3′-N-Alkylamino-3′-deoxy-ara-uridines: A new class of potential inhibitors of ribonuclease A and angiogenin (English)
- New search for: Maiti, Tushar K.
- New search for: Soumya De
- New search for: Dasgupta, Swagata
- New search for: Pathak, Tanmaya
- New search for: Maiti, Tushar K.
- New search for: Soumya De
- New search for: Dasgupta, Swagata
- New search for: Pathak, Tanmaya
In:
Bioorganic and Medicinal Chemistry
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14
, 4
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1221-1228
;
2005
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ISSN:
- Article (Journal) / Electronic Resource
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Title:3′-N-Alkylamino-3′-deoxy-ara-uridines: A new class of potential inhibitors of ribonuclease A and angiogenin
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Contributors:Maiti, Tushar K. ( author ) / Soumya De ( author ) / Dasgupta, Swagata ( author ) / Pathak, Tanmaya ( author )
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Published in:Bioorganic and Medicinal Chemistry ; 14, 4 ; 1221-1228
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Publisher:
- New search for: Elsevier Ltd
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Publication date:2005-09-20
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Size:8 pages
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ISSN:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Keywords:RNase A , ribonuclease A , HSA , human serum albumin , 2′-CMP , cytidine-2′-mono phosphate , 3′-CMP, cytidine-3′-mono phosphate , 2′,3′ cCMP , cytidine 2′,3′ cyclic monophosphate , tRNA , transfer ribonucleic acid , Mes , 4-morpholine ethanesulphonic acid , NMR , nuclear magnetic resonance , HRMS , high resolution mass spectrometry , PDB , Protein Data Bank , GA , genetic algorithm , Ribonuclease A , Angiogenin and angiogenesis , Aminonucleosides , Precipitation assay , AutoDock , Inhibition kinetics
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Source:
Table of contents – Volume 14, Issue 4
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 885
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Graphical contents list| 2005
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- 918
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Synthesis, molecular modelling and enzymatic evaluation of ((plus-minus))3,5-diphenyl-2-thioxoimidazolidin-4-ones as new potential cyclooxygenase inhibitorsGauthier, Marie P. et al. | 2006
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Versatile synthesis and biological evaluation of 1,3-diamino-substituted 1#945,25-dihydroxyvitamin D3 analoguesOves, Daniel et al. | 2006
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Versatile synthesis and biological evaluation of 1,3-diamino-substituted 1α,25-dihydroxyvitamin D3 analoguesOves, Daniel / Fernández, Susana / Ferrero, Miguel / Bouillon, Roger / Verstuyf, Annemieke / Gotor, Vicente et al. | 2005
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Tyrosinase inhibitory cycloartane type triterpenoids from the methanol extract of the whole plant of Amberboa ramosa Jafri and their structure#8211activity relationshipKhan, Mahmud Tareq Hassan et al. | 2006
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Microwave-assisted synthesis of antimicrobial dihydropyridines and tetrahydropyrimidin-2-ones: Novel compounds against aspergillosisChhillar, Anil K. / Arya, Pragya / Mukherjee, Chandrani / Kumar, Pankaj / Yadav, Yogesh / Sharma, Ajendra K. / Yadav, Vibha / Gupta, Jyotsana / Dabur, Rajesh / Jha, Hirday N. et al. | 2005
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A QSAR study on influenza neuraminidase inhibitorsVerma, Rajeshwar P. / Hansch, Corwin et al. | 2005
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Enaminones 9. Further studies on the anticonvulsant activity and potential type IV phosphodiesterase inhibitory activity of substituted vinylic benzamidesAnderson, Alan J. / Nicholson, Jesse M. / Bakare, Oladapo / Butcher, Ray J. / Wilson, Tiffany L. / Scott, K.R. et al. | 2005
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Structure#8211activity relationships and enzyme inhibition of pantothenamide-type pantothenate kinase inhibitorsVirga, Kristopher G. et al. | 2006
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Structure–activity relationships and enzyme inhibition of pantothenamide-type pantothenate kinase inhibitorsVirga, Kristopher G. / Zhang, Yong-Mei / Leonardi, Roberta / Ivey, Robert A. / Hevener, Kirk / Park, Hee-Won / Jackowski, Suzanne / Rock, Charles O. / Lee, Richard E. et al. | 2005
- 1021
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QSPR models for polychlorinated biphenyls: n-Octanol/water partition coefficientPadmanabhan, J. / Parthasarathi, R. / Subramanian, V. / Chattaraj, P.K. et al. | 2005
- 1029
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Synthesis and properties of 2′-O,4′-C-methyleneoxymethylene bridged nucleic acidHari, Yoshiyuki / Obika, Satoshi / Ohnishi, Ryo / Eguchi, Ken / Osaki, Tomohisa / Ohishi, Hirofumi / Imanishi, Takeshi et al. | 2005
- 1029
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Synthesis and properties of 2#8242-O,4#8242-C-methyleneoxymethylene bridged nucleic acidHari, Yoshiyuki et al. | 2006
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QSAR by LFER model of HIV protease inhibitor mannitol derivatives using FA-MLR, PCRA, and PLS techniquesLeonard, J. Thomas / Roy, Kunal et al. | 2005
- 1047
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Building a successful structural motif into sialylmimetics—cyclohexenephosphonate monoesters as pseudo-sialosides with promising inhibitory propertiesStreicher, Hansjörg / Busse, Heike et al. | 2005
- 1047
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Building a successful structural motif into sialylmimetics#8212cyclohexenephosphonate monoesters as pseudo-sialosides with promising inhibitory propertiesStreicher, Hansjörg et al. | 2006
- 1058
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Epoxide opening in water and screening in situ for rapid discovery of enzyme inhibitors in microtiter platesLiang, Fu-Sen / Brik, Ashraf / Lin, Ying-Chuan / Elder, John H. / Wong, Chi-Huey et al. | 2005
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Absolute stereochemistry and antitumor activity of iejimalidesNozawa, Kohei / Tsuda, Masashi / Ishiyama, Haruaki / Sasaki, Takuma / Tsuruo, Takashi / Kobayashi, Jun’ichi et al. | 2005
- 1068
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Combination of porphyrins and DNA-alkylation agents: Synthesis and tumor cell apoptosis inductionHe, Hanping / Zhou, Yan / Liang, Feng / Li, Dongqing / Wu, Juanjuan / Yang, Li / Zhou, Xiang / Zhang, Xiaolian / Cao, Xiaoping et al. | 2005
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Synthesis and biological evaluation of N-(7-indazolyl)benzenesulfonamide derivatives as potent cell cycle inhibitorsBouissane, L. / El Kazzouli, S. / Léonce, S. / Pfeiffer, B. / Rakib, E.M. / Khouili, M. / Guillaumet, G. et al. | 2005
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Guanaconetins, new antitumoral acetogenins, mitochondrial complex I and tumor cell growth inhibitorsChahboune, Nadia / Barrachina, Isabel / Royo, Inmaculada / Romero, Vanessa / Sáez, Jairo / Tormo, José R. / De Pedro, Nuria / Estornell, Ernesto / Zafra-Polo, M. Carmen / Peláez, Fernando et al. | 2005
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Stochastic entropy QSAR for the in silico discovery of anticancer compounds: Prediction, synthesis, and in vitro assay of new purine carbanucleosidesGonzález-Díaz, Humberto / Viña, Dolores / Santana, Lourdes / de Clercq, Erik / Uriarte, Eugenio et al. | 2005
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QSAR study on para-substituted aromatic sulfonamides as carbonic anhydrase II inhibitors using topological information indicesMelagraki, Georgia / Afantitis, Antreas / Sarimveis, Haralambos / Igglessi-Markopoulou, Olga / Supuran, Claudiu T. et al. | 2005
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Synthesis, radiosynthesis and in vivo preliminary evaluation of [11C]LBT-999, a selective radioligand for the visualisation of the dopamine transporter with PETDollé, Frédéric / Emond, Patrick / Mavel, Sylvie / Demphel, Stéphane / Hinnen, Françoise / Mincheva, Zoïa / Saba, Wadad / Valette, Heric / Chalon, Sylvie / Halldin, Christer et al. | 2005
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Improving the membrane permeability of sialic acid derivativesAltamore, Timothy M. / Duggan, Peter J. / Krippner, Guy Y. et al. | 2005
- 1134
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Development and optimization of a useful assay for determining Hsp90’s inherent ATPase activityAvila, Christopher / Kornilayev, Boris A. / Blagg, Brian S.J. et al. | 2005
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Development and optimization of a useful assay for determining Hsp90#8217s inherent ATPase activityAvila, Christopher et al. | 2006
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High-throughput screening of ecdysone agonists using a reporter gene assay followed by 3-D QSAR analysis of the molting hormonal activityWheelock, Craig E. / Nakagawa, Yoshiaki / Harada, Toshiyuki / Oikawa, Nobuhiro / Akamatsu, Miki / Smagghe, Guy / Stefanou, Dimitra / Iatrou, Kostas / Swevers, Luc et al. | 2005
- 1160
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Phenazine-1-carboxamides: Structure#8211cytotoxicity relationships for 9-substituents and changes in the H-bonding pattern of the cationic side chainGamage, Swarna A. et al. | 2006
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Phenazine-1-carboxamides: Structure–cytotoxicity relationships for 9-substituents and changes in the H-bonding pattern of the cationic side chainGamage, Swarna A. / Rewcastle, Gordon W. / Baguley, Bruce C. / Charlton, Peter A. / Denny, William A. et al. | 2005
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Identification of 12Cysβ on tubulin as the binding site of tubulyzineKim, Yeoun Jin / Sackett, Dan L. / Schapira, Matthieu / Walsh, Daniel P. / Min, Jaeki / Pannell, Lewis K. / Chang, Young-Tae et al. | 2005
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Identification of 12Cys#946 on tubulin as the binding site of tubulyzineKim, Yeoun Jin et al. | 2006
- 1176
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Effect of polycyclic cage amines on the transmembrane potential of neuronal cellsGrobler, Erika / Grobler, Anne / Van der Schyf, Cornelis J. / Malan, Sarel F. et al. | 2005
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C-Glycoside analogues of #946-galactosylceramide with a simple ceramide substitute: Synthesis and binding to HIV-1 gp120Augustin, Line A. et al. | 2006
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Induction of apoptosis in HeLa cells by 3#946-hydroxy-12-oleanen-27-oic acid from the rhizomes of Astilbe chinensisSun, Hong-Xiang et al. | 2006
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QSAR analysis of phenolic antioxidants using MOLMAP descriptors of local propertiesGupta, Sunil / Matthew, Susan / Abreu, Pedro M. / Aires-de-Sousa, João et al. | 2005
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A chemoenzymatic scalable route to optically active (R)-1-(pyridin-3-yl)-2-aminoethanol, valuable moiety of #9463-adrenergic receptor agonistsPerrone, Maria Grazia et al. | 2006
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A chemoenzymatic scalable route to optically active (R)-1-(pyridin-3-yl)-2-aminoethanol, valuable moiety of β3-adrenergic receptor agonistsPerrone, Maria Grazia / Santandrea, Ernesto / Giorgio, Erika / Bleve, Laura / Scilimati, Antonio / Tortorella, Paolo et al. | 2005
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Thioureido N-acetyllactosamine derivatives as potent galectin-7 and 9N inhibitorsSalameh, B.A. / Sundin, A. / Leffler, H. / Nilsson, U.J. et al. | 2005
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3′-N-Alkylamino-3′-deoxy-ara-uridines: A new class of potential inhibitors of ribonuclease A and angiogeninMaiti, Tushar K. / Soumya De / Dasgupta, Swagata / Pathak, Tanmaya et al. | 2005
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3#8242-N-Alkylamino-3#8242-deoxy-ara-uridines: A new class of potential inhibitors of ribonuclease A and angiogeninMaiti, Tushar K. et al. | 2006
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- 1274
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Reviews and Perspectives| 2005
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Editorial Board| 2005
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Instructions to contributors| 2005