Discovery of novel oridonin sulfamide derivatives as potent NLRP3 inhibitors by a visible-light photocatalysis-enabled peripheral editing (English)
- New search for: Li, Mochenxuan
- New search for: Wang, Chuanhao
- New search for: Ye, Shuang
- New search for: Li, Wei
- New search for: Zhang, Yanming
- New search for: Yan, Jianyu
- New search for: Wang, Yongchuang
- New search for: Yang, Hang
- New search for: Wu, Yuelin
- New search for: Zhang, Yongqiang
- New search for: Zhang, Huojun
- New search for: Miao, Zhenyuan
- New search for: Li, Mochenxuan
- New search for: Wang, Chuanhao
- New search for: Ye, Shuang
- New search for: Li, Wei
- New search for: Zhang, Yanming
- New search for: Yan, Jianyu
- New search for: Wang, Yongchuang
- New search for: Yang, Hang
- New search for: Wu, Yuelin
- New search for: Zhang, Yongqiang
- New search for: Zhang, Huojun
- New search for: Miao, Zhenyuan
In:
Bioorganic and Medicinal Chemistry Letters
;
99
;
2024
-
ISSN:
- Article (Journal) / Electronic Resource
-
Title:Discovery of novel oridonin sulfamide derivatives as potent NLRP3 inhibitors by a visible-light photocatalysis-enabled peripheral editing
-
Contributors:Li, Mochenxuan ( author ) / Wang, Chuanhao ( author ) / Ye, Shuang ( author ) / Li, Wei ( author ) / Zhang, Yanming ( author ) / Yan, Jianyu ( author ) / Wang, Yongchuang ( author ) / Yang, Hang ( author ) / Wu, Yuelin ( author ) / Zhang, Yongqiang ( author )
-
Published in:
-
Publication date:2024-01-15
-
ISSN:
-
DOI:
-
Type of media:Article (Journal)
-
Type of material:Electronic Resource
-
Language:English
-
Keywords:
-
Source:
Table of contents – Volume 99
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
-
Identification of 4-(6-((2-methoxyphenyl)amino)pyrazin-2-yl)benzoic acids as CSNK2A inhibitors with antiviral activity and improved selectivity over PIM3Galal, Kareem A. / Krämer, Andreas / Strickland, Benjamin G. / Smith, Jeffery L. / Dickmander, Rebekah J. / Moorman, Nathaniel J. / Willson, Timothy M. et al. | 2024
-
Therapeutic potential of Coumarin-polyphenolic acid hybrids in PD: Inhibition of α-Syn aggregation and disaggregation of preformed fibrils, leading to reduced neuronal inclusion formationWang, Zhen-Ping / Zhang, Wei / Xing, Li-Zi / Zhao, Ya-Dong / Xu, Ji / Zhang, Yun-Xiao et al. | 2024
-
Graphical abstract TOC| 2024
-
Design of cyclic peptides as novel inhibitors of ICOS/ICOSL interactionAbdel‐Rahman, Somaya A. / Santini, Brianda L / Calvo-Barreiro, Laura / Zacharias, Martin / Gabr, Moustafa et al. | 2024
-
Discovery of novel oridonin sulfamide derivatives as potent NLRP3 inhibitors by a visible-light photocatalysis-enabled peripheral editingLi, Mochenxuan / Wang, Chuanhao / Ye, Shuang / Li, Wei / Zhang, Yanming / Yan, Jianyu / Wang, Yongchuang / Yang, Hang / Wu, Yuelin / Zhang, Yongqiang et al. | 2024
-
Further structural optimization and SAR study of sungsanpin derivatives as cell-invasion inhibitorsChen, Shuai / Zhang, Kai / Zou, Jihua / Yu, Zhou / Gai, Conghao / Chai, Xiaoyun / Zhao, Qingjie / Zou, Yan et al. | 2024
-
Expanded library of novel 2,3-pyrrolidinedione analogues exhibit anti-biofilm activityNie, Minhua / Alejandro Valdes-Pena, M. / Frohock, Bram H. / Smits, Emma / Daiker, Jennifer C. / Gilbertie, Jessica M. / Schnabel, Lauren V. / Pierce, Joshua G. et al. | 2024
-
Design, synthesis and biological evaluation of 6-chloro-quinolin-2-one derivatives as novel FXIa inhibitorsWang, Yanshi / Yuan, Jianglin / Yan, Sida / Liu, Peng / Zheng, Zhichao / Zhang, Shijun / Meng, Fancui / Liu, Wei / Huang, Changjiang / Wei, Qunchao et al. | 2024
-
Editorial Board| 2024
-
Contents continued| 2024
-
Novel orexin receptor agonists based on arene- or pyridine-fused 1,3-dihydro-2H-imidazole-2-iminesWang, Wentian / Ranjan, Alok / Zhang, Wei / Liang, Qiren / MacMillan, Karen S. / Chapman, Karen / Wang, Xiaoyu / Chandrasekaran, Preethi / Williams, Noelle S. / Rosenbaum, Daniel M. et al. | 2024
-
Improved synthesis and evaluation of preclinical pharmacodynamic parameters of a new monocyclic β-lactam DPI-2016Zhai, Lijuan / Sun, Jian / Ji, Jingwen / He, Lili / Zhou, Pengjuan / Tang, Dong / Ji, Jinbo / Yang, Haikang / Iqbal, Zafar / Yang, Zhixiang et al. | 2024
-
Design, synthesis and bioactivity evaluation of the combination of evodiamine and erlotinib linked by indolequinoneWei, Binbin / Ma, Jingjing / Guo, Hui / Wang, Yuwei / Guo, Dongyan / Tang, Yuping et al. | 2024
-
Synthesis and biological evaluation of novel 18F-labeled 2,4-diaminopyrimidine derivatives for detection of ghrelin receptor in the brainSaito, Haruka / Watanabe, Hiroyuki / Ono, Masahiro et al. | 2024
-
Inhibition of dengue viruses by N-methylcytisine thio derivatives through targeting viral envelope protein and NS2B-NS3 proteaseLin, Chen-Sheng / Lu, Chih-Hao / Lin, Tsai-Hsiu / Kiu, Yan-Tung / Kan, Ju-Ying / Chang, Yu-Jen / Hung, Ping-Yi / Koval'skaya, Alena V. / Tsypyshev, Dmitry O. / Tsypysheva, Inna P. et al. | 2024
-
Synthetic assembly of α-O-linked-type GlcNAc using polymer chemistry affords sugar clusters, which effectively bind to lectinsNakada, Jyuichi / Matsushita, Takahiko / Koyama, Tetsuo / Hatano, Ken / Matsuoka, Koji et al. | 2024
-
Design and synthesis of unique morphinan-type molecules: Their application to the search for the unexplored binding domain between opioid receptors and morphinan ligandsMaeda, Kenta / Sugai, Tomoya / Tokuda, Akihisa / Kajino, Keita / Saitoh, Tsuyoshi / Nagase, Hiroshi / Kutsumura, Noriki et al. | 2024
-
Synthesis, biological activity evaluation and mechanism of action of novel bis-isatin derivatives as potential anti-liver cancer agentsLi, Zhifen / Ma, Jingbo / Tian, Ming / Xia, Peng / Lv, Xiannian / Hou, Rui / Jiang, Yuke / Xu, Xiaolong / Jia, Zhifang / Wang, Jigang et al. | 2024
-
Natural products fragment-based design and synthesis of a novel pentacyclic ring system as potential MAPK inhibitorHou, Bao-Long / Wu, Kenan / Liu, Rongrong / Liu, Jianli / Wang, Jinrui / Wang, Cuiling / Liang, Yanni / Wang, Zheng et al. | 2023
-
Structure-based design and synthesis of sulfonylureas as novel NLRP3 inhibitors for Alzheimer’s diseaseKim, Eun Young / Im, Jae Hong / Han, Jinhe / Cho, Won-Jea et al. | 2024