5-Chloro-2-thiophenyl-1,2,3-triazolylmethyldihydroquinolines as dual inhibitors of Mycobacterium tuberculosis and influenza virus: Synthesis and evaluation (English)
- New search for: Marvadi, Sandeep Kumar
- New search for: Krishna, Vagolu Siva
- New search for: Sinegubova, Ekaterina O.
- New search for: Volobueva, Alexandrina S.
- New search for: Esaulkova, Yana L.
- New search for: Muryleva, Anna A.
- New search for: Tentler, Dmitry G.
- New search for: Sriram, Dharmarajan
- New search for: Zarubaev, Vladimir V.
- New search for: Kantevari, Srinivas
- Further information on Kantevari, Srinivas:
- https://orcid.org/0000-0002-6837-5242
- New search for: Marvadi, Sandeep Kumar
- New search for: Krishna, Vagolu Siva
- New search for: Sinegubova, Ekaterina O.
- New search for: Volobueva, Alexandrina S.
- New search for: Esaulkova, Yana L.
- New search for: Muryleva, Anna A.
- New search for: Tentler, Dmitry G.
- New search for: Sriram, Dharmarajan
- New search for: Zarubaev, Vladimir V.
- New search for: Kantevari, Srinivas
In:
Bioorganic and Medicinal Chemistry Letters
;
29
, 18
;
2664-2669
;
2019
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ISSN:
- Article (Journal) / Electronic Resource
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Title:5-Chloro-2-thiophenyl-1,2,3-triazolylmethyldihydroquinolines as dual inhibitors of Mycobacterium tuberculosis and influenza virus: Synthesis and evaluation
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Contributors:Marvadi, Sandeep Kumar ( author ) / Krishna, Vagolu Siva ( author ) / Sinegubova, Ekaterina O. ( author ) / Volobueva, Alexandrina S. ( author ) / Esaulkova, Yana L. ( author ) / Muryleva, Anna A. ( author ) / Tentler, Dmitry G. ( author ) / Sriram, Dharmarajan ( author ) / Zarubaev, Vladimir V. ( author ) / Kantevari, Srinivas ( author )
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Published in:Bioorganic and Medicinal Chemistry Letters ; 29, 18 ; 2664-2669
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Publisher:
- New search for: Elsevier Ltd
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Publication date:2019-07-22
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Size:6 pages
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ISSN:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Keywords:
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Source:
Table of contents – Volume 29, Issue 18
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 2527
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Targeting TRAILIon, George Nicolae Daniel / Nitulescu, George Mihai / Popescu, Costin Ioan et al. | 2019
- 2535
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Applications of amide isosteres in medicinal chemistrySun, Shaoyi / Jia, Qi / Zhang, Zaihui et al. | 2019
- 2551
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Design, synthesis and biological evaluation of 2-(3,4-dimethoxyphenyl)-6 (1,2,3,6-tetrahydropyridin-4-yl)imidazo[1,2-a]pyridine analogues as antiproliferative agentsChitti, Surendar / Singireddi, SrinivasaRao / Santosh Kumar Reddy, Pochana / Trivedi, Prakruti / Bobde, Yamini / Kumar, Chandan / Rangan, Krishnan / Ghosh, Balaram / Sekhar, Kondapalli Venkata Gowri Chandra et al. | 2019
- 2559
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Discovery of small molecule inhibitors of human uridine-cytidine kinase 2 by high-throughput screeningOkesli-Armlovich, Ayse / Gupta, Amita / Jimenez, Marta / Auld, Douglas / Liu, Qi / Bassik, Michael C. / Khosla, Chaitan et al. | 2019
- 2565
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Potent HIV-1 protease inhibitors incorporating squaramide-derived P2 ligands: Design, synthesis, and biological evaluationGhosh, Arun K. / Williams, Jacqueline N. / Kovela, Satish / Takayama, Jun / Simpson, Hannah M. / Walters, D. Eric / Hattori, Shin-ichiro / Aoki, Manabu / Mitsuya, Hiroaki et al. | 2019
- 2571
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Phosphoramidate derivates as controlled-release prodrugs of l-DopaOlatunji, Feyisola P. / Kesic, Brittany N. / Choy, Cindy J. / Berkman, Clifford E. et al. | 2019
- 2575
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Design of selective PI3Kδ inhibitors using an iterative scaffold-hopping workflowFradera, Xavier / Methot, Joey L. / Achab, Abdelghani / Christopher, Matthew / Altman, Michael D. / Zhou, Hua / McGowan, Meredeth A. / Kattar, Sam D. / Wilson, Kevin / Garcia, Yudith et al. | 2019
- 2581
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Exploring hydroxamic acid inhibitors of HDAC1 and HDAC2 using small molecule tools and molecular or homology modellingDaniel, Lydia / Gotsbacher, Michael P. / Richardson-Sanchez, Tomas / Tieu, William / Codd, Rachel et al. | 2019
- 2587
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Synthesis and in vitro anticancer activity of new gemcitabine-nucleoside analogue dimers containing methyltriazole or ester-methyltriazole linkerTrznadel, Roksana / Singh, Aleksandra / Kleczewska, Natalia / Liberska, Joanna / Ruszkowski, Piotr / Celewicz, Lech et al. | 2019
- 2595
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Discovery of 1,8-disubstituted-[1,2,3]triazolo[4,5-c]quinoline derivatives as a new class of Hippo signaling pathway inhibitorsQiao, Jingxin / Lin, Guifeng / Xia, Anjie / Xiang, Zhiyu / Chen, Pei / Zhang, Guo / Li, Linli / Yang, Shengyong et al. | 2019
- 2604
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Synthesis of N-arylindazole-3-carboxamide and N-benzoylindazole derivatives and their evaluation against α-MSH-stimulated melanogenesisArepalli, Sateesh Kumar / Lee, Chaerim / Jung, Jae-Kyung / Kim, Youngsoo / Lee, Kiho / Lee, Heesoon et al. | 2019
- 2609
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A glycal-based photoaffinity probe that enriches sialic acid binding proteinsThuy-Boun, Peter S. / Wolan, Dennis W. et al. | 2019
- 2613
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Discovery of novel PTHR1 antagonists: Design, synthesis, and structure activity relationshipsArai, Yoshikazu / Kiyotsuka, Yohei / Shimada, Kousei / Oyama, Kazunori / Izumi, Masanori et al. | 2019
- 2617
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The synthesis of a novel Crizotinib heptamethine cyanine dye conjugate that potentiates the cytostatic and cytotoxic effects of Crizotinib in patient-derived glioblastoma cell linesChoi, Peter J. / Cooper, Elizabeth / Schweder, Patrick / Mee, Edward / Faull, Richard / Denny, William A. / Dragunow, Mike / Park, Thomas I.-H. / Jose, Jiney et al. | 2019
- 2622
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An investigation of targeted inhibition of transcription factor activity with pyrrole imidazole polyamide (PA) in chronic myeloid leukemia (CML) blast crisis cellsHayatigolkhatmi, K. / Padroni, G. / Su, W. / Fang, L. / Gómez-Castañeda, E. / Hsieh, Y.C. / Jackson, L. / Pellicano, F. / Burley, G.A. / Jørgensen, H.G. et al. | 2019
- 2626
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A fragment-like approach to PYCR1 inhibitionMilne, Kirsty / Sun, Jianhui / Zaal, Esther A. / Mowat, Jenna / Celie, Patrick H.N. / Fish, Alexander / Berkers, Celia R. / Forlani, Giuseppe / Loayza-Puch, Fabricio / Jamieson, Craig et al. | 2019
- 2632
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Synthesis and biological evaluation of 7-methoxy-1-(3,4,5-trimethoxyphenyl)-4,5-dihydro-2H-benzo[e]indazoles as new colchicine site inhibitorsJiang, Junhang / Zhang, Qingsen / Guo, Jiapeng / Fang, Shaoyu / Zhou, Ruolan / Zhu, Ju / Chen, Xin / Zhou, Youjun / Zheng, Canhui et al. | 2019
- 2635
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Ciprofloxacin-1,2,3-triazole-isatin hybrids tethered via amide: Design, synthesis, and in vitro anti-mycobacterial activity evaluationChen, Rongxing / Zhang, Hao / Ma, Tianwei / Xue, Huarui / Miao, Zhong / Chen, Liyan / Shi, Xiangkui et al. | 2019
- 2638
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Anti-tumor activity evaluation of novel tubulin and HDAC dual-targeting inhibitorsWang, Baolei / Chen, Xuehong / Gao, Jianjun / Su, Li / Zhang, Li / Xu, Hongwei / Luan, Yepeng et al. | 2019
- 2646
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A highly selective and sensitive 1,8-naphthalimide-based fluorescent sensor for Zn2+ imaging in living cellsLiu, Daying / Zhao, Ye / Shi, Jun / Zhu, Hualing / Zhang, Tingting / Qi, Pengpeng / Chen, Jiatong / Yang, Guangming / He, Huarui et al. | 2019
- 2650
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Synthesis and evaluation of 2′H-spiro[cyclohexane-1,3′-imidazo[1,5-a]pyridine]-1′,5′-dione derivatives as Mnk inhibitorsAbdelaziz, Ahmed M. / Basnet, Sunita K.C. / Islam, Saiful / Li, Manjun / Tadesse, Solomon / Albrecht, Hugo / Gerber, Cobus / Yu, Mingfeng / Wang, Shudong et al. | 2019
- 2655
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Essential structure of orexin 1 receptor antagonist YNT-707, Part IV: The role of D-ring in 4,5-epoxymorphinan on the orexin 1 receptor antagonistic activitySaitoh, Tsuyoshi / Seki, Kazunori / Nakajima, Ryo / Yamamoto, Naoshi / Kutsumura, Noriki / Nagumo, Yasuyuki / Irukayama-Tomobe, Yoko / Ogawa, Yasuhiro / Ishikawa, Yukiko / Tanimura, Ryuji et al. | 2019
- 2659
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Inhibition of β-amyloid–induced neurotoxicity by planar analogues of procyanidin B3Mizuno, Mirei / Mori, Kazunori / Misawa, Takashi / Takaki, Takashi / Demizu, Yosuke / Shibanuma, Motoko / Fukuhara, Kiyoshi et al. | 2019
- 2664
-
5-Chloro-2-thiophenyl-1,2,3-triazolylmethyldihydroquinolines as dual inhibitors of Mycobacterium tuberculosis and influenza virus: Synthesis and evaluationMarvadi, Sandeep Kumar / Krishna, Vagolu Siva / Sinegubova, Ekaterina O. / Volobueva, Alexandrina S. / Esaulkova, Yana L. / Muryleva, Anna A. / Tentler, Dmitry G. / Sriram, Dharmarajan / Zarubaev, Vladimir V. / Kantevari, Srinivas et al. | 2019
- 2670
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Further exploration of an N-aryl phenoxyethoxy pyridinone-based series of mGlu3 NAMs: Challenging SAR, enantiospecific activity and in vivo efficacyYamada, Yosuke / Yohn, Samantha E. / Gilliland, Kristen / Loch, Mathew T. / Schulte, Michael L. / Rodriguez, Alice L. / Blobaum, Anna L. / Niswender, Colleen M. / Conn, P. Jeffrey / Lindsley, Craig W. et al. | 2019
- 2675
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Incorporation of privileged structures into 3-O-β-chacotriosyl ursolic acid can enhance inhibiting the entry of the H5N1 virusLi, Hui / Chen, Lizhu / Li, Sumei / Liao, Yixian / Wang, Lei / Liu, Zhihao / Liu, Shuwen / Song, Gaopeng et al. | 2019
- 2681
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Design, synthesis and anticancer activity of constrained sphingolipid-phenoxazine/phenothiazine hybrid constructs targeting protein phosphatase 2AGarsi, Jean-Baptiste / Vece, Vito / Sernissi, Lorenzo / Auger-Morin, Catherine / Hanessian, Stephen / McCracken, Alison N. / Selwan, Elizabeth / Ramirez, Cuauhtemoc / Dahal, Amogha / Romdhane, Nadine Ben et al. | 2019
- 2686
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Incorporation of a chiral gem-disubstituted nitrogen heterocycle yields an oxazolidinone antibiotic with reduced mitochondrial toxicitySun, Alexander W. / Bulterys, Philip L. / Bartberger, Michael D. / Jorth, Peter A. / O'Boyle, Brendan M. / Virgil, Scott C. / Miller, Jeff F. / Stoltz, Brian M. et al. | 2019
- 2690
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Design, synthesis, and evaluation of N-(4-(4-phenyl piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamides as selective dopamine D3 receptor ligandsChen, Peng-Jen / Taylor, Michelle / Griffin, Suzy A. / Amani, Armaghan / Hayatshahi, Hamed / Korzekwa, Kenneth / Ye, Min / Mach, Robert H. / Liu, Jin / Luedtke, Robert R. et al. | 2019
- 2695
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Anti-tubercular activity of novel 4-anilinoquinolines and 4-anilinoquinazolinesAsquith, Christopher R.M. / Fleck, Neil / Torrice, Chad D. / Crona, Daniel J. / Grundner, Christoph / Zuercher, William J. et al. | 2019
- 2700
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Discovery and optimization of pyridyl-cycloalkyl-carboxylic acids as inhibitors of microsomal prostaglandin E synthase-1 for the treatment of endometriosisKoppitz, Marcus / Bräuer, Nico / Ter Laak, Antonius / Irlbacher, Horst / Rotgeri, Andrea / Coelho, Anne-Marie / Walter, Daryl / Steinmeyer, Andreas / Zollner, Thomas M. / Peters, Michaele et al. | 2019
- I
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Graphical abstract TOC continued| 2019
- IBC
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Graphical abstract TOC| 2019
- ii
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Editorial Board| 2019