Synthesis and in vitro biological evaluation of novel coumarin derivatives containing isoxazole moieties on melanin synthesis in B16 cells and inhibition on bacteria (English)
- New search for: Pang, Guang Xian
- New search for: Niu, Chao
- New search for: Mamat, Nuramina
- New search for: Aisa, Haji Akber
- New search for: Pang, Guang Xian
- New search for: Niu, Chao
- New search for: Mamat, Nuramina
- New search for: Aisa, Haji Akber
In:
Bioorganic and Medicinal Chemistry Letters
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27
, 12
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2674-2677
;
2017
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ISSN:
- Article (Journal) / Electronic Resource
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Title:Synthesis and in vitro biological evaluation of novel coumarin derivatives containing isoxazole moieties on melanin synthesis in B16 cells and inhibition on bacteria
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Contributors:Pang, Guang Xian ( author ) / Niu, Chao ( author ) / Mamat, Nuramina ( author ) / Aisa, Haji Akber ( author )
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Published in:Bioorganic and Medicinal Chemistry Letters ; 27, 12 ; 2674-2677
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Publisher:
- New search for: Elsevier Ltd
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Publication date:2017-04-12
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Size:4 pages
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ISSN:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Keywords:
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Source:
Table of contents – Volume 27, Issue 12
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 2645
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Evaluation of synthesized coumarin derivatives on aromatase inhibitory activityYamaguchi, Yuki / Nishizono, Naozumi / Kobayashi, Daisuke / Yoshimura, Teruki / Wada, Keiji / Oda, Kazuaki et al. | 2017
- 2650
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Neutral macrocyclic factor VIIa inhibitorsWurtz, Nicholas R. / Parkhurst, Brandon L. / DeLucca, Indawati / Glunz, Peter W. / Jiang, Wen / Zhang, Xiaojun / Cheney, Daniel L. / Bozarth, Jeffrey M. / Rendina, Alan R. / Wei, Anzhi et al. | 2017
- 2655
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Nucleobase azide–ethynylribose click chemistry contributes to stabilizing oligonucleotide duplexes and stem-loop structuresKitamura, Yoshiaki / Asakura, Ryo / Terazawa, Koki / Shibata, Aya / Ikeda, Masato / Kitade, Yukio et al. | 2017
- 2659
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Sulfoximines as ATR inhibitors: Analogs of VE-821Hendriks, Christine M.M. / Hartkamp, Jörg / Wiezorek, Stefan / Steinkamp, Anne-Dorothee / Rossetti, Giulia / Lüscher, Bernhard / Bolm, Carsten et al. | 2017
- 2663
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N-(1H-Pyrazol-3-yl)quinazolin-4-amines as a novel class of casein kinase 1δ/ε inhibitors: Synthesis, biological evaluation and molecular modeling studiesKarthikeyan, Chandrabose / Jharia, Pramod / Waiker, Digambar Kumar / Nusbaum, Amy Catherine / Amawi, Haneen / Kirwen, Erin Marie / Christman, Ryann / Arudra, Sri Krishna Chaitanya / Meijer, Laurent / Tiwari, Amit K. et al. | 2017
- 2668
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Design, synthesis, biological evaluation and molecular docking studies of novel 3-aryl-4-anilino-2H-chromen-2-one derivatives targeting ERα as anti-breast cancer agentsLuo, Guoshun / Chen, Mingqi / Lyu, Weiting / Zhao, Ruheng / Xu, Qian / You, Qidong / Xiang, Hua et al. | 2017
- 2674
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Synthesis and in vitro biological evaluation of novel coumarin derivatives containing isoxazole moieties on melanin synthesis in B16 cells and inhibition on bacteriaPang, Guang Xian / Niu, Chao / Mamat, Nuramina / Aisa, Haji Akber et al. | 2017
- 2678
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Discovery of potent and orally active 1,4-disubstituted indazoles as novel allosteric glucokinase activatorsCheruvallath, Zacharia S. / Gwaltney, Stephen L. II / Sabat, Mark / Tang, Mingnam / Wang, Haixia / Jennings, Andy / Hosfield, David / Lee, Bumsup / Wu, Yiqin / Halkowycz, Petro et al. | 2017
- 2683
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Benzoxazolinone aryl sulfonamides as potent, selective Nav1.7 inhibitors with in vivo efficacy in a preclinical pain modelPero, Joseph E. / Rossi, Michael A. / Lehman, Hannah D.G.F. / Kelly, Michael J. III / Mulhearn, James J. / Wolkenberg, Scott E. / Cato, Matthew J. / Clements, Michelle K. / Daley, Christopher J. / Filzen, Tracey et al. | 2017
- 2689
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Discovery of a novel and potent class of anti-HIV-1 maturation inhibitors with improved virology profile against gag polymorphismsTang, Jun / Jones, Stacey A. / Jeffrey, Jerry L. / Miranda, Sonia R. / Galardi, Cristin M. / Irlbeck, David M. / Brown, Kevin W. / McDanal, Charlene B. / Johns, Brian A. et al. | 2017
- 2695
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Design, synthesis and SAR of substituted indoles as selective TrkA inhibitorsHurzy, Danielle M. / Henze, Darrell A. / Cabalu, Tamara D. / Narayan, Kartik / Heller, Amanda / Cooke, Andrew J. et al. | 2017
- 2702
-
Optimization of a binding fragment targeting the “enlarged methionine pocket” leads to potent Trypanosoma brucei methionyl-tRNA synthetase inhibitorsHuang, Wenlin / Zhang, Zhongsheng / Ranade, Ranae M. / Gillespie, J. Robert / Barros-Álvarez, Ximena / Creason, Sharon A. / Shibata, Sayaka / Verlinde, Christophe L.M.J. / Hol, Wim G.J. / Buckner, Frederick S. et al. | 2017
- 2708
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Discovery of novel substituted benzo-anellated 4-benzylamino pyrrolopyrimidines as dual EGFR and VEGFR2 inhibitorsFischer, Tim / Krüger, Thomas / Najjar, Abdulkarim / Totzke, Frank / Schächtele, Christoph / Sippl, Wolfgang / Ritter, Christoph / Hilgeroth, Andreas et al. | 2017
- 2713
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Thio-functionalized carbohydrate thiosemicarbazones and evaluation of their anticancer activityCzubatka-Bieńkowska, Anna / Sarnik, Joanna / Macieja, Anna / Galita, Grzegorz / Witczak, Zbigniew J. / Poplawski, Tomasz et al. | 2017
- 2721
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Identification of quinazoline based inhibitors of IRAK4 for the treatment of inflammationSmith, Graham F. / Altman, Michael D. / Andresen, Brian / Baker, James / Brubaker, Jason D. / Chen, Hongmin / Chen, Yiping / Childers, Matthew / Donofrio, Anthony / Ferguson, Heidi et al. | 2017
- 2727
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Synthesis and preliminary biological evaluation of [11C]methyl (2-amino-5-(benzylthio)thiazolo[4,5-d]pyrimidin-7-yl)-d-leucinate for the fractalkine receptor (CX3CR1)Gao, Mingzhang / Wang, Min / Meyer, Jill A. / Peters, Jonathan S. / Zarrinmayeh, Hamideh / Territo, Paul R. / Hutchins, Gary D. / Zheng, Qi-Huang et al. | 2017
- 2731
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Antitubulin effects of aminobenzothiophene-substituted triethylated chromonesKobayashi, Yukiko / Saito, Yohei / Goto, Masuo / Nakagawa-Goto, Kyoko et al. | 2017
- 2736
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An unusual spinaceamine-bearing pregnane from a soft coral Scleronephthya sp. inhibits the migration of tumor cellsCheng, Wei / Liu, Zhen / Yu, Yang / van Ofwegen, Leen / Proksch, Peter / Yu, Siwang / Lin, Wenhan et al. | 2017
- 2742
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Novel delta opioid receptor agonists with oxazatricyclodecane structure showing potent agonistic activitiesHayashida, Kohei / Hirayama, Shigeto / Iwai, Takashi / Watanabe, Yoshikazu / Takahashi, Toshihiro / Sakai, Junichi / Nakata, Eriko / Yamakawa, Tomio / Fujii, Hideaki / Nagase, Hiroshi et al. | 2017
- 2746
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Synthesis and evaluation of phenylisoserine derivatives for the SARS-CoV 3CL protease inhibitorKonno, Hiroyuki / Onuma, Takumi / Nitanai, Ikumi / Wakabayashi, Masaki / Yano, Shigekazu / Teruya, Kenta / Akaji, Kenichi et al. | 2017
- 2752
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Design, synthesis and biological evaluation of fucose-truncated monosaccharide analogues of ipomoeassin FZong, Guanghui / Hirsch, Melissa / Mondrik, Collin / Hu, Zhijian / Shi, Wei Q. et al. | 2017
- 2757
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Investigation of the structural requirements of K-Ras(G12D) selective inhibitory peptide KRpep-2d using alanine scans and cysteine bridgingNiida, Ayumu / Sasaki, Shigekazu / Yonemori, Kazuko / Sameshima, Tomoya / Yaguchi, Masahiro / Asami, Taiji / Sakamoto, Kotaro / Kamaura, Masahiro et al. | 2017
- 2762
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Isolation of the antibiotic pseudopyronine B and SAR evaluation of C3/C6 alkyl analogsBouthillette, Leah M. / Darcey, Catherine A. / Handy, Tess E. / Seaton, Sarah C. / Wolfe, Amanda L. et al. | 2017
- 2766
-
Activity of resveratrol triesters against primary acute lymphoblastic leukemia cellsUrbaniak, Alicja / Delgado, Magdalena / Kacprzak, Karol / Chambers, Timothy C. et al. | 2017
- 2771
-
Design and synthesis of a fluorinated quinazoline-based type-II Trk inhibitor as a scaffold for PET radiotracer developmentBernard-Gauthier, Vadim / Mahringer, Anne / Vesnaver, Matthew / Fricker, Gert / Schirrmacher, Ralf et al. | 2017
- 2776
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Structure-activity relationships of rosiglitazone for peroxisome proliferator-activated receptor gamma transrepressionToyota, Yosuke / Nomura, Sayaka / Makishima, Makoto / Hashimoto, Yuichi / Ishikawa, Minoru et al. | 2017
- 2781
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Phenanthridin-6-one derivatives as the first class of non-steroidal pharmacological chaperones for Niemann-Pick disease type C1 proteinFukuda, Hiromitsu / Karaki, Fumika / Dodo, Kosuke / Noguchi-Yachide, Tomomi / Ishikawa, Minoru / Hashimoto, Yuichi / Ohgane, Kenji et al. | 2017
- 2788
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Drug-like property-driven optimization of 4-substituted 1,5-diarylanilines as potent HIV-1 non-nucleoside reverse transcriptase inhibitors against rilpivirine-resistant mutant virusWei, Lei / Wang, Hui-Ling / Huang, Li / Chen, Chin-Ho / Morris-Natschke, Susan L. / Lee, Kuo-Hsiung / Xie, Lan et al. | 2017
- 2793
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Cell line studies and analytical measurements of three paclitaxel complex variationsManning, Thomas / Plummer, Sydney / Woods, Rechelle / Wylie, Greg / Phillips, Dennis / Krajewski, Logan et al. | 2017
- 2800
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Flex-nucleoside analogues – Novel therapeutics against filovirusesYates, Mary K. / Raje, Mithun R. / Chatterjee, Payel / Spiropoulou, Christina F. / Bavari, Sina / Flint, Mike / Soloveva, Veronica / Seley-Radtke, Katherine L. et al. | 2017
- 2803
-
Design, synthesis, and biological evaluation of deuterated apalutamide with improved pharmacokinetic profilesPang, Xuehai / Wang, Yingwei / Chen, Yuanwei et al. | 2017
- 2807
-
Alkaloids from aerial parts of Houttuynia cordata and their anti-inflammatory activityAhn, Jongmin / Chae, Hee-Sung / Chin, Young-Won / Kim, Jinwoong et al. | 2017
- 2812
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Anti-atherosclerotic activities of flavonoids from the flowers of Helichrysum arenarium L. MOENCH through the pathway of anti-inflammationMao, Zhonghua / Gan, Chunli / Zhu, Jiuxin / Ma, Nan / Wu, Lijun / Wang, Libo / Wang, Xiaobo et al. | 2017
- 2818
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Synthesis and α-glucosidase inhibition activity of dihydroxy pyrrolidinesKasturi, Sivaprasad / Surarapu, Sujatha / Uppalanchi, Srinivas / Anireddy, Jaya Shree / Dwivedi, Shubham / Anantaraju, Hasitha Shilpa / Perumal, Yogeeswari / Sigalapalli, Dilep Kumar / Babu, Bathini Nagendra / Ethiraj, Krishna S. et al. | 2017
- IFC
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Editorial board| 2017