Design and synthesis of novel 7-aminoquinazoline derivatives: Antitumor and anticonvulsant activities (English)
- New search for: El-Azab, Adel S.
- New search for: El-Azab, Adel S.
- New search for: ElTahir, Kamal E.H.
In:
Bioorganic & medicinal chemistry letters
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22
, 5
; 1879-1886
;
2012
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ISSN:
- Article (Journal) / Print
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Title:Design and synthesis of novel 7-aminoquinazoline derivatives: Antitumor and anticonvulsant activities
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Contributors:El-Azab, Adel S. ( author ) / ElTahir, Kamal E.H.
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Published in:Bioorganic & medicinal chemistry letters ; 22, 5 ; 1879-1886
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2012
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.42
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Source:
Table of contents – Volume 22, Issue 5
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1831
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Graphical contents list| 2012
- 1846
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Synthesis of novel long wavelength cationic chlorins via stereoselective aldol-like condensationLi, Jia Zhu / Wang, Jin Jun / Yoon, Il / Cui, Bing Cun / Shim, Young Key et al. | 2012
- 1850
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Synthesis and biological evaluation of sulfonyl acrylonitriles as novel inhibitors to peritoneal carcinomatosisZificsak, Craig A. / Shen, Yi / Lisko, Joseph G. / Theroff, Jay P. / Lao, Xuegang / Bollt, Oana / Li, Xiufen / Dorsey, Bruce D. / Kuwada, Scott K. et al. | 2012
- 1854
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Aminoimidazoles as BACE-1 inhibitors: The challenge to achieve in vivo brain efficacySwahn, Britt-Marie / Holenz, Jörg / Kihlström, Jacob / Kolmodin, Karin / Lindström, Johan / Plobeck, Niklas / Rotticci, Didier / Sehgelmeble, Fernando / Sundström, Marie / Berg, Stefan von et al. | 2012
- 1860
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New aromatase inhibitors from the 3-pyridyl arylether and 1-aryl pyrrolo[2,3-c]pyridine seriesStauffer, Frédéric / Furet, Pascal / Floersheimer, Andreas / Lang, Marc et al. | 2012
- 1864
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Characterization of TAE684 as a potent LRRK2 kinase inhibitorZhang, Jinwei / Deng, Xianming / Choi, Hwan Geun / Alessi, Dario R. / Gray, Nathanael S. et al. | 2012
- 1870
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Identification of fused bicyclic heterocycles as potent and selective 5-HT2A receptor antagonists for the treatment of insomniaXiong, Yifeng / Ullman, Brett / Choi, Jin-Sun Karoline / Cherrier, Martin / Strah-Pleynet, Sonja / Decaire, Marc / Feichtinger, Konrad / Frazer, John M. / Yoon, Woo H. / Whelan, Kevin et al. | 2012
- 1874
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Imidazo[1,2-a]pyrazines as novel PI3K inhibitorsMartínez González, Sonia / Hernández, Ana Isabel / Varela, Carmen / Rodríguez-Arístegui, Sonsoles / Alvarez, Rosa María / García, Ana Belén / Lorenzo, Milagros / Rivero, Virginia / Oyarzabal, Julen / Rabal, Obdulia et al. | 2012
- 1879
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Design and synthesis of novel 7-aminoquinazoline derivatives: Antitumor and anticonvulsant activitiesEl-Azab, Adel S. / ElTahir, Kamal E.H. et al. | 2012
- 1886
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Inhibitors of human histone deacetylase with potent activity against the African trypanosome Trypanosoma bruceiKelly, John M. / Taylor, Martin C. / Horn, David / Loza, Einars / Kalvinsh, Ivars / Björkling, Fredrik et al. | 2012
- 1891
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Structure–activity relationship of the 7-hydroxy benzimidazole analogs as glycogen synthase kinase 3β inhibitorLee, Seung-Chul / Shin, Dongkyu / Cho, Joong Myung / Ro, Sunggu / Suh, Young-Ger et al. | 2012
- 1891
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Structure-activity relationship of the 7-hydroxy benzimidazole analogs as glycogen synthase kinase 3b inhibitorLee, S. C. / Shin, D. / Cho, J. M. / Ro, S. / Suh, Y. G. et al. | 2012
- 1895
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New antitumor compounds from Carya cathayensisWu, Wei / Bi, Xiu-Li / Cao, Jia-Qing / Zhang, Kai-Qing / Zhao, Yu-Qing et al. | 2012
- 1899
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Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the δ opioid receptor. Discovery of two highly potent and selective δ opioid agonistsBerezowska, Irena / Lemieux, Carole / Chung, Nga N. / Ding, Jinguo / Schiller, Peter W. et al. | 2012
- 1899
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Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the d opioid receptor. Discovery of two highly potent and selective d opioid agonistsBerezowska, I. / Lemieux, C. / Chung, N. N. / Ding, J. / Schiller, P. W. et al. | 2012
- 1903
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Discovery of vinylcycloalkyl-substituted benzimidazole TRPM8 antagonists effective in the treatment of cold allodyniaCalvo, Raul R. / Meegalla, Sanath K. / Parks, Daniel J. / Parsons, William H. / Ballentine, Shelley K. / Lubin, Mary Lou / Schneider, Craig / Colburn, Raymond W. / Flores, Christopher M. / Player, Mark R. et al. | 2012
- 1908
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New cyclic peptides with osteoblastic proliferative activity from Dianthus superbusTong, Yun / Luo, Jian-Guang / Wang, Rui / Wang, Xiao-Bing / Kong, Ling-Yi et al. | 2012
- 1912
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1,2,4-Oxadiazoles: A new class of anti-prostate cancer agentsKhatik, Gopal L. / Kaur, Jasmine / Kumar, Varun / Tikoo, Kulbhushan / Nair, Vipin A. et al. | 2012
- 1917
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Novel imidazo[2,1-b][1,3,4]thiadiazole carrying rhodanine-3-acetic acid as potential antitubercular agentsAlegaon, Shankar G. / Alagawadi, Kallanagouda R. / Sonkusare, Pranali V. / Chaudhary, Sagar M. / Dadwe, Dilip H. / Shah, Amol S. et al. | 2012
- 1922
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Synthesis and evaluation of cytotoxic effects of novel α-methylenelactone tetracyclic diterpenoidsZeng, Yao-fu / Wu, Jia-qiang / Shi, Lian-yong / Wang, Ke / Zhou, Bin / Tang, Yong / Zhang, Da-yong / Wu, Yang-chang / Hua, Wei-yi / Wu, Xiao-ming et al. | 2012
- 1922
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Synthesis and evaluation of cytotoxic effects of novel a-methylenelactone tetracyclic diterpenoidsZeng, Y. f. / Wu, J. q. / Shi, L. y. / Wang, K. / Zhou, B. / Tang, Y. / Zhang, D. y. / Wu, Y. c. / Hua, W. y. / Wu, X. m. et al. | 2012
- 1926
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Anti-tumor activity of new orally bioavailable 2-amino-5-(thiophen-2-yl)benzamide-series histone deacetylase inhibitors, possessing an aqueous soluble functional group as a surface recognition domainHirata, Yoshiyuki / Hirata, Masahiko / Kawaratani, Yasuyuki / Shibano, Makio / Taniguchi, Masahiko / Yasuda, Masahide / Ohmomo, Yoshiro / Nagaoka, Yasuo / Baba, Kimiye / Uesato, Shinichi et al. | 2012
- 1931
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Characterization of H2O-forming NADH oxidase from Streptococcus pyogenes and its application in l-rare sugar productionGao, Hui / Tiwari, Manish Kumar / Kang, Yun Chan / Lee, Jung-Kul et al. | 2012
- 1936
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Influence of ring size on the cognition-enhancing activity of DM235 and MN19, two potent nootropic drugsGuandalini, L. / Martini, E. / Di Cesare Mannelli, L. / Dei, S. / Manetti, D. / Scapecchi, S. / Teodori, E. / Ghelardini, C. / Romanelli, M.N. et al. | 2012
- 1940
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Aminopyrimidinone Cdc7 Kinase InhibitorsWoods, Keith W. / Lai, Chunqiu / Miyashiro, Julie M. / Tong, Yunsong / Florjancic, Alan S. / Han, Edward K. / Soni, Niru / Shi, Yan / Lasko, Loren / Leverson, Joel D. et al. | 2012
- 1944
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Discovery of 4-hydroxy-1,6-naphthyridine-3-carbonitrile derivatives as novel PDE10A inhibitorsBauer, Udo / Giordanetto, Fabrizio / Bauer, Martin / O’Mahony, Gavin / Johansson, Kjell E. / Knecht, Wolfgang / Hartleib-Geschwindner, Judith / Carlsson, Eva Töppner / Enroth, Cristofer et al. | 2012
- 1949
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Novel bisbenzimide-nitroxides for nuclear redox imaging in living cellsIkeda, Mamiko / Nakagawa, Hidehiko / Suzuki, Takayoshi / Miyata, Naoki et al. | 2012
- 1953
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3,4-Diarylpiperidines as potent renin inhibitorsLacombe, Patrick / Arbour, Mélissa / Aspiotis, Renée / Cauchon, Elizabeth / Chen, Austin / Dubé, Daniel / Falgueyret, Jean-Pierre / Fournier, Pierre-André / Gallant, Michel / Grimm, Erich et al. | 2012
- 1958
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Radiosynthesis of PET radiotracer as a prodrug for imaging group II metabotropic glutamate receptors in vivoWang, Ji-Quan / Zhang, Zhaoda / Kuruppu, Darshini / Brownell, Anna-Liisa et al. | 2012
- 1963
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Novel substituted 9-norbornylpurines and their activities against RNA virusesŠála, Michal / Hřebabecký, Hubert / Leyssen, Pieter / Dejmek, Milan / Dračínský, Martin / De Palma, Armando M. / Neyts, Johan / Nencka, Radim et al. | 2012
- 1969
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SAR-study on a new class of imidazo[1,2-a]pyridine-based inhibitors of 5-lipoxygenaseHieke, Martina / Rödl, Carmen B. / Wisniewska, Joanna M. / la Buscató, Estel. / Stark, Holger / Schubert-Zsilavecz, Manfred / Steinhilber, Dieter / Hofmann, Bettina / Proschak, Ewgenij et al. | 2012
- 1976
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Synthesis and biological evaluation of novel amprenavir-based P1-substituted bi-aryl derivatives as ultra-potent HIV-1 protease inhibitorsYan, Jianwei / Huang, Ning / Li, Shukun / Yang, Liu-Meng / Xing, Weiqiang / Zheng, Yong-Tang / Hu, Youhong et al. | 2012
- 1980
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3,5-Disubstituted indole derivatives as selective human neuronal nitric oxide synthase (nNOS) inhibitorsAnnedi, Subhash C. / Maddaford, Shawn P. / Ramnauth, Jailall / Renton, Paul / Speed, Joanne / Rakhit, Suman / Andrews, John S. / Porreca, Frank et al. | 2012
- 1985
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Structure–activity relationship study of selective benzimidazole-based inhibitors of Cryptosporidium parvum IMPDHKirubakaran, Sivapriya / Gorla, Suresh Kumar / Sharling, Lisa / Zhang, Minjia / Liu, Xiaoping / Ray, Soumya S. / MacPherson, Iain S. / Striepen, Boris / Hedstrom, Lizbeth / Cuny, Gregory D. et al. | 2012
- 1989
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5-Aryl-4-carboxamide-1,3-oxazoles: Potent and selective GSK-3 inhibitorsGentile, Gabriella / Merlo, Giancarlo / Pozzan, Alfonso / Bernasconi, Giovanni / Bax, Benjamin / Bamborough, Paul / Bridges, Angela / Carter, Paul / Neu, Margarete / Yao, Gang et al. | 2012
- 1995
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A domino Knoevenagel hetero-Diels–Alder reaction for the synthesis of polycyclic chromene derivatives and evaluation of their cytotoxicityReddy, B.V. Subba / Divya, Baddula / Swain, Manisha / Rao, T. Prabhakar / Yadav, J.S. / Vishnu Vardhan, M.V.P.S. et al. | 2012
- 2000
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A small molecule regulates hairpin structures in d(CGG) trinucleotide repeatsHagihara, Masaki / He, Hanping / Kimura, Maki / Nakatani, Kazuhiko et al. | 2012
- 2004
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Depigmenting activity of new kojic acid derivative obtained as a side product in the synthesis of cinnamate of kojic acidCho, Jun-Cheol / Rho, Ho Sik / Baek, Heung Soo / Ahn, Soo Mi / Woo, Byoung Young / Hong, Yong Deog / Cheon, Jong Woo / Heo, Jung Mi / Shin, Song Seok / Park, Young-Ho et al. | 2012
- 2008
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Design, synthesis, single-crystal and preliminary antitumor activity of novel arenesulfonylimidazolidin-2-onesAbdel-Aziz, Alaa A.-M. / El-Azab, Adel S. / El-Subbagh, Hussein I. / Al-Obaid, Abdulrahman M. / Alanazi, Amer M. / Al-Omar, Mohamed A. et al. | 2012
- 2015
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- 2020
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- IFC
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Editorial board| 2012