Facile synthesis of benzonitrile/nicotinonitrile based s-triazines as new potential antimycobacterial agents (English)
- New search for: Patel, A. B.
- New search for: Chikhalia, K. H.
- New search for: Kumari, P.
- New search for: Patel, A. B.
- New search for: Chikhalia, K. H.
- New search for: Kumari, P.
In:
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
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79
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57-65
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2014
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ISSN:
- Article (Journal) / Print
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Title:Facile synthesis of benzonitrile/nicotinonitrile based s-triazines as new potential antimycobacterial agents
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Contributors:
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Published in:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY ; 79 ; 57-65
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Publisher:
- New search for: Elsevier Science B.V., Amsterdam.
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Publication date:2014-01-01
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Size:9 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 615.1
- Further information on Dewey Decimal Classification
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Classification:
DDC: 615.1 -
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© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Table of contents – Volume 79
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1
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Novel merosesquiterpene exerts a potent antitumor activity against breast cancer cells in vitro and in vivoCarrasco, E. / Alvarez, P. J. / Melguizo, C. / Prados, J. / Alvarez-Manzaneda, E. / Chahboun, R. / Messouri, I. / Vazquez-Vazquez, M. I. / Aranega, A. / Rodriguez-Serrano, F. et al. | 2014
- 13
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Study of the binding interaction between fluorinated matrix metalloproteinase inhibitors and Human Serum AlbuminDigilio, G. / Tuccinardi, T. / Casalini, F. / Cassino, C. / Dias, D. M. / Geraldes, C. F. G. C. / Catanzaro, V. / Maiocchi, A. / Rossello, A. et al. | 2014
- 24
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Palladacycle (BPC) antitumour activity against resistant and metastatic cell lines: The relationship with cytosolic calcium mobilisation and cathepsin B activityBechara, A. / Barbosa, C. M. V. / Paredes-Gamero, E. J. / Garcia, D. M. / Silva, L. S. / Matsuo, A. L. / Nascimento, F. D. / Rodrigues, E. G. / Caires, A. C. F. / Smaili, S. S. et al. | 2014
- 34
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Synthesis and evaluation of several oleanolic acid glycoconjugates as protein tyrosine phosphatase 1B inhibitorsLiu, Q. / Guo, T. / Li, D. / Li, F. / Li, W. et al. | 2014
- 47
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Synthesis, crystal structures and characterization of late first row transition metal complexes derived from benzothiazole core: Anti-tuberculosis activity and special emphasis on DNA binding and cleavage propertyNetalkar, P. P. / Netalkar, S. P. / Budagumpi, S. / Revankar, V. K. et al. | 2014
- 57
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Facile synthesis of benzonitrile/nicotinonitrile based s-triazines as new potential antimycobacterial agentsPatel, A. B. / Chikhalia, K. H. / Kumari, P. et al. | 2014
- 66
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Synthesis, antiproliferative and anti-dengue virus evaluations of 2-aroyl-3-arylquinoline derivativesTseng, C. H. / Lin, C. K. / Chen, Y. L. / Hsu, C. Y. / Wu, H. N. / Tseng, C. K. / Lee, J. C. et al. | 2014
- 77
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Development of fluorescent double-strand probes labeled with 8-(p-CF"3-cinnamyl)-adenosine for the detection of cyclin D1 breast cancer markerZilbershtein-Shklanovsky, L. / Kafri, P. / Shav-Tal, Y. / Yavin, E. / Fischer, B. et al. | 2014
- 89
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Novel metronidazole-chalcone conjugates with potential to counter drug resistance in Trichomonas vaginalisAnthwal, A. / Rajesh, U. C. / Rawat, M. S. M. / Kushwaha, B. / Maikhuri, J. P. / Sharma, V. L. / Gupta, G. / Rawat, D. S. et al. | 2014
- 95
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Synthesis of 6-cinnamoyl-2H-benzo[b][1,4]oxazin-3(4H)-ones and their effects on A549 lung cancer cell growthZhou, X. W. / Ma, H. L. / Zhang, X. / Jing, S. Y. / Miao, J. Y. / Zhao, B. X. et al. | 2014
- 102
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In-vitro anti-proliferative and anti-oxidant activity of galangin, fisetin and quercetin: Role of localization and intermolecular interaction in model membraneSinha, R. / Srivastava, S. / Joshi, A. / Joshi, U. J. / Govil, G. et al. | 2014
- 110
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Novel R-(+)-limonene-based thiosemicarbazones and their antitumor activity against human tumor cell linesVandresen, F. / Falzirolli, H. / Almeida Batista, S. A. / da Silva-Giardini, A. P. B. / de Oliveira, D. N. / Catharino, R. R. / Ruiz, A. L. T. G. / de Carvalho, J. E. / Foglio, M. A. / da Silva, C. C. et al. | 2014
- 117
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Picolinic acid based Cu(II) complexes with heterocyclic bases - Crystal structure, DNA binding and cleavage studiesPulimamidi, R. R. / Nomula, R. / Pallepogu, R. / Shaik, H. et al. | 2014
- 128
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Pyrazole-5-carboxamides, novel inhibitors of receptor for advanced glycation end products (RAGE)Han, Y. T. / Kim, K. / Choi, G. I. / An, H. / Son, D. / Kim, H. / Ha, H. J. / Son, J. H. / Chung, S. J. / Park, H. J. et al. | 2014
- 143
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Discovery of small molecular (d)-leucinamides as potent, Notch-sparing @c-secretase modulatorsLiao, Y. F. / Tang, Y. C. / Chang, M. Y. / Wang, B. J. / Hu, M. K. et al. | 2014
- 152
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Synthesis, radiolabeling and in vivo evaluation of [^1^1C](R)-1-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT"7 receptorHansen, H. D. / Lacivita, E. / Di Pilato, P. / Herth, M. M. / Lehel, S. / Ettrup, A. / Andersen, V. L. / Dyssegaard, A. / De Giorgio, P. / Perrone, R. et al. | 2014
- 164
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Gold(I) complexes with alkylated PTA (1,3,5-triaza-7-phosphaadamantane) phosphanes as anticancer metallodrugsGarcia-Moreno, E. / Gascon, S. / Atrian-Blasco, E. / Rodriguez-Yoldi, M. J. / Cerrada, E. / Laguna, M. et al. | 2014
- 173
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Optimization of anti-virulence PqsR antagonists regarding aqueous solubility and biological properties resulting in new insights in structure-activity relationshipsLu, C. / Kirsch, B. / Maurer, C. K. / de Jong, J. C. / Braunshausen, A. / Steinbach, A. / Hartmann, R. W. et al. | 2014
- 184
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Imidazole-derived 2-[N-carbamoylmethyl-alkylamino]acetic acids, substrate-dependent modulators of insulin-degrading enzyme in amyloid-@b hydrolysisCharton, J. / Gauriot, M. / Guo, Q. / Hennuyer, N. / Marechal, X. / Dumont, J. / Hamdane, M. / Pottiez, V. / Landry, V. / Sperandio, O. et al. | 2014
- 194
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Synthesis, crystal studies, anti-tuberculosis and cytotoxic studies of 1-[(2E)-3-phenylprop-2-enoyl]-1H-benzimidazole derivativesKalalbandi, V. K. A. / Seetharamappa, J. / Katrahalli, U. / Bhat, K. G. et al. | 2014
- 203
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Synthesis and evaluation of cyclohexane carboxylic acid head group containing isoxazole and thiazole analogs as DGAT1 inhibitorsKandre, S. / Bhagat, P. R. / Kumar Reddy, M. M. / Dalal, R. / Dixit, A. / Deshmukh, N. J. / Anthony, J. / Bose, J. / Anupindi, R. / Sharma, R. et al. | 2014
- 216
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Synthesis and biological evaluation of a novel sigma-1 receptor antagonist based on 3,4-dihydro-2(1H)-quinolinone scaffold as a potential analgesicLan, Y. / Chen, Y. / Xu, X. / Qiu, Y. / Liu, S. / Liu, X. / Liu, B. F. / Zhang, G. et al. | 2014
- 231
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Cell-penetrating peptoids: Introduction of novel cationic side chainsKolmel, D. K. / Horner, A. / Ronicke, F. / Nieger, M. / Schepers, U. / Brase, S. et al. | 2014
- 244
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Synthesis and antiproliferative activity of ligerin and new fumagillin analogs against osteosarcomaBlanchet, E. / Vansteelandt, M. / Le Bot, R. / Egorov, M. / Guitton, Y. / Pouchus, Y. F. / Grovel, O. et al. | 2014
- 251
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Influence of the adamantyl moiety on the activity of biphenylacrylohydroxamic acid-based HDAC inhibitorsCincinelli, R. / Musso, L. / Giannini, G. / Zuco, V. / De Cesare, M. / Zunino, F. / Dallavalle, S. et al. | 2014
- 260
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Synthesis of novel building blocks of benzosuberone bearing coumarin moieties and their evaluation as potential anticancer agentsYadagiri, B. / Holagunda, U. D. / Bantu, R. / Nagarapu, L. / Kumar, C. G. / Pombala, S. / Sridhar, B. et al. | 2014
- 266
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Synthesis of novel spiropyrazoline oxindoles and evaluation of cytotoxicity in cancer cell linesMonteiro, A. / Goncalves, L. M. / Santos, M. M. M. et al. | 2014
- 273
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Targeting triple-negative breast cancer cells with 6,7-bis(hydroxymethyl)-1H,3H-pyrrolo[1,2-c]thiazolesSantos, K. / Laranjo, M. / Abrantes, A. M. / Brito, A. F. / Goncalves, C. / Sarmento Ribeiro, A. B. / Botelho, M. F. / Soares, M. I. L. / Oliveira, A. S. R. / Pinho e Melo, T. M. V. D. et al. | 2014
- 282
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Synthesis and biological activity of 4-aryl-3-benzoyl-5-phenylspiro[pyrrolidine-2.3'-indolin]-2'-one derivatives as novel potent inhibitors of advanced glycation end productKaur, A. / Singh, B. / Vyas, B. / Silakari, O. et al. | 2014
- 290
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Brominated polyunsaturated lipids from the Chinese sponge Xestospongia testudinaria as a new class of pancreatic lipase inhibitorsLiang, L. F. / Wang, T. / Cai, Y. S. / He, W. F. / Sun, P. / Li, Y. F. / Huang, Q. / Taglialatela-Scafati, O. / Wang, H. Y. / Guo, Y. W. et al. | 2014
- 298
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Prospective therapeutic agents for obesity: Molecular modification approaches of centrally and peripherally acting selective cannabinoid 1 receptor antagonistsSharma, M. K. / Murumkar, P. R. / Kanhed, A. M. / Giridhar, R. / Yadav, M. R. et al. | 2014
- 340
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Discovery, synthesis, and structure-activity relationships of 20(S)-protopanaxadiol (PPD) derivatives as a novel class of AMPK@a2@b1@c1 activatorsLiu, J. / Chen, D. / Liu, P. / He, M. / Li, J. / Hu, L. et al. | 2014
- 350
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Design, economical synthesis and antiplasmodial evaluation of vanillin derived allylated chalcones and their marked synergism with artemisinin against chloroquine resistant strains of Plasmodium falciparumSharma, N. / Mohanakrishnan, D. / Sharma, U. K. / Kumar, R. / Richa / Sinha, A. K. / Sahal, D. et al. | 2014
- 369
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Inhibition of tumor cell growth and angiogenesis by 7-Aminoalkoxy-4-aryloxy-quinazoline ureas, a novel series of multi-tyrosine kinase inhibitorsRavez, S. / Barczyk, A. / Six, P. / Cagnon, A. / Garofalo, A. / Goossens, L. / Depreux, P. et al. | 2014
- 382
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Substituted E-3-(3-indolylmethylene)1,3-dihydroindol-2-ones with antiproliferative activity. Study of the effects on HL-60 leukemia cellsLeoni, A. / Locatelli, A. / Morigi, R. / Rambaldi, M. / Cappadone, C. / Farruggia, G. / Iotti, S. / Merolle, L. / Zini, M. / Stefanelli, C. et al. | 2014
- 391
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Synthesis, characterization and anti-proliferative activity of heterocyclic hypervalent organoantimony compoundsChen, Y. / Yu, K. / Tan, N. Y. / Qiu, R. H. / Liu, W. / Luo, N. L. / Tong, L. / Au, C. T. / Luo, Z. Q. / Yin, S. F. et al. | 2014
- 399
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Identification and optimization of novel Hsp90 inhibitors with tetrahydropyrido[4,3-d]pyrimidines core through shape-based screeningSun, H. P. / Jia, J. M. / Jiang, F. / Xu, X. L. / Liu, F. / Guo, X. K. / Cherfaoui, B. / Huang, H. Z. / Pan, Y. / You, Q. D. et al. | 2014
- 413
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4-Oxo-1,4-dihydro-quinoline-3-carboxamides as BACE-1 inhibitors: Synthesis, biological evaluation and docking studiesLiu, P. / Niu, Y. / Wang, C. / Sun, Q. / Zhai, Y. / Yu, J. / Sun, J. / Xu, F. / Yan, G. / Huang, W. et al. | 2014
- 422
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Synthesis and biological evaluation of some novel pyrido[1,2-a]pyrimidin-4-ones as antimalarial agentsMane, U. R. / Mohanakrishnan, D. / Sahal, D. / Murumkar, P. R. / Giridhar, R. / Yadav, M. R. et al. | 2014
- 436
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Synthesis and biological evaluation of novel ^1^2^3I-labeled 4-(4-iodophenyl)butanoyl-l-prolyl-(2S)-pyrrolidines for imaging prolyl oligopeptidase in vivoKallinen, A. / Todorov, B. / Kallionpaa, R. / Back, S. / Sarparanta, M. / Raki, M. / Garcia-Horsman, J. A. / Bergstrom, K. A. / Wallen, E. A. A. / Mannisto, P. T. et al. | 2014
- 446
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Design, synthesis and biological evaluation of some novel substituted quinazolines as antitumor agentsAlanazi, A. M. / Abdel-Aziz, A. A. M. / Al-Suwaidan, I. A. / Abdel-Hamide, S. G. / Shawer, T. Z. / El-Azab, A. S. et al. | 2014