N-n-Propyl-Substituted 3-(Dimethylphenyl)piperidines Display Novel Discriminative Properties between Dopamine Receptor Subtypes: Synthesis and Receptor Binding Studies (English)
- New search for: Cervetto, L.
- New search for: Demontis, G. C.
- New search for: Giannaccini, G.
- New search for: Longoni, B.
- New search for: Macchia, B.
- New search for: Macchia, M.
- New search for: Martinelli, A.
- New search for: Orlandini, E.
- New search for: Cervetto, L.
- New search for: Demontis, G. C.
- New search for: Giannaccini, G.
- New search for: Longoni, B.
- New search for: Macchia, B.
- New search for: Macchia, M.
- New search for: Martinelli, A.
- New search for: Orlandini, E.
In:
JOURNAL OF MEDICINAL CHEMISTRY
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41
, 25
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4933-4938
;
1998
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ISSN:
- Article (Journal) / Print
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Title:N-n-Propyl-Substituted 3-(Dimethylphenyl)piperidines Display Novel Discriminative Properties between Dopamine Receptor Subtypes: Synthesis and Receptor Binding Studies
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Contributors:Cervetto, L. ( author ) / Demontis, G. C. ( author ) / Giannaccini, G. ( author ) / Longoni, B. ( author ) / Macchia, B. ( author ) / Macchia, M. ( author ) / Martinelli, A. ( author ) / Orlandini, E. ( author )
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Published in:JOURNAL OF MEDICINAL CHEMISTRY ; 41, 25 ; 4933-4938
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Publisher:
- New search for: ACS AMERICAN CHEMICAL SOCIETY
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Publication date:1998-01-01
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Size:6 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 615
- Further information on Dewey Decimal Classification
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Classification:
DDC: 615 -
Source:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Table of contents – Volume 41, Issue 25
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 4911
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Mutational Evidence for a Common kappa Antagonist Binding Pocket in the Wild-Type kappa and Mutant [K303E] Opioid ReceptorsJones, R. M. / Hjorth, S. A. / Schwartz, T. W. / Portoghese, P. S. et al. | 1998
- 4911
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Mutational Evidence for a Common κ Antagonist Binding Pocket in the Wild-Type κ and Mutant μ[K303E] Opioid Receptors †Jones, Robert M. / Hjorth, Siv A. / Schwartz, Thue W. / Portoghese, Philip S. et al. | 1998
- 4911
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COMMUNICATIONS TO THE EDITOR - Mutational Evidence for a Common K Antagonist Binding Pocket in the Wild-Type k and Mutant m(K303E) Opioid ReceptorsJones, Robert M. et al. | 1998
- 4915
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Dual D2-Receptor and β2-Adrenoceptor Agonists for the Treatment of Airway Diseases. 1. Discovery and Biological Evaluation of Some 7-(2-Aminoethyl)- 4-hydroxybenzothiazol-2(3H)-one AnaloguesBonnert, Roger V. / Brown, Roger C. / Chapman, David / Cheshire, David R. / Dixon, John / Ince, Francis / Kinchin, Elizabeth C. / Lyons, Amanda J. / Davis, Andrew M. / Hallam, Catherine et al. | 1998
- 4915
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COMMUNICATIONS TO THE EDITOR - Dual D2-Receptor and b2-Adrenoceptor Agonists for the Treatment of Airway Diseases. 1. Discovery and Biological Evaluation of Some 7-(2-Aminoethyl)-4-hydroxybenzothiazol-2(3H)-one AnaloguesBonnert, Roger V. et al. | 1998
- 4918
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Structure−Activity Relationships for Antiplasmodial Activity among 7-Substituted 4-AminoquinolinesDe, Dibyendu / Krogstad, Frances M. / Byers, Larry D. / Krogstad, Donald J. et al. | 1998
- 4918
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ARTICLES - Structure-Activity Relationships for Antiplasmodial Activity among 7-Substituted 4-AminoquinolinesDe, Dibyendu et al. | 1998
- 4927
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Polyanion Inhibitors of HIV and Other Viruses. 7. Polyanionic Compounds and Polyzwitterionic Compounds Derived from Cyclodextrins as Inhibitors of HIV TransmissionLeydet, Alain / Moullet, Céline / Roque, Jean Pierre / Witvrouw, Myriam / Pannecouque, Christophe / Andrei, Graciela / Snoeck, Robert / Neyts, Johan / Schols, Dominique / De Clercq, Erik et al. | 1998
- 4927
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ARTICLES - Polyanion Inhibitors of HIV and Other Viruses. 7. Polyanionic Compounds and Polyzwitterionic Compounds Derived from Cyclodextrins as Inhibitors of HIV TransmissionLeydet, Alain et al. | 1998
- 4933
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N-n-Propyl-Substituted 3-(Dimethylphenyl)piperidines Display Novel Discriminative Properties between Dopamine Receptor Subtypes: Synthesis and Receptor Binding StudiesCervetto, Luigi / Demontis, Gian Carlo / Giannaccini, Gino / Longoni, Biancamaria / Macchia, Bruno / Macchia, Marco / Martinelli, Adriano / Orlandini, Elisabetta et al. | 1998
- 4933
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ARTICLES - N-n-Propyl-Substituted 3-(Dimethylphenyl)piperidines Display Novel Discriminative Properties between Dopamine Receptor Subtypes: Synthesis and Receptor Binding StudiesCervetto, Luigi et al. | 1998
- 4939
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Correlation of Human Jejunal Permeability (in Vivo) of Drugs with Experimentally and Theoretically Derived Parameters. A Multivariate Data Analysis ApproachWiniwarter, Susanne / Bonham, Nicholas M. / Ax, Fredrik / Hallberg, Anders / Lennernäs, Hans / Karlén, Anders et al. | 1998
- 4939
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ARTICLES - Correlation of Human Jejunal Permeability (in Vivo) of Drugs with Experimentally and Theoretically Derived Parameters. A Multivariate Data Analysis ApproachWiniwarter, Susanne et al. | 1998
- 4950
-
ARTICLES - Characterization of Novel N,N'-Disubstituted Piperazines as s Receptor LigandsZhang, Ying et al. | 1998
- 4950
-
Characterization of Novel N,N‘-Disubstituted Piperazines as σ Receptor LigandsZhang, Ying / Williams, Wanda / Torrence-Campbell, Cheryl / Bowen, Wayne D. / Rice, Kenner C. et al. | 1998
- 4958
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Antiviral Oligo- and Polyribonucleotides Containing Selected Triazolo[2,3-]purinesTutonda, M. G. / Buckheit, R. W. / Agrawal, V. K. / Broom, A. D. et al. | 1998
- 4958
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Antiviral Oligo- and Polyribonucleotides Containing Selected Triazolo[2,3-a]purines ‖Tutonda, Mayoka G. / Buckheit,, Robert W. / Agrawal, Vijai K. / Broom, Arthur D. et al. | 1998
- 4958
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ARTICLES - Antiviral Oligo- and Polyribonucleotides Containing Selected Triazolo(2,3-a)purinesTutonda, Mayoka G. et al. | 1998
- 4965
-
ARTICLES - Methoxy-Substituted 3-Formyl-2-phenylindoles Inhibit Tubulin PolymerizationGastpar, Robert et al. | 1998
- 4965
-
Methoxy-Substituted 3-Formyl-2-phenylindoles Inhibit Tubulin PolymerizationGastpar, Robert / Goldbrunner, Michael / Marko, Doris / von Angerer, Erwin et al. | 1998
- 4973
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Synthesis and Biological Properties of New 2β-Alkyl- and 2β-Aryl-3-(substituted phenyl)tropane Derivatives: Stereochemical Effect of C-3 on Affinity and Selectivity for Neuronal Dopamine and Serotonin TransportersKozikowski, Alan P. / Araldi, Gian Luca / Prakash, K. R. C. / Zhang, Mei / Johnson, Kenneth M. et al. | 1998
- 4973
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ARTICLES - Synthesis and Biological Properties of New 2b-Alkyl- and 2b-Aryl-3-(substituted phenyl)tropane Derivatives: Stereochemical Effect of C-3 on Affinity and Selectivity for Neuronal Dopamine and Serotonin TransportersKozikowski, Alan P. et al. | 1998
- 4983
-
ARTICLES - Tetrahydro-isoquinoline-Based Factor Xa InhibitorsKucznierz, Ralf et al. | 1998
- 4983
-
Tetrahydro-isoquinoline-Based Factor Xa InhibitorsKucznierz, Ralf / Grams, Frank / Leinert, Herbert / Marzenell, Klaus / Engh, Richard A. / von der Saal, Wolfgang et al. | 1998
- 4995
-
ARTICLES - Synthesis and Serotonin Receptor Affinities of a Series of trans-2-(Indol-3-yl)cyclopropylamine DerivativesVangveravong, Suwanna et al. | 1998
- 4995
-
Synthesis and Serotonin Receptor Affinities of a Series of trans-2-(Indol-3-yl)cyclopropylamine DerivativesVangveravong, Suwanna / Kanthasamy, Arthi / Lucaites, Virginia L. / Nelson, David L. / Nichols, David E. et al. | 1998
- 5002
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Constrained Corticotropin-Releasing Factor (CRF) Agonists and Antagonists with i−(i+3) Glu-Xaa-dXbb-Lys Bridges †Koerber, Steven C. / Gulyas, Jozsef / Lahrichi, Sabine L. / Corrigan, Anne / Craig, A. Grey / Rivier, Catherine / Vale, Wylie / Rivier, Jean et al. | 1998
- 5002
-
ARTICLES - Constrained Corticotropin-Releasing Factor (CRF) Agonists and Antagonists with i-(i+3) Glu-Xaa-DXbb-Lys BridgesKoerber, Steven C. et al. | 1998
- 5012
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Astressin Analogues (Corticotropin-Releasing Factor Antagonists) with Extended Duration of Action in the Rat ‖Rivier, Jean / Gulyas, Jozsef / Corrigan, Anne / Martinez, Vicente / Craig, A. Grey / Taché, Yvette / Vale, Wylie / Rivier, Catherine et al. | 1998
- 5012
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ARTICLES - Astressin Analogues (Corticotropin-Releasing Factor Antagonists) with Extended Duration of Action in the RatRivier, Jean et al. | 1998
- 5020
-
N-(2-Benzoylphenyl)-l-tyrosine PPARγ Agonists. 1. Discovery of a Novel Series of Potent Antihyperglycemic and Antihyperlipidemic AgentsHenke, Brad R. / Blanchard, Steven G. / Brackeen, Marcus F. / Brown, Kathleen K. / Cobb, Jeff E. / Collins, Jon L. / Harrington,, W. Wallace / Hashim, Mir A. / Hull-Ryde, Emily A. / Kaldor, Istvan et al. | 1998
- 5020
-
ARTICLES - N-(2-Benzoylphenyl)-L-tyrosine PPARg Agonists. 1. Discovery of a Novel Series of Potent Antihyperglycemic and Antihyperlipidemic AgentsHenke, Brad R. et al. | 1998
- 5037
-
N-(2-Benzoylphenyl)-l-tyrosine PPARγ Agonists. 2. Structure−Activity Relationship and Optimization of the Phenyl Alkyl Ether MoietyCollins, Jon L. / Blanchard, Steven G. / Boswell, G. Evan / Charifson, Paul S. / Cobb, Jeff E. / Henke, Brad R. / Hull-Ryde, Emily A. / Kazmierski, Wieslaw M. / Lake, Debra H. / Leesnitzer, Lisa M. et al. | 1998
- 5037
-
ARTICLES - N-(2-Benzoylphenyl)-L-tyrosine PPARg Agonists. 2. Structure-Activity Relationship and Optimization of the Phenyl Alkyl Ether MoietyCollins, Jon L. et al. | 1998
- 5055
-
N-(2-Benzoylphenyl)-l-tyrosine PPARγ Agonists. 3. Structure−Activity Relationship and Optimization of the N-Aryl SubstituentCobb, Jeff E. / Blanchard, Steven G. / Boswell, Evan G. / Brown, Kathleen K. / Charifson, Paul S. / Cooper, Joel P. / Collins, Jon L. / Dezube, Milana / Henke, Brad R. / Hull-Ryde, Emily A. et al. | 1998
- 5055
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ARTICLES - N-(2-Benzoylphenyl)-L-tyrosine PPARg Agonists. 3. Structure-Activity Relationship and Optimization of the N-Aryl SubstituentCobb, Jeff E. et al. | 1998
- 5070
-
Design and Synthesis of a Series of 6-Substituted-2-pyridinylmethylamine Derivatives as Novel, High-Affinity, Selective Agonists at 5-HT1A ReceptorsVacher, Bernard / Bonnaud, Bernard / Funes, Philippe / Jubault, Nathalie / Koek, Wouter / Assié, Marie-Bernadette / Cosi, Cristina et al. | 1998
- 5070
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ARTICLES - Design and Synthesis of a Series of 6-Substituted-2-pyridinylmethylamine Derivatives as Novel, High-Affinity, Selective Agonists at 5-HT1A ReceptorsVacher, Bernard et al. | 1998
- 5084
-
ARTICLES - Spiperone: Influence of Spiro Ring Substituents on 5-HT2A Serotonin Receptor BindingMetwally, Kamel A. et al. | 1998
- 5084
-
Spiperone: Influence of Spiro Ring Substituents on 5-HT2A Serotonin Receptor BindingMetwally, Kamel A. / Dukat, Malgorzata / Egan, Christina T. / Smith, Carol / DuPre, Ann / Gauthier, Colleen B. / Herrick-Davis, Katharine / Teitler, Milt / Glennon, Richard A. et al. | 1998
- 5094
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Nucleosides and Nucleotides. 180. Synthesis and Antitumor Activity of Nucleosides That Have a Hydroxylamino Group Instead of a Hydroxyl Group at the 2‘- or 3‘-Position of the Sugar MoietyOgawa, Akira / Tanaka, Motohiro / Sasaki, Takuma / Matsuda, Akira et al. | 1998
- 5094
-
ARTICLES - Nucleosides and Nucleotides. 180. Synthesis and Antitumor Activity of Nucleosides That Have a Hydroxylamino Group Instead of a Hydroxyl Group at the 2'- or 3'-Position of the Sugar MoietyOgawa, Akira et al. | 1998
- 5108
-
Synthesis of Imidazo[1,2-a]pyridines as Antiviral AgentsGueiffier, Alain / Mavel, Sylvie / Lhassani, Mohammed / Elhakmaoui, Ahmed / Snoeck, Robert / Andrei, Graciela / Chavignon, Olivier / Teulade, Jean-Claude / Witvrouw, Myriam / Balzarini, Jan et al. | 1998
- 5108
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Synthesis of Imidazo[1,2-]pyridines as Antiviral AgentsGueiffier, A. / Mavel, S. / Lhassani, M. / Elhakmaoui, A. / Snoeck, R. / Andrei, G. / Chavignon, O. / Teulade, J.-C. / Witvrouw, M. / Balzarini, J. et al. | 1998
- 5108
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NOTES - Synthesis of Imidazo(1,2-a)pyridines as Antiviral AgentsGueiffier, Alain et al. | 1998
- 5113
-
NOTES - Stereoisomers of Cyclic Urea HIV-1 Protease Inhibitors: Synthesis and Binding AffinitiesKaltenbach III, Robert F. et al. | 1998
- 5113
-
Stereoisomers of Cyclic Urea HIV-1 Protease Inhibitors: Synthesis and Binding AffinitiesKaltenbach, Robert F. / Nugiel, David A. / Lam, Patrick Y. S. / Klabe, Ronald M. / Seitz, Steven P. et al. | 1998
- 5118
-
The Molecular and Supramolecular Chemistry of CarbohydratesLevy, D. E. et al. | 1998
- 5118
-
BOOK REVIEWS - The Molecular and Supramolecular Chemistry of CarbohydratesLevy, Daniel E. et al. | 1998
- 5118
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The Molecular and Supramolecular Chemistry of Carbohydrates By Serge David. Oxford University Press, New York. 1998. vii + 320 pp. 15.5 × 23 cm. ISBN 0-19-850046-7. $45.00.Levy, Daniel E. et al. | 1998