockerSeo, Han Na / Choi, Ja Youn / Choe, Yun Jeong et al. | 2007
- 5744
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Studies on the interactions between some flavonols and cyclodextrinsBergonzi, Maria Camilla / Bilia, Anna Rita / Bari, Lorenzo Di et al. | 2007
- 5749
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Two new phenylpiperazines with atypical antipsychotic potentialTomić, Mirko / Ignjatović, Djurdjica / Tovilović, Gordana et al. | 2007
- 5754
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Synthesis and identification of novel 11β-aryl-4′,5′-dihydrospiro[estra-4,9-diene-17β,4′-oxazole] analogs with dissociated antiprogesterone activitiesJin, Chunyang / Manikumar, G. / Kepler, John A. et al. | 2007
- 5754
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Synthesis and identification of novel 11b-aryl-4prime,5prime-dihydrospiro[estra-4,9-diene-17b,4prime-oxazole] analogs with dissociated antiprogesterone activitiesJin, C. / Manikumar, G. / Kepler, J. A. et al. | 2007
- 5758
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Design and evaluation of analogues of the bacterial cell-wall peptidoglycan motif l-Lys-d-Ala-d-Ala for use in a vancomycin biosensorHernout, Olivier / Berthoin, Karine / Delattre, Isabelle et al. | 2007
- 5763
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Convenient synthesis of indeno[1,2-c]isoquinolines as constrained forms of 3-arylisoquinolines and docking study of a topoisomerase I inhibitor into DNA–topoisomerase I complexVan, Hue Thi My / Le, Quynh Manh / Lee, Kwang Youl et al. | 2007
- 5768
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Design and synthesis of opioidmimetics containing 2′,6′-dimethyl-l-tyrosine and a pyrazinone-ring platformShiotani, Kimitaka / Li, Tingyou / Miyazaki, Anna et al. | 2007
- 5768
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Design and synthesis of opioidmimetics containing 2prime,6prime-dimethyl-l-tyrosine and a pyrazinone-ring platformShiotani, K. / Li, T. / Miyazaki, A. et al. | 2007
- 5772
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Design and synthesis of novel antibacterial peptide-resin conjugatesCho, Won-Mi / Joshi, Bishnu Prasad / Cho, Hyeongjin et al. | 2007
- 5777
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Pentacyclic triterpenes. Part 5: Synthesis and SAR study of corosolic acid derivatives as inhibitors of glycogen phosphorylasesWen, Xiaoan / Xia, Jun / Cheng, Keguang et al. | 2007
- 5783
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N4-Phenyl modifications of N2-(2-hydroxyl)ethyl-6-(pyrrolidin-1-yl)-1,3,5-triazine-2,4-diamines enhance glucocerebrosidase inhibition by small molecules with potential as chemical chaperones for Gaucher diseaseHuang, Wenwei / Zheng, Wei / Urban, Daniel J. et al. | 2007
- 5790
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Amino-caprolactam derivatives as γ-secretase inhibitorsParker, Michael F. / Bronson, Joanne J. / Barten, Donna M. et al. | 2007
- 5790
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Amino-caprolactam derivatives as g-secretase inhibitorsParker, M. F. / Bronson, J. J. / Barten, D. M. et al. | 2007
- 5796
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Identification and synthesis of major metabolites of Vasopressin V2-receptor agonist WAY-151932, and antagonist, Lixivaptan®Molinari, Albert J. / Trybulski, Eugene J. / Bagli, Jehan et al. | 2007
- 5801
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d-Phenylglycinol-derived non-covalent factor Xa inhibitors: Effect of non-peptidic S4 linkage elements on affinity and anticoagulant activityKlimkowski, Valentine J. / Watson, Brian M. / Wiley, Michael R. et al. | 2007
- 5806
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4-Arylcyclohexylalanine analogs as potent, selective, and orally active inhibitors of dipeptidyl peptidase IVKaelin, David E. / Smenton, Abigail L. / Eiermann, George J. et al. | 2007
- 5812
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The design and preliminary structure–activity relationship studies of benzotriazines as potent inhibitors of Abl and Abl-T315I enzymesCao, Jianguo / Fine, Richard / Gritzen, Colleen et al. | 2007
- 5819
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Synthesis and TNF expression inhibitory properties of new thalidomide analogues derived via Heck cross couplingStewart, Scott G. / Spagnolo, Daniel / Polomska, Marta E. et al. | 2007
- 5825
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Structure–activity relationship (SAR) investigations of substituted imidazole analogs as TRPV1 antagonistsGore, Vijay K. / Ma, Vu V. / Tamir, Rami et al. | 2007
- 5831
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Strategies toward improving the brain penetration of macrocyclic tertiary carbinamine BACE-1 inhibitorsMoore, Keith P. / Zhu, Hong / Rajapakse, Hemaka A. et al. | 2007
- 5836
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Quantitative structure–activity relationship studies for prediction of antimicrobial activity of synthesized 2,4-hexadienoic acid derivativesNarasimhan, Balasubramanian / Judge, Vikramjeet / Narang, Rakesh et al. | 2007
- 5846
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Effect of indole ethyl isothiocyanates on proliferation, apoptosis, and MAPK signaling in neuroblastoma cell linesSingh, Rakesh K. / Lange, Thilo S. / Kim, Kyukwang et al. | 2007
- 5853
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Imidazopiperidine amides as dipeptidyl peptidase IV inhibitors for the treatment of diabetesChen, Ping / Caldwell, Charles G. / Mathvink, Robert J. et al. | 2007
- 5858
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A novel class of potent NF-kB signaling inhibitorsLeban, J. / Baierl, M. / Mies, J. et al. | 2007
- 5858
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A novel class of potent NF-κB signaling inhibitorsLeban, Johann / Baierl, Marcel / Mies, Jan et al. | 2007
- 5863
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Synthesis and inhibitory activity of 4-alkynyl and 4-alkenylquinazolines: Identification of new scaffolds for potent EGFR tyrosine kinase inhibitorsKitano, Yasunori / Suzuki, Tsuyoshi / Kawahara, Eiji et al. | 2007
- 5868
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Taxodistines A and B, abietane-type diterpenes from Taxodium distichumHirasawa, Yusuke / Izawa, Emi / Matsuno, Yosuke et al. | 2007
- 5872
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Synthesis of poison-frog alkaloids 233A, 235U, and 251AA and their inhibitory effects on neuronal nicotinic acetylcholine receptorsToyooka, Naoki / Kobayashi, Soushi / Zhou, Dejun et al. | 2007
- 5876
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Structure-based design, synthesis, and biological evaluation of peptidomimetic SARS-CoV 3CLpro inhibitorsGhosh, Arun K. / Xi, Kai / Grum-Tokars, Valerie et al. | 2007
- 5881
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NO donors. Part 16: Investigations on structure–activity relationships of organic mononitrates reveal 2-nitrooxyethylammoniumnitrate as a high potent vasodilatorKoenig, Andreas / Roegler, Carolin / Lange, Kathrin et al. | 2007
- 5886
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The discovery of substituted 4-(3-hydroxyanilino)-quinolines as potent RET kinase inhibitorsGraham Robinett, R. / Freemerman, Alex J. / Skinner, Michael A. et al. | 2007
- 5894
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A straightforward stereoselective synthesis of meso-, (S,S)- and (R,R)-2,6-diaminopimelic acids from cis-1,4-diacetoxycyclohept-2-eneSaito, Yukako / Shinkai, Takumi / Yoshimura, Yuichi et al. | 2007
- 5897
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Design, synthesis, and biological testing of pyrazoline derivatives of combretastatin-A4Johnson, Marlie / Younglove, Brent / Lee, Lauren et al. | 2007
- 5902
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Inactivation of soybean sterol 24-C-methyltransferase by elongated sterol side chains at C26Song, Zhihong / Nes, W. David et al. | 2007
- 5907
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Fluorinated chloramphenicol acetyltransferase thermostability and activity profile: Improved thermostability by a single-isoleucine mutantVoloshchuk, Natalya / Lee, Man Xia / Zhu, Wan Wen et al. | 2007
- 5912
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Synthesis and biological activities of glycosphingolipid analogues from marine sponge Aplysinella rhaxHada, Noriyasu / Nakashima, Taishi / Shrestha, Suraj Prakash et al. | 2007
- 5916
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5′-Halogenated analogs of oxymorphindoleMetcalf, Matthew D. / Coop, Andrew et al. | 2007
- 5916
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5prime-Halogenated analogs of oxymorphindoleMetcalf, M. D. / Coop, A. et al. | 2007
- 5918
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Novel orally active, dibenzazepinone-based γ-secretase inhibitorsPeters, Jens-Uwe / Galley, Guido / Jacobsen, Helmut et al. | 2007
- 5918
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Novel orally active, dibenzazepinone-based g-secretase inhibitorsPeters, J. U. / Galley, G. / Jacobsen, H. et al. | 2007
- 5924
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Synthesis and in vitro evaluation of a selective antagonist and the corresponding radioligand for the prostaglandin D2 receptor CRTH2Ulven, Trond / Gallen, Michael J. / Nielsen, Mads C. et al. | 2007
- 5928
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Discovery, synthesis, and structure–activity studies of tetrazole based growth hormone secretagoguesHernández, Andrés S. / Cheng, Peter T.W. / Musial, Christa M. et al. | 2007
- 5934
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Design, synthesis, and biological evaluation of triazolopiperazine-based β-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitorsKowalchick, Jennifer E. / Leiting, Barbara / Pryor, KellyAnn D. et al. | 2007
- 5934
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Design, synthesis, and biological evaluation of triazolopiperazine-based b-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitorsKowalchick, J. E. / Leiting, B. / Pryor, K. D. et al. | 2007
- 5940
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Synthesis and screening of 3-substituted thioxanthen-9-one-10,10-dioxidesLory, Pedro M.J. / Estrella-Jimenez, Maria E. / Shashack, Matthew J. et al. | 2007
- 5944
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Discovery of 4′-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-benzonitriles and 4′-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-pyridine-2′-carbonitriles as potent checkpoint kinase 1 (Chk1) inhibitorsTao, Zhi-Fu / Li, Gaoquan / Tong, Yunsong et al. | 2007
- 5944
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Discovery of 4prime-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-benzonitriles and 4prime-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-pyridine-2prime-carbonitriles as potent checkpoint kinase 1 (Chk1) inhibitorsTao, Z. F. / Li, G. / Tong, Y. et al. | 2007
- 5952
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Amino(methyl) pyrrolidines as novel scaffolds for factor Xa inhibitorsShi, Yan / Sitkoff, Doree / Zhang, Jing et al. | 2007
- 5959
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Conformationally constrained analogues of 2-arachidonoylglycerolVadivel, Subramanian K. / Vardarajan, Sundararaman / Duclos, Richard I. Jr. et al. | 2007
- 5964
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Synthesis and biological evaluation of phenyl piperidine derivatives as CCR2 antagonistsXia, Mingde / Hou, Cuifen / Pollack, Scott et al. | 2007
- 5969
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An effective method for the in situ synthesis of DNA–CPG conjugates using chemical ligation technology as tools for SNP analysisOhkubo, Akihiro / Tanaka, Kunihiko / Taguchi, Haruhiko et al. | 2007
- 5974
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Arene cis-dihydrodiols: Useful precursors for the preparation of analogues of the anti-tumour agent, 2-crotonyloxymethyl-(4R,5R,6R)-4,5,6-trihydroxycyclohex-2-enone (COTC)Arthurs, Claire L. / Raftery, James / Whitby, Helen L. et al. | 2007
- 5978
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Synthesis and structure–activity relationship of 4-(2-aryl-cyclopropylamino)-quinoline-3-carbonitriles as EGFR tyrosine kinase inhibitorsPannala, Madhavi / Kher, Sunil / Wilson, Norma et al. | 2007
- 5983
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(1R,2S)-4-(2-Cyano-cyclohexyl-oxy)-2-trifluoromethyl-benzonitrile, a potent androgen receptor antagonist for stimulating hair growth and reducing sebum productionHu, Lain-Yen / Du, Daniel / Hoffman, Jennifer et al. | 2007
- 5989
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Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitorsBrnardic, Edward J. / Garbaccio, Robert M. / Fraley, Mark E. et al. | 2007
- 5995
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Design and synthesis of thiazole-5-hydroxamic acids as novel histone deacetylase inhibitorsAnandan, Sampath-Kumar / Ward, John S. / Brokx, Richard D. et al. | 2007
- 6000
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Expedient synthesis of N-Z-pyroglutamyl-amino acid derivativesKatritzky, Alan R. / Angrish, Parul / Todadze, Ekaterina et al. | 2007
- 6003
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Discovery of N-phenyl nicotinamides as potent inhibitors of KdrDominguez, Celia / Smith, Leon / Huang, Qi et al. | 2007
- 6009
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On the search of new I2-IBS aliphatic ligands: Bis-guanidino carbonyl derivativesCorcoran, Jonathan / Rodriguez, Fernando / Rozas, Isabel et al. | 2007
- 6013
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From ATP to AZD6140: The discovery of an orally active reversible P2Y12 receptor antagonist for the prevention of thrombosisSpringthorpe, Brian / Bailey, Andrew / Barton, Patrick et al. | 2007
- 6019
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High dopamine transporter selectivity can be displayed by remarkably simple non-nitrogen containing inhibitorsBoye, Søren V. / Ortega-Caballero, Fernando / Sinning, Steffen et al. | 2007
- 6026
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Solid-phase synthesis and thermal denaturation study of cyclic PNAs targeting the HIV-1 TAR RNA loopUpert, Gregory / Mehiri, Mohamed / Giorgio, Audrey Di et al. | 2007
- 6031
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Inhibitors of NF-kB derived from thalidomideCarcache de-Blanco, E. J. / Pandit, B. / Hu, Z. et al. | 2007
- 6031
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Inhibitors of NF-κB derived from thalidomideCarcache de-Blanco, Esperanza J. / Pandit, Bulbul / Hu, Zhigen et al. | 2007
- I
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Instructions to contributors| 2007
- IFC
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Editorial board| 2007