Disruption of Kv1.1 N-type inactivation by novel small molecule inhibitors (disinactivators) (English)
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In:
Bioorganic and Medicinal Chemistry
;
16
, 6
;
3067-3075
;
2007
-
ISSN:
- Article (Journal) / Electronic Resource
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Title:Disruption of Kv1.1 N-type inactivation by novel small molecule inhibitors (disinactivators)
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Contributors:Lu, Qiang ( author ) / Peevey, Joseph ( author ) / Jow, Flora ( author ) / Monaghan, Michael M. ( author ) / Mendoza, Grace ( author ) / Zhang, Howard ( author ) / Wu, Jerome ( author ) / Kim, Callain Y. ( author ) / Bicksler, James ( author ) / Greenblatt, Lynn ( author )
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Published in:Bioorganic and Medicinal Chemistry ; 16, 6 ; 3067-3075
-
Publisher:
- New search for: Elsevier Ltd
-
Publication date:2007-12-17
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Size:9 pages
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ISSN:
-
DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Keywords:
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Source:
Table of contents – Volume 16, Issue 6
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 2707
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Graphical contents list| 2008
- 2726
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A comparative density-functional study of the reaction mechanism of the O2-dependent coproporphyrinogen III oxidaseSilva, Pedro J. / Ramos, Maria João et al. | 2008
- 2734
-
Effect of five-membered sugar mimics on mammalian glycogen-degrading enzymes and various glucosidasesMinami, Yasuhiro / Kuriyama, Chinami / Ikeda, Kyoko / Kato, Atsushi / Takebayashi, Kenji / Adachi, Isao / Fleet, George W.J. / Kettawan, Aikkarach / Okamoto, Tadashi / Asano, Naoki et al. | 2008
- 2741
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A new generation of adenosine receptor antagonists: From di- to trisubstituted aminopyrimidinesvan Veldhoven, Jacobus P.D. / Chang, Lisa C.W. / von Frijtag Drabbe Künzel, Jacobien K. / Mulder-Krieger, Thea / Struensee-Link, Regina / Beukers, Margot W. / Brussee, Johannes / IJzerman, Adriaan P. et al. | 2008
- 2753
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11-(Pyridinylphenyl)steroids—A new class of mixed-profile progesterone agonists/antagonistsRewinkel, Jos / Enthoven, Mark / Golstein, Irene / van der Rijst, Marcel / Scholten, André / van Tilborg, Martin / de Weys, Dirk / Wisse, Jeffry / Hamersma, Hans et al. | 2008
- 2764
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Targeted inhibition of hedgehog signaling by cyclopamine prodrugs for advanced prostate cancerKumar, Srinivas K. / Roy, Indrajit / Anchoori, Ravi K. / Fazli, Sarah / Maitra, Anirban / Beachy, Philip A. / Khan, Saeed R. et al. | 2008
- 2769
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Further structural optimization of cis-(6-benzhydryl-piperidin-3-yl)-benzylamine and 1,4-diazabicyclo[3.3.1]nonane derivatives by introducing an exocyclic hydroxyl group: Interaction with dopamine, serotonin, and norepinephrine transportersMishra, Manoj / Kolhatkar, Rohit / Zhen, Juan / Parrington, Ingrid / Reith, Maarten E.A. / Dutta, Aloke K. et al. | 2008
- 2779
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Binding to human serum albumin of zidovudine (AZT) and novel AZT derivatives. Experimental and theoretical analysesQuevedo, Mario A. / Ribone, Sergio R. / Moroni, Guillermo N. / Briñón, Margarita C. et al. | 2008
- 2791
-
Structure–activity relationship analysis of N-benzoylpyrazoles for elastase inhibitory activity: A simplified approach using atom pair descriptorsKhlebnikov, Andrei I. / Schepetkin, Igor A. / Quinn, Mark T. et al. | 2008
- 2803
-
Interactive effects of polymethoxy flavones from Citrus on cell growth inhibition in human neuroblastoma SH-SY5Y cellsAkao, Yukihiro / itoh, Tomohiro / Ohguchi, Kenji / Iinuma, Munekazu / Nozawa, Yoshinori et al. | 2008
- 2811
-
Development of polymeric drug delivery system for recognizing vascular endothelial dysfunctionIkuta, Kenjiro / Mori, Takeshi / Yamamoto, Tatsurhiro / Niidome, Takuro / Shimokawa, Hiroaki / Katayama, Yoshiki et al. | 2008
- 2819
-
Exploring the potential of 3′-O-carboxy esters of thymidine as inhibitors of ribonuclease A and angiogeninGhosh, Kalyan S. / Debnath, Joy / Dutta, Palash / Sahoo, Bijaya K. / Dasgupta, Swagata et al. | 2008
- 2819
-
Exploring the potential of 3prime-O-carboxy esters of thymidine as inhibitors of ribonuclease A and angiogeninGhosh, K. S. / Debnath, J. / Dutta, P. / Sahoo, B. K. / Dasgupta, S. et al. | 2008
- 2829
-
Structure–activity relationships and CoMFA of N-3 substituted phenoxypropyl piperidine benzimidazol-2-one analogues as NOP receptor agonists with analgesic propertiesPalin, Ronald / Clark, John K. / Evans, Louise / Houghton, Andrea K. / Jones, Philip S. / Prosser, Alan / Wishart, Grant / Yoshiizumi, Kazuya et al. | 2008
- 2852
-
1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptorStefanachi, Angela / Brea, Jose Manuel / Cadavid, Maria Isabel / Centeno, Nuria B. / Esteve, Cristina / Loza, Maria Isabel / Martinez, Ana / Nieto, Rosa / Raviña, Enrique / Sanz, Ferran et al. | 2008
- 2870
-
Synthesis and pharmacological evaluation of bicyclic SNC80 analogues with separated benzhydryl moietyJung, Bettina / Englberger, Werner / Fröhlich, Roland / Schepmann, Dirk / Lehmkuhl, Kirstin / Wünsch, Bernhard et al. | 2008
- 2886
-
Biocatalytic and semisynthetic optimization of the anti-invasive tobacco (1S,2E,4R,6R,7E,11E)-2,7,11-cembratriene-4,6-diolEl Sayed, Khalid A. / Laphookhieo, Surat / Baraka, Hany N. / Yousaf, Muhammad / Hebert, Anne / Bagaley, Danielle / Rainey, Frederick A. / Muralidharan, A. / Thomas, Shibu / Shah, Girish V. et al. | 2007
- 2894
-
Synthesis and exploration of novel curcumin analogues as anti-malarial agentsMishra, Satyendra / Karmodiya, Krishanpal / Surolia, Namita / Surolia, Avadhesha et al. | 2007
- 2903
-
A genetic algorithm optimized fuzzy neural network analysis of the affinity of inhibitors for HIV-1 proteaseFabry-Asztalos, Levente / Andonie, Raˇzvan / Collar, Catharine J. / Abdul-Wahid, Sarah / Salim, Nicholas et al. | 2007
- 2912
-
New triterpenoid saponins with strong α-glucosidase inhibitory activity from the roots of Gypsophila oldhamianaLuo, Jian-Guang / Ma, Li / Kong, Ling-Yi et al. | 2007
- 2912
-
New triterpenoid saponins with strong a-glucosidase inhibitory activity from the roots of Gypsophila oldhamianaLuo, J. G. / Ma, L. / Kong, L. Y. et al. | 2008
- 2921
-
Synthesis of chemically functionalized superparamagnetic nanoparticles as delivery vectors for chemotherapeutic drugsHanessian, Stephen / Grzyb, Justyna A. / Cengelli, Feride / Juillerat-Jeanneret, Lucienne et al. | 2007
- 2932
-
Inhibitory property of the Piper betel phenolics against photosensitization-induced biological damagesMula, Soumyaditya / Banerjee, Debashish / Patro, Birija S. / Bhattacharya, Sayanti / Barik, Atanu / Bandyopadhyay, Sandip K. / Chattopadhyay, Subrata et al. | 2007
- 2939
-
1-Deoxyrubralactone, a novel specific inhibitor of families X and Y of eukaryotic DNA polymerases from a fungal strain derived from sea algaeNaganuma, Mitsuki / Nishida, Masayuki / Kuramochi, Kouji / Sugawara, Fumio / Yoshida, Hiromi / Mizushina, Yoshiyuki et al. | 2007
- 2945
-
Recognition of TA interruption by 2prime,4prime-BNAs bearing heteroaromatic nucleobases through parallel motif triplex formationObika, S. / Inohara, H. / Hari, Y. / Imanishi, T. et al. | 2008
- 2945
-
Recognition of T·A interruption by 2′,4′-BNAs bearing heteroaromatic nucleobases through parallel motif triplex formationObika, Satoshi / Inohara, Hiroyasu / Hari, Yoshiyuki / Imanishi, Takeshi et al. | 2007
- 2955
-
Hepatitis C virus NS3 protease inhibitors comprising a novel aromatic P1 moietyRönn, Robert / Lampa, Anna / Peterson, Shane D. / Gossas, Thomas / Åkerblom, Eva / Danielson, U. Helena / Karlén, Anders / Sandström, Anja et al. | 2007
- 2968
-
Lead identification of acetylcholinesterase inhibitors–histamine H3 receptor antagonists from molecular modelingBembenek, Scott D. / Keith, John M. / Letavic, Michael A. / Apodaca, Richard / Barbier, Ann J. / Dvorak, Lisa / Aluisio, Leah / Miller, Kirsten L. / Lovenberg, Timothy W. / Carruthers, Nicholas I. et al. | 2007
- 2974
-
Achiral, selective CCK2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione templateSpencer, John / Gaffen, John / Griffin, Eric / Harper, Elaine A. / Linney, Ian D. / McDonald, Iain M. / Roberts, Sonia P. / Shaxted, Mark E. / Adatia, Trushar / Bashall, Alan et al. | 2007
- 2984
-
Novel 1,3,4-thiadiazolium-2-phenylamine chlorides derived from natural piperine as trypanocidal agents: Chemical and biological studiesda Silva Ferreira, Welisson / Freire-de-Lima, Leonardo / Saraiva, Víctor Barbosa / Alisson-Silva, Frederico / Mendonça-Previato, Lucia / Previato, José Osvaldo / Echevarria, Aurea / de Lima, Marco Edilson Freire et al. | 2007
- 2992
-
Synthesis and structure–affinity relationships of novel spirocyclic σ receptor ligands with furopyrazole structureSchläger, Torsten / Schepmann, Dirk / Würthwein, Ernst-Ulrich / Wünsch, Bernhard et al. | 2007
- 3002
-
The 2α-(3-hydroxypropyl) group as an active motif in vitamin D3 analogues as agonists of the mutant vitamin D receptor (Arg274Leu)Honzawa, Shinobu / Yamamoto, Yasuhiro / Yamashita, Atsushi / Sugiura, Takayuki / Kurihara, Masaaki / Arai, Midori A. / Kato, Shigeaki / Kittaka, Atsushi et al. | 2007
- 3002
-
The 2a-(3-hydroxypropyl) group as an active motif in vitamin D3 analogues as agonists of the mutant vitamin D receptor (Arg274Leu)Honzawa, S. / Yamamoto, Y. / Yamashita, A. / Sugiura, T. / Kurihara, M. / Arai, M. A. / Kato, S. / Kittaka, A. et al. | 2008
- 3025
-
Conformations of 3-carboxylic esters essential for neurotoxicity in veratrum alkaloids are loosely restricted and fluctuateNiitsu, Ai / Harada, Masanori / Yamagaki, Tohru / Tachibana, Kazuo et al. | 2007
- 3032
-
Role of benzimidazole (Bid) in the δ-opioid agonist pseudopeptide H-Dmt-Tic-NH-CH2-Bid (UFP-502)Salvadori, Severo / Fiorini, Stella / Trapella, Claudio / Porreca, Frank / Davis, Peg / Sasaki, Yusuke / Ambo, Akihiro / Marczak, Ewa D. / Lazarus, Lawrence H. / Balboni, Gianfranco et al. | 2007
- 3032
-
Role of benzimidazole (Bid) in the d-opioid agonist pseudopeptide H-Dmt-Tic-NH-CH2-Bid (UFP-502)Salvadori, S. / Fiorini, S. / Trapella, C. / Porreca, F. / Davis, P. / Sasaki, Y. / Ambo, A. / Marczak, E. D. / Lazarus, L. H. / Balboni, G. et al. | 2008
- 3039
-
Molecular modeling studies of N-substituted pyrrole derivatives—Potential HIV-1 gp41 inhibitorsTeixeira, Cátia / Barbault, Florent / Rebehmed, Joseph / Liu, Kun / Xie, Lan / Lu, Hong / Jiang, Shibo / Fan, BoTao / Maurel, François et al. | 2007
- 3049
-
Docking analyses on human muscarinic receptors: Unveiling the subtypes peculiarities in agonists bindingVistoli, Giulio / Pedretti, Alessandro / Dei, Silvia / Scapecchi, Serena / Marconi, Cristina / Romanelli, Maria Novella et al. | 2007
- 3059
-
Synthesis and in silico biological activity evaluation of new N-substituted pyrazolo-oxazin-2-one systemsBenaamane, Nora / Nedjar-Kolli, Bellara / Bentarzi, Yamina / Hammal, Lamouri / Geronikaki, Athina / Eleftheriou, Phaedra / Lagunin, Alexey et al. | 2007
- 3067
-
Disruption of Kv1.1 N-type inactivation by novel small molecule inhibitors (disinactivators)Lu, Qiang / Peevey, Joseph / Jow, Flora / Monaghan, Michael M. / Mendoza, Grace / Zhang, Howard / Wu, Jerome / Kim, Callain Y. / Bicksler, James / Greenblatt, Lynn et al. | 2007
- 3076
-
Synthesis and antiviral activities of novel chiral cyanoacrylate derivatives with (E) configurationChen, Zhuo / Wang, Xianyou / Song, Baoan / Wang, Hua / Bhadury, Pinaki S. / Yan, Kai / Zhang, Huiping / Yang, Song / Jin, Linhong / Hu, Deyu et al. | 2007
- 3084
-
Effects of lipid constituents on membrane-permeabilizing activity of amphidinolsMorsy, Nagy / Houdai, Toshihiro / Konoki, Keiichi / Matsumori, Nobuaki / Oishi, Tohru / Murata, Michio et al. | 2007
- 3091
-
New anti-viral drugs for the treatment of the common coldMaugeri, Caterina / Alisi, Maria A. / Apicella, Claudia / Cellai, Luciano / Dragone, Patrizia / Fioravanzo, Elena / Florio, Saverio / Furlotti, Guido / Mangano, Giorgina / Ombrato, Rosella et al. | 2007
- 3108
-
Design and synthesis of biologically active analogues of vitamin K2: Evaluation of their biological activities with cultured human cell linesSuhara, Yoshitomo / Hirota, Yoshihisa / Nakagawa, Kimie / Kamao, Maya / Tsugawa, Naoko / Okano, Toshio et al. | 2007
- 3118
-
N-Phenethyl and N-naphthylmethyl isatins and analogues as in vitro cytotoxic agentsMatesic, Lidia / Locke, Julie M. / Bremner, John B. / Pyne, Stephen G. / Skropeta, Danielle / Ranson, Marie / Vine, Kara L. et al. | 2007
- 3125
-
Discovery of piperazinylimidazo[1,2-a]pyridines as novel S4 binding elements for orally active Factor Xa inhibitorsImaeda, Yasuhiro / Kawamoto, Tetsuji / Tobisu, Mamoru / Konishi, Noriko / Hiroe, Katsuhiko / Kawamura, Masaki / Tanaka, Toshimasa / Kubo, Keiji et al. | 2007
- 3141
-
Structure-activity relationship of uniconazole, a potent inhibitor of ABA 8prime-hydroxylase, with a focus on hydrophilic functional groups and conformationTodoroki, Y. / Kobayashi, K. / Yoneyama, H. / Hiramatsu, S. / Jin, M. H. / Watanabe, B. / Mizutani, M. / Hirai, N. et al. | 2008
- 3141
-
Structure–activity relationship of uniconazole, a potent inhibitor of ABA 8′-hydroxylase, with a focus on hydrophilic functional groups and conformationTodoroki, Yasushi / Kobayashi, Kyotaro / Yoneyama, Hidetaka / Hiramatsu, Saori / Jin, Mei-Hong / Watanabe, Bunta / Mizutani, Masaharu / Hirai, Nobuhiro et al. | 2007
- 3153
-
Synthesis and antiproliferative evaluation of certain indeno[1,2-c]quinoline derivativesTseng, Chih-Hua / Chen, Yeh-Long / Lu, Pei-Jung / Yang, Chia-Ning / Tzeng, Cherng-Chyi et al. | 2007
- 3163
-
Synthesis of insecticidal fluorinated anthranilic diamidesClark, David A. / Lahm, George P. / Smith, Ben K. / Barry, James D. / Clagg, Don G. et al. | 2007
- 3171
-
Core-modified porphyrins. Part 6: Effects of lipophilicity and core structures on physicochemical and biological properties in vitroNgen, Ethel J. / Daniels, Thalia S. / Murthy, Rajesh S. / Detty, Michael R. / You, Youngjae et al. | 2007
- 3184
-
Structure–reactivity relationships for electrophilic sugars in interaction with nucleophilic biological targetsCampodónico, Paola R. / Contreras, Renato et al. | 2007
- 3191
-
Synthesis and in vitro properties of trimethylamine- and phosphonate-substituted carboranylporphyrins for application in BNCTEasson, Michael W. / Fronczek, Frank R. / Jensen, Timothy J. / Vicente, M. Graça H. et al. | 2007
- 3209
-
Synthesis and cytotoxic activity of diosgenyl saponin analoguesKaskiw, Matthew J. / Tassotto, Mary Lynn / Th’ng, John / Jiang, Zi-Hua et al. | 2007
- 3218
-
Novel coumarin glycoside and phenethyl vanillate from Notopterygium forbesii and their binding affinities for opioid and dopamine receptorsMa, Zhongze / Xu, Wei / Liu-Chen, Lee-Yuan / Lee, David Y.W. et al. | 2007
- 3224
-
Synthesis and biological evaluation of novel dimiracetam derivatives useful for the treatment of neuropathic painFarina, Carlo / Gagliardi, Stefania / Ghelardini, Carla / Martinelli, Marisa / Norcini, Monica / Parini, Carlo / Petrillo, Paola / Ronzoni, Silvano et al. | 2007
- 3233
-
Synthesis, dopaminergic profile, and molecular dynamics calculations of N-aralkyl substituted 2-aminoindansAndujar, Sebastian A. / de Angel, Biagina Migliore / Charris, Jaime E. / Israel, Anita / Suárez-Roca, Heberto / López, Simon E. / Garrido, Maria R. / Cabrera, Elvia Victoria / Visbal, Gonzalo / Rosales, Cecire et al. | 2007
- 3245
-
Inhibition of 3(17)α-hydroxysteroid dehydrogenase (AKR1C21) by aldose reductase inhibitorsDhagat, Urmi / Endo, Satoshi / Hara, Akira / El-Kabbani, Ossama et al. | 2007
- 3245
-
Inhibition of 3(17)a-hydroxysteroid dehydrogenase (AKR1C21) by aldose reductase inhibitorsDhagat, U. / Endo, S. / Hara, A. / El-Kabbani, O. et al. | 2008
- 3255
-
Novel nitroheterocyclic hypoxic markers for solid tumor: Synthesis and biological evaluationZhu, Weiping / Dai, Min / Xu, Yufang / Qian, Xuhong et al. | 2007
- 3261
-
Synthesis, analgesic, anti-inflammatory, and antimicrobial activity of some novel pyrimido[4,5-b]quinolin-4-onesEl-Gazzar, Abdel-Rahman B.A. / El-Enany, Mervat M. / Mahmoud, Mahmoud N. et al. | 2007
- 3274
-
Synthesis of naphtho[2,3-a]phenoxazinium chlorides: Structure–activity relationships of these heterocycles and benzo[a]phenoxazinium chlorides as new antimicrobialsFrade, Vânia H.J. / Sousa, Maria J. / Moura, João C.V.P. / Gonçalves, M. Sameiro T. et al. | 2007
- 3283
-
Synthesis and biological evaluation of 2-alkylaminoethyl-1,1-bisphosphonic acids against Trypanosoma cruzi and Toxoplasma gondii targeting farnesyl diphosphate synthaseSzajnman, Sergio H. / Garcı´a Liñares, Guadalupe E. / Li, Zhu-Hong / Jiang, Cuiying / Galizzi, Melina / Bontempi, Esteban J. / Ferella, Marcela / Moreno, Silvia N.J. / Docampo, Roberto / Rodriguez, Juan B. et al. | 2007
- 3291
-
Pyrimidinone-peptoid hybrid molecules with distinct effects on molecular chaperone function and cell proliferationWright, Christine M. / Chovatiya, Raj J. / Jameson, Nora E. / Turner, David M. / Zhu, Guangyu / Werner, Stefan / Huryn, Donna M. / Pipas, James M. / Day, Billy W. / Wipf, Peter et al. | 2007
- 3302
-
Diazen-1-ium-1,2-diolated and nitrooxyethyl nitric oxide donor ester prodrugs of anti-inflammatory (E)-2-(aryl)-3-(4-methanesulfonylphenyl)acrylic acids: Synthesis, cyclooxygenase inhibition, and nitric oxide release studiesAbdellatif, Khaled R.A. / Chowdhury, Morshed Alam / Dong, Ying / Chen, Qiao-Hong / Knaus, Edward E. et al. | 2007
- 3309
-
Synthesis and structure–activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonistsShimada, Itsuro / Maeno, Kyoichi / Kondoh, Yutaka / Kaku, Hidetaka / Sugasawa, Keizo / Kimura, Yasuharu / Hatanaka, Ken-ichi / Naitou, Yuki / Wanibuchi, Fumikazu / Sakamoto, Shuichi et al. | 2007
- 3321
-
Synthesis and structure–activity relationships of thiadiazole-derivatives as potent and orally active peroxisome proliferator-activated receptors α/δ dual agonistsShen, Lan / Zhang, Yan / Wang, Aihua / Sieber-McMaster, Ellen / Chen, Xiaoli / Pelton, Patricia / Xu, June Z. / Yang, Maria / Zhu, Peifang / Zhou, Lubing et al. | 2007
- 3321
-
Synthesis and structure-activity relationships of thiadiazole-derivatives as potent and orally active peroxisome proliferator-activated receptors a/d dual agonistsShen, L. / Zhang, Y. / Wang, A. / Sieber-McMaster, E. / Chen, X. / Pelton, P. / Xu, J. Z. / Yang, M. / Zhu, P. / Zhou, L. et al. | 2008
- 3342
-
Oligo(tyrosine sulfate)s as heparin pentasaccharide mimic: Evaluation by surface noncovalent affinity mass spectrometryYamaguchi, Miyuki / Ohmori, Tsukasa / Sakata, Yoichi / Ueki, Masaaki et al. | 2007
- 3352
-
Improved synthesis of histone deacetylase inhibitors (HDIs) (MS-275 and CI-994) and inhibitory effects of HDIs alone or in combination with RAMBAs or retinoids on growth of human LNCaP prostate cancer cells and tumor xenograftsGediya, Lalji K. / Belosay, Aashvini / Khandelwal, Aakanksha / Purushottamachar, Puranik / Njar, Vincent C.O. et al. | 2007
- 3361
-
Synthesis of β- and γ-oxa isosteres of fosmidomycin and FR900098 as antimalarial candidatesHaemers, Timothy / Wiesner, Jochen / Gießmann, Dirk / Verbrugghen, Thomas / Hillaert, Ulrik / Ortmann, Regina / Jomaa, Hassan / Link, Andreas / Schlitzer, Martin / Van Calenbergh, Serge et al. | 2007
- 3361
-
Synthesis of b- and g-oxa isosteres of fosmidomycin and FR900098 as antimalarial candidatesHaemers, T. / Wiesner, J. / Giemann, D. / Verbrugghen, T. / Hillaert, U. / Ortmann, R. / Jomaa, H. / Link, A. / Schlitzer, M. / Van Calenbergh, S. et al. | 2008
- 3372
-
Thiahomoisocitrate: A highly potent inhibitor of homoisocitrate dehydrogenase involved in the α-aminoadipate pathwayYamamoto, Takashi / Eguchi, Tadashi et al. | 2007
- 3372
-
Thiahomoisocitrate: A highly potent inhibitor of homoisocitrate dehydrogenase involved in the a-aminoadipate pathwayYamamoto, T. / Eguchi, T. et al. | 2008
- 3377
-
Synthetic derivatives of the α- and β-amyrin triterpenes and their antinociceptive propertiesSoldi, Cristian / Pizzolatti, Moacir Geraldo / Luiz, Ana Paula / Marcon, Rodrigo / Meotti, Flavia Carla / Mioto, Letícia Adelia / Santos, Adair R.S. et al. | 2007
- 3377
-
Synthetic derivatives of the a- and b-amyrin triterpenes and their antinociceptive propertiesSoldi, C. / Pizzolatti, M. G. / Luiz, A. P. / Marcon, R. / Meotti, F. C. / Mioto, L. A. / Santos, A. R. et al. | 2008
- 3387
-
Structure and estrogenic activity of new lignans from Iryanthera lancifoliaMesa-Siverio, Dulce / Machín, Rubén P. / Estévez-Braun, Ana / Ravelo, Ángel. G. / Lock, Olga et al. | 2007
- 3395
-
QSAR modeling of the rodent carcinogenicity of nitrocompoundsHelguera, Aliuska Morales / Cordeiro, M. Natália D.S. / Pérez, Miguel Ángel Cabrera / Combes, Robert D. / González, Maykel Pérez et al. | 2007
- 3408
-
Antimycobacterial activities of novel 2-(sub)-3-fluoro/nitro-5,12-dihydro-5-oxobenzothiazolo[3,2-a]quinoline-6-carboxylic acidDinakaran, Murugesan / Senthilkumar, Palaniappan / Yogeeswari, Perumal / China, Arnab / Nagaraja, Valakunja / Sriram, Dharmarajan et al. | 2007
- 3419
-
Deoxygenated phosphorothioate inositol phosphate analogs: Synthesis, phosphatase stability, and binding affinityLiu, Xiaodan / Moody, Emily C. / Hecht, Stephen S. / Sturla, Shana J. et al. | 2007
- 3428
-
Synthesis and structure–activity relationship studies in peripheral benzodiazepine receptor ligands related to alpidemCappelli, Andrea / Giuliani, Germano / Valenti, Salvatore / Anzini, Maurizio / Vomero, Salvatore / Giorgi, Gianluca / Sogliano, Cristiana / Maciocco, Elisabetta / Biggio, Giovanni / Concas, Alessandra et al. | 2007
- 3438
-
A novel synthesis and pharmacological evaluation of a potential dopamine D1/D2 agonist: 1-Propyl-1,2,3,4,4a,5,10,10a-octahydrobenzo[g]quinoline-6,7-diolLiu, Danyang / Dijkstra, Durk / de Vries, Jan B. / Wikström, Håkan V. et al. | 2007
- 3445
-
Design, synthesis and cell growth inhibitory activity of a series of novel aminosubstituted xantheno[1,2-d]imidazoles in breast cancer cellsKostakis, Ioannis K. / Pouli, Nicole / Marakos, Panagiotis / Kousidou, Olga Ch. / Roussidis, Andreas / Tzanakakis, George N. / Karamanos, Nikos K. et al. | 2007
- 3456
-
3D-QSAR CoMFA studies on bis-coumarine analogues as urease inhibitors: A strategic design in anti-urease agentsZaheer-ul-Haq / Lodhi, M. Arif / Ahmad Nawaz, Sarfraz / Iqbal, Sajid / Mohammed Khan, Khalid / Rode, Bernd M. / Atta-ur-Rahman / Choudhary, M. Iqbal et al. | 2005
- 3462
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Corrigendum to “Virtual screening and bioassay study of novel inhibitors for dengue virus mRNA cap (nucleoside-2′O)-methyltransferase” [Bioorg. Med. Chem. 15 (2007) 7795–7802]Luzhkov, Victor B. / Selisko, Barbara / Nordqvist, Anneli / Peyrane, Frédéric / Decroly, Etienne / Alvarez, Karine / Karlen, Anders / Canard, Bruno / Åqvist, Johan et al. | 2007
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Corrigendum to "Virtual screening and bioassay study of novel inhibitors for dengue virus mRNA cap (nucleoside-2primeO)-methyltransferase" [Bioorg. Med. Chem. 15 (2007) 7795-7802]Luzhkov, V. B. / Selisko, B. / Nordqvist, A. / Peyrane, F. / Decroly, E. / Alvarez, K. / Karlen, A. / Canard, B. / angstqvist, J. et al. | 2008
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Instructions to contributors| 2008
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Editorial board| 2008