Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 1831
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Graphical contents list| 2012
- 1846
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Synthesis of novel long wavelength cationic chlorins via stereoselective aldol-like condensationLi, Jia Zhu / Wang, Jin Jun / Yoon, Il et al. | 2012
- 1850
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Synthesis and biological evaluation of sulfonyl acrylonitriles as novel inhibitors to peritoneal carcinomatosisZificsak, Craig A. / Shen, Yi / Lisko, Joseph G. et al. | 2012
- 1854
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Aminoimidazoles as BACE-1 inhibitors: The challenge to achieve in vivo brain efficacySwahn, Britt-Marie / Holenz, Jörg / Kihlström, Jacob et al. | 2012
- 1860
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New aromatase inhibitors from the 3-pyridyl arylether and 1-aryl pyrrolo[2,3-c]pyridine seriesStauffer, Frédéric / Furet, Pascal / Floersheimer, Andreas et al. | 2012
- 1864
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Characterization of TAE684 as a potent LRRK2 kinase inhibitorZhang, Jinwei / Deng, Xianming / Choi, Hwan Geun et al. | 2012
- 1870
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Identification of fused bicyclic heterocycles as potent and selective 5-HT2A receptor antagonists for the treatment of insomniaXiong, Yifeng / Ullman, Brett / Choi, Jin-Sun Karoline et al. | 2012
- 1874
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Imidazo[1,2-a]pyrazines as novel PI3K inhibitorsMartínez González, Sonia / Hernández, Ana Isabel / Varela, Carmen et al. | 2012
- 1879
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Design and synthesis of novel 7-aminoquinazoline derivatives: Antitumor and anticonvulsant activitiesEl-Azab, Adel S. / ElTahir, Kamal E.H. et al. | 2012
- 1886
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Inhibitors of human histone deacetylase with potent activity against the African trypanosome Trypanosoma bruceiKelly, John M. / Taylor, Martin C. / Horn, David et al. | 2012
- 1891
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Structure–activity relationship of the 7-hydroxy benzimidazole analogs as glycogen synthase kinase 3β inhibitorLee, Seung-Chul / Shin, Dongkyu / Cho, Joong Myung et al. | 2012
- 1891
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Structure-activity relationship of the 7-hydroxy benzimidazole analogs as glycogen synthase kinase 3b inhibitorLee, S. C. / Shin, D. / Cho, J. M. et al. | 2012
- 1895
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New antitumor compounds from Carya cathayensisWu, Wei / Bi, Xiu-Li / Cao, Jia-Qing et al. | 2012
- 1899
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Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the δ opioid receptor. Discovery of two highly potent and selective δ opioid agonistsBerezowska, Irena / Lemieux, Carole / Chung, Nga N. et al. | 2012
- 1899
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Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the d opioid receptor. Discovery of two highly potent and selective d opioid agonistsBerezowska, I. / Lemieux, C. / Chung, N. N. et al. | 2012
- 1903
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Discovery of vinylcycloalkyl-substituted benzimidazole TRPM8 antagonists effective in the treatment of cold allodyniaCalvo, Raul R. / Meegalla, Sanath K. / Parks, Daniel J. et al. | 2012
- 1908
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New cyclic peptides with osteoblastic proliferative activity from Dianthus superbusTong, Yun / Luo, Jian-Guang / Wang, Rui et al. | 2012
- 1912
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1,2,4-Oxadiazoles: A new class of anti-prostate cancer agentsKhatik, Gopal L. / Kaur, Jasmine / Kumar, Varun et al. | 2012
- 1917
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Novel imidazo[2,1-b][1,3,4]thiadiazole carrying rhodanine-3-acetic acid as potential antitubercular agentsAlegaon, Shankar G. / Alagawadi, Kallanagouda R. / Sonkusare, Pranali V. et al. | 2012
- 1922
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Synthesis and evaluation of cytotoxic effects of novel α-methylenelactone tetracyclic diterpenoidsZeng, Yao-fu / Wu, Jia-qiang / Shi, Lian-yong et al. | 2012
- 1922
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Synthesis and evaluation of cytotoxic effects of novel a-methylenelactone tetracyclic diterpenoidsZeng, Y. f. / Wu, J. q. / Shi, L. y. et al. | 2012
- 1926
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Anti-tumor activity of new orally bioavailable 2-amino-5-(thiophen-2-yl)benzamide-series histone deacetylase inhibitors, possessing an aqueous soluble functional group as a surface recognition domainHirata, Yoshiyuki / Hirata, Masahiko / Kawaratani, Yasuyuki et al. | 2012
- 1931
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Characterization of H2O-forming NADH oxidase from Streptococcus pyogenes and its application in l-rare sugar productionGao, Hui / Tiwari, Manish Kumar / Kang, Yun Chan et al. | 2012
- 1936
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Influence of ring size on the cognition-enhancing activity of DM235 and MN19, two potent nootropic drugsGuandalini, L. / Martini, E. / Di Cesare Mannelli, L. et al. | 2012
- 1940
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Aminopyrimidinone Cdc7 Kinase InhibitorsWoods, Keith W. / Lai, Chunqiu / Miyashiro, Julie M. et al. | 2012
- 1944
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Discovery of 4-hydroxy-1,6-naphthyridine-3-carbonitrile derivatives as novel PDE10A inhibitorsBauer, Udo / Giordanetto, Fabrizio / Bauer, Martin et al. | 2012
- 1949
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Novel bisbenzimide-nitroxides for nuclear redox imaging in living cellsIkeda, Mamiko / Nakagawa, Hidehiko / Suzuki, Takayoshi et al. | 2012
- 1953
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3,4-Diarylpiperidines as potent renin inhibitorsLacombe, Patrick / Arbour, Mélissa / Aspiotis, Renée et al. | 2012
- 1958
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Radiosynthesis of PET radiotracer as a prodrug for imaging group II metabotropic glutamate receptors in vivoWang, Ji-Quan / Zhang, Zhaoda / Kuruppu, Darshini et al. | 2012
- 1963
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Novel substituted 9-norbornylpurines and their activities against RNA virusesŠála, Michal / Hřebabecký, Hubert / Leyssen, Pieter et al. | 2012
- 1969
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SAR-study on a new class of imidazo[1,2-a]pyridine-based inhibitors of 5-lipoxygenaseHieke, Martina / Rödl, Carmen B. / Wisniewska, Joanna M. et al. | 2012
- 1976
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Synthesis and biological evaluation of novel amprenavir-based P1-substituted bi-aryl derivatives as ultra-potent HIV-1 protease inhibitorsYan, Jianwei / Huang, Ning / Li, Shukun et al. | 2012
- 1980
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3,5-Disubstituted indole derivatives as selective human neuronal nitric oxide synthase (nNOS) inhibitorsAnnedi, Subhash C. / Maddaford, Shawn P. / Ramnauth, Jailall et al. | 2012
- 1985
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Structure–activity relationship study of selective benzimidazole-based inhibitors of Cryptosporidium parvum IMPDHKirubakaran, Sivapriya / Gorla, Suresh Kumar / Sharling, Lisa et al. | 2012
- 1989
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5-Aryl-4-carboxamide-1,3-oxazoles: Potent and selective GSK-3 inhibitorsGentile, Gabriella / Merlo, Giancarlo / Pozzan, Alfonso et al. | 2012
- 1995
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A domino Knoevenagel hetero-Diels–Alder reaction for the synthesis of polycyclic chromene derivatives and evaluation of their cytotoxicityReddy, B.V. Subba / Divya, Baddula / Swain, Manisha et al. | 2012
- 2000
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A small molecule regulates hairpin structures in d(CGG) trinucleotide repeatsHagihara, Masaki / He, Hanping / Kimura, Maki et al. | 2012
- 2004
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Depigmenting activity of new kojic acid derivative obtained as a side product in the synthesis of cinnamate of kojic acidCho, Jun-Cheol / Rho, Ho Sik / Baek, Heung Soo et al. | 2012
- 2008
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Design, synthesis, single-crystal and preliminary antitumor activity of novel arenesulfonylimidazolidin-2-onesAbdel-Aziz, Alaa A.-M. / El-Azab, Adel S. / El-Subbagh, Hussein I. et al. | 2012
- 2015
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Structure–activity relationship study of beta-carboline derivatives as haspin kinase inhibitorsCuny, Gregory D. / Ulyanova, Natalia P. / Patnaik, Debasis et al. | 2012
- 2020
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Hit to lead SAR study on benzoxazole derivatives for an NPY Y5 antagonistOmori, Naoki / Kouyama, Naoki / Yukimasa, Akira et al. | 2012
- 2024
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Design, synthesis, and evaluation of novel 4-thiazolylimidazoles as inhibitors of transforming growth factor-β type I receptor kinaseAmada, Hideaki / Sekiguchi, Yoshinori / Ono, Naoya et al. | 2012
- 2024
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Design, synthesis, and evaluation of novel 4-thiazolylimidazoles as inhibitors of transforming growth factor-b type I receptor kinaseAmada, H. / Sekiguchi, Y. / Ono, N. et al. | 2012
- 2030
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The anomeric mixture of some O-galactolipid derivatives is more toxic against cancer cells than either anomer aloneSong, Shao-Xing / Wu, Ming-Li / He, Xiao-Peng et al. | 2012
- 2033
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The discovery of aminopyrazines as novel, potent Nav1.7 antagonists: Hit-to-lead identification and SARBregman, Howard / Nguyen, Hanh Nho / Feric, Elma et al. | 2012
- 2043
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The use of small molecule probes to study spatially separated stimulus-induced signaling pathwaysKravchenko, Vladimir V. / Gloeckner, Christian / Stowe, G. Neil et al. | 2012
- 2046
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Discovery of a new class of ghrelin receptor antagonistsMihalic, Jeffrey T. / Kim, Yong-Jae / Lizarzaburu, Mike et al. | 2012
- 2052
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Discovery and hit-to-lead optimization of pyrrolopyrimidines as potent, state-dependent Nav1.7 antagonistsChakka, Nagasree / Bregman, Howie / Du, Bingfan et al. | 2012
- 2063
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Discovery of azabenzimidazole derivatives as potent, selective inhibitors of TBK1/IKKε kinasesWang, Tao / Block, Michael A. / Cowen, Scott et al. | 2012
- 2070
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Synthesis, SAR and biological evaluation of 1,6-disubstituted-1H-pyrazolo[3,4-d]pyrimidines as dual inhibitors of Aurora kinases and CDK1Le Brazidec, Jean-Yves / Pasis, Angela / Tam, Betty et al. | 2012
- 2075
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Synthesis and structure–activity relationship (SAR) study of 4-azabenzoxazole analogues as H3 antagonistsShao, Ning / Aslanian, Robert / West, Robert E. Jr. et al. | 2012
- 2079
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Cytotoxic terpenoids from Juglans sinensis leaves and twigsYang, Heejung / Cho, Hyun-Jong / Sim, So Hee et al. | 2012
- 2084
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Identification of 3-acyl-2-phenylamino-1,4-dihydroquinolin-4-one derivatives as inhibitors of the phosphatase SerB653 in Porphyromonas gingivalis, implicated in periodontitisJung, Suk-Kyeong / Ko, Youngkyung / Yu, Keum Ran et al. | 2012
- 2089
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Syntheses of structurally-simplified and fluorescently-labeled neovibsanin derivatives and analysis of their neurite outgrowth activity in PC12 cellsImagawa, Hiroshi / Saijo, Hayato / Yamaguchi, Hitomi et al. | 2012
- 2094
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Discovery of the first small molecule inhibitor of human DDX3 specifically designed to target the RNA binding site: Towards the next generation HIV-1 inhibitorsRadi, Marco / Falchi, Federico / Garbelli, Anna et al. | 2011
- 2099
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Towards the preparation of radiolabeled 1-aryl-3-benzyl ureas: Radiosynthesis of [11C-carbonyl] AR-A014418 by [11C]CO2 fixationHicks, Justin W. / Wilson, Alan A. / Rubie, Elizabeth A. et al. | 2011
- 2102
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Two-step efficient synthesis of 5-methyluridine via two thermostable nucleoside phosphorylase from Aeropyrum pernixZhu, Shaozhou / Ren, Lu / Wang, Jianjun et al. | 2011
- 2105
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Methoxychalcone inhibitors of androgen receptor translocation and functionKim, Yeong Sang / Kumar, Vineet / Lee, Sunmin et al. | 2011
- 2110
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Adamantyl N-benzylbenzamide: New series of depigmentation agents with tyrosinase inhibitory activityBaek, Heung Soo / Hong, Yong Deog / Lee, Chang Seok et al. | 2011
- 2114
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A resveratrol analog, phoyunbene B, induces G2/M cell cycle arrest and apoptosis in HepG2 liver cancer cellsWang, Guanghui / Guo, Xiaoyu / Chen, Haifeng et al. | 2011
- 2119
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Discovery of 3,4-dihydropyrimidin-2(1H)-ones with inhibitory activity against HIV-1 replicationKim, Junwon / Park, Changmin / Ok, Taedong et al. | 2011
- 2125
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Small molecule inhibitors of the HPV16-E6 interaction with caspase 8Yuan, Chung-Hsiang / Filippova, Maria / Tungteakkhun, Sandy S. et al. | 2011
- 2130
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Erratum to “Potent mGluR5 antagonists: Pyridyl and thiazolyl-ethynyl-3,5-disubstituted-phenyl series” [Bioorg. Med. Chem. Lett. 21 (2011) 3243–3247]Alagille, David / DaCosta, Herve / Chen, Yelin et al. | 2012
- 2131
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Corrigendum to “Absolute configurations of tubulin inhibitors taltobulin (HTI-286) and HTI-042 characterized by X-ray diffraction analysis and NMR studies” [Bioorg. Med. Chem. Lett. 20 (2010) 1535–1538]Niu, Chuansheng / Ho, Douglas M. / Williamson, Robert Thomas et al. | 2012
- IFC
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Editorial board| 2012