Preparation of the HIV Attachment Inhibitor BMS-663068. Part 6. Friedel—Crafts Acylation/Hydrolysis and Amidation (English)
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- New search for: Silverman, Steven M.
- New search for: Steinhardt, Sarah E.
- New search for: Kolotuchin, Sergei
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- New search for: Fan, Junying
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- New search for: Zheng, Bin
- New search for: Silverman, Steven M.
- New search for: Steinhardt, Sarah E.
- New search for: Kolotuchin, Sergei
- New search for: Iyer, Vidya
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In:
Organic process research & development
;
21
, 8
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1145-1155
;
2017
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ISSN:
- Article (Journal) / Print
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Title:Preparation of the HIV Attachment Inhibitor BMS-663068. Part 6. Friedel—Crafts Acylation/Hydrolysis and Amidation
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Contributors:Zheng, Bin ( author ) / Silverman, Steven M. ( author ) / Steinhardt, Sarah E. ( author ) / Kolotuchin, Sergei ( author ) / Iyer, Vidya ( author ) / Fan, Junying ( author ) / Skliar, Dimitri ( author ) / McLeod, Douglas D. ( author ) / Bultman, Michael ( author ) / Tripp, Jonathan C. ( author )
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Published in:Organic process research & development ; 21, 8 ; 1145-1155
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Publisher:
- New search for: AMERICAN CHEMICAL SOCIETY & ROYAL SOCIETY OF
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Publication date:2017-01-01
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Size:11 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 661.8
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Classification:
DDC: 661.8 -
Source:
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Table of contents – Volume 21, Issue 8
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1091
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BMS-663068: Another Quiet Victory for ChemistryYan, Ming / Baran, Phil S. et al. | 2017
- 1095
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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 1. Evolution of Enabling StrategiesFox, Richard J. / Tripp, Jonathan C. / Schultz, Mitchell J. / Payack, Joseph F. / Fanfair, Dayne D. / Mudryk, Boguslaw M. / Murugesan, Saravanababu / Chen, Chung-Pin H. / La Cruz, Thomas E. / Ivy, Sabrina E. et al. | 2017
- 1110
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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 2. Strategic Selections in the Transition from an Enabling Route to a Commercial SynthesisChen, Ke / Risatti, Christina / Simpson, James / Soumeillant, Maxime / Soltani, Michelle / Bultman, Michael / Zheng, Bin / Mudryk, Boguslaw / Tripp, Jonathan C. / La Cruz, Thomas E. et al. | 2017
- 1122
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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 3. Mechanistic Studies Enable a Scale-Independent Friedel–Crafts AcylationBeutner, Gregory L. / Albrecht, Jacob / Fan, Junying / Fanfair, Dayne / Lawler, Michael J. / Bultman, Michael / Chen, Ke / Ivy, Sabrina / Schild, Richard L. / Tripp, Jonathan C. et al. | 2017
- 1131
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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 4. Synthesis of the 6‑Azaindole CoreBultman, Michael S. / Fan, Junying / Fanfair, Dayne / Soltani, Michelle / Simpson, James / Murugesan, Saravanababu / Soumeillant, Maxime / Chen, Ke / Risatti, Christina / La Cruz, Thomas E. et al. | 2017
- 1137
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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 5. Selective C‑7 Bromination of the 6‑Azaindole CoreGonzález-Bobes, Francisco / Hickey, Matthew R. / Cohen, Benjamin / Bultman, Michael / Chen, Ke / Fanfair, Dayne / Rosso, Victor W. / Strotman, Neil A. / Mudryk, Boguslaw / Murugesan, Saravanababu et al. | 2017
- 1145
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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 6. Friedel–Crafts Acylation/Hydrolysis and AmidationZheng, Bin / Silverman, Steven M. / Steinhardt, Sarah E. / Kolotuchin, Sergei / Iyer, Vidya / Fan, Junying / Skliar, Dimitri / McLeod, Douglas D. / Bultman, Michael / Tripp, Jonathan C. et al. | 2017
- 1156
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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 7. Development of a Regioselective Ullmann–Goldberg–Buchwald ReactionGallagher, William P. / Soumeillant, Maxime / Chen, Ke / Fox, Richard J. / Hsiao, Yi / Mack, Brendan / Iyer, Vidya / Fan, Junying / Zhu, Jason / Beutner, Gregory et al. | 2017
- 1166
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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 8. Installation of the Phosphonoxymethyl Prodrug MoietyFox, Richard J. / Cohen, Benjamin / La Cruz, Thomas E. / Simpson, James H. / Freitag, Adam / Saurer, Eric / Tripp, Jonathan C. / Chen, Chien-Kuang / Beutner, Gregory L. / Rosso, Victor W. et al. | 2017
- 1174
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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 9. Active Pharmaceutical Ingredient Process Development and Powder PropertiesLa Cruz, Thomas E. / Saurer, Eric M. / Engstrom, Joshua / Bultman, Michael S. / Forest, Robert / Akpinar, Fulya / Ferreira, Glenn / Ho, Jeanne W. / Huang, Masano / Soltani, Michelle et al. | 2017