Enzymic synthesis and comparative biological evaluation of a phosphonate analog of the lipid A precursor (English)
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- New search for: Scholz, Dieter
- New search for: Bednarik, Karl
- New search for: Ehn, Gerald
- New search for: Neruda, Wolfgang
- New search for: Janzek, Evelyne
- New search for: Loibner, Hans
- New search for: Briner, Karin
- New search for: Vasella, Andrea
- New search for: Scholz, Dieter
- New search for: Bednarik, Karl
- New search for: Ehn, Gerald
- New search for: Neruda, Wolfgang
- New search for: Janzek, Evelyne
- New search for: Loibner, Hans
- New search for: Briner, Karin
- New search for: Vasella, Andrea
In:
Journal of Medicinal Chemistry
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35
, 11
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2070-2074
;
1992
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ISSN:
- Article (Journal) / Electronic Resource
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Title:Enzymic synthesis and comparative biological evaluation of a phosphonate analog of the lipid A precursor
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Additional title:J. Med. Chem.
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Contributors:Scholz, Dieter ( author ) / Bednarik, Karl ( author ) / Ehn, Gerald ( author ) / Neruda, Wolfgang ( author ) / Janzek, Evelyne ( author ) / Loibner, Hans ( author ) / Briner, Karin ( author ) / Vasella, Andrea ( author )
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Published in:Journal of Medicinal Chemistry ; 35, 11 ; 2070-2074
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Publisher:
- New search for: American Chemical Society
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Publication date:1992-05-01
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ISSN:
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Coden:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Source:
Table of contents – Volume 35, Issue 11
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1927
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The role of concepts in structure-activity relationship studies of opioid ligandsPortoghese, Philip S. et al. | 1992
- 1938
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New thymidine triphosphate analog inhibitors of human immunodeficiency virus-1 reverse transcriptase.Ma, Qi Feng / Bathurst, Ian C. / Barr, Philip J. / Kenyon, George L. et al. | 1992
- 1942
-
2-Carboxytetrahydroquinolines. Conformational and stereochemical requirements for antagonism of the glycine site on the N-methyl-D-aspartate (NMDA) receptorCarling, Robert W. / Leeson, Paul D. / Moseley, Angela M. / Baker, Raymond / Foster, Alan C. / Grimwood, Sarah / Kemp, John A. / Marshall, George R. et al. | 1992
- 1954
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4-Amido-2-carboxytetrahydroquinolines. Structure-activity relationships for antagonism at the glycine site of the NMDA receptorLeeson, Paul D. / Carling, Robert W. / Moore, Kevin W. / Moseley, Angela M. / Smith, Julian D. / Stevenson, Graeme / Chan, Tony / Baker, Raymond / Foster, Alan C. / Grimwood, Sarah et al. | 1992
- 1969
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Structure and molecular modeling of GABAA receptor antagonistsRognan, Didier / Boulanger, Thierry / Hoffmann, Remy / Vercauteren, Daniel P. / Andre, Jean Marie / Durant, Francois / Wermuth, Camille Georges et al. | 1992
- 1978
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A nonpromoting phorbol from the Samoan medicinal plant Homalanthus nutans inhibits cell killing by HIV-1Gustafson, Kirk R. / Cardellina, John H. / McMahon, James B. / Gulakowski, Robert J. / Ishitoya, Junichi / Szallasi, Zoltan / Lewin, Nancy E. / Blumberg, Peter M. / Weislow, Owen S. et al. | 1992
- 1987
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Asymmetric synthesis of 1,3-dioxolane-pyrimidine nucleosides and their anti-HIV activity.Kim, Hea O. / Ahn, Soon K. / Alves, Antonio J. / Beach, J. Warren / Jeong, Lak S. / Choi, Bo G. / Van Roey, Patrick / Schinazi, Raymond F. / Chu, Chung K. et al. | 1992
- 1996
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Highly water-soluble lipophilic prodrugs of the anti-HIV nucleoside analog 2',3'-dideoxycytidine and its 3'-fluoro derivativeKerr, Stephen G. / Kalman, Thomas I. et al. | 1992
- 2002
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Synthesis and biological evaluation of N.alpha.-(5-deaza-5,6,7,8-tetrahydropteroyl)-L-ornithineSingh, Shyam K. / Singer, Sara C. / Ferone, Robert / Waters, Kathleen A. / Mullin, Robert J. / Hynes, John B. et al. | 1992
- 2007
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Development of potent and selective CCK-A receptor agonists from Boc-CCK-4: tetrapeptides containing Lys(N.epsilon.)-amide residuesShiosaki, Kazumi / Lin, Chun Wel / Kopecka, Hana / Craig, Richard A. / Bianchi, Bruce R. / Miller, Thomas R. / Witte, David G. / Stashko, Michael / Nadzan, Alex M. et al. | 1992
- 2015
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Studies on neurokinin antagonists. 1. The design of novel tripeptides possessing glutaminyl-D-tryptophylphenylalanine sequence as substance P antagonistsHagiwara, Daijiro / Miyake, Hiroshi / Morimoto, Hiroshi / Murai, Masako / Fujii, Takashi / Matsuo, Masaaki et al. | 1992
- 2025
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Benz[f]isoquinoline analogs as high-affinity .sigma. ligandsRussell, Michael G. N. / Baker, Raymond / Billington, David C. / Knight, Antony K. / Middlemiss, Derek N. / Noble, Alison J. et al. | 1992
- 2033
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Spiropiperidines as high-affinity, selective .sigma. ligands.Chambers, Mark S. / Baker, Raymond / Billington, David C. / Knight, Anthony K. / Middlemiss, D. N. / Wong, Eric H. F. et al. | 1992
- 2040
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Cyclic RGD peptide analogs as antiplatelet antithromboticsBarker, Peter L. / Bullens, Sherron / Bunting, Stuart / Burdick, Daniel J. / Chan, Kathryn S. / Deisher, Tracy / Eigenbrot, Charles / Gadek, Thomas R. / Gantzos, Robin et al. | 1992
- 2048
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Ester and amide derivatives of E64c as inhibitors of platelet calpainsHuang, Zhenya / McGowan, Eleanor B. / Detwiler, Thomas C. et al. | 1992
- 2055
-
Synthesis and structure-activity relationships of a series of novel benzopyran-containing platelet activating factor antagonistsGuinn, Denise E. / Summers, James B. / Heyman, H. Robin / Conway, Richard G. / Rhein, David A. / Albert, Daniel H. / Magoc, Terry / Carter, George W. et al. | 1992
- 2061
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Benzofuran bioisosteres of hallucinogenic tryptaminesTomaszewski, Zbigniew / Johnson, Michael P. / Huang, Xuemei / Nichols, David E. et al. | 1992
- 2065
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A novel probe for the cannabinoid receptorDevane, William A. / Breuer, Aviva / Sheskin, Tzviel / Jaerbe, Torbjoern U. C. / Eisen, Moris S. / Mechoulam, Raphael et al. | 1992
- 2070
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Enzymic synthesis and comparative biological evaluation of a phosphonate analog of the lipid A precursorScholz, Dieter / Bednarik, Karl / Ehn, Gerald / Neruda, Wolfgang / Janzek, Evelyne / Loibner, Hans / Briner, Karin / Vasella, Andrea et al. | 1992
- 2074
-
Synthesis and antiallergic activity of 11-(aminoalkylidene)-6,11-dihydrodibenz[b,e]oxepin derivativesOhshima, Etsuo / Otaki, Shizuo / Sato, Hideyuki / Kumazawa, Toshiaki / Obase, Hiroyuki / Ishii, Akio / Ishii, Hidee / Ohmori, Kenji / Hirayama, Noriaki et al. | 1992
- 2085
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Biological activities and quantitative structure-activity relationships of spiro[imidazolidine-4,4'(1'H)-quinazoline]-2,2',5(3'H)-triones as aldose reductase inhibitorsYamagishi, Masafumi / Yamada, Yoshihisa / Ozaki, Kenichi / Asao, Masaaki / Shimizu, Ryo / Suzuki, Mamoru / Matsumoto, Mamoru / Matsuoka, Yuzo / Matsumoto, Kazuo et al. | 1992
- 2095
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Inhibitors of cholesterol biosynthesis. 6. trans-6-[2-(2-N-heteroaryl-3,5-disubstituted-pyrazol-4-yl)ethyl/ethenyl]tetrahydro-4-hydroxy-2H-pyran-2-onesSliskovic, D. R. / Blankley, C. J. / Krause, B. R. / Newton, R. S. / Picard, J. A. / Roark, W. H. / Roth, B. D. / Sekerke, C. / Shaw, M. K. / Stanfield, R. L. et al. | 1992
- 2103
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Renin inhibitors containing C-termini derived from mercaptoheterocyclesAshton, Wallace T. / Cantone, Christine L. / Meurer, Laura C. / Tolman, Richard L. / Greenlee, William J. / Patchett, Arthur A. / Lynch, Robert J. / Schorn, Terry W. / Strouse, John F. / Siegl, Peter K. S. et al. | 1992
- 2113
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Synthesis of high-affinity fluorine-substituted ligands for the androgen receptor. Potential agents for imaging prostatic cancer by positron emission tomographyLiu, Aijun / Carlson, Kathryn E. / Katzenellenbogen, John A. et al. | 1992
- 2129
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Bisquinolines. 1. N,N-bis(7-chloroquinolin-4-yl)alkanediamines with potential against chloroquine-resistant malariaVennerstrom, Jonathan L. / Ellis, William Y. / Ager, Arba L. / Andersen, Steven L. / Gerena, Lucia / Milhous, Wilbur K. et al. | 1992
- 2134
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Clinical analysis by proton spin-echo NMR. 2. Oxidation of intracellular glutathione as a consequence of penicillamine therapy in rheumatoid arthritisReglinski, J. / Smith, W. E. / Brzeski, M. / Marabani, M. / Sturrock, R. D. et al. | 1992
- 2137
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p-(Methylsulfinyl)phenyl nitrogen mustard as a novel bioreductive prodrug selective against hypoxic tumorsKwon, Chul Hoon / Blanco, Daria R. / Baturay, Nesrine et al. | 1992
- 2139
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Cyclic pentapeptide endothelin antagonists with high ETA selectivity. Potency- and solubility-enhancing modificationsIshikawa, Kiyofumi / Fukami, Takehiro / Nagase, Toshio / Fujita, Kagari / Hayama, Takashi / Niiyama, Kenji / Mase, Toshiaki / Ihara, Masaki / Yano, Mitsuo et al. | 1992
- 2142
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Book Reviews| 1992
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Masthead| 1992