Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 3987
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Graphical contents list| 2010
- 4004
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Synthesis and SAR of potent inhibitors of the Hepatitis C virus NS3/4A protease: Exploration of P2 quinazoline substituentsNilsson, Magnus / Belfrage, Anna Karin / Lindström, Stefan et al. | 2010
- 4012
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Studies on the structure–activity relationship of 1,3,3,4-tetra-substituted pyrrolidine embodied CCR5 receptor antagonists. Part 1: Tuning the N-substituentsBen, Li / Jones, Eric Dale / Zhou, Enkun et al. | 2010
- 4015
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One unique steroidal sapogenin obtained through the microbial transformation of ruscogenin by Phytophthora cactorum ATCC 32134 and its potential inhibitory effect on tissue factor (TF) procoagulant activityChen, Nai-Dong / Yue, Lei / Zhang, Jian et al. | 2010
- 4018
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Synthesis and biological activity of 2-hydroxynicotinoyl-serine-butyl esters related to antibiotic UK-3AArsianti, Ade / Hanafi, Muhammad / Saepudin, Endang et al. | 2010
- 4021
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Exploring structural requirements of 1-N-substituted thiocarbamoyl-3-phenyl-2-pyrazolines as antiamoebic agents using comparative QSAR modellingAdhikari, Nilanjan / Maiti, Milan Kumar / Jha, Tarun et al. | 2010
- 4027
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Discovery of novel 1H-imidazol-2-yl-pyrimidine-4,6-diamines as potential antimalarialsDeng, Xianming / Nagle, Advait / Wu, Tao et al. | 2010
- 4032
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A novel organogermanium protected atopic dermatitis induced by oxazoloneLim, Doo Hyeon / Li, Minghua / Seo, Jung-A et al. | 2010
- 4035
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1,5-Diarylimidazoles with strong inhibitory activity against COX-2 catalyzed PGE2 production from LPS-induced RAW 264.7 cellsChe, Haiyan / Tuyen, Truong Ngoc / Kim, Hyun Pyo et al. | 2010
- 4038
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Subtype-selectivity of metal-dependent methionine aminopeptidase inhibitorsAltmeyer, Markus A. / Marschner, Aline / Schiffmann, Rolf et al. | 2010
- 4045
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Design and evaluation of 3,6-di(hetero)aryl imidazo[1,2-a]pyrazines as inhibitors of checkpoint and other kinasesMatthews, Thomas P. / McHardy, Tatiana / Klair, Suki et al. | 2010
- 4050
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Synthesis of isosteric selenium analog of the PPARb/d agonist GW501516 and comparison of biological activitySharma, A. K. / Sk, U. H. / He, P. et al. | 2010
- 4050
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Synthesis of isosteric selenium analog of the PPARβ/δ agonist GW501516 and comparison of biological activitySharma, Arun K. / Sk, Ugir Hossain / He, Pengfei et al. | 2010
- 4053
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Synthesis and anti-HIV activity of 2prime-deoxy-2prime-fluoro-4prime-C-ethynyl nucleoside analogsWang, Q. / Li, Y. / Song, C. et al. | 2010
- 4053
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Synthesis and anti-HIV activity of 2′-deoxy-2′-fluoro-4′-C-ethynyl nucleoside analogsWang, Qiang / Li, Yanfeng / Song, Chuanjun et al. | 2010
- 4057
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7′,8′-Dihydroobolactone, a typanocidal α-pyrone from the rainforest tree Cryptocarya obovataDavis, Rohan A. / Demirkiran, Ozlem / Sykes, Melissa L. et al. | 2010
- 4057
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7prime,8prime-Dihydroobolactone, a typanocidal a-pyrone from the rainforest tree Cryptocarya obovataDavis, R. A. / Demirkiran, O. / Sykes, M. L. et al. | 2010
- 4060
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Diazinones as P2 replacements for pyrazole-based cathepsin S inhibitorsAmeriks, Michael K. / Bembenek, Scott D. / Burdett, Matthew T. et al. | 2010
- 4065
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Epsilon substituted lysinol derivatives as HIV-1 protease inhibitorsJones, Kristen L.G. / Holloway, M. Katharine / Su, Hua-Poo et al. | 2010
- 4069
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Structure–activity relationships and hepatic safety risks of thiazole agonists of the thrombopoietin receptorAntipas, Amy S. / Blumberg, Laura C. / Brissette, William H. et al. | 2010
- 4073
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Monastrol analogs: A synthesis of pyrazolopyridine, benzopyranopyrazolopyridine, and oxygen-bridged azolopyrimidine derivatives and their biological screeningSvetlik, Jan / Veizerová, Lucia / Mayer, Thomas U. et al. | 2010
- 4077
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Synthesis and biological evaluation of novel biotin–iminoalditol conjugatesPototschnig, Gerit / De Csáky, Christian Morales / Montenegro Burke, Jose R. et al. | 2010
- 4080
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Design and synthesis of trivalent ligands targeting opioid, cholecystokinin, and melanocortin receptors for the treatment of painLee, Yeon Sun / Fernandes, Steve / Kulkarani, Vinod et al. | 2010
- 4085
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Antitumor agents 278. 4-Amino-2H-benzo[h]chromen-2-one (ABO) analogs as potent in vitro anti-cancer agentsDong, Yizhou / Nakagawa-Goto, Kyoko / Lai, Chin-Yu et al. | 2010
- 4088
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Betulin and ursolic acid synthetic derivatives as inhibitors of Papilloma virusKazakova, Oxana B. / Giniyatullina, Gul’nara V. / Yamansarov, Emil Yu. et al. | 2010
- 4091
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Antitumor agents 273. Design and synthesis of N-alkyl-thiocolchicinoids as potential antitumor agentsKozaka, Takashi / Nakagawa-Goto, Kyoko / Shi, Qian et al. | 2010
- 4095
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Structure-based optimization of potent PDK1 inhibitorsAngiolini, Mauro / Banfi, Patrizia / Casale, Elena et al. | 2010
- 4100
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Eudistomidin G, a new β-carboline alkaloid from the Okinawan marine tunicate Eudistoma glaucus and structure revision of eudistomidin BTakahashi, Yohei / Ishiyama, Haruaki / Kubota, Takaaki et al. | 2010
- 4100
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Eudistomidin G, a new b-carboline alkaloid from the Okinawan marine tunicate Eudistoma glaucus and structure revision of eudistomidin BTakahashi, Y. / Ishiyama, H. / Kubota, T. et al. | 2010
- 4104
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Benzofuran-substituted urea derivatives as novel P2Y1 receptor antagonistsThalji, Reema K. / Aiyar, Nambi / Davenport, Elizabeth A. et al. | 2010
- 4108
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Motualevic acids and analogs: Synthesis and antimicrobial structure–activity relationshipsCheruku, Pradeep / Keffer, Jessica L. / Dogo-Isonagie, Cajetan et al. | 2010
- 4112
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Acid-catalyzed synthesis of 10-substituted triazolyl artemisinins and their growth inhibitory activity against various cancer cellsOh, Sangtae / Shin, Woon-Seob / Ham, Jungyeob et al. | 2010
- 4116
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Recombination of diterpenoid structure units: Synthesis of antitumor amides bearing functionalized bicyclo[3.2.1]octane ringMao, Zewei / Li, Yan / Chen, Jingbo et al. | 2010
- 4120
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Hydroxysafflor Yellow A suppresses thrombin generation and inflammatory responses following focal cerebral ischemia–reperfusion in ratsSun, Xia / Wei, Xinbing / Qu, Sifeng et al. | 2010
- 4125
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Efficient synthesis of 5′-O-laurate of 1-β-d-arabinofuranosylcytosine via highly regioselective enzymatic acylation in binary solvent mixturesLi, Xiao-feng / Zong, Min-hua / Zhao, Guang-lei et al. | 2010
- 4125
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Efficient synthesis of 5prime-O-laurate of 1-b-d-arabinofuranosylcytosine via highly regioselective enzymatic acylation in binary solvent mixturesLi, X. f. / Zong, M. h. / Zhao, G. l. et al. | 2010
- 4128
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AMP-activated protein kinase (AMPK) activators from Myristica fragrans (nutmeg) and their anti-obesity effectNguyen, Phi Hung / Le, Thi Van Thu / Kang, Hu Won et al. | 2010
- 4132
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Synthesis and biological activity of halophenols as potent antioxidant and cytoprotective agentsZhao, Wanyi / Feng, Xiue / Ban, Shurong et al. | 2010
- 4135
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An analysis of the ‘legal high’ mephedroneGibbons, Simon / Zloh, Mire et al. | 2010
- 4140
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4-Substituted-7-N-alkyl-N-acetyl 2-aminobenzothiazole amides: Drug-like and non-xanthine based A2B adenosine receptor antagonistsCheung, Adrian Wai-Hing / Brinkman, John / Firooznia, Fariborz et al. | 2010
- 4147
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Synthesis, characterization and preliminary analysis of in vivo biological activity of chitosan/celecoxib microcapsulesCheng, Shuk-Yan / Yuen, Marcus Chun-Wah / Lam, Pik-Ling et al. | 2010
- 4152
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Probe molecule equipped with boronic acid moiety as a reversible cross-linking group improves its binding affinityKotoku, Naoyuki / Guo, Xiu-Han / Arai, Masayoshi et al. | 2010
- 4156
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Structure-based design and synthesis of pyrrole derivatives as MEK inhibitorsWallace, Michael B. / Adams, Mark E. / Kanouni, Toufike et al. | 2010
- 4159
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Folacin C60 derivative exerts a protective activity against oxidative stress-induced apoptosis in rat pheochromocytoma cellsHu, Zhen / Guan, Wenchao / Wang, Wei et al. | 2010
- 4163
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Synthesis and molecular docking studies of novel 2-chloro-pyridine derivatives containing flavone moieties as potential antitumor agentsLiu, Xin-Hua / Liu, Hui-Feng / Shen, Xu et al. | 2010
- 4168
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Novel semicarbazones based 2,5-disubstituted-1,3,4-oxadiazoles: One more step towards establishing four binding site pharmacophoric model hypothesis for anticonvulsant activityRajak, Harish / Deshmukh, Ravitas / Veerasamy, Ravichandran et al. | 2010
- 4173
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In vitro antituberculosis activities of the constituents isolated from Haloxylon salicornicumBibi, Nazia / Tanoli, Sheraz Ahmad. K. / Farheen, Sadia et al. | 2010
- 4177
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Synthesis and characterization of multifunctional hyperbranched polyesters as prospective contrast agents for targeted MRISideratou, Zili / Tsiourvas, Dimitris / Theodossiou, Theodossis et al. | 2010
- 4182
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Interaction of aminoadamantane derivatives with the influenza A virus M2 channel-Docking using a pore blocking modelEleftheratos, Stelios / Spearpoint, Philip / Ortore, Gabriella et al. | 2010
- 4188
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High-throughput sequencing for the identification of binding molecules from DNA-encoded chemical librariesBuller, Fabian / Steiner, Martina / Scheuermann, Jörg et al. | 2010
- 4193
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Synthesis of diaryl-azo derivatives as potential antifungal agentsXu, Hui / Zeng, Xiwen et al. | 2010
- 4196
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Broad spectrum alkynyl inhibitors of T315I Bcr-AblDeng, Xianming / Lim, Sang Min / Zhang, Jianming et al. | 2010
- 4201
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Discovery of 3,9-diazabicyclo[4.2.1]nonanes as potent dual orexin receptor antagonists with sleep-promoting activity in the ratColeman, Paul J. / Schreier, John D. / Roecker, Anthony J. et al. | 2010
- 4206
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Synthesis of two marine farnesylacetones that dilate the basilar arteries of rabbitsOh, Sangtae / Park, Byong-Gon / Ham, Jungyeob et al. | 2010
- 4210
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Pre-clinical characterization of aryloxypyridine amides as histamine H3 receptor antagonists: Identification of candidates for clinical developmentLetavic, Michael A. / Aluisio, Leah / Atack, John R. et al. | 2010
- 4215
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Discovery of piperidin-4-yl-aminopyrimidines as HIV-1 reverse transcriptase inhibitors. N-Benzyl derivatives with broad potency against resistant mutant virusesKertesz, Denis J. / Brotherton-Pleiss, Christine / Yang, Minmin et al. | 2010
- 4219
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Synthesis and biological evaluation of oxazole derivatives as T-type calcium channel blockersLee, Jie Eun / Koh, Hun Yeong / Seo, Seon Hee et al. | 2010
- 4223
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Discovery of aminopyridines substituted with benzoxazole as orally active c-Met kinase inhibitorsCho, Sung Yun / Han, Sun-Young / Ha, Jae Du et al. | 2010
- 4228
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Synthesis and biological evaluation of 2-pyridyl-substituted pyrazoles and imidazoles as transforming growth factor-β type 1 receptor kinase inhibitorsDewang, Purushottam M. / Kim, Dae-Kee et al. | 2010
- 4228
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Synthesis and biological evaluation of 2-pyridyl-substituted pyrazoles and imidazoles as transforming growth factor-b type 1 receptor kinase inhibitorsDewang, P. M. / Kim, D. K. et al. | 2010
- 4233
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In vitro and in vivo antimalarial evaluation of semi-synthetic derivatives of gomphosteninSathe, Manisha / Kaushik, M.P. et al. | 2010
- 4237
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Chemoselective regulation of TREK2 channel: Activation by sulfonate chalcones and inhibition by sulfonamide chalconesKim, Eun-Jin / Ryu, Hyung Won / Curtis-Long, Marcus J. et al. | 2010
- 4240
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Synthesis of Tc-99m labeled 1,2,3-triazole-4-yl c-met binding peptide as a potential c-met receptor kinase positive tumor imaging agentKim, Eun-Mi / Joung, Min-Hee / Lee, Chang-Moon et al. | 2010
- 4244
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Montmorillonite K-10 catalyzed cyclization of N-ethoxycarbonyl-N′-arylguanidines: Access to pyrimido[4,5-c]carbazole and pyrimido[5,4-b]indole derivativesDebray, Julien / Zeghida, Walid / Baldeyrou, Brigitte et al. | 2010
- 4244
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Montmorillonite K-10 catalyzed cyclization of N-ethoxycarbonyl-Nprime-arylguanidines: Access to pyrimido[4,5-c]carbazole and pyrimido[5,4-b]indole derivativesDebray, J. / Zeghida, W. / Baldeyrou, B. et al. | 2010
- 4248
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Novel coumarin derivatives as potential antidyslipidemic agentsSashidhara, Koneni V. / Kumar, Abdhesh / Kumar, Manoj et al. | 2010
- 4252
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One-pot multicomponent synthesis and anti-microbial evaluation of 2prime-(indol-3-yl)-2-oxospiro(indoline-3,4prime-pyran) derivativesNandakumar, A. / Thirumurugan, P. / Perumal, P. T. et al. | 2010
- 4252
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One-pot multicomponent synthesis and anti-microbial evaluation of 2′-(indol-3-yl)-2-oxospiro(indoline-3,4′-pyran) derivativesNandakumar, A. / Thirumurugan, Prakasam / Perumal, Paramasivan T. et al. | 2010
- 4259
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Screening and characterization of an inhibitory chemical specific to Arabidopsis gibberellin 2-oxidasesOtani, Masato / Yoon, Jung-Min / Park, Seung-Hyun et al. | 2010
- 4263
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Synthesis and biological activity of glycosyl-1H-1,2,3-triazolesSlámová, Kristýna / Marhol, Petr / Bezouška, Karel et al. | 2010
- 4266
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Antioxidative activities of histidine containing caffeic acid-dipeptidesSeo, Hyo-Suk / Kwak, Seon-Yeong / Lee, Yoon-Sik et al. | 2010
- 4273
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Design and synthesis of 1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazoles and pyrazolo[3,4-b]pyridines for Aurora-A kinase inhibitorsShi, Jianyou / Xu, Guobin / Zhu, Wei et al. | 2010
- 4279
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A new approach for PEGylation of dendrimersKhambete, Hemant / Gautam, Surya P. / Karthikeyan, C. et al. | 2010
- 4282
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Corrigendum to “Synthesis and pharmacological evaluation of condensed heterocyclic 6-substituted-1,2,4-triazolo[3,4-b]-1,3,4-thiadiazole derivatives of naproxen” [Bioorg. Med. Chem. Lett. 17 (2007) 4504]Amir, Mohammad / Kumar, Harish / Javed, Sadique A. et al. | 2010
- IFC
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Editorial board| 2010