Correction to “Discovery and Structure-Based Optimization of Novel Atg4B Inhibitors for the Treatment of Castration-Resistant Prostate Cancer” (English)
- New search for: Kudo, Yudai
- New search for: Endo, Satoshi
- Further information on Endo, Satoshi:
- https://orcid.org/0000-0003-0578-9672
- New search for: Fujita, Mei
- New search for: Ota, Atsumi
- New search for: Kamatari, Yuji O.
- New search for: Tanaka, Yoshimasa
- New search for: Ishikawa, Takeshi
- Further information on Ishikawa, Takeshi:
- https://orcid.org/0000-0002-3187-1381
- New search for: Ikeda, Hayato
- New search for: Okada, Takuya
- New search for: Toyooka, Naoki
- Further information on Toyooka, Naoki:
- https://orcid.org/0000-0002-9568-1528
- New search for: Fujimoto, Naohiro
- New search for: Matsunaga, Toshiyuki
- New search for: Ikari, Akira
- New search for: Kudo, Yudai
- New search for: Endo, Satoshi
- Further information on Endo, Satoshi:
- https://orcid.org/0000-0003-0578-9672
- New search for: Fujita, Mei
- New search for: Ota, Atsumi
- New search for: Kamatari, Yuji O.
- New search for: Tanaka, Yoshimasa
- New search for: Ishikawa, Takeshi
- Further information on Ishikawa, Takeshi:
- https://orcid.org/0000-0002-3187-1381
- New search for: Ikeda, Hayato
- New search for: Okada, Takuya
- New search for: Toyooka, Naoki
- Further information on Toyooka, Naoki:
- https://orcid.org/0000-0002-9568-1528
- New search for: Fujimoto, Naohiro
- New search for: Matsunaga, Toshiyuki
- New search for: Ikari, Akira
In:
Journal of Medicinal Chemistry
;
65
, 11
;
8062-8063
;
2022
- Article (Journal) / Electronic Resource
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Title:Correction to “Discovery and Structure-Based Optimization of Novel Atg4B Inhibitors for the Treatment of Castration-Resistant Prostate Cancer”
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Additional title:J. Med. Chem.
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Contributors:Kudo, Yudai ( author ) / Endo, Satoshi ( author ) / Fujita, Mei ( author ) / Ota, Atsumi ( author ) / Kamatari, Yuji O. ( author ) / Tanaka, Yoshimasa ( author ) / Ishikawa, Takeshi ( author ) / Ikeda, Hayato ( author ) / Okada, Takuya ( author ) / Toyooka, Naoki ( author )
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Published in:Journal of Medicinal Chemistry ; 65, 11 ; 8062-8063
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Publisher:
- New search for: American Chemical Society
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Publication date:2022-06-09
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ISSN:
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Coden:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Source:
Table of contents – Volume 65, Issue 11
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 7415
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Medicinal Chemistry Strategies for the Development of Bruton’s Tyrosine Kinase Inhibitors against ResistanceSun, Shan-Liang / Wu, Shi-Han / Kang, Ji-Bo / Ma, Yi-Yuan / Chen, Lu / Cao, Peng / Chang, Liang / Ding, Ning / Xue, Xin / Li, Nian-Guang et al. | 2022
- 7438
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Peptidomimetics: An Overview of Recent Medicinal Chemistry Efforts toward the Discovery of Novel Small Molecule InhibitorsLi Petri, Giovanna / Di Martino, Simona / De Rosa, Maria et al. | 2022
- 7476
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Electrostatic Complementarity in Structure-Based Drug DesignCons, Benjamin D. / Twigg, David G. / Kumar, Rajendra / Chessari, Gianni et al. | 2022
- 7489
-
Tuberculosis Drug Discovery: Challenges and New HorizonsFernandes, Guilherme F. S. / Thompson, Andrew M. / Castagnolo, Daniele / Denny, William A. / Dos Santos, Jean L. et al. | 2022
- 7532
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Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small MoleculesNizi, Maria Giulia / Maksimainen, Mirko M. / Lehtiö, Lari / Tabarrini, Oriana et al. | 2022
- 7561
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Progress and Challenges in Targeting the SARS-CoV‑2 Papain-like ProteaseTan, Haozhou / Hu, Yanmei / Jadhav, Prakash / Tan, Bin / Wang, Jun et al. | 2022
- 7581
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The Dawn of Allosteric BCR-ABL1 Drugs: From a Phenotypic Screening Hit to an Approved DrugTeng, Mingxing / Luskin, Marlise R. / Cowan-Jacob, Sandra W. / Ding, Qiang / Fabbro, Doriano / Gray, Nathanael S. et al. | 2022
- 7595
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Discovery of 1,6-Naphthyridin-2(1H)‑one Derivatives as Novel, Potent, and Selective FGFR4 Inhibitors for the Treatment of Hepatocellular CarcinomaZhang, Xiaomeng / Wang, Yazhou / Ji, Jianfeng / Si, Dongjuan / Bao, Xueting / Yu, Zhuangzhuang / Zhu, Yueyue / Zhao, Liwen / Li, Wei / Liu, Jian et al. | 2022
- 7619
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Ispinesib as an Effective Warhead for the Design of Autophagosome-Tethering Chimeras: Discovery of Potent Degraders of Nicotinamide Phosphoribosyltransferase (NAMPT)Dong, Guoqiang / Wu, Ying / Cheng, Junfei / Chen, Long / Liu, Rui / Ding, Yu / Wu, Shanchao / Ma, Junhui / Sheng, Chunquan et al. | 2022
- 7629
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Discovery of a Novel Series of Imipridone Compounds as Homo sapiens Caseinolytic Protease P Agonists with Potent Antitumor Activities In Vitro and In VivoHuang, Jiasheng / Zhang, Jiangnan / Luo, Baozhu / Qiao, Wenliang / Qiu, Zhiqiang / Song, Rao / Dai, Zhengyi / Sui, Jing / Xu, Xin / Ruan, Shihua et al. | 2022
- 7656
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Discovery of In Vivo Active Sphingosine-1-phosphate Transporter (Spns2) InhibitorsFritzemeier, Russell / Foster, Daniel / Peralta, Ashley / Payette, Michael / Kharel, Yugesh / Huang, Tao / Lynch, Kevin R. / Santos, Webster L. et al. | 2022
- 7682
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Penicillin Derivatives Inhibit the SARS-CoV‑2 Main Protease by Reaction with Its Nucleophilic CysteineMalla, Tika R. / Brewitz, Lennart / Muntean, Dorian-Gabriel / Aslam, Hiba / Owen, C. David / Salah, Eidarus / Tumber, Anthony / Lukacik, Petra / Strain-Damerell, Claire / Mikolajek, Halina et al. | 2022
- 7697
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Novel Sphingosine Kinase 1 Inhibitor Suppresses Growth of Solid Tumor and Inhibits the Lung Metastasis of Triple-Negative Breast CancerZhang, Shurui / Chen, Xiaoxu / Wu, Chenglin / Xu, Hui / Xie, Xiong / Feng, Mingshun / Hu, Shulei / Bai, Hudagula / Gao, Feng / Tong, Linjiang et al. | 2022
- 7717
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Long Residence Time at the Vasopressin V2 Receptor Translates into Superior Inhibitory Effects in Ex Vivo and In Vivo Models of Autosomal Dominant Polycystic Kidney DiseaseZhang, Haoran / Yan, Wenzhong / Sun, Yongzhan / Yuan, Haoxing / Su, Limin / Cao, Xudong / Wang, Peng / Xu, Zhou / Hu, Youhui / Wang, Zhongjian et al. | 2022
- 7729
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Structure–Activity Relationships of 8‑Hydroxyquinoline-Derived Mannich Bases with Tertiary Amines Targeting Multidrug-Resistant CancerPape, Veronika F. S. / Palkó, Roberta / Tóth, Szilárd / Szabó, Miklós J. / Sessler, Judit / Dormán, György / Enyedy, Éva A. / Soós, Tibor / Szatmári, István / Szakács, Gergely et al. | 2022
- 7746
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Discovery of Small Molecules Simultaneously Targeting NAD(P)H:Quinone Oxidoreductase 1 and Nicotinamide Phosphoribosyltransferase: Treatment of Drug-Resistant Non-small-Cell Lung CancerZhang, Kuojun / Wang, Kaizhen / Zhang, Xiangyu / Qian, Zhenlong / Zhang, Wenbo / Zheng, Xiao / Wang, Jiaying / Jiang, Yin / Zhang, Wanheng / Lu, Zhiyu et al. | 2022
- 7770
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Design, Synthesis, and Biological Evaluations of DOT1L Peptide Mimetics Targeting the Protein–Protein Interactions between DOT1L and MLL-AF9/MLL-ENLYuan, Yinan / Du, Lei / Tan, Rongliang / Yu, Yifan / Jiang, Jinxin / Yao, Aihong / Luo, Jiajun / Tang, Rui / Xiao, Yibei / Sun, Haiying et al. | 2022
- 7786
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Platinum-Based Two-Photon Photosensitizer Responsive to NIR Light in Tumor Hypoxia MicroenvironmentWang, Yanjun / Shi, Xiangchao / Fang, Hongbao / Han, Zhong / Yuan, Hao / Zhu, Zhenzhu / Dong, Lei / Guo, Zijian / Wang, Xiaoyong et al. | 2022
- 7799
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Illuminating the Dark: Highly Selective Inhibition of Serine/Threonine Kinase 17A with Pyrazolo[1,5‑a]pyrimidine-Based MacrocyclesKurz, Christian G. / Preuss, Franziska / Tjaden, Amelie / Cusack, Martin / Amrhein, Jennifer Alisa / Chatterjee, Deep / Mathea, Sebastian / Berger, Lena Marie / Berger, Benedict-Tilman / Krämer, Andreas et al. | 2022
- 7818
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Structure-Guided Design of Potent Spirocyclic Inhibitors of Severe Acute Respiratory Syndrome Coronavirus‑2 3C-like ProteaseDampalla, Chamandi S. / Rathnayake, Athri D. / Galasiti Kankanamalage, Anushka C. / Kim, Yunjeong / Perera, Krishani Dinali / Nguyen, Harry Nhat / Miller, Matthew J. / Madden, Trent K. / Picard, Hunter R. / Thurman, Hayden A. et al. | 2022
- 7833
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Discovery of 8‑(6-Methoxypyridin-3-yl)-1-(4-(piperazin-1-yl)-3-(trifluoromethyl)phenyl)-1,5-dihydro-4H-[1,2,3]triazolo[4,5‑c]quinolin-4-one (CQ211) as a Highly Potent and Selective RIOK2 InhibitorOuyang, Yifan / Si, Hongfei / Zhu, Chengjun / Zhong, Liang / Ma, Haowen / Li, Zongyang / Xiong, Huilan / Liu, Tongzheng / Liu, Zhong / Zhang, Zhang et al. | 2022
- 7843
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Structural Basis for Binding of Potassium-Competitive Acid Blockers to the Gastric Proton PumpTanaka, Saki / Morita, Mikio / Yamagishi, Tatsuya / Madapally, Hridya Valia / Hayashida, Kenichi / Khandelia, Himanshu / Gerle, Christoph / Shigematsu, Hideki / Oshima, Atsunori / Abe, Kazuhiro et al. | 2022
- 7854
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Structure-Aided Design, Synthesis, and Biological Evaluation of Potent and Selective Non-Nucleoside Inhibitors Targeting Protein Arginine Methyltransferase 5Rong, Deqin / Zhou, Kaixin / Fang, Wei / Yang, Hong / Zhang, Yi / Shi, Qiongyu / Huang, Yuting / Li, Jiayi / Dong, Hui / Li, Lanlan et al. | 2022
- 7876
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Multiparameter Optimization of Naphthyridine Derivatives as Selective α5-GABAA Receptor Negative Allosteric ModulatorsSzabó, György / Éliás, Olivér / Erdélyi, Péter / Potor, Attila / Túrós, György I. / Károlyi, Benedek I. / Varró, Gábor / Vaskó, Ágnes Gy. / Bata, Imre / Kapus, Gábor L. et al. | 2022
- 7896
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Scaffold Hopping Strategy to Identify Prostanoid EP4 Receptor Antagonists for Cancer ImmunotherapyWang, Wei / He, Jiacheng / Yang, Junjie / Zhang, Chan / Cheng, Zhiyuan / Zhang, Yao / Zhang, Qiansen / Wang, Peili / Tang, Shuowen / Wang, Xin et al. | 2022
- 7918
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TocoDecoy: A New Approach to Design Unbiased Datasets for Training and Benchmarking Machine-Learning Scoring FunctionsZhang, Xujun / Shen, Chao / Liao, Ben / Jiang, Dejun / Wang, Jike / Wu, Zhenxing / Du, Hongyan / Wang, Tianyue / Huo, Wenbo / Xu, Lei et al. | 2022
- 7933
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Platinum(IV) Prodrugs with Cancer Stem Cell Inhibitory Effects on Lung Cancer for Overcoming Drug ResistanceWang, Xinyi / Liu, Zhikun / Wang, Yuanjiang / Gou, Shaohua et al. | 2022
- 7946
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On the Frustration to Predict Binding Affinities from Protein–Ligand Structures with Deep Neural NetworksVolkov, Mikhail / Turk, Joseph-André / Drizard, Nicolas / Martin, Nicolas / Hoffmann, Brice / Gaston-Mathé, Yann / Rognan, Didier et al. | 2022
- 7959
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Discovery and Characterization of the First Nonpeptide Antagonists for the Relaxin-3/RXFP3 SystemGay, Elaine A. / Guan, Dongliang / Van Voorhies, Kalynn / Vasukuttan, Vineetha / Mathews, Kelly M. / Besheer, Joyce / Jin, Chunyang et al. | 2022
- 7975
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Design, Synthesis, and Biological Evaluation of Novel Evodiamine Derivatives as Potential Antihepatocellular Carcinoma AgentsLei, Fang / Xiong, Yongxia / Wang, Yuqing / Zhang, Honghua / Liang, Ziyi / Li, Junfang / Feng, Yiyue / Hao, Xiangyong / Wang, Zhen et al. | 2022
- 7993
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Discovery of Novel Bicyclic Phenylselenyl-Containing Hybrids: An Orally Bioavailable, Potential, and Multiacting Class of Estrogen Receptor Modulators against Endocrine-Resistant Breast CancerDeng, Xiangping / Xie, Baohua / Li, Qiuzi / Xiao, Yuan / Hu, Zhiye / Deng, Xiaofei / Fang, Pingping / Dong, Chune / Zhou, Hai-Bing / Huang, Jian et al. | 2022
- 8011
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Design and Optimization of Thienopyrimidine Derivatives as Potent and Selective PI3Kδ Inhibitors for the Treatment of B‑Cell MalignanciesZhang, Jingbo / Jiang, Huimin / Lin, Songwen / Wu, Deyu / Tian, Hua / Jiang, Lin / Cui, Yiman / Jin, Jing / Chen, Xiaoguang / Xu, Heng et al. | 2022
- 8029
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Development of Lipo-γ-AA Peptides as Potent Antifungal AgentsZhang, Xing / Wang, Minghui / Zhu, Xiaodi / Peng, Yan / Fu, Tiwei / Hu, Chang-Hua / Cai, Jianfeng / Liao, Guojian et al. | 2022
- 8040
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Optimization of the Natural Product Calothrixin A to Discover Novel Dual Topoisomerase I and II Inhibitors with Improved Anticancer ActivityYang, Xiaohong / Wang, Zhi-Peng / Xiang, Sichuan / Wang, Daoqiang / Zhao, Yi / Luo, Dong / Qiu, Yanfei / Huang, Chao / Guo, Jian / Dai, Yuanwei et al. | 2022
- 8062
-
Correction to “Discovery and Structure-Based Optimization of Novel Atg4B Inhibitors for the Treatment of Castration-Resistant Prostate Cancer”Kudo, Yudai / Endo, Satoshi / Fujita, Mei / Ota, Atsumi / Kamatari, Yuji O. / Tanaka, Yoshimasa / Ishikawa, Takeshi / Ikeda, Hayato / Okada, Takuya / Toyooka, Naoki et al. | 2022