Dopamine D3 Receptor Antagonists. 1. Synthesis and Structure−Activity Relationships of 5,6-Dimethoxy-N-alkyl- and N-Alkylaryl-Substituted 2-Aminoindans (Unknown)
- New search for: Haadsma-Svensson, Susanne R.
- New search for: Cleek, Kerry A.
- New search for: Dinh, Dac M.
- New search for: Duncan, J. Neil
- New search for: Haber, Christopher L.
- New search for: Huff, Rita M.
- New search for: Lajiness, Mary E.
- New search for: Nichols, Nanette F.
- New search for: Smith, Martin W.
- New search for: Svensson, Kjell A.
- New search for: Zaya, Matt J.
- New search for: Carlsson, Arvid
- New search for: Lin, Chiu-Hong
- New search for: Haadsma-Svensson, Susanne R.
- New search for: Cleek, Kerry A.
- New search for: Dinh, Dac M.
- New search for: Duncan, J. Neil
- New search for: Haber, Christopher L.
- New search for: Huff, Rita M.
- New search for: Lajiness, Mary E.
- New search for: Nichols, Nanette F.
- New search for: Smith, Martin W.
- New search for: Svensson, Kjell A.
- New search for: Zaya, Matt J.
- New search for: Carlsson, Arvid
- New search for: Lin, Chiu-Hong
In:
Journal of Medicinal Chemistry
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44
, 26
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4716-4732
;
2001
- Article (Journal) / Electronic Resource
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Title:Dopamine D3 Receptor Antagonists. 1. Synthesis and Structure−Activity Relationships of 5,6-Dimethoxy-N-alkyl- and N-Alkylaryl-Substituted 2-Aminoindans
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Additional title:J. Med. Chem.
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Contributors:Haadsma-Svensson, Susanne R. ( author ) / Cleek, Kerry A. ( author ) / Dinh, Dac M. ( author ) / Duncan, J. Neil ( author ) / Haber, Christopher L. ( author ) / Huff, Rita M. ( author ) / Lajiness, Mary E. ( author ) / Nichols, Nanette F. ( author ) / Smith, Martin W. ( author ) / Svensson, Kjell A. ( author )
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Published in:Journal of Medicinal Chemistry ; 44, 26 ; 4716-4732
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Publisher:
- New search for: American Chemical Society
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Publication date:2001-12-20
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ISSN:
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Coden:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:Unknown
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Source:
Table of contents – Volume 44, Issue 26
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 4497
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Synthesis and Biological Evaluation of Myoseverin Derivatives: Microtubule Assembly InhibitorsChang, Young-Tae / Wignall, Sarah M. / Rosania, Gustavo R. / Gray, Nathanael S. / Hanson, Sarah R. / Su, Andrew I. / Merlie,, John / Moon, Ho-Sang / Sangankar, Sameep B. / Perez, Omar et al. | 2001
- 4501
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Characterization of the 1H-Cyclopentapyrimidine-2,4(1H,3H)-dione Derivative (S)-CPW399 as a Novel, Potent, and Subtype-Selective AMPA Receptor Full Agonist with Partial Desensitization PropertiesCampiani, Giuseppe / Morelli, Elena / Nacci, Vito / Fattorusso, Caterina / Ramunno, Anna / Novellino, Ettore / Greenwood, Jeremy / Liljefors, Tommy / Griffiths, Roger / Sinclair, Colin et al. | 2001
- 4505
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Design, Synthesis and Biological Evaluation of Novel Arachidonic Acid Derivatives as Highly Potent and Selective Endocannabinoid Transporter InhibitorsLópez-Rodríguez, María L. / Viso, Alma / Ortega-Gutiérrez, Silvia / Lastres-Becker, Isabel / González, Sara / Fernández-Ruiz, Javier / Ramos, José A. et al. | 2001
- 4509
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Quadruplex-Interactive Agents as Telomerase Inhibitors: Synthesis of Porphyrins and Structure−Activity Relationship for the Inhibition of TelomeraseShi, Dong-Fang / Wheelhouse, Richard T. / Sun, Daekyu / Hurley, Laurence H. et al. | 2001
- 4524
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Identification of Dipeptidyl Nitriles as Potent and Selective Inhibitors of Cathepsin B through Structure-Based Drug DesignGreenspan, Paul D. / Clark, Kirk L. / Tommasi, Ruben A. / Cowen, Scott D. / McQuire, Leslie W. / Farley, David L. / van Duzer, John H. / Goldberg, Ronald L. / Zhou, Huanghai / Du, Zhengming et al. | 2001
- 4535
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Synthetic 2-Aroylindole Derivatives as a New Class of Potent Tubulin-Inhibitory, Antimitotic Agents ‖Mahboobi, Siavosh / Pongratz, Herwig / Hufsky, Harald / Hockemeyer, Jörg / Frieser, Markus / Lyssenko, Alexei / Paper, Dietrich H. / Bürgermeister, Jutta / Böhmer, Frank-D. / Fiebig, Heinz-Herbert et al. | 2001
- 4554
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Synthesis, Biological Evaluation, and Pharmacophore Generation of Uracil, 4(3H)-Pyrimidinone, and Uridine Derivatives as Potent and Selective Inhibitors of Parainfluenza 1 (Sendai) VirusSaladino, Raffaele / Crestini, Claudia / Palamara, Anna Teresa / Danti, Maria Chiara / Manetti, Fabrizio / Corelli, Federico / Garaci, E. / Botta, Maurizio et al. | 2001
- 4563
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Design, Synthesis, and Biological Characterization of Bivalent 1-Methyl-1,2,5,6-tetrahydropyridyl-1,2,5-thiadiazole Derivatives as Selective Muscarinic AgonistsRajeswaran, W. G. / Cao, Yang / Huang, Xi-Ping / Wroblewski, Mary Elizabeth / Colclough, Tracy / Lee, Selina / Liu, Fenghua / Nagy, Peter I. / Ellis, James / Levine, Beth A. et al. | 2001
- 4577
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Synthesis and Antitumor Activity of Novel C-7 Paclitaxel Ethers: Discovery of BMS-184476Altstadt, Thomas J. / Fairchild, Craig R. / Golik, Jerzy / Johnston, Kathy A. / Kadow, John F. / Lee, Francis Y. / Long, Byron H. / Rose, William C. / Vyas, Dolatrai M. / Wong, Henry et al. | 2001
- 4584
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Structure of Protein Tyrosine Phosphatase 1B in Complex with Inhibitors Bearing Two Phosphotyrosine MimeticsJia, Zongchao / Ye, Qilu / Dinaut, A. Nicole / Wang, Qingping / Waddleton, Deena / Payette, Paul / Ramachandran, Chidambaram / Kennedy, Brian / Hum, Gabriel / Taylor, Scott D. et al. | 2001
- 4595
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Dimerization of G-Protein-Coupled ReceptorsDean, Mark K. / Higgs, Christopher / Smith, Richard E. / Bywater, Robert P. / Snell, Christopher R. / Scott, Paul D. / Upton, Graham J. G. / Howe, Trevor J. / Reynolds, Christopher A. et al. | 2001
- 4615
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Structure-Based Generation of a New Class of Potent Cdk4 Inhibitors: New de Novo Design Strategy and Library DesignHonma, Teruki / Hayashi, Kyoko / Aoyama, Tetsuya / Hashimoto, Noriaki / Machida, Takumitsu / Fukasawa, Kazuhiro / Iwama, Toshiharu / Ikeura, Chinatsu / Ikuta, Mari / Suzuki-Takahashi, Ikuko et al. | 2001
- 4628
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A Novel Approach for the Development of Selective Cdk4 Inhibitors: Library Design Based on Locations of Cdk4 Specific Amino Acid ResiduesHonma, Teruki / Yoshizumi, Takashi / Hashimoto, Noriaki / Hayashi, Kyoko / Kawanishi, Nobuhiko / Fukasawa, Kazuhiro / Takaki, Tohru / Ikeura, Chinatsu / Ikuta, Mari / Suzuki-Takahashi, Ikuko et al. | 2001
- 4641
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Oxindole Derivatives as Orally Active Potent Growth Hormone SecretagoguesTokunaga, Teruhisa / Hume, W. Ewan / Umezome, Takashi / Okazaki, Kazuhiko / Ueki, Yasuyuki / Kumagai, Kazuo / Hourai, Shinji / Nagamine, Jun / Seki, Hitoshi / Taiji, Mutsuo et al. | 2001
- 4650
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Structural Basis for the Binding Affinity of Xanthines with the DNA Intercalator Acridine OrangeLyles, Mark B. / Cameron, Ivan L. / Rawls, H. Ralph et al. | 2001
- 4661
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Mononuclear Platinum(II) Complex with 2-Phenylpyridine Ligands Showing High Cytotoxicity against Mouse Sarcoma 180 Cells Acquiring High Cisplatin ResistanceOkada, Tomoko / El-Mehasseb, Ibrahim M. / Kodaka, Masato / Tomohiro, Takenori / Okamoto, Ken-ichi / Okuno, Hiroaki et al. | 2001
- 4668
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Chemosensitization of a Multidrug-Resistant Leishmania tropica Line by New Sesquiterpenes from Maytenus magellanica and Maytenus chubutensisKennedy, María L. / Cortés-Selva, Fernando / Pérez-Victoria, José M. / Jiménez, Ignacio A. / González, Antonio G. / Muñoz, Orlando M. / Gamarro, Francisco / Castanys, Santiago / Ravelo, Angel G. et al. | 2001
- 4677
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Diaminoindanes as Microsomal Triglyceride Transfer Protein InhibitorsKsander, Gary M. / deJesus, Reynalda / Yuan, Andrew / Fink, Cynthia / Moskal, Michael / Carlson, Eric / Kukkola, Paivi / Bilci, Natalie / Wallace, Eli / Neubert, Alan et al. | 2001
- 4688
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C-16 Artemisinin Derivatives and Their Antimalarial and Cytotoxic Activities: Syntheses of Artemisinin Monomers, Dimers, Trimers, and Tetramers by Nucleophilic Additions to ArtemisiteneEkthawatchai, Sanchai / Kamchonwongpaisan, Sumalee / Kongsaeree, Palangpon / Tarnchompoo, Bongkoch / Thebtaranonth, Yodhathai / Yuthavong, Yongyuth et al. | 2001
- 4696
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Design, Synthesis, and Pharmacological Evaluation of Thapsigargin Analogues for Targeting Apoptosis to Prostatic Cancer CellsJakobsen, Carsten M. / Denmeade, Samuel R. / Isaacs, John T. / Gady, Alyssa / Olsen, Carl E. / Christensen, Søren Brøgger et al. | 2001
- 4704
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2-(2-Piperidyl)- and 2-(2-Pyrrolidyl)chromans as Nicotine Agonists: Synthesis and Preliminary Pharmacological CharacterizationEfange, Simon M. N. / Tu, Zhude / von Hohenberg, Krystyna / Francesconi, Lynn / Howell, Robertha C. / Rampersad, Marilyn V. / Todaro, Louis J. / Papke, Roger L. / Kung, Mei-Ping et al. | 2001
- 4716
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Dopamine D3 Receptor Antagonists. 1. Synthesis and Structure−Activity Relationships of 5,6-Dimethoxy-N-alkyl- and N-Alkylaryl-Substituted 2-AminoindansHaadsma-Svensson, Susanne R. / Cleek, Kerry A. / Dinh, Dac M. / Duncan, J. Neil / Haber, Christopher L. / Huff, Rita M. / Lajiness, Mary E. / Nichols, Nanette F. / Smith, Martin W. / Svensson, Kjell A. et al. | 2001
- 4733
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Synthesis, in Vitro Pharmacology, and Molecular Modeling of syn-Huprines as Acetylcholinesterase InhibitorsCamps, Pelayo / Gómez, Elena / Muñoz-Torrero, Diego / Badia, Albert / Vivas, Nuria María / Barril, Xavier / Orozco, Modesto / Luque, Francisco Javier et al. | 2001
- 4737
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Design and Synthesis of Non-peptidic Inhibitors for the Syk C-Terminal SH2 Domain Based on Structure-Based In-Silico ScreeningNiimi, Tatsuya / Orita, Masaya / Okazawa-Igarashi, Miwa / Sakashita, Hitoshi / Kikuchi, Kazumi / Ball, Evelyn / Ichikawa, Atsushi / Yamagiwa, Yoko / Sakamoto, Shuichi / Tanaka, Akihiro et al. | 2001
- 4741
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Principles and Applications of Asymmetric Synthesis By Guo-Qiang Lin, Yue-Ming Li, and Albert S. C. Chan. Wiley Interscience, New York. 2001. xvii + 515 pp. 16 x 24 cm. ISBN 0-471-40027-0. 89.95.Aube, J. et al. | 2001
- 4741
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Synthesis and Applications of Isotopically Labelled Compounds. Volume 7. Proceedings of the Seventh International Symposium, Dresden, Germany, June 18−22, 2000 Edited by U. Pleiss and R. Voges. Wiley, New York. 2001. xxv + 702 pp. 17 × 25 cm. ISBN 0-471-49501-8. $220.00.Filer, Crist N. et al. | 2001
- 4741
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Synthesis and Applications of Isotopically Labelled Compounds. Volume 7. Proceedings of the Seventh International Symposium, Dresden, Germany, June 18-22, 2000 Edited by U. Pleiss and R. Voges. Wiley, New York. 2001. xxv + 702 pp. 17 x 25 cm. ISBN 0-471-49501-8. 220.00.Filer, C.N. et al. | 2001
- 4741
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Principles and Applications of Asymmetric Synthesis By Guo-Qiang Lin, Yue-Ming Li, and Albert S. C. Chan. Wiley Interscience, New York. 2001. xvii + 515 pp. 16 × 24 cm. ISBN 0-471-40027-0. $89.95.Aubé, Jeffrey et al. | 2001