-Phosphonosulfonic Acids: Potent and Selective Inhibitors of Squalene Synthase (English)
- New search for: Magnin, D. R.
- New search for: Biller, S. A.
- New search for: Chen, Y.
- New search for: Dickson, J. K.
- New search for: Fryszman, O. M.
- New search for: Lawrence, R. M.
- New search for: Logan, J. V. H.
- New search for: Sieber-McMaster, E. S.
- New search for: Sulsky, R. B.
- New search for: Traeger, S. C.
- New search for: Magnin, D. R.
- New search for: Biller, S. A.
- New search for: Chen, Y.
- New search for: Dickson, J. K.
- New search for: Fryszman, O. M.
- New search for: Lawrence, R. M.
- New search for: Logan, J. V. H.
- New search for: Sieber-McMaster, E. S.
- New search for: Sulsky, R. B.
- New search for: Traeger, S. C.
In:
JOURNAL OF MEDICINAL CHEMISTRY
;
39
, 3
;
657-660
;
1996
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ISSN:
- Article (Journal) / Print
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Title:-Phosphonosulfonic Acids: Potent and Selective Inhibitors of Squalene Synthase
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Contributors:Magnin, D. R. ( author ) / Biller, S. A. ( author ) / Chen, Y. ( author ) / Dickson, J. K. ( author ) / Fryszman, O. M. ( author ) / Lawrence, R. M. ( author ) / Logan, J. V. H. ( author ) / Sieber-McMaster, E. S. ( author ) / Sulsky, R. B. ( author ) / Traeger, S. C. ( author )
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Published in:JOURNAL OF MEDICINAL CHEMISTRY ; 39, 3 ; 657-660
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Publisher:
- New search for: ACS AMERICAN CHEMICAL SOCIETY
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Publication date:1996-01-01
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Size:4 pages
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ISSN:
-
Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 615
- Further information on Dewey Decimal Classification
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Classification:
DDC: 615 -
Source:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Table of contents – Volume 39, Issue 3
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 625
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Nonpeptide Angiotensin II Receptor Antagonists: The Next Generation in Antihypertensive TherapyWexler, Ruth R. / Greenlee, William J. / Irvin, John D. / Goldberg, Michael R. / Prendergast, Kristine / Smith, Ronald D. / Timmermans, Pieter B. M. W. M. et al. | 1996
- 657
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a-Phosphonosulfonic Acids: Potent and Selective Inhibitors of Squalene SynthaseMagnin, David R. et al. | 1996
- 657
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α-Phosphonosulfonic Acids: Potent and Selective Inhibitors of Squalene SynthaseMagnin, David R. / Biller, Scott A. / Chen, Ying / Dickson,, John K. / Fryszman, Olga M. / Lawrence, R. Michael / Logan, Janette V. H. / Sieber-McMaster, Ellen S. / Sulsky, Richard B. / Traeger, Sarah C. et al. | 1996
- 661
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Orally Active Squalene Synthase Inhibitors: Bis((acyloxy)alkyl) Prodrugs of the a-Phosphonosulfonic Acid MoietyDickson Jr, John K. et al. | 1996
- 661
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Orally Active Squalene Synthase Inhibitors: Bis((acyloxy)alkyl) Prodrugs of the α-Phosphonosulfonic Acid MoietyDickson,, John K. / Biller, Scott A. / Magnin, David R. / Petrillo,, Edward W. / Hillyer, John W. / Hsieh, Dolly C. / Lan, Shih-Jung / Rinehart, J. Kent / Gregg, Richard E. / Harrity, Thomas W. et al. | 1996
- 665
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The Structure-Activity Relationship between Peroxisome Proliferator-Activated Receptor gamma Agonism and the Antihyperglycemic Activity of ThiazolidinedionesWillson, T. M. / Cobb, J. E. / Cowan, D. J. / Wiethe, R. W. / Correa, I. D. / Prakash, S. R. / Beck, K. D. / Moore, L. B. / Kliever, S. A. / Lehmann, J. M. et al. | 1996
- 665
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The Structure-Activity Relationship between Peroxisome Proliferator-Activated Receptor g Agonism and the Antihyperglycemic Activity of ThiazolidinedionesWillson, Timothy M. et al. | 1996
- 665
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The Structure−Activity Relationship between Peroxisome Proliferator-Activated Receptor γ Agonism and the Antihyperglycemic Activity of ThiazolidinedionesWillson, Timothy M. / Cobb, Jeffery E. / Cowan, David J. / Wiethe, Robert W. / Correa, Itzela D. / Prakash, Shimoga R. / Beck, Kelli D. / Moore, Linda B. / Kliewer, Steven A. / Lehmann, Jürgen M. et al. | 1996
- 669
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2-Iminopiperidine and Other 2-Iminoazaheterocycles as Potent Inhibitors of Human Nitric Oxide Synthase Isoforms †Moore, William M. / Webber, R. Keith / Fok, Kam F. / Jerome, Gina M. / Connor, Jane R. / Manning, Pamela T. / Wyatt, Pamela S. / Misko, Thomas P. / Tjoeng, Foe S. / Currie, Mark G. et al. | 1996
- 673
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Synthesis and Antibacterial Activity of U-100592 and U-100766, Two Oxazolidinone Antibacterial Agents for the Potential Treatment of Multidrug-Resistant Gram-Positive Bacterial InfectionsBrickner, Steven J. / Hutchinson, Douglas K. / Barbachyn, Michael R. / Manninen, Peter R. / Ulanowicz, Debra A. / Garmon, Stuart A. / Grega, Kevin C. / Hendges, Susan K. / Toops, Dana S. / Ford, Charles W. et al. | 1996
- 680
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Identification of a Novel Oxazolidinone (U-100480) with Potent Antimycobacterial ActivityBarbachyn, Michael R. / Hutchinson, Douglas K. / Brickner, Steven J. / Cynamon, Michael H. / Kilburn, James O. / Klemens, Sally P. / Glickman, Suzanne E. / Grega, Kevin C. / Hendges, Susan K. / Toops, Dana S. et al. | 1996
- 686
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Slow-Binding Inhibition of g-Aminobutyric Acid Aminotransferase by Hydrazine AnaloguesLightcap, Eric S. et al. | 1996
- 686
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Slow-Binding Inhibition of γ-Aminobutyric Acid Aminotransferase by Hydrazine Analogues † , ‡Lightcap, Eric S. / Silverman, Richard B. et al. | 1996
- 686
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Slow-Binding Inhibition of gamma-Aminobutyric Acid Aminotransferase by Hydrazine AnaloguesLightcap, E. S. / Silverman, R. B. et al. | 1996
- 695
-
Quinazoline Antifolates Thymidylate Synthase Inhibitors: Lipophilic Analogues with Modification to the C2-Methyl SubstituentHennequin, Laurent F. / Boyle, F. Thomas / Wardleworth, J. Michael / Marsham, Peter R. / Kimbell, Rosemary / Jackman, Ann L. et al. | 1996
- 705
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An Approach to Rapid Estimation of Relative Binding Affinities of Enzyme Inhibitors: Application to Peptidomimetic Inhibitors of the Human Immunodeficiency Virus Type 1 ProteaseViswanadhan, Vellarkad N. / Reddy, M. Rami / Wlodawer, Alexander / Varney, Michael D. / Weinstein, John N. et al. | 1996
- 713
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Water Soluble Inhibitors of Topoisomerase I: Quaternary Salt Derivatives of CamptothecinLackey, Karen / Sternbach, Daniel D. / Croom, Dallas K. / Emerson, David L. / Evans, Michael G. / Leitner, Peter L. / Luzzio, Michael J. / McIntyre, Gordon / Vuong, Alain / Yates, Julie et al. | 1996
- 720
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In Vivo Activity and Hydrophobicity of Cytostatic Aziridinyl QuinonesMoret, Ed E. / de Boer, Mark / Hilbers, Hans W. / Tollenaere, Jan P. / Janssen, Lambert H. M. / Holthuis, Joost J. M. / Driebergen, Reinoud J. / Verboom, Willem / Reinhoudt, David N. et al. | 1996
- 729
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Structure−Activity Relationships of the Quinolone Antibacterials against Mycobacteria: Effect of Structural Changes at N-1 and C-7 †Renau, Thomas E. / Sanchez, Joseph P. / Gage, Jeffrey W. / Dever, Julie A. / Shapiro, Martin A. / Gracheck, Stephen J. / Domagala, John M. et al. | 1996
- 736
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3-Aryl-1,2-diacetamidopropane Derivatives as Novel and Potent NK-1 Receptor AntagonistsHipskind, Philip A. / Howbert, J. Jeffry / Bruns, Robert F. / Cho, Steven S. Y. / Crowell, Thomas A. / Foreman, Mark M. / Gehlert, Donald R. / Iyengar, Smriti / Johnson, Kirk W. / Krushinski, Joseph H. et al. | 1996
- 749
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Structure−Activity Relationship Studies of Novel 4-[2-[Bis(4-fluorophenyl)methoxy]ethyl]-1-(3-phenylpropyl)piperidine Analogs: Synthesis and Biological Evaluation at the Dopamine and Serotonin Transporter SitesDutta, Aloke K. / Xu, Cen / Reith, Maarten E. A. et al. | 1996
- 749
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Structure-Activity Relationship Studies of Novel 4-[2-[Bis(4-fluorophenyl)methoxyl)-ethyl]-1-(3-phenylpropyl)piperidine Analogs: Synthesis and Biological Evaluation at the Dopamine and Serotonin Transporter SitesDutta, A. K. / Xu, C. / Reith, M. E. A. et al. | 1996
- 757
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Structure−Activity Relationships of a New Family of Steroidal Aromatase Inhibitors. 1. Synthesis and Evaluation of a Series of Analogs Related to 19-[(Methylthio)methyl]androstenedione (RU54115)Lesuisse, Dominique / Gourvest, Jean-François / Benslimane, Ouafae / Canu, Frank / Delaisi, Christine / Doucet, Bernard / Hartmann, Catherine / Lefrançois, Jean-Michel / Tric, Bernadette / Mansuy, Daniel et al. | 1996
- 773
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Design and Synthesis of 1-Aminocycloalkane-1-carboxylic Acid-Substituted Deltorphin Analogues: Unique δ and μ Opioid Activity in Modified PeptidesBreveglieri, Angela / Guerrini, Remo / Salvadori, Severo / Bianchi, Clementina / Bryant, Sharon D. / Attila, Martti / Lazarus, Lawrence H. et al. | 1996
- 773
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Design and Synthesis of 1-Aminocycloalkane-1-carboxylic Acid-Substituted Deltorphin Analogues: Unique d and m Opioid Activity in Modified PeptidesBreveglieri, Angela et al. | 1996
- 781
-
Interactions of Flavonoids and Other Phytochemicals with Adenosine ReceptorsJi, Xiao-duo / Melman, Neli / Jacobson, Kenneth A. et al. | 1996
- 789
-
Synthesis and Anti-Herpes Virus Activity of 2‘-Deoxy-4‘-thiopyrimidine NucleosidesRahim, S. George / Trivedi, Naimisha / Bogunovic-Batchelor, Mirjana V. / Hardy, George W. / Mills, Gail / Selway, John W. T. / Snowden, Wendy / Littler, Edward / Coe, Paul L. / Basnak, Ivan et al. | 1996
- 796
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Antitumor 2-(Aminocarbonyl)-1,2-bis(methylsulfonyl)-1-(2-chloroethyl)- hydrazinesShyam, Krishnamurthy / Penketh, Philip G. / Loomis, Regina H. / Rose, William C. / Sartorelli, Alan C. et al. | 1996
- 802
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Novel N 6-(Substituted-phenylcarbamoyl)adenosine-5‘-uronamides as Potent Agonists for A3 Adenosine ReceptorsBaraldi, Pier Giovanni / Cacciari, Barbara / Spalluto, Giampiero / Ji, Xiao-duo / Olah, Mark E. / Stiles, Gary / Dionisotti, Silvio / Zocchi, Cristina / Ongini, Ennio / Jacobson, Kenneth A. et al. | 1996
- 807
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Cancer Chemotherapeutic AgentsBrueggemeier, Robert W. et al. | 1996
- 807
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Cancer Chemotherapeutic Agents William O. Foye, Editor. American Chemical Society, Washington, D.C. 1995. xx + 698 pp. 18.5 × 26 cm. ISBN 0-8412-2920-1. $149.95.Brueggemeier, Robert W. et al. | 1996
- 807
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Taxol: Science and ApplicationsOjima, Iwao et al. | 1996
- 807
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Taxol®: Science and Applications Edited by Matthew Suffness. CRC Press, Boca Raton, FL. 1995. 426 pp. 18.5 × 26 cm. ISBN 0-8493-8382-X. $129.95.Ojima, Iwao et al. | 1996
- 808
-
Percutaneous Penetration EnhancersChasin, Mark et al. | 1996
- 808
-
CNS Neurotransmitters and Neuromodulators Glutamate Edited by Trevor W. Stone. CRC Press, Boca Raton, FL. 1995. 380 pp. 18.5 × 26 cm. ISBN 0-8493-7631-9. $159.95.Ferkany, John Wm. et al. | 1996
- 808
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CNS Neurotransmitters and Neuromodulators GlutamateFerkany, John Wm et al. | 1996
- 808
-
Percutaneous Penetration Enhancers Edited by Eric W. Smith and Howard I. Maibach. CRC Press, New York. 1995. 500 pp. 16.5 × 24 cm. ISBN 0-8493-2605-2. $125.00.Chasin, Mark et al. | 1996
- 809
-
Antibiotics. A Multidisciplinary ApproachElliott, Richard L. et al. | 1996
- 809
-
Endothelin Receptors. From the Gene to the HumanCody, Wayne L. et al. | 1996
- 809
-
Annual Reports in Medicinal Chemistry. Volume 30 - Staff| 1996
- 809
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Antibiotics. A Multidisciplinary Approach By Giancarlo Lancini, Francesco Parenti, and Gian Gualberto Gallo. Plenum Press, New York. 1995. ix + 278 pp. 15.5 × 23.5 cm. ISBN 0-306-44924-2. $59.50.Elliott, Richard L. et al. | 1996
- 809
-
Annual Reports in Medicinal Chemistry. Volume 30 Editor-in-Chief: James A. Bristol. Academic Press, Inc., San Diego, CA. 1995. xi + 387 pp. 17 × 25 cm. ISBN 0-12-040530-X. $70.00 (pbk).| 1996
- 809
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Endothelin Receptors. From the Gene to the Human Edited by Robert R. Ruffolo, Jr. CRC Press Inc., Boca Raton, FL. 1995. 285 pp. 16 × 24 cm. ISBN 0-8493-5938-4. $169.95.Cody, Wayne L. et al. | 1996